Compound & Protein features
Download training file (ECFP)
Download training file (Checkmol)
Download training file (Checkmol+AC10)
Download training file (Checkmol+AC10+ECFP)
Download example training file (ECFP)

Active :  <=  10 μM      Inactive :  >=  20 μM

Kinases: 131
Compounds: 56,690
Pairs: 147,583
Kinase Family Group Uniprot Active_num Inactive_num Download (ECFP features)
PKChPKCAGCP24723168168Image
DLKMLKTKLQ12852519519Image
PLK4PLKOtherO00444106106Image
ZAP70SykTKP43403163163Image
FGFR3FGFRTKP22607427427Image
FMSPDGFRTKP07333700700Image
FLT4VEGFRTKP35916222222Image
COTSTE-UniqueSTEP41279132132Image
Erk2MAPKCMGCP28482901901Image
FGFR2FGFRTKP21802223223Image
TTKTTKOtherP33981311311Image
HCKSrcTKP08631274274Image
PIM2PIMCAMKQ9P1W9930930Image
IGF1RInsRTKP0806912541254Image
IRAK4IRAKTKLQ9NWZ3291291Image
p70S6KRSKAGCP23443554554Image
CHK2RAD53CAMKO96017214214Image
PKCePKCAGCQ02156252252Image
FLT1VEGFRTKP17948534534Image
NIKSTE-UniqueSTEQ99558469469Image
JAK1JakTKP2345813141314Image
Wee1WEEOtherP30291234234Image
PIM3PIMCAMKQ86V86634634Image
MERAxlTKQ12866160160Image
TYRO3AxlTKQ06418171171Image
ACKAckTKQ07912358358Image
PKCbPKCAGCP05771450450Image
CDK9CDKCMGCP50750374374Image
FGFR1FGFRTKP11362786786Image
PKCaPKCAGCP17252578578Image
JAK2JakTKO6067422442244Image
TYK2JakTKP29597394394Image
TGFbR1STKRTKLP36897530530Image
PKCtPKCAGCQ04759450450Image
CK1dCK1CK1P48730131131Image
INSRInsRTKP06213443443Image
SYKSykTKP4340516741674Image
FLT3PDGFRTKP36888995995Image
CDC7CDC7OtherO00311252252Image
BTKTecTKQ06187525525Image
KDRVEGFRTKP3596840492699Image
PKCdPKCAGCQ05655453453Image
CDK7CDKCMGCP50613100100Image
METMetTKP0858120592059Image
PIM1PIMCAMKP1130914201420Image
JAK3JakTKP5233314381438Image
FAKFAKTKQ05397834834Image
ErbB2EGFRTKP04626979979Image
KITPDGFRTKP10721659659Image
JNK1MAPKCMGCP45983972972Image
p38aMAPKCMGCQ1653927232723Image
PLK3PLKOtherQ9H4B48383Image
p38bMAPKCMGCQ15759125125Image
MAPKAPK2MAPKAPKCAMKP49137566566Image
ALKALKTKQ9UM73743743Image
CHK1CAMKLCAMKO1475713371337Image
BRKSrcTKQ13882106106Image
TRKATrkTKP04629928928Image
AXLAxlTKP30530172172Image
CDK6CDKCMGCQ00534228228Image
SRCSrcTKP1293119301930Image
AKT1AktAGCP3174916491649Image
RETRetTKP07949339339Image
LYNSrcTKP07948191191Image
CaMK2dCAMK2CAMKQ135579595Image
PDGFRbPDGFRTKP09619693693Image
LIMK1LISKTKLP53667184184Image
Erk1MAPKCMGCP273618282Image
MAP2K1STE7STEQ02750490490Image
PYK2FAKTKQ14289154154Image
EphB4EphTKP54760307307Image
AurBAurOtherQ96GD410921092Image
YESSrcTKP07947101101Image
PKCgPKCAGCP05129145145Image
LRRK2LRRKTKLQ5S007601601Image
ROCK2DMPKAGCO75116996996Image
NEK1NEKOtherQ96PY6192192Image
JNK2MAPKCMGCP45984410410Image
PKD1PKDCAMKQ15139101101Image
CK2a2CK2CMGCP19784145145Image
CDK4CDKCMGCP11802821821Image
RAF1RAFTKLP04049457457Image
CDK2CDKCMGCP2494110521052Image
BRAFRAFTKLP1505613991399Image
PDGFRaPDGFRTKP16234238238Image
LCKSrcTKP0623911121112Image
EGFREGFRTKP0053333072462Image
ROCK1DMPKAGCQ13464411411Image
ITKTecTKQ08881489489Image
CDC2CDKCMGCP06493734734Image
FYNSrcTKP06241150150Image
DYRK1ADYRKCMGCQ13627278278Image
GSK3BGSKCMGCP4984114981498Image
PKCiPKCAGCP41743394394Image
TNIKSTE20STEQ9UKE5126126Image
MAP3K5STE11STEQ996839696Image
PDK1PDK1AGCO15530544544Image
MNK2MAPKAPKCAMKQ9HBH9211211Image
TIE2TieTKQ02763475475Image
LIMK2LISKTKLP53671159159Image
ABL1AblTKP0051910921092Image
PAK1STE20STEQ13153149149Image
HGKSTE20STEO958199696Image
CDK5CDKCMGCQ00535128128Image
PKACaPKAAGCP176128888Image
MNK1MAPKAPKCAMKQ9BUB59090Image
IRE1IREOtherO75460239239Image
PLK1PLKOtherP53350428428Image
PAK4STE20STEO96013138138Image
AurAAurOtherO1496518021802Image
GSK3AGSKCMGCP49840214214Image
RPS6KA3RSKAGCP51812250250Image
CLK4CLKCMGCQ9HAZ1124124Image
CLK1CLKCMGCP49759246246Image
CDK8CDKCMGCP49336118118Image
TRKBTrkTKQ16620127127Image
DYRK1BDYRKCMGCQ9Y463162162Image
JNK3MAPKCMGCP53779679679Image
IKKeIKKOtherQ14164146146Image
IKKbIKKOtherO14920650650Image
ILKMLKTKLQ13418130130Image
PBKTOPKOtherQ96KB58383Image
TBK1IKKOtherQ9UHD2183183Image
AKT2AktAGCP31751634634Image
AKT3AktAGCQ9Y243162162Image
TAK1MLKTKLO43318102102Image
BARK1GRKAGCP25098139139Image
IKKaIKKOtherO15111224224Image
DYRK2DYRKCMGCQ926308686Image
CK2a1CK2CMGCP68400403403Image
MELKCAMKLCAMKQ14680614614Image