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ECFP
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Compound features (1048)
Protein features (1700)
Compound & Protein features
Download independent file (ECFP)
Download independent file (Checkmol)
Download independent file (Checkmol+AC10)
Download independent file (Checkmol+AC10+ECFP)
Download example independent file (ECFP)
Active : <= 10 μM Inactive : >= 20 μM
Kinases: 131
Compounds: 38,468
Pairs: 57,383
Kinase
Family
Group
Uniprot
Active_num
Inactive_num
Download (ECFP features)
PKCh
PKC
AGC
P24723
168
168
DLK
MLK
TKL
Q12852
519
519
PLK4
PLK
Other
O00444
106
106
ZAP70
Syk
TK
P43403
163
163
FGFR3
FGFR
TK
P22607
427
427
FMS
PDGFR
TK
P07333
700
700
FLT4
VEGFR
TK
P35916
222
222
COT
STE-Unique
STE
P41279
132
132
Erk2
MAPK
CMGC
P28482
901
901
FGFR2
FGFR
TK
P21802
223
223
TTK
TTK
Other
P33981
311
311
HCK
Src
TK
P08631
274
274
PIM2
PIM
CAMK
Q9P1W9
930
930
IGF1R
InsR
TK
P08069
1254
1254
IRAK4
IRAK
TKL
Q9NWZ3
291
291
p70S6K
RSK
AGC
P23443
554
554
CHK2
RAD53
CAMK
O96017
214
214
PKCe
PKC
AGC
Q02156
252
252
FLT1
VEGFR
TK
P17948
534
534
NIK
STE-Unique
STE
Q99558
469
469
JAK1
Jak
TK
P23458
1314
1314
Wee1
WEE
Other
P30291
234
234
PIM3
PIM
CAMK
Q86V86
634
634
MER
Axl
TK
Q12866
160
160
TYRO3
Axl
TK
Q06418
171
171
ACK
Ack
TK
Q07912
358
358
PKCb
PKC
AGC
P05771
450
450
CDK9
CDK
CMGC
P50750
374
374
FGFR1
FGFR
TK
P11362
786
786
PKCa
PKC
AGC
P17252
578
578
JAK2
Jak
TK
O60674
2244
2244
TYK2
Jak
TK
P29597
394
394
TGFbR1
STKR
TKL
P36897
530
530
PKCt
PKC
AGC
Q04759
450
450
CK1d
CK1
CK1
P48730
131
131
INSR
InsR
TK
P06213
443
443
SYK
Syk
TK
P43405
1674
1674
FLT3
PDGFR
TK
P36888
995
995
CDC7
CDC7
Other
O00311
252
252
BTK
Tec
TK
Q06187
525
525
KDR
VEGFR
TK
P35968
4049
2699
PKCd
PKC
AGC
Q05655
453
453
CDK7
CDK
CMGC
P50613
100
100
MET
Met
TK
P08581
2059
2059
PIM1
PIM
CAMK
P11309
1420
1420
JAK3
Jak
TK
P52333
1438
1438
FAK
FAK
TK
Q05397
834
834
ErbB2
EGFR
TK
P04626
979
979
KIT
PDGFR
TK
P10721
659
659
JNK1
MAPK
CMGC
P45983
972
972
p38a
MAPK
CMGC
Q16539
2723
2723
PLK3
PLK
Other
Q9H4B4
83
83
p38b
MAPK
CMGC
Q15759
125
125
MAPKAPK2
MAPKAPK
CAMK
P49137
566
566
ALK
ALK
TK
Q9UM73
743
743
CHK1
CAMKL
CAMK
O14757
1337
1337
BRK
Src
TK
Q13882
106
106
TRKA
Trk
TK
P04629
928
928
AXL
Axl
TK
P30530
172
172
CDK6
CDK
CMGC
Q00534
228
228
SRC
Src
TK
P12931
1930
1930
AKT1
Akt
AGC
P31749
1649
1649
RET
Ret
TK
P07949
339
339
LYN
Src
TK
P07948
191
191
CaMK2d
CAMK2
CAMK
Q13557
95
95
PDGFRb
PDGFR
TK
P09619
693
693
LIMK1
LISK
TKL
P53667
184
184
Erk1
MAPK
CMGC
P27361
82
82
MAP2K1
STE7
STE
Q02750
490
490
PYK2
FAK
TK
Q14289
154
154
EphB4
Eph
TK
P54760
307
307
AurB
Aur
Other
Q96GD4
1092
1092
YES
Src
TK
P07947
101
101
PKCg
PKC
AGC
P05129
145
145
LRRK2
LRRK
TKL
Q5S007
601
601
ROCK2
DMPK
AGC
O75116
996
996
NEK1
NEK
Other
Q96PY6
192
192
JNK2
MAPK
CMGC
P45984
410
410
PKD1
PKD
CAMK
Q15139
101
101
CK2a2
CK2
CMGC
P19784
145
145
CDK4
CDK
CMGC
P11802
821
821
RAF1
RAF
TKL
P04049
457
457
CDK2
CDK
CMGC
P24941
1052
1052
BRAF
RAF
TKL
P15056
1399
1399
PDGFRa
PDGFR
TK
P16234
238
238
LCK
Src
TK
P06239
1112
1112
EGFR
EGFR
TK
P00533
3307
2462
ROCK1
DMPK
AGC
Q13464
411
411
ITK
Tec
TK
Q08881
489
489
CDC2
CDK
CMGC
P06493
734
734
FYN
Src
TK
P06241
150
150
DYRK1A
DYRK
CMGC
Q13627
278
278
GSK3B
GSK
CMGC
P49841
1498
1498
PKCi
PKC
AGC
P41743
394
394
TNIK
STE20
STE
Q9UKE5
126
126
MAP3K5
STE11
STE
Q99683
96
96
PDK1
PDK1
AGC
O15530
544
544
MNK2
MAPKAPK
CAMK
Q9HBH9
211
211
TIE2
Tie
TK
Q02763
475
475
LIMK2
LISK
TKL
P53671
159
159
ABL1
Abl
TK
P00519
1092
1092
PAK1
STE20
STE
Q13153
149
149
HGK
STE20
STE
O95819
96
96
CDK5
CDK
CMGC
Q00535
128
128
PKACa
PKA
AGC
P17612
88
88
MNK1
MAPKAPK
CAMK
Q9BUB5
90
90
IRE1
IRE
Other
O75460
239
239
PLK1
PLK
Other
P53350
428
428
PAK4
STE20
STE
O96013
138
138
AurA
Aur
Other
O14965
1802
1802
GSK3A
GSK
CMGC
P49840
214
214
RPS6KA3
RSK
AGC
P51812
250
250
CLK4
CLK
CMGC
Q9HAZ1
124
124
CLK1
CLK
CMGC
P49759
246
246
CDK8
CDK
CMGC
P49336
118
118
TRKB
Trk
TK
Q16620
127
127
DYRK1B
DYRK
CMGC
Q9Y463
162
162
JNK3
MAPK
CMGC
P53779
679
679
IKKe
IKK
Other
Q14164
146
146
IKKb
IKK
Other
O14920
650
650
ILK
MLK
TKL
Q13418
130
130
PBK
TOPK
Other
Q96KB5
83
83
TBK1
IKK
Other
Q9UHD2
183
183
AKT2
Akt
AGC
P31751
634
634
AKT3
Akt
AGC
Q9Y243
162
162
TAK1
MLK
TKL
O43318
102
102
BARK1
GRK
AGC
P25098
139
139
IKKa
IKK
Other
O15111
224
224
DYRK2
DYRK
CMGC
Q92630
86
86
CK2a1
CK2
CMGC
P68400
403
403
MELK
CAMKL
CAMK
Q14680
614
614