P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Ki |
- |
- |
- |
P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
IC50 |
- |
- |
- |
P23975 |
BXGT008935 |
Sodium-dependent noradrenaline transporter |
reviewed |
Transporter |
SLC6A2 |
IC50 |
- |
- |
- |
P30411 |
BXGT009424 |
B2 bradykinin receptor |
reviewed |
G-protein coupled receptor |
BDKRB2 |
Ki |
- |
- |
- |
P41597 |
BXGT010268 |
C-C chemokine receptor type 2 |
reviewed |
- |
CCR2 |
Ki |
- |
- |
- |
P25025 |
BXGT009006 |
C-X-C chemokine receptor type 2 |
reviewed |
G-protein coupled receptor |
CXCR2 |
IC50 |
- |
- |
- |
P05181 |
BXGT006337 |
Cytochrome P450 2E1 |
reviewed |
- |
CYP2E1 |
Ki |
- |
- |
- |
P29477 |
BXGT009355 |
Nitric oxide synthase, inducible |
reviewed |
- |
Nos2 |
Ki |
- |
- |
- |
P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
Ki |
- |
- |
- |
P21452 |
BXGT008653 |
Substance-K receptor |
reviewed |
G-protein coupled receptor |
TACR2 |
Ki |
- |
- |
- |
P11229 |
BXGT007676 |
Muscarinic acetylcholine receptor M1 |
reviewed |
G-protein coupled receptor |
CHRM1 |
Ki |
- |
- |
- |
P20309 |
BXGT008562 |
Muscarinic acetylcholine receptor M3 |
reviewed |
G-protein coupled receptor |
CHRM3 |
Ki |
- |
- |
- |
P35372 |
BXGT009823 |
Mu-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRM1 |
IC50 |
- |
- |
- |
P08246 |
BXGT006756 |
Neutrophil elastase |
reviewed |
Enzyme |
ELANE |
Ki |
- |
- |
- |
P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
IC50 |
- |
- |
- |
Q690N0 |
BXGT016199 |
Progesterone receptor |
unreviewed |
- |
PGR |
Ki |
- |
- |
- |
P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
Ki |
- |
- |
- |
P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
IC50 |
- |
- |
- |
P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
- |
- |
- |
P17948 |
BXGT008358 |
Vascular endothelial growth factor receptor 1 |
reviewed |
Kinase |
FLT1 |
IC50 |
- |
- |
- |
P11229 |
BXGT007676 |
Muscarinic acetylcholine receptor M1 |
reviewed |
G-protein coupled receptor |
CHRM1 |
IC50 |
- |
- |
- |
P29476 |
BXGT009354 |
Nitric oxide synthase, brain |
reviewed |
- |
Nos1 |
Ki |
- |
- |
- |
O76074 |
BXGT005174 |
cGMP-specific 3',5'-cyclic phosphodiesterase |
reviewed |
- |
PDE5A |
IC50 |
- |
- |
- |
Q690N0 |
BXGT016199 |
Progesterone receptor |
unreviewed |
- |
PGR |
IC50 |
- |
- |
- |
P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
IC50 |
- |
- |
- |
P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
Ki |
- |
- |
- |
P21554 |
BXGT008662 |
Cannabinoid receptor 1 |
reviewed |
G-protein coupled receptor |
CNR1 |
Ki |
- |
- |
- |
P51681 |
BXGT010878 |
C-C chemokine receptor type 5 |
reviewed |
G-protein coupled receptor |
CCR5 |
Ki |
- |
- |
- |
P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
IC50 |
- |
- |
- |
P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Ki |
- |
- |
- |
P15127 |
BXGT008085 |
Insulin receptor |
reviewed |
- |
Insr |
IC50 |
- |
- |
- |
P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
Ki |
- |
- |
- |
P33032 |
BXGT009689 |
Melanocortin receptor 5 |
reviewed |
G-protein coupled receptor |
MC5R |
IC50 |
- |
- |
- |
P08912 |
BXGT006840 |
Muscarinic acetylcholine receptor M5 |
reviewed |
G-protein coupled receptor |
CHRM5 |
Ki |
- |
- |
- |
P49146 |
BXGT010681 |
Neuropeptide Y receptor type 2 |
reviewed |
G-protein coupled receptor |
NPY2R |
Ki |
- |
- |
- |
P41143 |
BXGT010223 |
Delta-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRD1 |
IC50 |
- |
- |
- |
P25105 |
BXGT009021 |
Platelet-activating factor receptor |
reviewed |
G-protein coupled receptor |
PTAFR |
IC50 |
- |
- |
- |
P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
IC50 |
- |
- |
- |
P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
- |
- |
- |
P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
- |
- |
- |
P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
IC50 |
- |
- |
- |
P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
- |
- |
- |
P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Ki |
- |
- |
- |
P21452 |
BXGT008653 |
Substance-K receptor |
reviewed |
G-protein coupled receptor |
TACR2 |
IC50 |
- |
- |
- |
P17948 |
BXGT008358 |
Vascular endothelial growth factor receptor 1 |
reviewed |
Kinase |
FLT1 |
Ki |
- |
- |
- |
P32241 |
BXGT009613 |
Vasoactive intestinal polypeptide receptor 1 |
reviewed |
G-protein coupled receptor |
VIPR1 |
IC50 |
- |
- |
- |
P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Ki |
- |
- |
- |
P41143 |
BXGT010223 |
Delta-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRD1 |
Ki |
- |
- |
- |
P12822 |
BXGT007850 |
Angiotensin-converting enzyme |
reviewed |
- |
ACE |
IC50 |
- |
- |
- |
P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
Ki |
- |
- |
- |
Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
Ki |
- |
- |
- |
Q08209 |
BXGT012968 |
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform |
reviewed |
- |
PPP3CA |
IC50 |
- |
- |
- |
P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
Ki |
- |
- |
- |
P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
IC50 |
- |
- |
- |
P08575 |
BXGT006793 |
Receptor-type tyrosine-protein phosphatase C |
reviewed |
Enzyme |
PTPRC |
Ki |
- |
- |
- |
O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
Ki |
- |
- |
- |
P31645 |
BXGT009558 |
Sodium-dependent serotonin transporter |
reviewed |
Transporter |
SLC6A4 |
Ki |
- |
- |
- |
Q99720 |
BXGT019955 |
Sigma non-opioid intracellular receptor 1 |
reviewed |
- |
SIGMAR1 |
IC50 |
- |
- |
- |
P25929 |
BXGT009078 |
Neuropeptide Y receptor type 1 |
reviewed |
G-protein coupled receptor |
NPY1R |
Ki |
- |
- |
- |
P08311 |
BXGT006762 |
Cathepsin G |
reviewed |
Enzyme |
CTSG |
Ki |
- |
- |
- |
Q08209 |
BXGT012968 |
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform |
reviewed |
- |
PPP3CA |
Ki |
- |
- |
- |
Q99720 |
BXGT019955 |
Sigma non-opioid intracellular receptor 1 |
reviewed |
- |
SIGMAR1 |
Ki |
- |
- |
- |
P24557 |
BXGT008976 |
Thromboxane-A synthase |
reviewed |
- |
TBXAS1 |
Ki |
- |
- |
- |
P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Ki |
- |
- |
- |
Q01959 |
BXGT012624 |
Sodium-dependent dopamine transporter |
reviewed |
Transporter |
SLC6A3 |
IC50 |
- |
- |
- |
P25101 |
BXGT009018 |
Endothelin-1 receptor |
reviewed |
G-protein coupled receptor |
EDNRA |
IC50 |
- |
- |
- |
Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
- |
- |
- |
P41968 |
BXGT010275 |
Melanocortin receptor 3 |
reviewed |
G-protein coupled receptor |
MC3R |
Ki |
- |
- |
- |
P29477 |
BXGT009355 |
Nitric oxide synthase, inducible |
reviewed |
- |
Nos2 |
IC50 |
- |
- |
- |
P31645 |
BXGT009558 |
Sodium-dependent serotonin transporter |
reviewed |
Transporter |
SLC6A4 |
IC50 |
- |
- |
- |
P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
- |
- |
- |
P50052 |
BXGT010768 |
Type-2 angiotensin II receptor |
reviewed |
G-protein coupled receptor |
AGTR2 |
Ki |
- |
- |
- |
P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
IC50 |
- |
- |
- |
P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
IC50 |
- |
- |
- |
Q01959 |
BXGT012624 |
Sodium-dependent dopamine transporter |
reviewed |
Transporter |
SLC6A3 |
Ki |
- |
- |
- |
P20781 |
BXGT008598 |
Glycine receptor subunit beta |
reviewed |
- |
Glrb |
IC50 |
- |
- |
- |
P07727 |
BXGT006662 |
Glycine receptor subunit alpha-1 |
reviewed |
- |
Glra1 |
IC50 |
- |
- |
- |
P24524 |
BXGT008974 |
Glycine receptor subunit alpha-3 |
reviewed |
- |
Glra3 |
IC50 |
- |
- |
- |
P22771 |
BXGT008806 |
Glycine receptor subunit alpha-2 |
reviewed |
- |
Glra2 |
IC50 |
- |
- |
- |
P15127 |
BXGT008085 |
Insulin receptor |
reviewed |
- |
Insr |
Ki |
- |
- |
- |
P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
IC50 |
- |
- |
- |
P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
IC50 |
- |
- |
- |
P37288 |
BXGT009977 |
Vasopressin V1a receptor |
reviewed |
G-protein coupled receptor |
AVPR1A |
Ki |
- |
- |
- |
P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Ki |
- |
- |
- |
P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
IC50 |
- |
- |
- |
P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
- |
- |
- |
P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
Potency |
'=' |
5623 |
nM |
P41968 |
BXGT010275 |
Melanocortin receptor 3 |
reviewed |
G-protein coupled receptor |
MC3R |
IC50 |
- |
- |
- |
P32245 |
BXGT009614 |
Melanocortin receptor 4 |
reviewed |
G-protein coupled receptor |
MC4R |
Ki |
- |
- |
- |
Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
IC50 |
- |
- |
- |
P08575 |
BXGT006793 |
Receptor-type tyrosine-protein phosphatase C |
reviewed |
Enzyme |
PTPRC |
IC50 |
- |
- |
- |
P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
Ki |
- |
- |
- |
P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
IC50 |
- |
- |
- |
P08246 |
BXGT006756 |
Neutrophil elastase |
reviewed |
Enzyme |
ELANE |
IC50 |
- |
- |
- |
P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
Ki |
- |
- |
- |
P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
IC50 |
- |
- |
- |
P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
Ki |
- |
- |
- |
P24557 |
BXGT008976 |
Thromboxane-A synthase |
reviewed |
- |
TBXAS1 |
IC50 |
- |
- |
- |
P32241 |
BXGT009613 |
Vasoactive intestinal polypeptide receptor 1 |
reviewed |
G-protein coupled receptor |
VIPR1 |
Ki |
- |
- |
- |
P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
Ki |
- |
- |
- |
P15207 |
BXGT008096 |
Androgen receptor |
reviewed |
- |
Ar |
IC50 |
- |
- |
- |
P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
IC50 |
- |
- |
- |
P20309 |
BXGT008562 |
Muscarinic acetylcholine receptor M3 |
reviewed |
G-protein coupled receptor |
CHRM3 |
IC50 |
- |
- |
- |
P08173 |
BXGT006738 |
Muscarinic acetylcholine receptor M4 |
reviewed |
G-protein coupled receptor |
CHRM4 |
Ki |
- |
- |
- |
P08912 |
BXGT006840 |
Muscarinic acetylcholine receptor M5 |
reviewed |
G-protein coupled receptor |
CHRM5 |
IC50 |
- |
- |
- |
P25105 |
BXGT009021 |
Platelet-activating factor receptor |
reviewed |
G-protein coupled receptor |
PTAFR |
Ki |
- |
- |
- |
P08311 |
BXGT006762 |
Cathepsin G |
reviewed |
Enzyme |
CTSG |
IC50 |
- |
- |
- |
P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
IC50 |
- |
- |
- |
P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Ki |
- |
- |
- |
P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ki |
- |
- |
- |
P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
- |
- |
- |
P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
IC50 |
- |
- |
- |
Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Ki |
- |
- |
- |
P04035 |
BXGT006129 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
reviewed |
- |
HMGCR |
IC50 |
- |
- |
- |
P08172 |
BXGT006737 |
Muscarinic acetylcholine receptor M2 |
reviewed |
G-protein coupled receptor |
CHRM2 |
IC50 |
- |
- |
- |
P29476 |
BXGT009354 |
Nitric oxide synthase, brain |
reviewed |
- |
Nos1 |
IC50 |
- |
- |
- |
P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
- |
- |
- |
P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
IC50 |
- |
- |
- |
P35372 |
BXGT009823 |
Mu-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRM1 |
Ki |
- |
- |
- |
Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
IC50 |
- |
- |
- |
P03956 |
BXGT006120 |
Interstitial collagenase |
reviewed |
Enzyme |
MMP1 |
Ki |
- |
- |
- |
P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
IC50 |
- |
- |
- |
P12822 |
BXGT007850 |
Angiotensin-converting enzyme |
reviewed |
- |
ACE |
Ki |
- |
- |
- |
P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
IC50 |
- |
- |
- |
P23975 |
BXGT008935 |
Sodium-dependent noradrenaline transporter |
reviewed |
Transporter |
SLC6A2 |
Ki |
- |
- |
- |
P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
IC50 |
- |
- |
- |
P30988 |
BXGT009491 |
Calcitonin receptor |
reviewed |
G-protein coupled receptor |
CALCR |
IC50 |
- |
- |
- |
P30988 |
BXGT009491 |
Calcitonin receptor |
reviewed |
G-protein coupled receptor |
CALCR |
Ki |
- |
- |
- |
P21554 |
BXGT008662 |
Cannabinoid receptor 1 |
reviewed |
G-protein coupled receptor |
CNR1 |
IC50 |
- |
- |
- |
P51679 |
BXGT010877 |
C-C chemokine receptor type 4 |
reviewed |
G-protein coupled receptor |
CCR4 |
Ki |
- |
- |
- |
P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
IC50 |
- |
- |
- |
P11509 |
BXGT007716 |
Cytochrome P450 2A6 |
reviewed |
- |
CYP2A6 |
IC50 |
- |
- |
- |
P05181 |
BXGT006337 |
Cytochrome P450 2E1 |
reviewed |
- |
CYP2E1 |
IC50 |
- |
- |
- |
P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
IC50 |
- |
- |
- |
P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
- |
- |
- |
P04035 |
BXGT006129 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
reviewed |
- |
HMGCR |
Ki |
- |
- |
- |
Q9Y271 |
BXGT022222 |
Cysteinyl leukotriene receptor 1 |
reviewed |
G-protein coupled receptor |
CYSLTR1 |
IC50 |
- |
- |
- |
P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
Ki |
- |
- |
- |
P32238 |
BXGT009611 |
Cholecystokinin receptor type A |
reviewed |
G-protein coupled receptor |
CCKAR |
IC50 |
- |
- |
- |
P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
IC50 |
- |
- |
- |
P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
IC50 |
- |
- |
- |
P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
IC50 |
- |
- |
- |
P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
IC50 |
- |
- |
- |
A6XA80 |
BXGT001522 |
Leukotriene C4 synthase |
reviewed |
- |
LTC4S |
IC50 |
- |
- |
- |
P30411 |
BXGT009424 |
B2 bradykinin receptor |
reviewed |
G-protein coupled receptor |
BDKRB2 |
IC50 |
- |
- |
- |
P41145 |
BXGT010225 |
Kappa-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRK1 |
IC50 |
- |
- |
- |
O76074 |
BXGT005174 |
cGMP-specific 3',5'-cyclic phosphodiesterase |
reviewed |
- |
PDE5A |
Ki |
- |
- |
- |
P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
Ki |
- |
- |
- |
P25025 |
BXGT009006 |
C-X-C chemokine receptor type 2 |
reviewed |
G-protein coupled receptor |
CXCR2 |
Ki |
- |
- |
- |
O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Potency |
- |
16360 |
nM |
P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
Ki |
- |
- |
- |
P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Ki |
- |
- |
- |
P11509 |
BXGT007716 |
Cytochrome P450 2A6 |
reviewed |
- |
CYP2A6 |
Ki |
- |
- |
- |
P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
IC50 |
- |
- |
- |
P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Ki |
- |
- |
- |
P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Ki |
- |
- |
- |
P35367 |
BXGT009821 |
Histamine H1 receptor |
reviewed |
G-protein coupled receptor |
HRH1 |
Ki |
- |
- |
- |
P20781 |
BXGT008598 |
Glycine receptor subunit beta |
reviewed |
- |
Glrb |
Ki |
- |
- |
- |
P07727 |
BXGT006662 |
Glycine receptor subunit alpha-1 |
reviewed |
- |
Glra1 |
Ki |
- |
- |
- |
P24524 |
BXGT008974 |
Glycine receptor subunit alpha-3 |
reviewed |
- |
Glra3 |
Ki |
- |
- |
- |
P22771 |
BXGT008806 |
Glycine receptor subunit alpha-2 |
reviewed |
- |
Glra2 |
Ki |
- |
- |
- |
P25021 |
BXGT009004 |
Histamine H2 receptor |
reviewed |
G-protein coupled receptor |
HRH2 |
IC50 |
- |
- |
- |
P25021 |
BXGT009004 |
Histamine H2 receptor |
reviewed |
G-protein coupled receptor |
HRH2 |
Ki |
- |
- |
- |
P12530 |
BXGT007827 |
Arachidonate 15-lipoxygenase |
reviewed |
- |
ALOX15 |
Ki |
- |
- |
- |
P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
Ki |
- |
- |
- |
O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
112 |
nM |
P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
IC50 |
- |
- |
- |
P25103 |
BXGT009020 |
Substance-P receptor |
reviewed |
G-protein coupled receptor |
TACR1 |
IC50 |
- |
- |
- |
P08172 |
BXGT006737 |
Muscarinic acetylcholine receptor M2 |
reviewed |
G-protein coupled receptor |
CHRM2 |
Ki |
- |
- |
- |
P08173 |
BXGT006738 |
Muscarinic acetylcholine receptor M4 |
reviewed |
G-protein coupled receptor |
CHRM4 |
IC50 |
- |
- |
- |
P49146 |
BXGT010681 |
Neuropeptide Y receptor type 2 |
reviewed |
G-protein coupled receptor |
NPY2R |
IC50 |
- |
- |
- |
P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Ki |
- |
- |
- |
P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Ki |
- |
- |
- |
P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
Ki |
- |
- |
- |
P33032 |
BXGT009689 |
Melanocortin receptor 5 |
reviewed |
G-protein coupled receptor |
MC5R |
Ki |
- |
- |
- |
P03956 |
BXGT006120 |
Interstitial collagenase |
reviewed |
Enzyme |
MMP1 |
IC50 |
- |
- |
- |
P41597 |
BXGT010268 |
C-C chemokine receptor type 2 |
reviewed |
- |
CCR2 |
IC50 |
- |
- |
- |
P32238 |
BXGT009611 |
Cholecystokinin receptor type A |
reviewed |
G-protein coupled receptor |
CCKAR |
Ki |
- |
- |
- |
P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
Ki |
- |
- |
- |
P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
Ki |
- |
- |
- |
P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
IC50 |
- |
- |
- |
P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
IC50 |
- |
- |
- |
P12530 |
BXGT007827 |
Arachidonate 15-lipoxygenase |
reviewed |
- |
ALOX15 |
IC50 |
- |
- |
- |
P51681 |
BXGT010878 |
C-C chemokine receptor type 5 |
reviewed |
G-protein coupled receptor |
CCR5 |
IC50 |
- |
- |
- |
P25024 |
BXGT009005 |
C-X-C chemokine receptor type 1 |
reviewed |
G-protein coupled receptor |
CXCR1 |
IC50 |
- |
- |
- |
P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Ki |
- |
- |
- |
P41145 |
BXGT010225 |
Kappa-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRK1 |
Ki |
- |
- |
- |
Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
Ki |
- |
- |
- |
P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
IC50 |
- |
- |
- |
P15207 |
BXGT008096 |
Androgen receptor |
reviewed |
- |
Ar |
Ki |
- |
- |
- |
P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
Ki |
- |
- |
- |
P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
IC50 |
- |
- |
- |
P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
IC50 |
- |
- |
- |
P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
IC50 |
- |
- |
- |
P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
Ki |
- |
- |
- |
P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
Ki |
- |
- |
- |
P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
Ki |
- |
- |
- |
P51679 |
BXGT010877 |
C-C chemokine receptor type 4 |
reviewed |
G-protein coupled receptor |
CCR4 |
IC50 |
- |
- |
- |
P25024 |
BXGT009005 |
C-X-C chemokine receptor type 1 |
reviewed |
G-protein coupled receptor |
CXCR1 |
Ki |
- |
- |
- |
P25101 |
BXGT009018 |
Endothelin-1 receptor |
reviewed |
G-protein coupled receptor |
EDNRA |
Ki |
- |
- |
- |
P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
- |
- |
- |
A6XA80 |
BXGT001522 |
Leukotriene C4 synthase |
reviewed |
- |
LTC4S |
Ki |
- |
- |
- |
P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
IC50 |
- |
- |
- |
P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
Ki |
- |
- |
- |
P32245 |
BXGT009614 |
Melanocortin receptor 4 |
reviewed |
G-protein coupled receptor |
MC4R |
IC50 |
- |
- |
- |
P25929 |
BXGT009078 |
Neuropeptide Y receptor type 1 |
reviewed |
G-protein coupled receptor |
NPY1R |
IC50 |
- |
- |
- |
P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
IC50 |
- |
- |
- |
O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
IC50 |
- |
- |
- |
P25103 |
BXGT009020 |
Substance-P receptor |
reviewed |
G-protein coupled receptor |
TACR1 |
Ki |
- |
- |
- |
P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
IC50 |
- |
- |
- |
Q9Y271 |
BXGT022222 |
Cysteinyl leukotriene receptor 1 |
reviewed |
G-protein coupled receptor |
CYSLTR1 |
Ki |
- |
- |
- |
P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Ki |
- |
- |
- |
P37288 |
BXGT009977 |
Vasopressin V1a receptor |
reviewed |
G-protein coupled receptor |
AVPR1A |
IC50 |
- |
- |
- |
P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
Ki |
- |
- |
- |
P50052 |
BXGT010768 |
Type-2 angiotensin II receptor |
reviewed |
G-protein coupled receptor |
AGTR2 |
IC50 |
- |
- |
- |
P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Ki |
- |
- |
- |
P35367 |
BXGT009821 |
Histamine H1 receptor |
reviewed |
G-protein coupled receptor |
HRH1 |
IC50 |
- |
- |
- |