Compound Information
Test on : DRx, Metz
Compound Name
DRx : Ruboxistaurin
Metz : Kinome_3136
Inchikey
Same : ZCBUQCWBWNUWSU-N
DRx : ZCBUQCWBWNUWSU-SFHVURJKSA-N
Metz : ZCBUQCWBWNUWSU-UHFFFAOYSA-N
ChemSpider
DRx : 135727
Metz : 8068036
Pubchem CID
DRx : 153999
Metz : 9892366
ChEMBL
DRx : CHEMBL432130
Metz : CHEMBL360847
DRx | Metz |
| |
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
Other
Other - NAK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
AAK1 | active (900nM) | - |
BIKE | active (430nM) | - |
GAK | active (1100nM) | - |
MPSK1 | inactive (10001nM) | - |
Other - Aur
Bioactivity |
---|
Kinase | DRx | Metz |
---|
AurA | inactive (10001nM) | inactive (>1584.89nM) |
AurB | inactive (10001nM) | inactive (>3981.07nM) |
AurC | inactive (10001nM) | - |
Other - CAMKK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
CaMKK1 | inactive (5000nM) | - |
CaMKK2 | active (2400nM) | - |
Other - PEK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
HRI | inactive (10001nM) | - |
PKR | inactive (10001nM) | - |
Other - IRE
Bioactivity |
---|
Kinase | DRx | Metz |
---|
IRE1 | inactive (10001nM) | - |
Other - IKK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
IKKa | inactive (10001nM) | - |
IKKb | inactive (10001nM) | - |
IKKe | inactive (10001nM) | inactive (>3162.28nM) |
TBK1 | active (970nM) | active (501.19nM) |
Other - NEK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
NEK1 | inactive (10001nM) | - |
NEK11 | inactive (10001nM) | - |
NEK2 | inactive (10001nM) | inactive (>3162.28nM) |
NEK3 | inactive (10001nM) | - |
NEK4 | inactive (10001nM) | - |
NEK5 | inactive (10001nM) | - |
NEK6 | inactive (10001nM) | - |
NEK7 | inactive (10001nM) | - |
NEK9 | inactive (10001nM) | - |
Other - WEE
Bioactivity |
---|
Kinase | DRx | Metz |
---|
MYT1 | inactive (10001nM) | - |
Wee1 | inactive (10001nM) | - |
Wee1B | inactive (10001nM) | - |
Other - PLK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
PLK1 | inactive (10001nM) | - |
PLK2 | inactive (10001nM) | - |
PLK3 | inactive (10001nM) | - |
PLK4 | inactive (4700nM) | - |
Other - SgK496
Bioactivity |
---|
Kinase | DRx | Metz |
---|
SgK496 | inactive (10001nM) | - |
Other - NKF1
Bioactivity |
---|
Kinase | DRx | Metz |
---|
SBK | inactive (10001nM) | - |
SgK110 | inactive (10001nM) | - |
Other - NKF4
Bioactivity |
---|
Kinase | DRx | Metz |
---|
CLIK1 | inactive (10001nM) | - |
Other - ULK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
Fused | inactive (10001nM) | - |
ULK1 | inactive (10001nM) | - |
ULK2 | inactive (10001nM) | - |
ULK3 | inactive (10001nM) | - |
Other - TLK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
TLK1 | active (2100nM) | - |
TLK2 | inactive (10001nM) | - |
Other - TTK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
TTK | inactive (10001nM) | - |
Other - CDC7
Bioactivity |
---|
Kinase | DRx | Metz |
---|
CDC7 | - | - |
Other - TOPK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
PBK | - | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | DRx | Metz |
---|
ABL1 | inactive (10001nM) | inactive (>2511.89nM) |
ABL2 | inactive (10001nM) | - |
TK - ALK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
ALK | inactive (10001nM) | inactive (3162.28nM) |
LTK | inactive (10001nM) | inactive (>2511.89nM) |
TK - Axl
Bioactivity |
---|
Kinase | DRx | Metz |
---|
AXL | inactive (10001nM) | - |
MER | inactive (10001nM) | - |
TYRO3 | inactive (10001nM) | inactive (>3162.28nM) |
TK - Src
Bioactivity |
---|
Kinase | DRx | Metz |
---|
BLK | inactive (10001nM) | - |
BRK | inactive (10001nM) | - |
FGR | inactive (10001nM) | - |
FRK | inactive (10001nM) | - |
FYN | inactive (10001nM) | inactive (>6309.57nM) |
HCK | inactive (10001nM) | - |
LCK | inactive (10001nM) | inactive (>6309.57nM) |
LYN | inactive (10001nM) | - |
SRC | inactive (10001nM) | - |
SRM | inactive (10001nM) | - |
YES | inactive (10001nM) | - |
TK - Tec
Bioactivity |
---|
Kinase | DRx | Metz |
---|
BMX | inactive (10001nM) | - |
BTK | inactive (10001nM) | inactive (>6309.57nM) |
ITK | inactive (10001nM) | - |
TEC | inactive (10001nM) | - |
TXK | inactive (10001nM) | - |
TK - PDGFR
Bioactivity |
---|
Kinase | DRx | Metz |
---|
FMS | inactive (10001nM) | inactive (>2511.89nM) |
FLT3 | active (1900nM) | inactive (>3162.28nM) |
KIT | inactive (10001nM) | - |
PDGFRa | inactive (10001nM) | inactive (>2511.89nM) |
PDGFRb | inactive (10001nM) | inactive (>1995.26nM) |
TK - Csk
Bioactivity |
---|
Kinase | DRx | Metz |
---|
CSK | inactive (10001nM) | - |
CTK | inactive (10001nM) | - |
TK - DDR
Bioactivity |
---|
Kinase | DRx | Metz |
---|
DDR1 | inactive (10001nM) | - |
DDR2 | inactive (10001nM) | - |
TK - EGFR
Bioactivity |
---|
Kinase | DRx | Metz |
---|
EGFR | inactive (10001nM) | - |
ErbB2 | inactive (10001nM) | - |
ErbB3 | inactive (10001nM) | - |
ErbB4 | inactive (10001nM) | - |
TK - Eph
Bioactivity |
---|
Kinase | DRx | Metz |
---|
EphA1 | inactive (10001nM) | - |
EphA2 | inactive (10001nM) | - |
EphA3 | inactive (10001nM) | - |
EphA4 | inactive (10001nM) | - |
EphA5 | inactive (10001nM) | - |
EphA6 | inactive (10001nM) | - |
EphA7 | inactive (10001nM) | - |
EphA8 | inactive (10001nM) | - |
EphB1 | inactive (10001nM) | - |
EphB2 | inactive (10001nM) | - |
EphB3 | inactive (10001nM) | - |
EphB4 | inactive (10001nM) | - |
EphB6 | inactive (10001nM) | - |
TK - FAK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
FAK | inactive (10001nM) | inactive (>6309.57nM) |
PYK2 | inactive (10001nM) | - |
TK - Fer
Bioactivity |
---|
Kinase | DRx | Metz |
---|
FER | inactive (10001nM) | - |
FES | inactive (10001nM) | - |
TK - FGFR
Bioactivity |
---|
Kinase | DRx | Metz |
---|
FGFR1 | inactive (10001nM) | inactive (>3981.07nM) |
FGFR2 | inactive (10001nM) | - |
FGFR3 | inactive (10001nM) | - |
FGFR4 | inactive (10001nM) | - |
TK - VEGFR
Bioactivity |
---|
Kinase | DRx | Metz |
---|
FLT1 | inactive (10001nM) | inactive (>3981.07nM) |
FLT4 | inactive (10001nM) | - |
KDR | inactive (10001nM) | inactive (1995.26nM) |
TK - InsR
Bioactivity |
---|
Kinase | DRx | Metz |
---|
IGF1R | inactive (10001nM) | inactive (>2511.89nM) |
INSR | inactive (10001nM) | - |
IRR | inactive (10001nM) | - |
TK - JakA
Bioactivity |
---|
Kinase | DRx | Metz |
---|
JAK1 | inactive (10001nM) | - |
JAK2 | inactive (10001nM) | inactive (>2511.89nM) |
JAK3 | active (1200nM) | inactive (1995.26nM) |
TYK2 | inactive (10001nM) | - |
TK - Met
Bioactivity |
---|
Kinase | DRx | Metz |
---|
MET | inactive (10001nM) | inactive (>2511.89nM) |
RON | inactive (10001nM) | active (199.53nM) |
TK - Musk
Bioactivity |
---|
Kinase | DRx | Metz |
---|
MUSK | inactive (10001nM) | - |
TK - Ret
Bioactivity |
---|
Kinase | DRx | Metz |
---|
RET | inactive (10001nM) | inactive (>3162.28nM) |
TK - Sev
Bioactivity |
---|
Kinase | DRx | Metz |
---|
ROS | inactive (5800nM) | - |
TK - Syk
Bioactivity |
---|
Kinase | DRx | Metz |
---|
SYK | inactive (10001nM) | - |
ZAP70 | inactive (10001nM) | - |
TK - Tie
Bioactivity |
---|
Kinase | DRx | Metz |
---|
TIE1 | inactive (10001nM) | - |
TIE2 | inactive (10001nM) | - |
TK - Ack
Bioactivity |
---|
Kinase | DRx | Metz |
---|
TNK1 | inactive (10001nM) | - |
ACK | inactive (10001nM) | inactive (>3981.07nM) |
TK - Trk
Bioactivity |
---|
Kinase | DRx | Metz |
---|
TRKA | inactive (10001nM) | inactive (>3162.28nM) |
TRKB | inactive (10001nM) | inactive (>3981.07nM) |
TRKC | inactive (10001nM) | inactive (>3162.28nM) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | DRx | Metz |
---|
ALK2 | inactive (10001nM) | inactive (>3981.07nM) |
ALK4 | inactive (10001nM) | - |
ACTR2 | inactive (10001nM) | - |
ACTR2B | inactive (10001nM) | - |
ALK1 | inactive (10001nM) | - |
BMPR1A | inactive (10001nM) | - |
BMPR1B | inactive (10001nM) | - |
BMPR2 | inactive (10001nM) | - |
TGFbR1 | inactive (10001nM) | - |
TGFbR2 | inactive (10001nM) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
SgK288 | inactive (10001nM) | - |
RIPK1 | inactive (10001nM) | - |
RIPK2 | inactive (10001nM) | - |
ANKRD3 | inactive (10001nM) | - |
TKL - RAF
Bioactivity |
---|
Kinase | DRx | Metz |
---|
BRAF | inactive (10001nM) | - |
RAF1 | inactive (10001nM) | - |
TKL - MLK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
DLK | inactive (10001nM) | - |
LZK | inactive (10001nM) | - |
MLK1 | active (1400nM) | - |
MLK2 | inactive (10001nM) | - |
MLK3 | inactive (10001nM) | - |
TAK1 | inactive (10001nM) | - |
HH498 | inactive (10001nM) | - |
ZAK | inactive (10001nM) | - |
TKL - IRAK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
IRAK1 | inactive (10001nM) | - |
IRAK3 | inactive (10001nM) | - |
IRAK4 | inactive (10001nM) | - |
TKL - LISK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
LIMK1 | inactive (10001nM) | inactive (>3162.28nM) |
LIMK2 | inactive (10001nM) | - |
TESK1 | inactive (10001nM) | - |
TKL - LRRK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
LRRK2 | inactive (10001nM) | inactive (>2511.89nM) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | Metz |
---|
ABC1 | 5 | 2 | - |
PIKK | 6 | 1 | - |
RIO | 3 | 3 | - |
Alpha | 6 | 1 | 1 |
Atypical - ABC1
Bioactivity |
---|
Kinase | DRx | Metz |
---|
ADCK3 | inactive (10001nM) | - |
ADCK4 | inactive (10001nM) | - |
Atypical - PIKK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
FRAP | inactive (10001nM) | - |
Atypical - RIO
Bioactivity |
---|
Kinase | DRx | Metz |
---|
RIOK1 | active (810nM) | - |
RIOK2 | inactive (10001nM) | - |
RIOK3 | active (650nM) | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | DRx | Metz |
---|
ChaK2 | inactive (10001nM) | - |
eEF2K | - | - |
AGC
AGC - Akt
Bioactivity |
---|
Kinase | DRx | Metz |
---|
AKT1 | inactive (10001nM) | - |
AKT2 | inactive (8700nM) | - |
AKT3 | active (1400nM) | - |
AGC - DMPK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
CRIK | active (1400nM) | - |
DMPK1 | active (280nM) | - |
DMPK2 | inactive (10001nM) | - |
MRCKa | inactive (10001nM) | - |
MRCKb | inactive (10001nM) | - |
ROCK1 | inactive (10001nM) | inactive (>3981.07nM) |
ROCK2 | inactive (10001nM) | - |
AGC - GRK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
RHOK | active (800nM) | - |
GPRK4 | active (590nM) | - |
GPRK7 | active (310nM) | - |
GPRK5 | - | inactive (3162.28nM) |
AGC - NDR
Bioactivity |
---|
Kinase | DRx | Metz |
---|
LATS1 | active (2600nM) | - |
LATS2 | active (640nM) | - |
NDR1 | inactive (10001nM) | - |
NDR2 | inactive (10001nM) | - |
AGC - MAST
Bioactivity |
---|
Kinase | DRx | Metz |
---|
MAST1 | inactive (10001nM) | - |
AGC - PDK1
Bioactivity |
---|
Kinase | DRx | Metz |
---|
PDK1 | active (700nM) | - |
AGC - PKA
Bioactivity |
---|
Kinase | DRx | Metz |
---|
PKACa | inactive (5400nM) | active (630.96nM) |
PKACb | inactive (3200nM) | - |
PRKX | inactive (10001nM) | inactive (>3162.28nM) |
AGC - PKN
Bioactivity |
---|
Kinase | DRx | Metz |
---|
PKN1 | active (350nM) | - |
PKN2 | active (1500nM) | - |
AGC - PKC
Bioactivity |
---|
Kinase | DRx | Metz |
---|
PKCd | active (3.6nM) | - |
PKCe | active (11nM) | - |
PKCh | active (1800nM) | - |
PKCi | active (1400nM) | - |
PKCt | active (2.5nM) | active (1.58nM) |
PKCg | - | - |
PKCz | - | - |
AGC - PKG
Bioactivity |
---|
Kinase | DRx | Metz |
---|
PKG1 | inactive (10001nM) | - |
PKG2 | inactive (3100nM) | - |
AGC - RSK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
p70S6K | active (210nM) | - |
RSK2 | - | active (19.95nM) |
MSK1 | - | - |
MSK2 | - | - |
AGC - SGK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
SGK3 | active (1400nM) | - |
SGK1 | - | - |
AGC - YANK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
YANK1 | inactive (10001nM) | - |
YANK2 | inactive (10001nM) | - |
YANK3 | inactive (10001nM) | - |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | DRx | Metz |
---|
AMPKa1 | inactive (10001nM) | inactive (>3162.28nM) |
AMPKa2 | inactive (10001nM) | - |
NuaK1 | active (1800nM) | - |
BRSK1 | inactive (10001nM) | - |
BRSK2 | inactive (10001nM) | - |
CHK1 | active (540nM) | active (316.23nM) |
HUNK | inactive (10001nM) | - |
LKB1 | inactive (5900nM) | - |
MARK1 | inactive (10001nM) | - |
MARK2 | inactive (10001nM) | - |
MARK3 | inactive (10001nM) | - |
MARK4 | inactive (10001nM) | - |
MELK | inactive (10001nM) | - |
NIM1 | inactive (10001nM) | - |
QSK | inactive (10001nM) | - |
SIK | inactive (10001nM) | - |
QIK | inactive (10001nM) | - |
NuaK2 | active (320nM) | - |
SNRK | inactive (10001nM) | - |
PASK | - | - |
CAMK - CAMK1
Bioactivity |
---|
Kinase | DRx | Metz |
---|
CaMK1a | inactive (10001nM) | - |
CaMK1d | inactive (4500nM) | inactive (>2511.89nM) |
CaMK1g | inactive (10001nM) | - |
CaMK4 | inactive (10001nM) | - |
CAMK - CAMK2
Bioactivity |
---|
Kinase | DRx | Metz |
---|
CaMK2a | inactive (4500nM) | inactive (>3981.07nM) |
CaMK2b | inactive (10001nM) | - |
CaMK2d | inactive (4600nM) | - |
CaMK2g | inactive (7800nM) | - |
CAMK - CASK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
CASK | inactive (10001nM) | - |
CAMK - RAD53
Bioactivity |
---|
Kinase | DRx | Metz |
---|
CHK2 | inactive (3700nM) | - |
CAMK - DAPK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
DAPK1 | active (970nM) | - |
DAPK2 | inactive (10001nM) | - |
DAPK3 | inactive (8000nM) | inactive (>5011.87nM) |
DRAK1 | inactive (10001nM) | - |
DRAK2 | inactive (10001nM) | - |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | DRx | Metz |
---|
DCLK1 | inactive (10001nM) | - |
DCLK2 | inactive (10001nM) | - |
DCLK3 | inactive (10001nM) | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
MAPKAPK2 | inactive (10001nM) | - |
MAPKAPK5 | inactive (10001nM) | - |
MNK1 | inactive (7100nM) | - |
MNK2 | inactive (10001nM) | - |
MAPKAPK3 | - | - |
CAMK - MLCK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
caMLCK | inactive (10001nM) | - |
smMLCK | active (290nM) | - |
skMLCK | inactive (10001nM) | - |
SgK085 | inactive (10001nM) | - |
CAMK - PHK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
PHKg1 | inactive (3700nM) | - |
PHKg2 | inactive (10001nM) | - |
CAMK - PIM
Bioactivity |
---|
Kinase | DRx | Metz |
---|
PIM1 | active (270nM) | active (19.95nM) |
PIM2 | active (1700nM) | - |
PIM3 | active (12nM) | - |
CAMK - PKD
Bioactivity |
---|
Kinase | DRx | Metz |
---|
PKD1 | inactive (10001nM) | - |
PKD2 | active (890nM) | - |
PKD3 | inactive (10001nM) | inactive (>3981.07nM) |
CAMK - STK33
Bioactivity |
---|
Kinase | DRx | Metz |
---|
STK33 | active (2600nM) | - |
CAMK - TSSK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
TSSK1 | inactive (10001nM) | - |
TSSK2 | - | - |
STE
STE
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | Metz |
---|
STE11 | 8 | 8 | - |
STE20 | 31 | 27 | 9 |
STE7 | 7 | 7 | 2 |
STE - STE11
Bioactivity |
---|
Kinase | DRx | Metz |
---|
MAP3K5 | inactive (10001nM) | - |
MAP3K6 | inactive (10001nM) | - |
MAP3K1 | inactive (10001nM) | - |
MAP3K7 | inactive (10001nM) | - |
MAP3K2 | active (710nM) | - |
MAP3K3 | active (170nM) | - |
MAP3K4 | inactive (10001nM) | - |
MAP3K8 | active (48nM) | - |
STE - STE20
Bioactivity |
---|
Kinase | DRx | Metz |
---|
HPK1 | active (2600nM) | - |
LOK | active (280nM) | - |
GCK | active (290nM) | inactive (>2511.89nM) |
KHS2 | inactive (8400nM) | - |
HGK | inactive (10001nM) | inactive (>5011.87nM) |
KHS1 | inactive (10001nM) | - |
MINK | active (310nM) | - |
MST1 | inactive (10001nM) | - |
MST2 | active (960nM) | - |
MST3 | inactive (10001nM) | - |
MST4 | inactive (10001nM) | - |
MYO3A | inactive (10001nM) | - |
MYO3B | inactive (10001nM) | - |
OSR1 | inactive (10001nM) | - |
PAK1 | inactive (10001nM) | - |
PAK2 | inactive (10001nM) | - |
PAK3 | inactive (10001nM) | - |
PAK4 | inactive (10001nM) | inactive (>5011.87nM) |
PAK6 | inactive (10001nM) | - |
PAK5 | inactive (10001nM) | - |
SLK | active (400nM) | - |
STLK3 | inactive (10001nM) | - |
TAO1 | active (1800nM) | inactive (2511.89nM) |
TAO2 | inactive (3900nM) | - |
TAO3 | active (97nM) | - |
TNIK | inactive (10001nM) | - |
YSK1 | inactive (10001nM) | - |
STE - STE7
Bioactivity |
---|
Kinase | DRx | Metz |
---|
MAP2K1 | inactive (10001nM) | inactive (>3162.28nM) |
MAP2K2 | inactive (10001nM) | inactive (>3981.07nM) |
MAP2K3 | inactive (10001nM) | - |
MAP2K4 | active (930nM) | - |
MAP2K5 | active (1100nM) | - |
MAP2K6 | inactive (3900nM) | - |
MAP2K7 | inactive (10001nM) | - |
CMGC
CMGC - CDK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
PITSLRE | inactive (10001nM) | - |
CHED | inactive (10001nM) | - |
CDK11 | inactive (10001nM) | - |
PCTAIRE1 | active (2600nM) | - |
PCTAIRE2 | inactive (10001nM) | - |
PCTAIRE3 | inactive (10001nM) | - |
PFTAIRE2 | inactive (10001nM) | - |
PFTAIRE1 | inactive (10001nM) | - |
CDC2 | - | - |
CDK2 | - | - |
CDK5 | - | inactive (>3162.28nM) |
CDK8 | - | inactive (>3981.07nM) |
CDK7 | - | inactive (2511.89nM) |
CDK9 | - | inactive (>1584.89nM) |
CMGC - CDKL
Bioactivity |
---|
Kinase | DRx | Metz |
---|
CDKL1 | inactive (10001nM) | - |
CDKL2 | inactive (10001nM) | - |
CDKL3 | inactive (10001nM) | - |
CDKL5 | inactive (4100nM) | - |
CMGC - CLK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
CLK1 | active (910nM) | - |
CLK2 | active (420nM) | active (158.49nM) |
CLK3 | inactive (10001nM) | - |
CLK4 | active (1900nM) | active (125.89nM) |
CMGC - CK2
Bioactivity |
---|
Kinase | DRx | Metz |
---|
CK2a1 | inactive (10001nM) | - |
CK2a2 | inactive (6700nM) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
DYRK1A | active (250nM) | inactive (>1995.26nM) |
DYRK1B | inactive (5400nM) | active (794.33nM) |
DYRK2 | inactive (10001nM) | - |
HIPK1 | active (230nM) | - |
HIPK2 | active (140nM) | - |
HIPK3 | active (77nM) | - |
HIPK4 | inactive (10001nM) | - |
PRP4 | active (1600nM) | - |
DYRK3 | - | - |
DYRK4 | - | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
Erk1 | inactive (10001nM) | - |
Erk2 | inactive (10001nM) | - |
Erk3 | inactive (10001nM) | - |
Erk4 | inactive (10001nM) | - |
Erk5 | inactive (10001nM) | - |
Erk7 | active (88nM) | - |
JNK1 | inactive (10001nM) | inactive (>5011.87nM) |
JNK2 | inactive (10001nM) | inactive (>3981.07nM) |
JNK3 | inactive (10001nM) | - |
NLK | inactive (10001nM) | - |
p38a | inactive (10001nM) | inactive (>3981.07nM) |
p38b | inactive (10001nM) | - |
p38d | inactive (10001nM) | - |
p38g | inactive (10001nM) | - |
CMGC - GSK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
GSK3A | inactive (10001nM) | inactive (1995.26nM) |
GSK3B | active (2600nM) | active (794.33nM) |
CMGC - RCK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
ICK | active (240nM) | - |
MAK | inactive (10001nM) | - |
CMGC - SRPK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
SRPK1 | active (1200nM) | - |
SRPK2 | active (1100nM) | - |
MSSK1 | active (1600nM) | - |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | Metz |
---|
CK1 | 7 | 7 | 5 |
VRK | 3 | 1 | - |
CK1 - CK1
Bioactivity |
---|
Kinase | DRx | Metz |
---|
CK1a | inactive (10001nM) | inactive (>3981.07nM) |
CK1a2 | inactive (10001nM) | - |
CK1d | inactive (10001nM) | - |
CK1e | inactive (10001nM) | - |
CK1g1 | inactive (10001nM) | - |
CK1g2 | inactive (10001nM) | - |
CK1g3 | inactive (10001nM) | - |
CK1 - VRK
Bioactivity |
---|
Kinase | DRx | Metz |
---|
VRK2 | inactive (10001nM) | - |