Compound Information
Test on : DRx, RBC, Metz
Compound Name
DRx, RBC, Metz : Dasatinib
Inchikey
Same : ZBNZXTGUTAYRHI-N
DRx, RBC, Metz : ZBNZXTGUTAYRHI-UHFFFAOYSA-N
ChemSpider
DRx, RBC, Metz : 2323020
Pubchem CID
DRx, RBC, Metz : 3062316
ChEMBL
DRx, RBC, Metz : CHEMBL1421
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
Other
Other - NAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AAK1 | inactive (10001nM) | - | - |
BIKE | inactive (10001nM) | - | - |
GAK | active (2.6nM) | - | - |
MPSK1 | inactive (10001nM) | inactive (96.9%) | - |
Other - Aur
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AurA | inactive (9300nM) | inactive (93.22%) | inactive (>1000nM) |
AurB | inactive (10001nM) | inactive (92.53%) | inactive (1258.93nM) |
AurC | inactive (10001nM) | inactive (84.82%) | - |
Other - CAMKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CaMKK1 | inactive (10001nM) | inactive (99.75%) | - |
CaMKK2 | inactive (10001nM) | inactive (101.46%) | inactive (>2511.89nM) |
Other - PEK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
HRI | inactive (10001nM) | - | - |
PKR | inactive (10001nM) | - | - |
Other - IRE
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IRE1 | inactive (10001nM) | - | - |
Other - IKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IKKa | inactive (10001nM) | inactive (95.05%) | inactive (>3981.07nM) |
IKKb | inactive (10001nM) | inactive (94.03%) | inactive (>3162.28nM) |
IKKe | inactive (10001nM) | inactive (90.01%) | inactive (>3162.28nM) |
TBK1 | inactive (10001nM) | inactive (90.77%) | inactive (>3162.28nM) |
Other - NEK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
NEK1 | inactive (10001nM) | inactive (89.81%) | - |
NEK11 | active (470nM) | active (21.66%) | - |
NEK2 | inactive (6500nM) | inactive (102.56%) | inactive (>6309.57nM) |
NEK3 | inactive (10001nM) | inactive (94.1%) | - |
NEK4 | inactive (10001nM) | inactive (90.71%) | inactive (>6309.57nM) |
NEK5 | inactive (10001nM) | - | - |
NEK6 | inactive (10001nM) | inactive (86.19%) | - |
NEK7 | inactive (10001nM) | inactive (90.99%) | - |
NEK9 | inactive (10001nM) | inactive (98.3%) | - |
Other - WEE
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MYT1 | active (130nM) | - | - |
Wee1 | inactive (7000nM) | inactive (92.61%) | - |
Wee1B | active (200nM) | - | - |
Other - PLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PLK1 | inactive (10001nM) | inactive (98.05%) | inactive (>7943.28nM) |
PLK2 | inactive (10001nM) | inactive (97.99%) | - |
PLK3 | inactive (10001nM) | inactive (105.02%) | inactive (>7943.28nM) |
PLK4 | inactive (10001nM) | - | inactive (1995.26nM) |
Other - SgK496
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SgK496 | inactive (10001nM) | inactive (99.35%) | - |
Other - NKF1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SBK | active (1200nM) | - | - |
SgK110 | inactive (10001nM) | - | - |
Other - NKF4
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CLIK1 | active (770nM) | - | - |
Other - ULK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Fused | active (210nM) | - | - |
ULK1 | inactive (10001nM) | inactive (85.49%) | - |
ULK2 | inactive (10001nM) | inactive (94.18%) | - |
ULK3 | inactive (4600nM) | inactive (102.87%) | - |
Other - TLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TLK1 | inactive (10001nM) | - | - |
TLK2 | inactive (10001nM) | inactive (94.4%) | - |
Other - TTK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TTK | inactive (10001nM) | inactive (104.91%) | - |
Other - Haspin
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Haspin | - | inactive (91.94%) | - |
Other - TOPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PBK | - | inactive (101.05%) | inactive (>10000nM) |
Other - WNK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Wnk2 | - | inactive (83.9%) | - |
Wnk3 | - | inactive (88.07%) | - |
Other - CDC7
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CDC7 | - | - | inactive (>1258.93nM) |
TK
TK - Abl
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ABL1 | active (0.03nM) | active (2.77%) | - |
ABL2 | active (0.17nM) | active (2.74%) | - |
TK - ALK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ALK | inactive (10001nM) | inactive (109.91%) | inactive (>5011.87nM) |
LTK | inactive (10001nM) | inactive (97.75%) | inactive (>2511.89nM) |
TK - Axl
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AXL | inactive (10001nM) | inactive (61.36%) | inactive (1995.26nM) |
MER | inactive (10001nM) | inactive (103.38%) | - |
TYRO3 | inactive (10001nM) | inactive (87.6%) | inactive (>1258.93nM) |
TK - Src
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
BLK | active (0.21nM) | active (3.04%) | - |
BRK | active (7.8nM) | active (4.59%) | active (5.01nM) |
FGR | active (0.5nM) | active (1.7%) | - |
FRK | active (0.31nM) | active (-0.88%) | - |
FYN | active (0.79nM) | active (1.96%) | - |
HCK | active (0.35nM) | active (0.79%) | active (0.32nM) |
LCK | active (0.2nM) | active (0.31%) | - |
LYN | active (0.57nM) | active (0.43%) | - |
SRC | active (0.21nM) | active (3.52%) | - |
SRM | active (13nM) | active (16.98%) | active (0.63nM) |
YES | active (0.3nM) | active (1.94%) | - |
TK - Tec
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
BMX | active (1.4nM) | active (2.53%) | - |
BTK | active (1.4nM) | active (2.09%) | - |
ITK | inactive (10001nM) | inactive (102.72%) | inactive (>1584.89nM) |
TEC | active (13nM) | active (11.28%) | - |
TXK | active (2.1nM) | active (1.37%) | - |
TK - PDGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FMS | active (0.58nM) | active (0.77%) | inactive (>6.31nM) |
FLT3 | inactive (4800nM) | inactive (71.02%) | inactive (>1995.26nM) |
KIT | active (0.81nM) | active (3.27%) | inactive (>3162.28nM) |
PDGFRa | active (0.47nM) | active (1.82%) | active (10nM) |
PDGFRb | active (0.63nM) | active (2.48%) | active (1.26nM) |
TK - Csk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CSK | active (1nM) | active (7.11%) | - |
CTK | inactive (10001nM) | inactive (79.03%) | inactive (>1995.26nM) |
TK - DDR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DDR1 | active (0.69nM) | - | - |
DDR2 | active (3.2nM) | active (0.24%) | - |
TK - EGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
EGFR | active (120nM) | active (21.08%) | inactive (>1000nM) |
ErbB2 | active (1400nM) | inactive (79.85%) | active (158.49nM) |
ErbB3 | active (18nM) | - | - |
ErbB4 | active (55nM) | active (4.03%) | active (39.81nM) |
TK - Eph
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
EphA1 | active (4.1nM) | active (2.72%) | - |
EphA2 | active (0.85nM) | active (6.82%) | active (3.98nM) |
EphA3 | active (0.09nM) | active (3.46%) | - |
EphA4 | active (1.2nM) | active (1.63%) | - |
EphA5 | active (0.24nM) | active (0.24%) | - |
EphA6 | active (2100nM) | inactive (50.45%) | - |
EphA7 | inactive (10001nM) | inactive (94.32%) | - |
EphA8 | active (0.24nM) | active (4.13%) | - |
EphB1 | active (0.45nM) | active (4.8%) | - |
EphB2 | active (0.39nM) | active (-0.19%) | - |
EphB3 | active (6.9nM) | active (0.99%) | - |
EphB4 | active (0.34nM) | active (1.17%) | - |
EphB6 | active (0.04nM) | - | - |
TK - FAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FAK | inactive (10001nM) | inactive (103.4%) | inactive (>3981.07nM) |
PYK2 | inactive (10001nM) | inactive (97.74%) | inactive (>1584.89nM) |
TK - Fer
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FER | inactive (10001nM) | inactive (95.86%) | inactive (>1584.89nM) |
FES | inactive (10001nM) | inactive (110.14%) | inactive (1995.26nM) |
TK - FGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FGFR1 | inactive (3700nM) | inactive (88.45%) | inactive (1995.26nM) |
FGFR2 | active (1400nM) | inactive (73.67%) | - |
FGFR3 | inactive (3900nM) | inactive (86.17%) | inactive (1258.93nM) |
FGFR4 | inactive (10001nM) | inactive (91.11%) | - |
TK - VEGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FLT1 | inactive (5000nM) | inactive (97.29%) | inactive (>1995.26nM) |
FLT4 | inactive (10001nM) | inactive (92.08%) | inactive (>5011.87nM) |
KDR | active (2900nM) | inactive (102.69%) | inactive (1258.93nM) |
TK - InsR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IGF1R | inactive (10001nM) | inactive (97.48%) | inactive (>1995.26nM) |
INSR | inactive (10001nM) | inactive (97.23%) | inactive (>5011.87nM) |
IRR | inactive (10001nM) | inactive (96.89%) | - |
TK - JakA
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
JAK1 | inactive (10001nM) | inactive (100.97%) | - |
JAK2 | active (1000nM) | inactive (98.1%) | inactive (1258.93nM) |
JAK3 | active (640nM) | inactive (93.43%) | inactive (>3981.07nM) |
TYK2 | active (1800nM) | inactive (95.56%) | inactive (>1995.26nM) |
TK - Met
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MET | inactive (10001nM) | inactive (88.05%) | inactive (>3162.28nM) |
RON | inactive (10001nM) | inactive (105.71%) | inactive (>3162.28nM) |
TK - Musk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MUSK | inactive (10001nM) | inactive (105.64%) | - |
TK - Ret
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
RET | active (730nM) | active (45.99%) | inactive (>1000nM) |
TK - Sev
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ROS | inactive (10001nM) | inactive (88.88%) | inactive (>2511.89nM) |
TK - Syk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SYK | active (2900nM) | inactive (65.46%) | active (199.53nM) |
ZAP70 | inactive (10001nM) | inactive (117.42%) | - |
TK - Tie
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TIE1 | inactive (10001nM) | - | - |
TIE2 | inactive (10001nM) | inactive (91.28%) | - |
TK - Ack
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TNK1 | inactive (10001nM) | - | - |
ACK | active (5.6nM) | active (2.62%) | active (2.51nM) |
TK - Trk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TRKA | inactive (10001nM) | inactive (97.19%) | inactive (>2511.89nM) |
TRKB | inactive (10001nM) | inactive (96.45%) | inactive (>3981.07nM) |
TRKC | inactive (10001nM) | inactive (65.29%) | inactive (>2511.89nM) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ALK2 | active (620nM) | inactive (196.97%) | active (79.43nM) |
ALK4 | active (330nM) | inactive (108.71%) | - |
ACTR2 | active (210nM) | - | - |
ACTR2B | active (570nM) | - | - |
ALK1 | active (460nM) | active (15.93%) | - |
BMPR1A | inactive (7000nM) | - | - |
BMPR1B | active (53nM) | - | - |
BMPR2 | inactive (10001nM) | - | - |
TGFbR1 | active (230nM) | inactive (76.74%) | - |
TGFbR2 | active (2900nM) | inactive (98.29%) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SgK288 | inactive (10001nM) | - | - |
RIPK1 | inactive (10001nM) | - | - |
RIPK2 | active (31nM) | active (25.2%) | - |
ANKRD3 | inactive (10001nM) | - | - |
TKL - RAF
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
BRAF | active (500nM) | inactive (52.13%) | - |
RAF1 | active (570nM) | active (39.66%) | - |
ARAF | - | active (33.76%) | - |
TKL - MLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DLK | inactive (10001nM) | - | - |
LZK | inactive (5300nM) | - | - |
MLK1 | inactive (10001nM) | inactive (99.56%) | - |
MLK2 | inactive (10001nM) | inactive (93.68%) | inactive (2511.89nM) |
MLK3 | inactive (10001nM) | inactive (87.5%) | - |
TAK1 | inactive (3700nM) | inactive (87.31%) | - |
HH498 | active (11nM) | - | - |
ZAK | active (45nM) | active (8.63%) | active (50.12nM) |
TKL - IRAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IRAK1 | inactive (10001nM) | inactive (98.15%) | inactive (>7943.28nM) |
IRAK3 | inactive (10001nM) | - | - |
IRAK4 | inactive (10001nM) | inactive (88.46%) | inactive (5011.87nM) |
TKL - LISK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
LIMK1 | active (570nM) | active (16.71%) | active (251.19nM) |
LIMK2 | active (86nM) | - | - |
TESK1 | active (33nM) | - | - |
TKL - LRRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
LRRK2 | inactive (10001nM) | inactive (99.42%) | inactive (>2511.89nM) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz |
---|
ABC1 | 5 | 2 | - | - |
PIKK | 6 | 1 | - | - |
RIO | 3 | 3 | - | - |
Alpha | 6 | 1 | - | 1 |
PDHK | 5 | - | 1 | - |
Atypical - ABC1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ADCK3 | active (190nM) | - | - |
ADCK4 | inactive (10001nM) | - | - |
Atypical - PIKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FRAP | inactive (10001nM) | - | - |
Atypical - RIO
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
RIOK1 | inactive (10001nM) | - | - |
RIOK2 | inactive (10001nM) | - | - |
RIOK3 | inactive (10001nM) | - | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ChaK2 | inactive (10001nM) | - | - |
eEF2K | - | - | inactive (>3981.07nM) |
Atypical - PDHK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PDHK1 | - | inactive (94.13%) | - |
AGC
AGC - Akt
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AKT1 | inactive (10001nM) | inactive (96.7%) | inactive (>7943.28nM) |
AKT2 | inactive (10001nM) | inactive (94.1%) | inactive (>7943.28nM) |
AKT3 | inactive (10001nM) | inactive (89.91%) | inactive (>10000nM) |
AGC - DMPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CRIK | inactive (10001nM) | - | - |
DMPK1 | active (1300nM) | inactive (106.83%) | - |
DMPK2 | active (1200nM) | - | - |
MRCKa | active (2000nM) | inactive (99.22%) | inactive (6309.57nM) |
MRCKb | active (2100nM) | inactive (98.84%) | - |
ROCK1 | inactive (10001nM) | inactive (105.37%) | inactive (>6309.57nM) |
ROCK2 | inactive (10001nM) | inactive (90.06%) | inactive (>6309.57nM) |
AGC - GRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
RHOK | inactive (10001nM) | - | - |
GPRK4 | inactive (10001nM) | inactive (94.15%) | - |
GPRK7 | inactive (10001nM) | inactive (102.6%) | - |
BARK1 | - | inactive (96.96%) | - |
BARK2 | - | inactive (101.53%) | - |
GPRK5 | - | inactive (105.6%) | inactive (>3981.07nM) |
GPRK6 | - | inactive (100.73%) | - |
AGC - NDR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
LATS1 | inactive (10001nM) | - | - |
LATS2 | inactive (10001nM) | - | - |
NDR1 | inactive (10001nM) | inactive (101.48%) | - |
NDR2 | inactive (10001nM) | - | - |
AGC - MAST
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAST1 | inactive (10001nM) | - | - |
AGC - PDK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PDK1 | inactive (10001nM) | inactive (94.13%) | inactive (>3981.07nM) |
AGC - PKA
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKACa | inactive (10001nM) | inactive (101.59%) | inactive (>3981.07nM) |
PKACb | inactive (10001nM) | - | - |
PRKX | inactive (10001nM) | inactive (105.03%) | inactive (>2511.89nM) |
PKACg | - | inactive (114.3%) | - |
AGC - PKN
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKN1 | inactive (10001nM) | inactive (90.01%) | - |
PKN2 | inactive (10001nM) | inactive (103.29%) | inactive (5011.87nM) |
AGC - PKC
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKCd | inactive (10001nM) | inactive (99.57%) | inactive (>7943.28nM) |
PKCe | inactive (10001nM) | inactive (102.31%) | - |
PKCh | inactive (10001nM) | inactive (105.8%) | - |
PKCi | inactive (10001nM) | inactive (100.83%) | inactive (>5011.87nM) |
PKCt | inactive (10001nM) | inactive (97.28%) | inactive (>2511.89nM) |
PKCa | - | inactive (103.01%) | - |
PKCg | - | inactive (86.19%) | inactive (>7943.28nM) |
PKCz | - | inactive (100.58%) | inactive (>7943.28nM) |
PKCb | - | inactive (88.86%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKG1 | inactive (10001nM) | inactive (84.62%) | inactive (>1995.26nM) |
PKG2 | inactive (10001nM) | inactive (104.4%) | inactive (>1584.89nM) |
AGC - RSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
p70S6K | inactive (10001nM) | inactive (102.41%) | inactive (>6309.57nM) |
MSK1 | - | inactive (100.61%) | inactive (>1995.26nM) |
MSK2 | - | inactive (106.81%) | - |
p70S6Kb | - | inactive (101.47%) | - |
RSK2 | - | inactive (99.83%) | inactive (>3981.07nM) |
RSK4 | - | inactive (101.23%) | - |
RSK1 | - | inactive (96.24%) | - |
RSK3 | - | inactive (93.9%) | - |
AGC - SGK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SGK3 | inactive (10001nM) | inactive (101.99%) | - |
SGK1 | - | inactive (131.93%) | inactive (>7943.28nM) |
SGK2 | - | inactive (106.62%) | - |
AGC - YANK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
YANK1 | inactive (10001nM) | - | - |
YANK2 | inactive (10001nM) | - | - |
YANK3 | inactive (10001nM) | - | - |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AMPKa1 | inactive (10001nM) | - | inactive (>5011.87nM) |
AMPKa2 | inactive (10001nM) | - | - |
NuaK1 | inactive (10001nM) | inactive (110.42%) | - |
BRSK1 | inactive (10001nM) | inactive (102.96%) | inactive (>10000nM) |
BRSK2 | inactive (10001nM) | inactive (99.18%) | - |
CHK1 | inactive (10001nM) | inactive (95.99%) | inactive (>6309.57nM) |
HUNK | inactive (10001nM) | - | - |
LKB1 | inactive (10001nM) | inactive (107.79%) | - |
MARK1 | inactive (10001nM) | inactive (106.86%) | - |
MARK2 | inactive (10001nM) | inactive (109.6%) | inactive (>7943.28nM) |
MARK3 | inactive (10001nM) | inactive (97.78%) | inactive (>5011.87nM) |
MARK4 | inactive (10001nM) | inactive (90.93%) | inactive (>5011.87nM) |
MELK | inactive (10001nM) | inactive (81.38%) | inactive (>1995.26nM) |
NIM1 | inactive (10001nM) | - | - |
QSK | active (28nM) | - | - |
SIK | active (3.9nM) | - | - |
QIK | active (6.4nM) | active (1.91%) | active (0.79nM) |
NuaK2 | inactive (10001nM) | inactive (100.84%) | - |
SNRK | inactive (10001nM) | - | - |
PASK | - | inactive (109.65%) | - |
CAMK - CAMK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CaMK1a | inactive (10001nM) | inactive (105.77%) | inactive (>6309.57nM) |
CaMK1d | inactive (10001nM) | inactive (104.74%) | inactive (>2511.89nM) |
CaMK1g | inactive (10001nM) | inactive (104.01%) | - |
CaMK4 | inactive (10001nM) | inactive (91.32%) | - |
CaMK1b | - | inactive (102.39%) | - |
CAMK - CAMK2
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CaMK2a | inactive (10001nM) | inactive (103.21%) | inactive (>5011.87nM) |
CaMK2b | inactive (10001nM) | inactive (97.31%) | inactive (>7943.28nM) |
CaMK2d | inactive (10001nM) | inactive (109.11%) | inactive (>6309.57nM) |
CaMK2g | inactive (10001nM) | inactive (103.32%) | inactive (>6309.57nM) |
CAMK - CASK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CASK | inactive (10001nM) | - | - |
CAMK - RAD53
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CHK2 | inactive (10001nM) | inactive (103.19%) | inactive (>5011.87nM) |
CAMK - DAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DAPK1 | inactive (10001nM) | inactive (121.98%) | - |
DAPK2 | inactive (10001nM) | inactive (91.22%) | - |
DAPK3 | inactive (10001nM) | inactive (106.96%) | inactive (>2511.89nM) |
DRAK1 | inactive (10001nM) | inactive (106.96%) | inactive (>3981.07nM) |
DRAK2 | inactive (10001nM) | - | - |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DCLK1 | inactive (10001nM) | - | inactive (>10000nM) |
DCLK2 | inactive (10001nM) | inactive (99.83%) | - |
DCLK3 | inactive (10001nM) | - | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAPKAPK2 | inactive (10001nM) | inactive (99.53%) | inactive (>7943.28nM) |
MAPKAPK5 | inactive (10001nM) | inactive (94.94%) | inactive (>1584.89nM) |
MNK1 | inactive (10001nM) | inactive (91.34%) | - |
MNK2 | inactive (10001nM) | inactive (100.27%) | inactive (>10000nM) |
MAPKAPK3 | - | inactive (100.9%) | inactive (>10000nM) |
CAMK - MLCK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
caMLCK | inactive (10001nM) | - | - |
smMLCK | inactive (10001nM) | inactive (92.29%) | - |
skMLCK | inactive (3500nM) | inactive (97.31%) | - |
SgK085 | inactive (10001nM) | - | - |
CAMK - PHK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PHKg1 | inactive (10001nM) | inactive (94.33%) | - |
PHKg2 | inactive (10001nM) | inactive (101.21%) | inactive (>5011.87nM) |
CAMK - PIM
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PIM1 | inactive (10001nM) | inactive (102.17%) | inactive (>6309.57nM) |
PIM2 | inactive (10001nM) | inactive (112.82%) | inactive (>1584.89nM) |
PIM3 | inactive (10001nM) | inactive (96.26%) | inactive (>7943.28nM) |
CAMK - PKD
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKD1 | inactive (10001nM) | inactive (98.94%) | - |
PKD2 | inactive (10001nM) | inactive (93.01%) | inactive (>10000nM) |
PKD3 | inactive (10001nM) | inactive (89.94%) | inactive (>3981.07nM) |
CAMK - STK33
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
STK33 | inactive (10001nM) | inactive (88.69%) | - |
CAMK - TSSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TSSK1 | inactive (10001nM) | inactive (93.77%) | inactive (>1584.89nM) |
TSSK2 | - | inactive (93.88%) | inactive (>1584.89nM) |
STE
STE - STE11
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAP3K5 | inactive (10001nM) | inactive (97.25%) | - |
MAP3K6 | inactive (10001nM) | - | - |
MAP3K1 | inactive (10001nM) | - | - |
MAP3K7 | inactive (10001nM) | - | - |
MAP3K2 | active (140nM) | inactive (100.02%) | - |
MAP3K3 | active (280nM) | inactive (87.79%) | - |
MAP3K4 | active (310nM) | - | - |
MAP3K8 | active (79nM) | - | - |
STE - STE20
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
HPK1 | active (980nM) | - | - |
LOK | active (1200nM) | inactive (51.97%) | - |
GCK | active (1300nM) | inactive (79.44%) | inactive (>1584.89nM) |
KHS2 | active (640nM) | - | - |
HGK | inactive (3100nM) | active (49.2%) | inactive (>3162.28nM) |
KHS1 | active (45nM) | active (3.07%) | active (15.85nM) |
MINK | active (430nM) | active (46.54%) | active (794.33nM) |
MST1 | inactive (3800nM) | inactive (96.32%) | - |
MST2 | inactive (10001nM) | inactive (90.65%) | inactive (>6309.57nM) |
MST3 | inactive (10001nM) | inactive (103.89%) | - |
MST4 | active (1900nM) | inactive (84.13%) | - |
MYO3A | inactive (10001nM) | - | - |
MYO3B | inactive (10001nM) | inactive (84.82%) | - |
OSR1 | inactive (10001nM) | inactive (99.86%) | - |
PAK1 | inactive (10001nM) | inactive (102.2%) | inactive (>10000nM) |
PAK2 | inactive (10001nM) | inactive (113%) | - |
PAK3 | inactive (10001nM) | inactive (104.62%) | - |
PAK4 | inactive (10001nM) | inactive (98.71%) | inactive (>5011.87nM) |
PAK6 | inactive (10001nM) | inactive (135.67%) | - |
PAK5 | inactive (10001nM) | inactive (91.06%) | - |
SLK | active (720nM) | inactive (81.1%) | active (630.96nM) |
STLK3 | inactive (10001nM) | inactive (92.8%) | - |
TAO1 | inactive (10001nM) | inactive (101.17%) | active (1000nM) |
TAO2 | inactive (5400nM) | inactive (86.68%) | - |
TAO3 | active (2300nM) | inactive (95.32%) | - |
TNIK | active (2000nM) | - | - |
YSK1 | inactive (3400nM) | inactive (83.83%) | - |
STE - STE7
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAP2K1 | active (1000nM) | inactive (119.91%) | active (630.96nM) |
MAP2K2 | active (1400nM) | inactive (102.09%) | inactive (1584.89nM) |
MAP2K3 | inactive (10001nM) | - | - |
MAP2K4 | inactive (10001nM) | - | - |
MAP2K5 | active (3.3nM) | - | - |
MAP2K6 | inactive (10001nM) | inactive (95.15%) | - |
MAP2K7 | inactive (10001nM) | - | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
COT | - | inactive (97.56%) | - |
NIK | - | inactive (97.49%) | - |
CMGC
CMGC - CDK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PITSLRE | inactive (10001nM) | - | - |
CHED | inactive (10001nM) | - | - |
CDK11 | inactive (10001nM) | - | - |
PCTAIRE1 | inactive (10001nM) | - | - |
PCTAIRE2 | inactive (10001nM) | - | - |
PCTAIRE3 | inactive (10001nM) | - | - |
PFTAIRE2 | inactive (10001nM) | - | - |
PFTAIRE1 | inactive (10001nM) | - | - |
CDC2 | - | - | inactive (>7943.28nM) |
CDK2 | - | - | inactive (>7943.28nM) |
CDK5 | - | - | inactive (>7943.28nM) |
CDK8 | - | - | inactive (>3981.07nM) |
CDK7 | - | - | inactive (>3981.07nM) |
CDK9 | - | - | inactive (>1584.89nM) |
CMGC - CDKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CDKL1 | inactive (10001nM) | - | - |
CDKL2 | inactive (10001nM) | - | - |
CDKL3 | inactive (10001nM) | - | - |
CDKL5 | inactive (10001nM) | - | - |
CMGC - CLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CLK1 | inactive (10001nM) | inactive (102.24%) | - |
CLK2 | inactive (10001nM) | inactive (87.18%) | inactive (>3162.28nM) |
CLK3 | inactive (10001nM) | inactive (95.25%) | - |
CLK4 | inactive (10001nM) | inactive (91.44%) | inactive (>2511.89nM) |
CMGC - CK2
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CK2a1 | inactive (10001nM) | inactive (105.07%) | inactive (>6309.57nM) |
CK2a2 | inactive (10001nM) | inactive (103.46%) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DYRK1A | inactive (10001nM) | inactive (105.65%) | inactive (>3981.07nM) |
DYRK1B | inactive (10001nM) | inactive (98.39%) | inactive (>2511.89nM) |
DYRK2 | inactive (10001nM) | inactive (113.47%) | - |
HIPK1 | inactive (10001nM) | inactive (99.48%) | - |
HIPK2 | inactive (10001nM) | inactive (97.11%) | inactive (>3162.28nM) |
HIPK3 | inactive (10001nM) | inactive (100.21%) | - |
HIPK4 | inactive (10001nM) | inactive (98.36%) | inactive (>7943.28nM) |
PRP4 | inactive (10001nM) | - | - |
DYRK3 | - | inactive (108.74%) | inactive (1258.93nM) |
DYRK4 | - | inactive (100.49%) | inactive (>7943.28nM) |
CMGC - MAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Erk1 | inactive (10001nM) | inactive (100.46%) | - |
Erk2 | inactive (10001nM) | inactive (93.25%) | inactive (>7943.28nM) |
Erk3 | inactive (10001nM) | - | - |
Erk4 | inactive (10001nM) | - | - |
Erk5 | inactive (10001nM) | - | - |
Erk7 | inactive (10001nM) | - | - |
JNK1 | inactive (10001nM) | inactive (105.91%) | inactive (>3981.07nM) |
JNK2 | inactive (10001nM) | inactive (109.51%) | inactive (>3981.07nM) |
JNK3 | inactive (10001nM) | inactive (100.47%) | inactive (>3162.28nM) |
NLK | active (260nM) | active (27.49%) | - |
p38a | active (27nM) | active (36.53%) | active (31.62nM) |
p38b | active (410nM) | inactive (76.58%) | - |
p38d | inactive (10001nM) | inactive (99.26%) | inactive (>7943.28nM) |
p38g | inactive (10001nM) | inactive (99.88%) | inactive (>6309.57nM) |
CMGC - GSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
GSK3A | inactive (10001nM) | inactive (103.41%) | inactive (>6309.57nM) |
GSK3B | inactive (10001nM) | inactive (97.33%) | inactive (>5011.87nM) |
CMGC - RCK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ICK | inactive (10001nM) | - | - |
MAK | inactive (10001nM) | - | - |
CMGC - SRPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SRPK1 | inactive (10001nM) | inactive (100.55%) | inactive (>7943.28nM) |
SRPK2 | inactive (10001nM) | inactive (103.76%) | - |
MSSK1 | inactive (10001nM) | inactive (101.86%) | - |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz |
---|
CK1 | 7 | 7 | 6 | 5 |
VRK | 3 | 1 | 1 | - |
CK1 - CK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CK1a | inactive (10001nM) | inactive (98.25%) | inactive (>5011.87nM) |
CK1a2 | inactive (10001nM) | - | - |
CK1d | inactive (10001nM) | inactive (84.09%) | inactive (>7943.28nM) |
CK1e | active (1500nM) | inactive (89.5%) | - |
CK1g1 | inactive (10001nM) | inactive (96.56%) | inactive (>6309.57nM) |
CK1g2 | inactive (10001nM) | inactive (97.24%) | inactive (>7943.28nM) |
CK1g3 | inactive (10001nM) | inactive (97.19%) | inactive (>6309.57nM) |
CK1 - VRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
VRK2 | inactive (3200nM) | - | - |
VRK1 | - | inactive (97.72%) | - |