Compound Information
Test on : RBC
Compound Name : dorsomorphin
Inchikey : XHBVYDAKJHETMP-UHFFFAOYSA-N
ChemSpider : 9698930
Pubchem CID : 11524144
ChEMBL : CHEMBL478629
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC |
---|
PDK1 | inactive (110.45%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC |
---|
AKT1 | inactive (103.96%) |
AKT2 | inactive (87.63%) |
AKT3 | inactive (104.38%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC |
---|
DMPK1 | inactive (99.28%) |
MRCKa | inactive (100.37%) |
MRCKb | inactive (95.69%) |
ROCK1 | inactive (92.16%) |
ROCK2 | inactive (100.42%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC |
---|
BARK1 | inactive (81.77%) |
BARK2 | inactive (93.3%) |
GPRK4 | inactive (97.94%) |
GPRK5 | inactive (111.48%) |
GPRK6 | inactive (90.16%) |
GPRK7 | inactive (92.78%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC |
---|
MSK1 | inactive (82.98%) |
MSK2 | inactive (89.22%) |
p70S6K | inactive (82.22%) |
p70S6Kb | inactive (94.86%) |
RSK2 | inactive (85.35%) |
RSK4 | inactive (74.28%) |
RSK1 | inactive (79.22%) |
RSK3 | inactive (80.99%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC |
---|
PKACg | - |
PRKX | inactive (58.23%) |
PKACa | inactive (81.21%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC |
---|
PKCa | inactive (90.39%) |
PKCd | inactive (93.93%) |
PKCe | inactive (105.71%) |
PKCh | inactive (94.98%) |
PKCg | inactive (89.63%) |
PKCi | inactive (98.09%) |
PKCt | inactive (104.19%) |
PKCz | inactive (101.41%) |
PKCb | inactive (127.39%) |
AGC - PKG
Bioactivity |
---|
Kinase | RBC |
---|
PKG2 | inactive (77.43%) |
PKG1 | inactive (57.6%) |
AGC - PKN
Bioactivity |
---|
Kinase | RBC |
---|
PKN1 | active (44.65%) |
PKN2 | inactive (69.17%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC |
---|
SGK1 | inactive (55.22%) |
SGK2 | inactive (83.96%) |
SGK3 | inactive (93.9%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC |
---|
NDR1 | active (0%) |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC |
---|
ABL1 | active (7.87%) |
ABL2 | active (13.59%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC |
---|
ACK | inactive (82.17%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC |
---|
ALK | inactive (84.48%) |
LTK | inactive (95.43%) |
TK - Axl
Bioactivity |
---|
Kinase | RBC |
---|
AXL | inactive (91.09%) |
MER | inactive (82.19%) |
TYRO3 | inactive (91.63%) |
TK - Src
Bioactivity |
---|
Kinase | RBC |
---|
BLK | inactive (84.48%) |
BRK | active (37.25%) |
SRC | active (5.82%) |
FGR | active (27.51%) |
FRK | inactive (66.46%) |
FYN | active (20.87%) |
HCK | inactive (62.63%) |
LCK | inactive (51.8%) |
SRM | inactive (98%) |
YES | active (15.94%) |
LYN | active (12.85%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC |
---|
BMX | inactive (95.41%) |
BTK | active (42.83%) |
ITK | active (39.86%) |
TEC | inactive (151.81%) |
TXK | inactive (54.39%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC |
---|
KIT | active (21.4%) |
FLT3 | active (0.16%) |
FMS | active (19.75%) |
PDGFRb | active (20.38%) |
PDGFRa | active (3.7%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC |
---|
CSK | inactive (59.11%) |
CTK | inactive (103.69%) |
TK - DDR
Bioactivity |
---|
Kinase | RBC |
---|
DDR2 | inactive (90.24%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC |
---|
EGFR | inactive (100.12%) |
ErbB2 | inactive (94.6%) |
ErbB4 | inactive (95.44%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC |
---|
EphA1 | active (31.37%) |
EphA2 | active (36.2%) |
EphA3 | inactive (55.7%) |
EphA4 | active (37.71%) |
EphA5 | inactive (66.4%) |
EphA6 | - |
EphA7 | inactive (79.81%) |
EphA8 | inactive (79.83%) |
EphB1 | active (17.03%) |
EphB2 | active (33.59%) |
EphB3 | inactive (96.98%) |
EphB4 | active (37.68%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC |
---|
FAK | inactive (109.95%) |
PYK2 | inactive (105.97%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC |
---|
FER | inactive (93.25%) |
FES | inactive (76.79%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC |
---|
FGFR1 | inactive (59.88%) |
FGFR2 | inactive (80.39%) |
FGFR3 | inactive (70.92%) |
FGFR4 | inactive (89.05%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC |
---|
FLT1 | inactive (59.53%) |
FLT4 | active (16.28%) |
KDR | active (22.23%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC |
---|
IGF1R | inactive (93.98%) |
IRR | inactive (90.13%) |
INSR | inactive (94.88%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC |
---|
JAK1 | inactive (101.38%) |
JAK2 | inactive (102.96%) |
JAK3 | inactive (97.74%) |
TYK2 | inactive (69.75%) |
TK - Musk
Bioactivity |
---|
Kinase | RBC |
---|
MUSK | active (47.31%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC |
---|
RET | active (32.17%) |
TK - Met
Bioactivity |
---|
Kinase | RBC |
---|
RON | inactive (101.79%) |
MET | inactive (91.07%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC |
---|
ROS | inactive (93.55%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC |
---|
SYK | inactive (87.45%) |
ZAP70 | inactive (94.47%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC |
---|
TIE2 | inactive (99.34%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC |
---|
TRKA | inactive (104.55%) |
TRKB | active (26.06%) |
TRKC | active (7.7%) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC |
---|
ALK1 | active (21.58%) |
ALK2 | active (15.38%) |
ALK4 | inactive (112.07%) |
TGFbR1 | inactive (107.46%) |
TGFbR2 | active (18.72%) |
TKL - RAF
Bioactivity |
---|
Kinase | RBC |
---|
ARAF | inactive (55.63%) |
BRAF | inactive (93.28%) |
RAF1 | inactive (102%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC |
---|
IRAK1 | active (15.29%) |
IRAK4 | inactive (105.1%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC |
---|
LIMK1 | inactive (66.38%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC |
---|
LRRK2 | inactive (103.21%) |
TKL - MLK
Bioactivity |
---|
Kinase | RBC |
---|
MLK1 | inactive (70.53%) |
MLK2 | inactive (95.84%) |
MLK3 | inactive (57.5%) |
TAK1 | active (49.74%) |
ZAK | active (11.66%) |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC |
---|
RIPK2 | active (15.93%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC |
---|
NuaK1 | active (26.55%) |
BRSK1 | inactive (74.46%) |
BRSK2 | inactive (67.91%) |
CHK1 | inactive (86.4%) |
LKB1 | inactive (85.31%) |
MARK1 | inactive (58.73%) |
MARK3 | inactive (58.42%) |
MARK4 | active (48.34%) |
MELK | active (6.63%) |
PASK | inactive (86.28%) |
QIK | active (46.37%) |
NuaK2 | inactive (82.01%) |
MARK2 | inactive (53.06%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC |
---|
CaMK1a | inactive (90.81%) |
CaMK1b | inactive (100.02%) |
CaMK1d | inactive (95.39%) |
CaMK1g | inactive (99.85%) |
CaMK4 | inactive (92%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC |
---|
CaMK2a | inactive (69.09%) |
CaMK2b | inactive (67.17%) |
CaMK2d | inactive (54.45%) |
CaMK2g | inactive (74.84%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC |
---|
CHK2 | inactive (92.69%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC |
---|
DAPK1 | inactive (89.62%) |
DAPK2 | inactive (90.2%) |
DRAK1 | active (48.77%) |
DAPK3 | inactive (91.63%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC |
---|
DCLK2 | inactive (94.05%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC |
---|
MAPKAPK2 | inactive (86.63%) |
MAPKAPK3 | inactive (94.17%) |
MAPKAPK5 | inactive (91.26%) |
MNK1 | active (40.44%) |
MNK2 | inactive (65.4%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC |
---|
smMLCK | inactive (91.62%) |
skMLCK | active (9.29%) |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC |
---|
PHKg1 | active (13.66%) |
PHKg2 | active (31.19%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC |
---|
PIM1 | inactive (96.72%) |
PIM2 | inactive (111.6%) |
PIM3 | inactive (83.79%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC |
---|
PKD1 | inactive (81.91%) |
PKD3 | inactive (73.17%) |
PKD2 | inactive (88.33%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC |
---|
TSSK1 | inactive (81.11%) |
TSSK2 | inactive (99.01%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC |
---|
STK33 | active (37.41%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC |
---|
MAP3K5 | inactive (98.41%) |
MAP3K2 | inactive (92.14%) |
MAP3K3 | inactive (102.5%) |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC |
---|
COT | inactive (103.58%) |
NIK | inactive (110.87%) |
STE - STE20
Bioactivity |
---|
Kinase | RBC |
---|
GCK | active (10.79%) |
HGK | active (28.98%) |
KHS1 | active (7.24%) |
LOK | active (41.76%) |
MINK | inactive (59.42%) |
MST1 | inactive (86.81%) |
MST2 | inactive (93.88%) |
MST3 | inactive (95.46%) |
MST4 | inactive (87.29%) |
OSR1 | inactive (99.37%) |
PAK1 | inactive (89.84%) |
PAK2 | inactive (105.07%) |
PAK3 | inactive (102.16%) |
PAK4 | inactive (109.3%) |
PAK5 | inactive (93.22%) |
PAK6 | inactive (94.16%) |
SLK | inactive (74.86%) |
YSK1 | inactive (91.13%) |
STLK3 | inactive (76.83%) |
TAO1 | inactive (84.83%) |
TAO2 | inactive (90.33%) |
TAO3 | inactive (104.39%) |
MYO3B | active (0%) |
STE - STE7
Bioactivity |
---|
Kinase | RBC |
---|
MAP2K1 | inactive (98.77%) |
MAP2K2 | inactive (81.86%) |
MAP2K6 | inactive (87.8%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC |
---|
AurA | inactive (74.83%) |
AurB | inactive (54.97%) |
AurC | inactive (70.42%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC |
---|
CaMKK1 | inactive (59.24%) |
CaMKK2 | active (30.45%) |
Other - Haspin
Bioactivity |
---|
Kinase | RBC |
---|
Haspin | inactive (64.05%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC |
---|
IKKa | inactive (103.95%) |
IKKb | inactive (103.9%) |
IKKe | inactive (71.92%) |
TBK1 | inactive (57.21%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC |
---|
NEK1 | inactive (88.95%) |
NEK11 | inactive (96.68%) |
NEK2 | inactive (101.51%) |
NEK4 | inactive (82.55%) |
NEK6 | inactive (109.02%) |
NEK7 | inactive (87.25%) |
NEK9 | inactive (96.37%) |
NEK3 | inactive (111.28%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC |
---|
PBK | inactive (79.74%) |
Other - PLK
Bioactivity |
---|
Kinase | RBC |
---|
PLK1 | inactive (107.02%) |
PLK2 | inactive (97.12%) |
PLK3 | inactive (93.96%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC |
---|
SgK496 | inactive (98.27%) |
Other - NAK
Bioactivity |
---|
Kinase | RBC |
---|
MPSK1 | active (40.89%) |
Other - TTK
Bioactivity |
---|
Kinase | RBC |
---|
TTK | inactive (82.83%) |
Other - ULK
Bioactivity |
---|
Kinase | RBC |
---|
ULK1 | active (44.29%) |
ULK2 | inactive (72.29%) |
ULK3 | active (0%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC |
---|
Wee1 | inactive (75.44%) |
Other - WNK
Bioactivity |
---|
Kinase | RBC |
---|
Wnk2 | inactive (119.54%) |
Wnk3 | inactive (78.07%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC |
---|
TLK2 | active (0%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
CK1 | 7 | 6 |
VRK | 3 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC |
---|
CK1d | active (22.64%) |
CK1g1 | inactive (88.73%) |
CK1g2 | inactive (74.42%) |
CK1g3 | inactive (86.26%) |
CK1a | inactive (55.12%) |
CK1e | inactive (51.63%) |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC |
---|
VRK1 | inactive (86.04%) |
CMGC
CMGC - CK2
Bioactivity |
---|
Kinase | RBC |
---|
CK2a1 | inactive (87.46%) |
CK2a2 | active (34.63%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC |
---|
CLK1 | active (20.03%) |
CLK2 | active (21.34%) |
CLK3 | inactive (92.18%) |
CLK4 | active (5.73%) |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC |
---|
DYRK1A | active (20.67%) |
DYRK1B | active (26.16%) |
DYRK2 | active (47.05%) |
DYRK3 | inactive (76.8%) |
DYRK4 | inactive (92.98%) |
HIPK1 | inactive (97.06%) |
HIPK2 | inactive (70.83%) |
HIPK3 | inactive (89.41%) |
HIPK4 | inactive (114.96%) |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC |
---|
Erk1 | inactive (109.78%) |
Erk2 | inactive (99.26%) |
JNK3 | inactive (103.57%) |
NLK | inactive (58.09%) |
p38a | inactive (92.24%) |
p38b | inactive (96.92%) |
p38d | inactive (96.87%) |
p38g | inactive (100.42%) |
JNK1 | inactive (91.51%) |
JNK2 | inactive (87.84%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC |
---|
GSK3A | inactive (80.74%) |
GSK3B | inactive (79.61%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC |
---|
MSSK1 | inactive (94.84%) |
SRPK1 | inactive (97.88%) |
SRPK2 | inactive (103.1%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
PDHK | 5 | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC |
---|
PDHK1 | inactive (110.45%) |