Compound Information
Test on : DRx, RBC
Compound Name
DRx, RBC : Gefitinib
Inchikey
Same : XGALLCVXEZPNRQ-N
DRx, RBC : XGALLCVXEZPNRQ-UHFFFAOYSA-N
ChemSpider
DRx, RBC : 110217
Pubchem CID
DRx, RBC : 123631
ChEMBL
DRx, RBC : CHEMBL939
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
Other
Other - NAK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
AAK1 | inactive (10001nM) | - |
BIKE | inactive (10001nM) | - |
GAK | active (13nM) | - |
MPSK1 | inactive (10001nM) | inactive (96.84%) |
Other - Aur
Bioactivity |
---|
Kinase | DRx | RBC |
---|
AurA | inactive (10001nM) | inactive (95.27%) |
AurB | inactive (10001nM) | inactive (105.68%) |
AurC | inactive (10001nM) | inactive (89.74%) |
Other - CAMKK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CaMKK1 | inactive (10001nM) | inactive (93.77%) |
CaMKK2 | inactive (10001nM) | inactive (102.66%) |
Other - PEK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
HRI | inactive (10001nM) | - |
PKR | inactive (10001nM) | - |
Other - IRE
Bioactivity |
---|
Kinase | DRx | RBC |
---|
IRE1 | inactive (10001nM) | - |
Other - IKK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
IKKa | inactive (10001nM) | inactive (94.87%) |
IKKb | inactive (10001nM) | inactive (86.54%) |
IKKe | inactive (10001nM) | inactive (89.85%) |
TBK1 | inactive (10001nM) | inactive (83.12%) |
Other - NEK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
NEK1 | inactive (10001nM) | inactive (90.42%) |
NEK11 | inactive (10001nM) | inactive (108.83%) |
NEK2 | inactive (10001nM) | inactive (98.44%) |
NEK3 | inactive (10001nM) | inactive (94.44%) |
NEK4 | inactive (10001nM) | inactive (103.13%) |
NEK5 | inactive (10001nM) | - |
NEK6 | inactive (10001nM) | inactive (89.9%) |
NEK7 | inactive (10001nM) | inactive (96.9%) |
NEK9 | inactive (10001nM) | inactive (99.33%) |
Other - WEE
Bioactivity |
---|
Kinase | DRx | RBC |
---|
MYT1 | inactive (10001nM) | - |
Wee1 | inactive (10001nM) | inactive (93.76%) |
Wee1B | inactive (10001nM) | - |
Other - PLK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PLK1 | inactive (10001nM) | inactive (96.99%) |
PLK2 | inactive (10001nM) | inactive (100.48%) |
PLK3 | inactive (10001nM) | inactive (103.02%) |
PLK4 | inactive (10001nM) | - |
Other - SgK496
Bioactivity |
---|
Kinase | DRx | RBC |
---|
SgK496 | inactive (10001nM) | inactive (101.21%) |
Other - NKF1
Bioactivity |
---|
Kinase | DRx | RBC |
---|
SBK | active (560nM) | - |
SgK110 | inactive (10001nM) | - |
Other - NKF4
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CLIK1 | inactive (10001nM) | - |
Other - ULK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
Fused | inactive (5700nM) | - |
ULK1 | inactive (10001nM) | inactive (93%) |
ULK2 | inactive (10001nM) | inactive (103.63%) |
ULK3 | inactive (10001nM) | inactive (107.59%) |
Other - TLK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
TLK1 | inactive (10001nM) | - |
TLK2 | inactive (10001nM) | inactive (80.44%) |
Other - TTK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
TTK | inactive (10001nM) | inactive (96.32%) |
Other - Haspin
Bioactivity |
---|
Kinase | DRx | RBC |
---|
Haspin | - | inactive (84.05%) |
Other - TOPK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PBK | - | inactive (101.69%) |
Other - WNK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
Wnk2 | - | inactive (97.23%) |
Wnk3 | - | inactive (102.14%) |
TK
TK - Abl
Bioactivity |
---|
Kinase | DRx | RBC |
---|
ABL1 | active (2200nM) | inactive (86.35%) |
ABL2 | active (1600nM) | inactive (71.98%) |
TK - ALK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
ALK | inactive (10001nM) | inactive (98.75%) |
LTK | inactive (5500nM) | inactive (90.35%) |
TK - Axl
Bioactivity |
---|
Kinase | DRx | RBC |
---|
AXL | active (1800nM) | inactive (88.8%) |
MER | inactive (10001nM) | inactive (95.91%) |
TYRO3 | inactive (10001nM) | inactive (94.86%) |
TK - Src
Bioactivity |
---|
Kinase | DRx | RBC |
---|
BLK | active (1200nM) | inactive (87.71%) |
BRK | inactive (10001nM) | inactive (77.22%) |
FGR | active (2600nM) | inactive (70.15%) |
FRK | active (2000nM) | inactive (97.87%) |
FYN | inactive (10001nM) | inactive (92.17%) |
HCK | inactive (4400nM) | inactive (73.33%) |
LCK | active (630nM) | inactive (68.44%) |
LYN | active (990nM) | inactive (57.09%) |
SRC | inactive (3800nM) | inactive (79%) |
SRM | inactive (10001nM) | inactive (96.36%) |
YES | inactive (10001nM) | inactive (74.36%) |
TK - Tec
Bioactivity |
---|
Kinase | DRx | RBC |
---|
BMX | inactive (10001nM) | inactive (102.44%) |
BTK | inactive (10001nM) | inactive (60.56%) |
ITK | inactive (10001nM) | inactive (99.94%) |
TEC | inactive (10001nM) | inactive (103.98%) |
TXK | inactive (6000nM) | inactive (83.21%) |
TK - PDGFR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
FMS | inactive (10001nM) | inactive (110.38%) |
FLT3 | inactive (3100nM) | inactive (56.47%) |
KIT | inactive (10001nM) | inactive (96.04%) |
PDGFRa | inactive (10001nM) | inactive (97%) |
PDGFRb | inactive (10001nM) | inactive (93.89%) |
TK - Csk
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CSK | inactive (10001nM) | inactive (95.4%) |
CTK | inactive (10001nM) | inactive (86.38%) |
TK - DDR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
DDR1 | inactive (10001nM) | - |
DDR2 | inactive (10001nM) | inactive (116.76%) |
TK - EGFR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
EGFR | active (1nM) | active (2.97%) |
ErbB2 | inactive (3500nM) | active (34.2%) |
ErbB3 | active (790nM) | - |
ErbB4 | active (410nM) | active (24.15%) |
TK - Eph
Bioactivity |
---|
Kinase | DRx | RBC |
---|
EphA1 | inactive (4000nM) | inactive (87.38%) |
EphA2 | inactive (10001nM) | inactive (85.71%) |
EphA3 | inactive (5500nM) | inactive (94.45%) |
EphA4 | inactive (10001nM) | inactive (90.23%) |
EphA5 | active (1500nM) | inactive (95.8%) |
EphA6 | active (590nM) | active (28.94%) |
EphA7 | inactive (10001nM) | inactive (74.31%) |
EphA8 | active (1800nM) | inactive (84.51%) |
EphB1 | active (1300nM) | inactive (94.76%) |
EphB2 | inactive (10001nM) | inactive (87.65%) |
EphB3 | inactive (10001nM) | inactive (57.52%) |
EphB4 | active (2500nM) | inactive (70.85%) |
EphB6 | inactive (3200nM) | - |
TK - FAK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
FAK | inactive (10001nM) | inactive (102.59%) |
PYK2 | inactive (10001nM) | inactive (98.87%) |
TK - Fer
Bioactivity |
---|
Kinase | DRx | RBC |
---|
FER | inactive (10001nM) | inactive (94.11%) |
FES | inactive (10001nM) | inactive (110.93%) |
TK - FGFR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
FGFR1 | inactive (10001nM) | inactive (96.4%) |
FGFR2 | inactive (10001nM) | inactive (98.73%) |
FGFR3 | inactive (10001nM) | inactive (79.32%) |
FGFR4 | inactive (10001nM) | inactive (92.38%) |
TK - VEGFR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
FLT1 | inactive (10001nM) | inactive (98.32%) |
FLT4 | inactive (10001nM) | inactive (92.15%) |
KDR | inactive (10001nM) | inactive (95.24%) |
TK - InsR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
IGF1R | inactive (10001nM) | inactive (92.33%) |
INSR | inactive (10001nM) | inactive (106.69%) |
IRR | inactive (10001nM) | inactive (111.76%) |
TK - JakA
Bioactivity |
---|
Kinase | DRx | RBC |
---|
JAK1 | inactive (10001nM) | inactive (101.53%) |
JAK2 | inactive (10001nM) | inactive (99.85%) |
JAK3 | inactive (10001nM) | inactive (96.64%) |
TYK2 | inactive (10001nM) | inactive (101.66%) |
TK - Met
Bioactivity |
---|
Kinase | DRx | RBC |
---|
MET | inactive (10001nM) | inactive (92.36%) |
RON | inactive (10001nM) | inactive (97.71%) |
TK - Musk
Bioactivity |
---|
Kinase | DRx | RBC |
---|
MUSK | inactive (10001nM) | inactive (98.12%) |
TK - Ret
Bioactivity |
---|
Kinase | DRx | RBC |
---|
RET | inactive (10001nM) | inactive (76.94%) |
TK - Sev
Bioactivity |
---|
Kinase | DRx | RBC |
---|
ROS | inactive (10001nM) | inactive (92.33%) |
TK - Syk
Bioactivity |
---|
Kinase | DRx | RBC |
---|
SYK | inactive (10001nM) | inactive (104.18%) |
ZAP70 | inactive (10001nM) | inactive (96.47%) |
TK - Tie
Bioactivity |
---|
Kinase | DRx | RBC |
---|
TIE1 | inactive (10001nM) | - |
TIE2 | inactive (10001nM) | inactive (96.18%) |
TK - Ack
Bioactivity |
---|
Kinase | DRx | RBC |
---|
TNK1 | inactive (10001nM) | - |
ACK | inactive (10001nM) | inactive (72.8%) |
TK - Trk
Bioactivity |
---|
Kinase | DRx | RBC |
---|
TRKA | inactive (10001nM) | inactive (103.32%) |
TRKB | inactive (10001nM) | inactive (98.16%) |
TRKC | inactive (10001nM) | inactive (102.82%) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
ALK2 | inactive (10001nM) | inactive (105.63%) |
ALK4 | inactive (10001nM) | inactive (99.64%) |
ACTR2 | inactive (10001nM) | - |
ACTR2B | inactive (10001nM) | - |
ALK1 | inactive (10001nM) | inactive (96.86%) |
BMPR1A | inactive (10001nM) | - |
BMPR1B | inactive (10001nM) | - |
BMPR2 | inactive (10001nM) | - |
TGFbR1 | inactive (10001nM) | inactive (99.58%) |
TGFbR2 | inactive (10001nM) | inactive (93.77%) |
TKL - RIPK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
SgK288 | inactive (10001nM) | - |
RIPK1 | inactive (10001nM) | - |
RIPK2 | active (530nM) | active (33.98%) |
ANKRD3 | inactive (10001nM) | - |
TKL - RAF
Bioactivity |
---|
Kinase | DRx | RBC |
---|
BRAF | inactive (10001nM) | inactive (95.81%) |
RAF1 | inactive (10001nM) | inactive (90.93%) |
ARAF | - | inactive (95.27%) |
TKL - MLK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
DLK | inactive (10001nM) | - |
LZK | inactive (10001nM) | - |
MLK1 | inactive (10001nM) | inactive (109.52%) |
MLK2 | inactive (10001nM) | inactive (108.75%) |
MLK3 | inactive (10001nM) | inactive (102.32%) |
TAK1 | inactive (10001nM) | inactive (91.33%) |
HH498 | inactive (10001nM) | - |
ZAK | inactive (10001nM) | inactive (96.17%) |
TKL - IRAK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
IRAK1 | active (69nM) | inactive (57.64%) |
IRAK3 | active (1500nM) | - |
IRAK4 | active (540nM) | inactive (78.79%) |
TKL - LISK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
LIMK1 | inactive (10001nM) | inactive (89.98%) |
LIMK2 | inactive (10001nM) | - |
TESK1 | inactive (10001nM) | - |
TKL - LRRK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
LRRK2 | inactive (10001nM) | inactive (107.6%) |
Atypical
Atypical - ABC1
Bioactivity |
---|
Kinase | DRx | RBC |
---|
ADCK3 | inactive (10001nM) | - |
ADCK4 | inactive (10001nM) | - |
Atypical - PIKK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
FRAP | inactive (10001nM) | - |
Atypical - RIO
Bioactivity |
---|
Kinase | DRx | RBC |
---|
RIOK1 | inactive (10001nM) | - |
RIOK2 | inactive (10001nM) | - |
RIOK3 | inactive (10001nM) | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | DRx | RBC |
---|
ChaK2 | inactive (10001nM) | - |
Atypical - PDHK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PDHK1 | - | inactive (88.16%) |
AGC
AGC - Akt
Bioactivity |
---|
Kinase | DRx | RBC |
---|
AKT1 | inactive (10001nM) | inactive (94.14%) |
AKT2 | inactive (10001nM) | inactive (111.08%) |
AKT3 | inactive (10001nM) | inactive (84.59%) |
AGC - DMPK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CRIK | active (1300nM) | - |
DMPK1 | inactive (6900nM) | inactive (90.09%) |
DMPK2 | inactive (10001nM) | - |
MRCKa | inactive (10001nM) | inactive (87.78%) |
MRCKb | inactive (10001nM) | inactive (98.96%) |
ROCK1 | inactive (10001nM) | inactive (105.65%) |
ROCK2 | inactive (10001nM) | inactive (90.75%) |
AGC - GRK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
RHOK | inactive (10001nM) | - |
GPRK4 | inactive (10001nM) | inactive (91.01%) |
GPRK7 | inactive (10001nM) | inactive (96.18%) |
BARK1 | - | inactive (93.33%) |
BARK2 | - | inactive (97.93%) |
GPRK5 | - | inactive (94.88%) |
GPRK6 | - | inactive (99.6%) |
AGC - NDR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
LATS1 | inactive (10001nM) | - |
LATS2 | inactive (10001nM) | - |
NDR1 | inactive (10001nM) | inactive (105.13%) |
NDR2 | inactive (10001nM) | - |
AGC - MAST
Bioactivity |
---|
Kinase | DRx | RBC |
---|
MAST1 | inactive (10001nM) | - |
AGC - PDK1
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PDK1 | inactive (10001nM) | inactive (88.16%) |
AGC - PKA
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PKACa | inactive (10001nM) | inactive (96.28%) |
PKACb | inactive (10001nM) | - |
PRKX | inactive (10001nM) | inactive (110.5%) |
PKACg | - | inactive (107.18%) |
AGC - PKN
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PKN1 | inactive (10001nM) | inactive (105.11%) |
PKN2 | inactive (10001nM) | inactive (93.08%) |
AGC - PKC
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PKCd | inactive (10001nM) | inactive (106%) |
PKCe | inactive (10001nM) | inactive (97.3%) |
PKCh | inactive (10001nM) | inactive (110.93%) |
PKCi | inactive (10001nM) | inactive (96.87%) |
PKCt | inactive (10001nM) | inactive (85.88%) |
PKCa | - | inactive (93.63%) |
PKCg | - | inactive (84.15%) |
PKCz | - | inactive (92.47%) |
PKCb | - | inactive (100.44%) |
AGC - PKG
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PKG1 | inactive (10001nM) | inactive (87.53%) |
PKG2 | inactive (10001nM) | inactive (94.76%) |
AGC - RSK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
p70S6K | inactive (10001nM) | inactive (93.87%) |
MSK1 | - | inactive (100.45%) |
MSK2 | - | inactive (104.47%) |
p70S6Kb | - | inactive (100.6%) |
RSK2 | - | inactive (100.01%) |
RSK4 | - | inactive (95.25%) |
RSK1 | - | inactive (97.28%) |
RSK3 | - | inactive (82.35%) |
AGC - SGK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
SGK3 | inactive (10001nM) | inactive (98.35%) |
SGK1 | - | inactive (131.23%) |
SGK2 | - | inactive (117.01%) |
AGC - YANK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
YANK1 | inactive (10001nM) | - |
YANK2 | inactive (10001nM) | - |
YANK3 | inactive (10001nM) | - |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | DRx | RBC |
---|
AMPKa1 | inactive (10001nM) | - |
AMPKa2 | inactive (10001nM) | - |
NuaK1 | inactive (10001nM) | inactive (99.06%) |
BRSK1 | inactive (10001nM) | inactive (92.5%) |
BRSK2 | inactive (10001nM) | inactive (103.09%) |
CHK1 | inactive (10001nM) | inactive (95.27%) |
HUNK | inactive (10001nM) | - |
LKB1 | inactive (10001nM) | inactive (106.26%) |
MARK1 | inactive (10001nM) | inactive (116.22%) |
MARK2 | inactive (10001nM) | inactive (119.2%) |
MARK3 | inactive (10001nM) | inactive (94.55%) |
MARK4 | inactive (10001nM) | inactive (94.21%) |
MELK | inactive (10001nM) | inactive (77.75%) |
NIM1 | inactive (10001nM) | - |
QSK | inactive (10001nM) | - |
SIK | inactive (10001nM) | - |
QIK | active (2100nM) | active (49.34%) |
NuaK2 | inactive (4600nM) | inactive (96.03%) |
SNRK | inactive (10001nM) | - |
PASK | - | inactive (97.94%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CaMK1a | inactive (10001nM) | inactive (101.56%) |
CaMK1d | inactive (10001nM) | inactive (88.64%) |
CaMK1g | inactive (10001nM) | inactive (103.44%) |
CaMK4 | inactive (10001nM) | inactive (93.3%) |
CaMK1b | - | inactive (108.09%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CaMK2a | inactive (10001nM) | inactive (94.45%) |
CaMK2b | inactive (10001nM) | inactive (95.43%) |
CaMK2d | inactive (10001nM) | inactive (92.43%) |
CaMK2g | inactive (10001nM) | inactive (128.23%) |
CAMK - CASK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CASK | inactive (10001nM) | - |
CAMK - RAD53
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CHK2 | active (800nM) | inactive (83.95%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
DAPK1 | inactive (10001nM) | inactive (108.61%) |
DAPK2 | inactive (10001nM) | inactive (93.17%) |
DAPK3 | inactive (5700nM) | inactive (95.66%) |
DRAK1 | active (2000nM) | inactive (95.96%) |
DRAK2 | inactive (3800nM) | - |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | DRx | RBC |
---|
DCLK1 | inactive (10001nM) | - |
DCLK2 | inactive (10001nM) | inactive (100.85%) |
DCLK3 | active (2900nM) | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
MAPKAPK2 | inactive (10001nM) | inactive (97.5%) |
MAPKAPK5 | inactive (10001nM) | inactive (92.66%) |
MNK1 | active (290nM) | active (41.86%) |
MNK2 | active (1200nM) | inactive (54.09%) |
MAPKAPK3 | - | inactive (99.61%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
caMLCK | inactive (10001nM) | - |
smMLCK | inactive (10001nM) | inactive (89.7%) |
skMLCK | active (1900nM) | inactive (99.24%) |
SgK085 | inactive (10001nM) | - |
CAMK - PHK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PHKg1 | inactive (3700nM) | inactive (68.81%) |
PHKg2 | active (2700nM) | inactive (93.88%) |
CAMK - PIM
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PIM1 | inactive (10001nM) | inactive (86.45%) |
PIM2 | inactive (10001nM) | inactive (96.22%) |
PIM3 | inactive (5800nM) | inactive (74.62%) |
CAMK - PKD
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PKD1 | inactive (3500nM) | inactive (85.4%) |
PKD2 | inactive (10001nM) | inactive (73.78%) |
PKD3 | inactive (10001nM) | inactive (76.27%) |
CAMK - STK33
Bioactivity |
---|
Kinase | DRx | RBC |
---|
STK33 | inactive (10001nM) | inactive (90.43%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
TSSK1 | inactive (10001nM) | inactive (89.98%) |
TSSK2 | - | inactive (91.51%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | DRx | RBC |
---|
MAP3K5 | inactive (10001nM) | inactive (102.87%) |
MAP3K6 | inactive (10001nM) | - |
MAP3K1 | inactive (10001nM) | - |
MAP3K7 | inactive (10001nM) | - |
MAP3K2 | inactive (3300nM) | inactive (108.9%) |
MAP3K3 | active (2100nM) | inactive (106.57%) |
MAP3K4 | inactive (10001nM) | - |
MAP3K8 | active (240nM) | - |
STE - STE20
Bioactivity |
---|
Kinase | DRx | RBC |
---|
HPK1 | inactive (10001nM) | - |
LOK | active (470nM) | active (38.59%) |
GCK | inactive (10001nM) | inactive (103.53%) |
KHS2 | inactive (10001nM) | - |
HGK | inactive (10001nM) | inactive (97.78%) |
KHS1 | inactive (10001nM) | inactive (79.95%) |
MINK | active (1800nM) | inactive (102.32%) |
MST1 | inactive (10001nM) | inactive (100.73%) |
MST2 | inactive (10001nM) | inactive (93.57%) |
MST3 | inactive (10001nM) | inactive (102.15%) |
MST4 | inactive (10001nM) | inactive (106.07%) |
MYO3A | inactive (10001nM) | - |
MYO3B | inactive (10001nM) | inactive (91.41%) |
OSR1 | inactive (10001nM) | inactive (101.19%) |
PAK1 | inactive (10001nM) | inactive (104.06%) |
PAK2 | inactive (10001nM) | inactive (100.18%) |
PAK3 | inactive (10001nM) | inactive (105.75%) |
PAK4 | inactive (10001nM) | inactive (90.22%) |
PAK6 | inactive (10001nM) | inactive (104.59%) |
PAK5 | inactive (10001nM) | inactive (97.39%) |
SLK | active (920nM) | inactive (83.71%) |
STLK3 | inactive (10001nM) | inactive (93.52%) |
TAO1 | inactive (10001nM) | inactive (103.35%) |
TAO2 | inactive (10001nM) | inactive (106.16%) |
TAO3 | inactive (10001nM) | inactive (99.52%) |
TNIK | inactive (6900nM) | - |
YSK1 | inactive (10001nM) | inactive (97.38%) |
STE - STE7
Bioactivity |
---|
Kinase | DRx | RBC |
---|
MAP2K1 | inactive (10001nM) | inactive (106.69%) |
MAP2K2 | inactive (10001nM) | inactive (101.76%) |
MAP2K3 | inactive (10001nM) | - |
MAP2K4 | inactive (10001nM) | - |
MAP2K5 | active (600nM) | - |
MAP2K6 | inactive (10001nM) | inactive (90.13%) |
MAP2K7 | inactive (10001nM) | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | DRx | RBC |
---|
COT | - | inactive (95.73%) |
NIK | - | inactive (103.54%) |
CMGC
CMGC - CDK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PITSLRE | inactive (10001nM) | - |
CHED | inactive (10001nM) | - |
CDK11 | inactive (10001nM) | - |
PCTAIRE1 | inactive (10001nM) | - |
PCTAIRE2 | inactive (10001nM) | - |
PCTAIRE3 | inactive (10001nM) | - |
PFTAIRE2 | inactive (10001nM) | - |
PFTAIRE1 | inactive (10001nM) | - |
CMGC - CDKL
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CDKL1 | inactive (10001nM) | - |
CDKL2 | inactive (10001nM) | - |
CDKL3 | inactive (10001nM) | - |
CDKL5 | inactive (10001nM) | - |
CMGC - CLK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CLK1 | inactive (10001nM) | inactive (105.34%) |
CLK2 | inactive (10001nM) | inactive (94.8%) |
CLK3 | inactive (10001nM) | inactive (105.68%) |
CLK4 | inactive (10001nM) | inactive (106.81%) |
CMGC - CK2
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CK2a1 | inactive (10001nM) | inactive (113.94%) |
CK2a2 | inactive (10001nM) | inactive (88.61%) |
CMGC - DYRK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
DYRK1A | inactive (10001nM) | inactive (101.21%) |
DYRK1B | inactive (10001nM) | inactive (91.87%) |
DYRK2 | inactive (10001nM) | inactive (98.2%) |
HIPK1 | inactive (10001nM) | inactive (97.55%) |
HIPK2 | inactive (10001nM) | inactive (99.71%) |
HIPK3 | inactive (10001nM) | inactive (102.72%) |
HIPK4 | active (310nM) | inactive (90.36%) |
PRP4 | inactive (10001nM) | - |
DYRK3 | - | inactive (84.98%) |
DYRK4 | - | inactive (104.94%) |
CMGC - MAPK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
Erk1 | inactive (10001nM) | inactive (100.48%) |
Erk2 | inactive (10001nM) | inactive (103.1%) |
Erk3 | active (1600nM) | - |
Erk4 | inactive (3100nM) | - |
Erk5 | inactive (10001nM) | - |
Erk7 | inactive (10001nM) | - |
JNK1 | inactive (10001nM) | inactive (93.07%) |
JNK2 | active (1700nM) | inactive (95.46%) |
JNK3 | inactive (3200nM) | inactive (101.5%) |
NLK | inactive (4200nM) | inactive (91.1%) |
p38a | inactive (10001nM) | inactive (74.59%) |
p38b | inactive (10001nM) | inactive (95.15%) |
p38d | inactive (10001nM) | inactive (94.68%) |
p38g | inactive (10001nM) | inactive (97.45%) |
CMGC - GSK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
GSK3A | inactive (10001nM) | inactive (99.73%) |
GSK3B | inactive (10001nM) | inactive (100.3%) |
CMGC - RCK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
ICK | inactive (10001nM) | - |
MAK | inactive (10001nM) | - |
CMGC - SRPK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
SRPK1 | inactive (10001nM) | inactive (98.31%) |
SRPK2 | inactive (10001nM) | inactive (99.49%) |
MSSK1 | inactive (10001nM) | inactive (102.83%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC |
---|
CK1 | 7 | 7 | 6 |
VRK | 3 | 1 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CK1a | inactive (10001nM) | inactive (98.63%) |
CK1a2 | inactive (10001nM) | - |
CK1d | inactive (3200nM) | inactive (90.37%) |
CK1e | active (430nM) | inactive (106.23%) |
CK1g1 | inactive (10001nM) | inactive (99.48%) |
CK1g2 | inactive (10001nM) | inactive (98.09%) |
CK1g3 | inactive (10001nM) | inactive (103.42%) |
CK1 - VRK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
VRK2 | inactive (10001nM) | - |
VRK1 | - | inactive (99.26%) |