Compound Information
Test on : RBC
Compound Name : -
Inchikey : XFXDYDZBKXMGBX-HOTGVXAUSA-N
CANNOT FIND
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC |
---|
PDK1 | inactive (95.96%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC |
---|
AKT1 | - |
AKT2 | inactive (100.47%) |
AKT3 | inactive (100.96%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC |
---|
DMPK1 | inactive (102.23%) |
MRCKa | inactive (96.27%) |
MRCKb | inactive (107.97%) |
ROCK1 | inactive (104.53%) |
ROCK2 | inactive (100.93%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC |
---|
BARK1 | inactive (100.81%) |
BARK2 | inactive (98.37%) |
GPRK4 | inactive (99.35%) |
GPRK5 | inactive (107.43%) |
GPRK6 | inactive (102.96%) |
GPRK7 | inactive (100.78%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC |
---|
MSK1 | inactive (107.12%) |
MSK2 | inactive (98.64%) |
p70S6K | inactive (98.41%) |
p70S6Kb | inactive (95.57%) |
RSK2 | inactive (98.67%) |
RSK4 | inactive (110.53%) |
RSK1 | inactive (105.55%) |
RSK3 | inactive (99.14%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC |
---|
PKACg | inactive (102.53%) |
PRKX | inactive (93.29%) |
PKACa | inactive (100.1%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC |
---|
PKCa | inactive (107.05%) |
PKCd | inactive (98.48%) |
PKCe | inactive (100.87%) |
PKCh | inactive (93.02%) |
PKCg | inactive (95.48%) |
PKCi | inactive (100.78%) |
PKCt | inactive (121.3%) |
PKCz | inactive (107.24%) |
PKCb | inactive (109.42%) |
AGC - PKG
Bioactivity |
---|
Kinase | RBC |
---|
PKG2 | inactive (91.94%) |
PKG1 | inactive (81.04%) |
AGC - PKN
Bioactivity |
---|
Kinase | RBC |
---|
PKN1 | inactive (97%) |
PKN2 | inactive (95.67%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC |
---|
SGK1 | inactive (103.96%) |
SGK2 | inactive (103.07%) |
SGK3 | inactive (99.26%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC |
---|
NDR1 | inactive (102.25%) |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC |
---|
ABL1 | inactive (101.38%) |
ABL2 | inactive (98.27%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC |
---|
ACK | inactive (100.32%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC |
---|
ALK | inactive (105.99%) |
LTK | inactive (105.99%) |
TK - Axl
Bioactivity |
---|
Kinase | RBC |
---|
AXL | inactive (99.92%) |
MER | inactive (92.12%) |
TYRO3 | inactive (97.91%) |
TK - Src
Bioactivity |
---|
Kinase | RBC |
---|
BLK | inactive (105.23%) |
BRK | inactive (88.53%) |
SRC | inactive (95.29%) |
FGR | inactive (97.16%) |
FRK | inactive (101.22%) |
FYN | inactive (95.05%) |
HCK | inactive (95.14%) |
LCK | inactive (99.26%) |
SRM | inactive (105.85%) |
YES | inactive (95.06%) |
LYN | inactive (103.47%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC |
---|
BMX | inactive (93.4%) |
BTK | inactive (106.32%) |
ITK | inactive (97.43%) |
TEC | inactive (109.06%) |
TXK | inactive (100.06%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC |
---|
KIT | inactive (92.71%) |
FLT3 | inactive (91.39%) |
FMS | inactive (100.42%) |
PDGFRb | inactive (104.55%) |
PDGFRa | inactive (96.31%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC |
---|
CSK | inactive (100.58%) |
CTK | inactive (94.1%) |
TK - DDR
Bioactivity |
---|
Kinase | RBC |
---|
DDR2 | inactive (96.12%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC |
---|
EGFR | inactive (102.62%) |
ErbB2 | inactive (98.89%) |
ErbB4 | inactive (86.8%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC |
---|
EphA1 | inactive (116.32%) |
EphA2 | inactive (101.73%) |
EphA3 | inactive (100.26%) |
EphA4 | inactive (105.17%) |
EphA5 | inactive (100.11%) |
EphA6 | inactive (103.8%) |
EphA7 | inactive (91.56%) |
EphA8 | inactive (93.51%) |
EphB1 | inactive (104.16%) |
EphB2 | inactive (111.28%) |
EphB3 | inactive (106.64%) |
EphB4 | inactive (90.31%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC |
---|
FAK | inactive (100.77%) |
PYK2 | inactive (94.62%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC |
---|
FER | inactive (96.37%) |
FES | inactive (100.05%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC |
---|
FGFR1 | inactive (88.14%) |
FGFR2 | inactive (103.6%) |
FGFR3 | inactive (99.79%) |
FGFR4 | inactive (95.92%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC |
---|
FLT1 | inactive (90.19%) |
FLT4 | inactive (123.49%) |
KDR | inactive (102.57%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC |
---|
IGF1R | inactive (99.49%) |
IRR | inactive (102.39%) |
INSR | inactive (84.98%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC |
---|
JAK1 | inactive (110.21%) |
JAK2 | inactive (96.65%) |
JAK3 | inactive (96.1%) |
TYK2 | inactive (105.65%) |
TK - Musk
Bioactivity |
---|
Kinase | RBC |
---|
MUSK | inactive (85.86%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC |
---|
RET | inactive (99.18%) |
TK - Met
Bioactivity |
---|
Kinase | RBC |
---|
RON | inactive (100.92%) |
MET | inactive (97.74%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC |
---|
ROS | inactive (91.8%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC |
---|
SYK | inactive (98.72%) |
ZAP70 | inactive (100.56%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC |
---|
TIE2 | inactive (99.08%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC |
---|
TRKA | inactive (106.27%) |
TRKB | inactive (104.63%) |
TRKC | inactive (102.77%) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC |
---|
ALK1 | inactive (100.74%) |
ALK2 | inactive (95.76%) |
ALK4 | inactive (86.5%) |
TGFbR1 | inactive (98.18%) |
TGFbR2 | inactive (139.72%) |
TKL - RAF
Bioactivity |
---|
Kinase | RBC |
---|
ARAF | inactive (99.62%) |
BRAF | inactive (101.55%) |
RAF1 | inactive (93.38%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC |
---|
IRAK1 | inactive (128.28%) |
IRAK4 | inactive (110.87%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC |
---|
LIMK1 | inactive (94.92%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC |
---|
LRRK2 | inactive (96.72%) |
TKL - MLK
Bioactivity |
---|
Kinase | RBC |
---|
MLK1 | inactive (88.08%) |
MLK2 | inactive (102.02%) |
MLK3 | inactive (96.68%) |
TAK1 | inactive (96.65%) |
ZAK | inactive (106.44%) |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC |
---|
RIPK2 | inactive (94.95%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC |
---|
NuaK1 | inactive (92.82%) |
BRSK1 | inactive (101.35%) |
BRSK2 | inactive (104.79%) |
CHK1 | inactive (98.63%) |
LKB1 | inactive (89.46%) |
MARK1 | inactive (99.18%) |
MARK3 | inactive (101.34%) |
MARK4 | inactive (96.44%) |
MELK | inactive (110.27%) |
PASK | inactive (96.31%) |
QIK | inactive (88.26%) |
NuaK2 | inactive (129.44%) |
MARK2 | inactive (99.36%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC |
---|
CaMK1a | inactive (108.34%) |
CaMK1b | inactive (102%) |
CaMK1d | inactive (103.91%) |
CaMK1g | inactive (98.02%) |
CaMK4 | inactive (97.48%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC |
---|
CaMK2a | inactive (105.14%) |
CaMK2b | inactive (97.08%) |
CaMK2d | inactive (96.39%) |
CaMK2g | inactive (105.71%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC |
---|
CHK2 | inactive (102.2%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC |
---|
DAPK1 | inactive (97.35%) |
DAPK2 | inactive (103.85%) |
DRAK1 | inactive (96.08%) |
DAPK3 | inactive (95.81%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC |
---|
DCLK2 | inactive (102.55%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC |
---|
MAPKAPK2 | inactive (100.05%) |
MAPKAPK3 | inactive (101.74%) |
MAPKAPK5 | inactive (95.17%) |
MNK1 | inactive (114.62%) |
MNK2 | inactive (88.15%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC |
---|
smMLCK | inactive (103.76%) |
skMLCK | inactive (101.26%) |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC |
---|
PHKg1 | inactive (97%) |
PHKg2 | inactive (110.64%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC |
---|
PIM1 | inactive (103.95%) |
PIM2 | inactive (104.64%) |
PIM3 | inactive (111.83%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC |
---|
PKD1 | inactive (100.01%) |
PKD3 | inactive (97.09%) |
PKD2 | inactive (101.61%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC |
---|
TSSK1 | inactive (105.64%) |
TSSK2 | inactive (98.73%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC |
---|
STK33 | inactive (100.65%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC |
---|
MAP3K5 | inactive (104.54%) |
MAP3K2 | inactive (98.17%) |
MAP3K3 | inactive (99.02%) |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC |
---|
COT | inactive (94.98%) |
NIK | inactive (117.75%) |
STE - STE20
Bioactivity |
---|
Kinase | RBC |
---|
GCK | inactive (105.58%) |
HGK | inactive (91.91%) |
KHS1 | inactive (105.52%) |
LOK | inactive (96.77%) |
MINK | inactive (103.25%) |
MST1 | inactive (106.12%) |
MST2 | inactive (104.47%) |
MST3 | inactive (93.22%) |
MST4 | inactive (106.06%) |
OSR1 | inactive (97.67%) |
PAK1 | inactive (99.28%) |
PAK2 | inactive (90.65%) |
PAK3 | inactive (103.49%) |
PAK4 | inactive (118.3%) |
PAK5 | inactive (101.46%) |
PAK6 | inactive (101.85%) |
SLK | inactive (99.69%) |
YSK1 | inactive (115.81%) |
STLK3 | inactive (94.19%) |
TAO1 | inactive (103.51%) |
TAO2 | inactive (98.16%) |
TAO3 | inactive (107.12%) |
MYO3B | inactive (106.82%) |
STE - STE7
Bioactivity |
---|
Kinase | RBC |
---|
MAP2K1 | inactive (97.77%) |
MAP2K2 | inactive (104.59%) |
MAP2K6 | inactive (109.72%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC |
---|
AurA | inactive (93.71%) |
AurB | inactive (100.74%) |
AurC | inactive (97.38%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC |
---|
CaMKK1 | inactive (121.86%) |
CaMKK2 | inactive (109.27%) |
Other - Haspin
Bioactivity |
---|
Kinase | RBC |
---|
Haspin | inactive (55.9%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC |
---|
IKKa | inactive (104.14%) |
IKKb | inactive (106.39%) |
IKKe | inactive (99.78%) |
TBK1 | inactive (99.69%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC |
---|
NEK1 | inactive (98.92%) |
NEK11 | inactive (77.41%) |
NEK2 | inactive (100.38%) |
NEK4 | inactive (95.24%) |
NEK6 | inactive (95.31%) |
NEK7 | inactive (99.83%) |
NEK9 | inactive (100.94%) |
NEK3 | inactive (92.41%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC |
---|
PBK | inactive (103.55%) |
Other - PLK
Bioactivity |
---|
Kinase | RBC |
---|
PLK1 | inactive (102.74%) |
PLK2 | inactive (101.49%) |
PLK3 | inactive (96.91%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC |
---|
SgK496 | inactive (99.63%) |
Other - NAK
Bioactivity |
---|
Kinase | RBC |
---|
MPSK1 | inactive (108.2%) |
Other - TTK
Bioactivity |
---|
Kinase | RBC |
---|
TTK | inactive (104.68%) |
Other - ULK
Bioactivity |
---|
Kinase | RBC |
---|
ULK1 | inactive (84.47%) |
ULK2 | inactive (97.96%) |
ULK3 | inactive (83.36%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC |
---|
Wee1 | inactive (89.06%) |
Other - WNK
Bioactivity |
---|
Kinase | RBC |
---|
Wnk2 | inactive (103.98%) |
Wnk3 | inactive (97.32%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC |
---|
TLK2 | inactive (101.62%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
CK1 | 7 | 6 |
VRK | 3 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC |
---|
CK1d | inactive (95.09%) |
CK1g1 | inactive (100.69%) |
CK1g2 | inactive (97.69%) |
CK1g3 | inactive (106.35%) |
CK1a | inactive (99.41%) |
CK1e | inactive (94.97%) |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC |
---|
VRK1 | inactive (103.8%) |
CMGC
CMGC - CK2
Bioactivity |
---|
Kinase | RBC |
---|
CK2a1 | inactive (95.27%) |
CK2a2 | inactive (95.25%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC |
---|
CLK1 | inactive (105.27%) |
CLK2 | inactive (105.6%) |
CLK3 | inactive (95.56%) |
CLK4 | inactive (99.27%) |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC |
---|
DYRK1A | inactive (97.69%) |
DYRK1B | inactive (105.62%) |
DYRK2 | inactive (85.77%) |
DYRK3 | inactive (95.47%) |
DYRK4 | inactive (100.44%) |
HIPK1 | inactive (97.73%) |
HIPK2 | inactive (93.58%) |
HIPK3 | inactive (105.54%) |
HIPK4 | inactive (89.99%) |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC |
---|
Erk1 | inactive (99.9%) |
Erk2 | inactive (97.17%) |
JNK3 | inactive (100.35%) |
NLK | inactive (102.63%) |
p38a | inactive (112.7%) |
p38b | inactive (103.52%) |
p38d | inactive (111.59%) |
p38g | inactive (104.09%) |
JNK1 | inactive (98.86%) |
JNK2 | inactive (100.87%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC |
---|
GSK3A | inactive (99.09%) |
GSK3B | inactive (107.73%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC |
---|
MSSK1 | inactive (101.99%) |
SRPK1 | inactive (105.93%) |
SRPK2 | inactive (100.56%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
PDHK | 5 | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC |
---|
PDHK1 | inactive (95.96%) |