Compound Information
Test on : RBC, Millipore
Compound Name
RBC, Millipore : -
Inchikey
Same : WXUJAQBSBZLVEV-N
RBC, Millipore : WXUJAQBSBZLVEV-UHFFFAOYSA-N
ChemSpider
RBC, Millipore : 4925373
Pubchem CID
RBC, Millipore : 6419741
ChEMBL
RBC, Millipore : -
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDK1 | inactive (89.04%) | inactive (56%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AKT1 | inactive (101.79%) | inactive (110%) |
AKT2 | inactive (120.66%) | inactive (96%) |
AKT3 | inactive (94.31%) | inactive (84%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DMPK1 | inactive (101.2%) | inactive (110%) |
MRCKa | inactive (92.7%) | inactive (99%) |
MRCKb | inactive (94.77%) | inactive (82%) |
ROCK1 | inactive (95.87%) | inactive (109%) |
ROCK2 | inactive (93.16%) | inactive (88%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BARK1 | inactive (107.14%) | - |
BARK2 | inactive (108.62%) | - |
GPRK4 | inactive (100.8%) | - |
GPRK5 | inactive (94.43%) | inactive (83%) |
GPRK6 | inactive (82.11%) | inactive (82%) |
GPRK7 | inactive (96.24%) | inactive (84%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSK1 | inactive (87.6%) | inactive (63%) |
MSK2 | inactive (61.29%) | inactive (53%) |
p70S6K | inactive (70.6%) | inactive (68%) |
p70S6Kb | inactive (74.71%) | - |
RSK2 | active (47.41%) | inactive (57%) |
RSK4 | active (33.37%) | active (37%) |
RSK1 | active (31.08%) | active (33%) |
RSK3 | active (32.73%) | inactive (58%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKACg | - | - |
PRKX | inactive (87.77%) | inactive (80%) |
PKACa | inactive (98.2%) | inactive (82%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKCa | inactive (66.55%) | inactive (97%) |
PKCd | inactive (64.97%) | inactive (79%) |
PKCe | inactive (84.9%) | inactive (105%) |
PKCh | inactive (74.81%) | inactive (85%) |
PKCg | inactive (116.7%) | inactive (71%) |
PKCi | inactive (82.28%) | inactive (102%) |
PKCt | inactive (88.94%) | inactive (71%) |
PKCz | inactive (84.76%) | inactive (113%) |
PKCb | inactive (94.66%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKG2 | inactive (64.12%) | - |
PKG1 | inactive (93.82%) | - |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKN1 | inactive (76.43%) | - |
PKN2 | inactive (95.47%) | inactive (69%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SGK1 | inactive (69.02%) | inactive (66%) |
SGK2 | inactive (75.25%) | inactive (52%) |
SGK3 | inactive (110.72%) | inactive (87%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NDR1 | active (0%) | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ABL1 | inactive (85.62%) | inactive (80%) |
ABL2 | inactive (79.94%) | inactive (91%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ACK | active (41.31%) | active (38%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK | inactive (84.62%) | inactive (77%) |
LTK | inactive (80.81%) | - |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AXL | inactive (91.74%) | inactive (86%) |
MER | inactive (53.92%) | active (37%) |
TYRO3 | inactive (88.83%) | inactive (95%) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BLK | inactive (73.95%) | inactive (57%) |
BRK | inactive (88.95%) | inactive (81%) |
SRC | inactive (88.4%) | inactive (100%) |
FGR | inactive (94.82%) | inactive (75%) |
FRK | inactive (96.8%) | inactive (87%) |
FYN | inactive (97.74%) | inactive (51%) |
HCK | inactive (94.55%) | inactive (54%) |
LCK | inactive (87.11%) | inactive (61%) |
SRM | inactive (100.33%) | - |
YES | inactive (79.94%) | inactive (90%) |
LYN | inactive (94.81%) | inactive (57%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BMX | inactive (91.71%) | inactive (54%) |
BTK | inactive (83.9%) | inactive (70%) |
ITK | inactive (71.36%) | inactive (85%) |
TEC | inactive (96.67%) | - |
TXK | inactive (76.44%) | inactive (71%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
KIT | active (38.05%) | active (11%) |
FLT3 | active (9.86%) | active (18%) |
FMS | inactive (64.86%) | active (26%) |
PDGFRb | inactive (68.44%) | inactive (88%) |
PDGFRa | inactive (84.42%) | inactive (96%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CSK | inactive (83.29%) | inactive (97%) |
CTK | inactive (99.81%) | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DDR2 | inactive (96.45%) | inactive (85%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EGFR | inactive (92.65%) | inactive (108%) |
ErbB2 | inactive (109.16%) | - |
ErbB4 | inactive (101.76%) | inactive (87%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EphA1 | inactive (72.45%) | inactive (74%) |
EphA2 | inactive (102.23%) | inactive (87%) |
EphA3 | inactive (105.06%) | inactive (91%) |
EphA4 | inactive (98.61%) | inactive (98%) |
EphA5 | inactive (92.04%) | inactive (105%) |
EphA6 | - | - |
EphA7 | inactive (78.81%) | inactive (86%) |
EphA8 | inactive (97.52%) | inactive (88%) |
EphB1 | inactive (93.96%) | inactive (90%) |
EphB2 | inactive (86.12%) | inactive (112%) |
EphB3 | inactive (79.71%) | inactive (121%) |
EphB4 | inactive (105.41%) | inactive (82%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FAK | inactive (56.91%) | inactive (57%) |
PYK2 | inactive (70.14%) | active (32%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FER | active (47.9%) | inactive (78%) |
FES | inactive (117.27%) | inactive (79%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FGFR1 | inactive (55.2%) | active (41%) |
FGFR2 | inactive (91.31%) | inactive (72%) |
FGFR3 | inactive (85.03%) | inactive (76%) |
FGFR4 | inactive (78.55%) | inactive (102%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FLT1 | inactive (57.99%) | active (16%) |
FLT4 | inactive (56.65%) | active (0%) |
KDR | inactive (66.6%) | active (10%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IGF1R | inactive (76.76%) | active (9%) |
IRR | active (20.7%) | active (5%) |
INSR | active (17.85%) | active (10%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
JAK1 | inactive (101.76%) | - |
JAK2 | inactive (116.64%) | inactive (97%) |
JAK3 | inactive (140.11%) | inactive (83%) |
TYK2 | inactive (85.37%) | - |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MUSK | inactive (54.43%) | inactive (72%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RET | active (41.97%) | inactive (59%) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RON | inactive (102.32%) | inactive (73%) |
MET | inactive (93.38%) | inactive (146%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ROS | inactive (76.96%) | inactive (97%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SYK | inactive (84.94%) | inactive (60%) |
ZAP70 | inactive (87.85%) | inactive (97%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TIE2 | inactive (78.94%) | inactive (98%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TRKA | inactive (89.78%) | active (21%) |
TRKB | active (49.03%) | active (48%) |
TRKC | active (26.12%) | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK1 | inactive (108.79%) | - |
ALK2 | inactive (103.46%) | - |
ALK4 | inactive (102.83%) | inactive (97%) |
TGFbR1 | inactive (96.29%) | inactive (91%) |
TGFbR2 | inactive (95.85%) | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ARAF | inactive (93.8%) | - |
BRAF | inactive (101%) | - |
RAF1 | inactive (108.07%) | inactive (68%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IRAK1 | inactive (83.13%) | inactive (76%) |
IRAK4 | inactive (84.84%) | inactive (61%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LIMK1 | inactive (74.71%) | inactive (71%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LRRK2 | inactive (61.31%) | - |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MLK1 | inactive (72.5%) | active (33%) |
MLK2 | inactive (82.47%) | - |
MLK3 | inactive (57.48%) | - |
TAK1 | inactive (63.38%) | inactive (55%) |
ZAK | inactive (78.73%) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RIPK2 | inactive (67.52%) | inactive (79%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NuaK1 | active (12.1%) | active (15%) |
BRSK1 | active (22.55%) | active (32%) |
BRSK2 | active (29.72%) | active (23%) |
CHK1 | active (24.64%) | active (18%) |
LKB1 | active (45.22%) | inactive (84%) |
MARK1 | active (36.72%) | active (25%) |
MARK3 | active (29.82%) | - |
MARK4 | active (26.82%) | - |
MELK | active (32.6%) | active (27%) |
PASK | active (33.63%) | inactive (57%) |
QIK | inactive (91.86%) | - |
NuaK2 | inactive (80.13%) | - |
MARK2 | active (34.69%) | active (40%) |
AMPKa1 | - | active (49%) |
AMPKa2 | - | active (38%) |
SIK | - | inactive (83%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK1a | inactive (83.34%) | inactive (61%) |
CaMK1b | inactive (105.24%) | - |
CaMK1d | inactive (91.91%) | inactive (71%) |
CaMK1g | inactive (94.66%) | - |
CaMK4 | inactive (89.75%) | inactive (61%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK2a | inactive (55.08%) | - |
CaMK2b | inactive (58.22%) | active (22%) |
CaMK2d | active (36.73%) | active (12%) |
CaMK2g | inactive (52.32%) | active (15%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CHK2 | active (21.23%) | active (23%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DAPK1 | active (26.61%) | inactive (57%) |
DAPK2 | active (43.83%) | active (9%) |
DRAK1 | active (36.56%) | active (10%) |
DAPK3 | active (29.61%) | active (27%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DCLK2 | inactive (82.28%) | inactive (96%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAPKAPK2 | inactive (98.94%) | inactive (79%) |
MAPKAPK3 | inactive (88.73%) | inactive (86%) |
MAPKAPK5 | inactive (123.19%) | inactive (97%) |
MNK1 | inactive (56.26%) | - |
MNK2 | active (35.04%) | active (32%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
smMLCK | active (15.53%) | active (11%) |
skMLCK | active (33.71%) | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PHKg1 | inactive (70.79%) | - |
PHKg2 | inactive (108.31%) | inactive (95%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PIM1 | active (1.43%) | active (6%) |
PIM2 | active (34.43%) | active (5%) |
PIM3 | active (4.48%) | active (14%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKD1 | inactive (61.42%) | active (41%) |
PKD3 | active (47.67%) | - |
PKD2 | inactive (69.38%) | inactive (90%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TSSK1 | inactive (84.44%) | inactive (83%) |
TSSK2 | inactive (99.13%) | inactive (83%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
STK33 | inactive (52.26%) | inactive (79%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP3K5 | inactive (97.85%) | inactive (99%) |
MAP3K2 | inactive (97.87%) | - |
MAP3K3 | inactive (86.92%) | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
COT | inactive (100.24%) | - |
NIK | inactive (83.01%) | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GCK | inactive (51.79%) | inactive (58%) |
HGK | active (21.23%) | - |
KHS1 | active (13.47%) | - |
LOK | inactive (69%) | inactive (70%) |
MINK | active (48.19%) | inactive (77%) |
MST1 | active (42.66%) | active (40%) |
MST2 | active (41.02%) | inactive (68%) |
MST3 | active (48.37%) | inactive (56%) |
MST4 | inactive (69.44%) | - |
OSR1 | inactive (97.17%) | - |
PAK1 | inactive (93.92%) | - |
PAK2 | inactive (99.04%) | inactive (98%) |
PAK3 | inactive (100.1%) | inactive (96%) |
PAK4 | inactive (97.06%) | inactive (81%) |
PAK5 | inactive (79.99%) | inactive (109%) |
PAK6 | inactive (85.49%) | inactive (98%) |
SLK | inactive (87.83%) | - |
YSK1 | inactive (72.51%) | - |
STLK3 | inactive (103.98%) | - |
TAO1 | inactive (134.62%) | inactive (78%) |
TAO2 | inactive (89.36%) | inactive (88%) |
TAO3 | inactive (66.9%) | inactive (69%) |
MYO3B | active (0%) | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP2K1 | inactive (101.61%) | inactive (59%) |
MAP2K2 | inactive (85.91%) | - |
MAP2K6 | inactive (65.72%) | inactive (69%) |
MAP2K7 | - | active (42%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AurA | active (34.84%) | active (14%) |
AurB | active (25.18%) | active (3%) |
AurC | active (47.6%) | active (37%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMKK1 | inactive (63.53%) | - |
CaMKK2 | inactive (77.18%) | - |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Haspin | active (33.51%) | active (8%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IKKa | inactive (100.28%) | inactive (63%) |
IKKb | inactive (95.85%) | inactive (94%) |
IKKe | inactive (102.88%) | - |
TBK1 | inactive (81.89%) | inactive (53%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NEK1 | inactive (75.19%) | - |
NEK11 | inactive (99.02%) | active (36%) |
NEK2 | inactive (87.49%) | inactive (77%) |
NEK4 | inactive (88.43%) | - |
NEK6 | inactive (88.71%) | inactive (98%) |
NEK7 | inactive (80.32%) | inactive (100%) |
NEK9 | inactive (77.4%) | - |
NEK3 | inactive (89.28%) | inactive (77%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PBK | inactive (72.38%) | - |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PLK1 | inactive (50.79%) | inactive (62%) |
PLK2 | inactive (63.76%) | active (38%) |
PLK3 | active (48.22%) | inactive (55%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SgK496 | inactive (105.92%) | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MPSK1 | inactive (70.91%) | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TTK | inactive (79.04%) | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ULK1 | inactive (97.2%) | - |
ULK2 | inactive (95.45%) | inactive (103%) |
ULK3 | active (0%) | inactive (80%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wee1 | inactive (94.65%) | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wnk2 | inactive (86.64%) | inactive (82%) |
Wnk3 | inactive (79.1%) | inactive (74%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TLK2 | active (0%) | inactive (74%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK1 | 7 | 6 | 4 |
VRK | 3 | 1 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK1d | active (17.19%) | active (15%) |
CK1g1 | inactive (68.36%) | inactive (58%) |
CK1g2 | inactive (63.42%) | active (40%) |
CK1g3 | inactive (87%) | active (46%) |
CK1a | inactive (51.59%) | - |
CK1e | active (18.88%) | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
VRK1 | inactive (78.08%) | - |
VRK2 | - | inactive (93%) |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK2 | 3 | 2 | 2 |
CLK | 4 | 4 | 2 |
DYRK | 10 | 9 | 4 |
MAPK | 14 | 10 | 10 |
GSK | 2 | 2 | 2 |
SRPK | 3 | 3 | 3 |
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK2a1 | inactive (52.61%) | inactive (60%) |
CK2a2 | inactive (53.37%) | inactive (81%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CLK1 | inactive (84%) | - |
CLK2 | inactive (94.7%) | inactive (51%) |
CLK3 | active (48.17%) | inactive (70%) |
CLK4 | inactive (99.01%) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DYRK1A | inactive (89.1%) | - |
DYRK1B | inactive (65.9%) | - |
DYRK2 | inactive (64.12%) | inactive (68%) |
DYRK3 | inactive (85.8%) | - |
DYRK4 | inactive (106.54%) | - |
HIPK1 | inactive (82.63%) | inactive (77%) |
HIPK2 | inactive (94.38%) | active (30%) |
HIPK3 | inactive (66.93%) | inactive (61%) |
HIPK4 | inactive (98.49%) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Erk1 | inactive (87.83%) | inactive (86%) |
Erk2 | inactive (124.65%) | inactive (109%) |
JNK3 | inactive (96.03%) | active (25%) |
NLK | inactive (87.92%) | inactive (89%) |
p38a | inactive (100.68%) | inactive (93%) |
p38b | inactive (94.53%) | inactive (90%) |
p38d | inactive (106.92%) | inactive (93%) |
p38g | inactive (85.93%) | inactive (95%) |
JNK1 | inactive (83.93%) | inactive (89%) |
JNK2 | inactive (65.3%) | inactive (67%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GSK3A | active (10.37%) | active (7%) |
GSK3B | active (30.83%) | active (26%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSSK1 | inactive (75.73%) | inactive (82%) |
SRPK1 | inactive (95.42%) | inactive (91%) |
SRPK2 | inactive (80.22%) | inactive (103%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
PDHK | 5 | 1 | - |
Alpha | 6 | - | 1 |
PIKK | 6 | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDHK1 | inactive (89.04%) | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
eEF2K | - | inactive (78%) |
Atypical - PIKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FRAP | - | inactive (75%) |