Compound Information
Test on : RBC, Metz, Millipore
Compound Name
RBC, Metz : Z-Semaxanib
Millipore : Semaxanib
Inchikey
Same : WUWDLXZGHZSWQZ-N
RBC, Metz : WUWDLXZGHZSWQZ-UHFFFAOYSA-N
Millipore : WUWDLXZGHZSWQZ-WQLSENKSSA-N
ChemSpider
RBC, Metz : 109638
Millipore : 4486260
Pubchem CID
RBC, Metz : 123015
Millipore : 5329098
ChEMBL
RBC, Metz : CHEMBL2002702
Millipore : CHEMBL276711
RBC, Metz | Millipore |
| |
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PDK1 | inactive (94.21%) | inactive (1995.26nM) | inactive (95%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
AKT1 | inactive (90.09%) | inactive (>7943.28nM) | inactive (89%) |
AKT2 | inactive (93.46%) | inactive (>7943.28nM) | inactive (114%) |
AKT3 | inactive (99.36%) | inactive (>10000nM) | inactive (101%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DMPK1 | inactive (101.12%) | - | inactive (84%) |
MRCKa | inactive (92.3%) | inactive (>10000nM) | inactive (119%) |
MRCKb | inactive (116.04%) | - | inactive (99%) |
ROCK1 | inactive (100.32%) | inactive (5011.87nM) | inactive (110%) |
ROCK2 | inactive (92.71%) | inactive (>7943.28nM) | inactive (88%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
BARK1 | inactive (92.01%) | - | - |
BARK2 | inactive (98.92%) | - | - |
GPRK4 | inactive (81.85%) | - | - |
GPRK5 | inactive (101.17%) | - | inactive (93%) |
GPRK6 | inactive (84.55%) | - | inactive (81%) |
GPRK7 | inactive (76.33%) | - | inactive (74%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MSK1 | inactive (76.61%) | inactive (>1995.26nM) | inactive (95%) |
MSK2 | inactive (78.42%) | - | inactive (61%) |
p70S6K | inactive (78.11%) | active (125.89nM) | active (38%) |
p70S6Kb | inactive (106.11%) | - | - |
RSK2 | inactive (50.91%) | active (158.49nM) | active (26%) |
RSK4 | active (39%) | - | active (38%) |
RSK1 | active (44.05%) | - | active (27%) |
RSK3 | active (35.25%) | - | inactive (51%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKACg | inactive (87.63%) | - | - |
PRKX | inactive (101%) | inactive (>1584.89nM) | inactive (94%) |
PKACa | inactive (93.13%) | inactive (>7943.28nM) | inactive (89%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKCa | inactive (95.62%) | - | inactive (100%) |
PKCd | inactive (91.67%) | inactive (>7943.28nM) | inactive (95%) |
PKCe | inactive (102.65%) | - | inactive (82%) |
PKCh | inactive (94.66%) | - | inactive (96%) |
PKCg | inactive (106.73%) | inactive (>7943.28nM) | inactive (106%) |
PKCi | inactive (97.5%) | - | inactive (79%) |
PKCt | inactive (98.51%) | - | inactive (103%) |
PKCz | inactive (89.88%) | inactive (>7943.28nM) | inactive (103%) |
PKCb | inactive (109%) | - | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKG2 | inactive (92.68%) | inactive (>1584.89nM) | - |
PKG1 | inactive (76.15%) | inactive (>1995.26nM) | - |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKN1 | inactive (96.39%) | - | - |
PKN2 | inactive (95.62%) | inactive (1258.93nM) | inactive (108%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
SGK1 | inactive (82.63%) | inactive (1995.26nM) | inactive (84%) |
SGK2 | inactive (94.43%) | - | inactive (80%) |
SGK3 | inactive (97.22%) | - | inactive (91%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
NDR1 | inactive (101.01%) | - | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ABL1 | inactive (95.24%) | inactive (>630.96nM) | inactive (81%) |
ABL2 | inactive (90.32%) | - | inactive (88%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ACK | inactive (75.85%) | - | inactive (52%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ALK | active (47.41%) | active (199.53nM) | active (37%) |
LTK | active (28.19%) | - | - |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
AXL | inactive (77.2%) | active (39.81nM) | active (31%) |
MER | inactive (68.34%) | - | active (4%) |
TYRO3 | inactive (81.02%) | inactive (>1995.26nM) | inactive (68%) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
BLK | inactive (71.53%) | active (100nM) | inactive (65%) |
BRK | inactive (83.59%) | inactive (>2511.89nM) | inactive (103%) |
SRC | inactive (86.54%) | inactive (1995.26nM) | inactive (78%) |
FGR | inactive (69.6%) | - | inactive (53%) |
FRK | inactive (92.58%) | inactive (1584.89nM) | inactive (89%) |
FYN | inactive (92.09%) | active (794.33nM) | inactive (75%) |
HCK | inactive (85.47%) | - | inactive (60%) |
LCK | inactive (81.03%) | active (1000nM) | inactive (83%) |
SRM | inactive (96.14%) | inactive (>1584.89nM) | - |
YES | inactive (53.64%) | - | inactive (58%) |
LYN | inactive (84.22%) | active (501.19nM) | active (46%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
BMX | inactive (94.18%) | - | inactive (87%) |
BTK | inactive (90.85%) | inactive (>1258.93nM) | inactive (89%) |
ITK | inactive (89.88%) | active (398.11nM) | inactive (66%) |
TEC | inactive (125.37%) | - | - |
TXK | inactive (93.41%) | - | inactive (103%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
KIT | active (31.52%) | inactive (>1258.93nM) | active (11%) |
FLT3 | active (3.07%) | active (5.01nM) | active (1%) |
FMS | active (28.53%) | active (19.95nM) | active (2%) |
PDGFRb | inactive (64.84%) | - | active (43%) |
PDGFRa | inactive (83.22%) | - | active (15%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CSK | inactive (99.39%) | - | inactive (121%) |
CTK | inactive (104.76%) | inactive (>1995.26nM) | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DDR2 | inactive (100.6%) | - | inactive (110%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
EGFR | inactive (91.7%) | inactive (>1995.26nM) | inactive (114%) |
ErbB2 | inactive (103.04%) | inactive (>1584.89nM) | - |
ErbB4 | inactive (80.75%) | inactive (>3981.07nM) | inactive (105%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
EphA1 | inactive (95.16%) | - | inactive (90%) |
EphA2 | inactive (103.8%) | inactive (>3162.28nM) | inactive (95%) |
EphA3 | inactive (95.93%) | - | inactive (101%) |
EphA4 | inactive (90.84%) | - | inactive (107%) |
EphA5 | inactive (87.38%) | - | inactive (99%) |
EphA6 | inactive (81.05%) | - | - |
EphA7 | inactive (86.92%) | - | inactive (85%) |
EphA8 | inactive (90.72%) | - | inactive (113%) |
EphB1 | inactive (88.77%) | - | inactive (102%) |
EphB2 | inactive (82.11%) | - | inactive (108%) |
EphB3 | inactive (92.83%) | - | inactive (113%) |
EphB4 | inactive (89.18%) | - | inactive (121%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FAK | inactive (61.48%) | inactive (>1584.89nM) | inactive (52%) |
PYK2 | inactive (66%) | active (316.23nM) | active (34%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FER | inactive (53.39%) | active (316.23nM) | inactive (100%) |
FES | inactive (90.52%) | inactive (>1995.26nM) | inactive (92%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FGFR1 | inactive (77.21%) | inactive (1258.93nM) | inactive (65%) |
FGFR2 | inactive (85.5%) | - | inactive (66%) |
FGFR3 | inactive (75.29%) | active (794.33nM) | inactive (80%) |
FGFR4 | inactive (69.27%) | - | inactive (124%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FLT1 | inactive (69.87%) | active (19.95nM) | active (3%) |
FLT4 | inactive (64.43%) | active (316.23nM) | active (1%) |
KDR | inactive (67.4%) | active (100nM) | active (4%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
IGF1R | inactive (80.97%) | inactive (>1000nM) | inactive (119%) |
IRR | inactive (74.16%) | - | inactive (65%) |
INSR | inactive (78.18%) | active (158.49nM) | active (30%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
JAK1 | inactive (84.9%) | - | - |
JAK2 | inactive (84.47%) | active (199.53nM) | inactive (108%) |
JAK3 | inactive (93.99%) | active (630.96nM) | inactive (98%) |
TYK2 | inactive (86.94%) | active (1000nM) | - |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MUSK | inactive (85.35%) | - | inactive (76%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
RET | active (17.64%) | active (31.62nM) | active (12%) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
RON | inactive (90.51%) | - | inactive (105%) |
MET | inactive (83.81%) | inactive (>3162.28nM) | inactive (101%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ROS | inactive (91.37%) | inactive (>1995.26nM) | inactive (100%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
SYK | inactive (92.46%) | active (794.33nM) | inactive (121%) |
ZAP70 | inactive (93.5%) | - | inactive (95%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TIE2 | inactive (89.94%) | - | inactive (74%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TRKA | active (42.83%) | active (251.19nM) | active (1%) |
TRKB | active (23.68%) | active (501.19nM) | active (40%) |
TRKC | active (6.15%) | active (19.95nM) | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ALK1 | inactive (104.23%) | - | - |
ALK2 | inactive (96.14%) | - | - |
ALK4 | inactive (100.54%) | - | inactive (112%) |
TGFbR1 | inactive (96.99%) | - | inactive (95%) |
TGFbR2 | inactive (113.87%) | - | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ARAF | inactive (115.89%) | - | - |
BRAF | inactive (111.24%) | - | - |
RAF1 | inactive (113.34%) | - | inactive (92%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
IRAK1 | inactive (98.66%) | inactive (1995.26nM) | inactive (76%) |
IRAK4 | active (45.85%) | active (1000nM) | active (39%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
LIMK1 | inactive (99.33%) | inactive (>10000nM) | inactive (112%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
LRRK2 | active (13.95%) | - | - |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MLK1 | active (39.5%) | - | active (10%) |
MLK2 | inactive (101.89%) | - | - |
MLK3 | active (17.59%) | - | - |
TAK1 | inactive (75.4%) | - | inactive (76%) |
ZAK | inactive (94.7%) | inactive (>7943.28nM) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
RIPK2 | inactive (81.38%) | - | inactive (94%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
NuaK1 | active (26.44%) | - | active (35%) |
BRSK1 | inactive (83.89%) | inactive (2511.89nM) | inactive (75%) |
BRSK2 | inactive (87.14%) | - | inactive (100%) |
CHK1 | inactive (71.87%) | inactive (>7943.28nM) | inactive (72%) |
LKB1 | inactive (87.61%) | - | inactive (103%) |
MARK1 | inactive (83.36%) | - | inactive (65%) |
MARK3 | inactive (80.26%) | inactive (1995.26nM) | - |
MARK4 | inactive (85.77%) | - | - |
MELK | inactive (77.94%) | inactive (>1584.89nM) | inactive (56%) |
PASK | inactive (99.68%) | - | inactive (111%) |
QIK | inactive (89.44%) | - | - |
NuaK2 | inactive (126.46%) | - | - |
MARK2 | inactive (88.07%) | inactive (1584.89nM) | inactive (78%) |
AMPKa1 | - | inactive (>7943.28nM) | inactive (55%) |
AMPKa2 | - | - | inactive (70%) |
SIK | - | - | inactive (115%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CaMK1a | inactive (103.86%) | inactive (5011.87nM) | inactive (86%) |
CaMK1b | inactive (91.08%) | - | - |
CaMK1d | inactive (94.56%) | - | inactive (102%) |
CaMK1g | inactive (100.75%) | - | - |
CaMK4 | inactive (96.51%) | - | inactive (104%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CaMK2a | inactive (84.54%) | - | - |
CaMK2b | inactive (93.98%) | inactive (6309.57nM) | inactive (81%) |
CaMK2d | inactive (83.79%) | active (630.96nM) | active (38%) |
CaMK2g | inactive (84.81%) | active (794.33nM) | active (32%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CHK2 | active (21.48%) | active (79.43nM) | active (18%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DAPK1 | inactive (108.93%) | - | inactive (95%) |
DAPK2 | inactive (101.31%) | - | inactive (91%) |
DRAK1 | inactive (52.94%) | active (125.89nM) | active (26%) |
DAPK3 | inactive (91.78%) | inactive (>1258.93nM) | inactive (88%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DCLK2 | inactive (95.81%) | - | inactive (90%) |
DCLK1 | - | inactive (>10000nM) | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MAPKAPK2 | inactive (100.28%) | inactive (>7943.28nM) | inactive (100%) |
MAPKAPK3 | inactive (99.04%) | inactive (>10000nM) | inactive (140%) |
MAPKAPK5 | inactive (88.87%) | inactive (>1584.89nM) | inactive (78%) |
MNK1 | inactive (105.14%) | - | - |
MNK2 | inactive (76.89%) | inactive (>10000nM) | inactive (100%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
smMLCK | inactive (68.73%) | - | active (32%) |
skMLCK | active (43.02%) | - | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PHKg1 | active (44.56%) | - | - |
PHKg2 | inactive (88.97%) | active (1000nM) | inactive (70%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PIM1 | inactive (95.75%) | inactive (>10000nM) | inactive (83%) |
PIM2 | inactive (100.76%) | inactive (>1584.89nM) | inactive (121%) |
PIM3 | inactive (87.93%) | inactive (>7943.28nM) | inactive (100%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKD1 | inactive (85.33%) | - | inactive (78%) |
PKD3 | inactive (81.64%) | inactive (5011.87nM) | - |
PKD2 | inactive (90.82%) | inactive (5011.87nM) | inactive (94%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TSSK1 | inactive (87.21%) | inactive (>1584.89nM) | inactive (91%) |
TSSK2 | inactive (94.06%) | inactive (>1584.89nM) | inactive (97%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
STK33 | inactive (72.09%) | - | inactive (69%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MAP3K5 | inactive (98.28%) | - | inactive (82%) |
MAP3K2 | inactive (95.84%) | - | - |
MAP3K3 | inactive (94.18%) | - | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
COT | inactive (116.22%) | - | - |
NIK | inactive (99%) | - | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
GCK | inactive (71.32%) | inactive (1584.89nM) | inactive (57%) |
HGK | active (48.78%) | active (199.53nM) | - |
KHS1 | active (39.69%) | active (501.19nM) | - |
LOK | inactive (71.86%) | - | inactive (86%) |
MINK | inactive (80.31%) | inactive (1258.93nM) | inactive (71%) |
MST1 | active (46.5%) | - | inactive (51%) |
MST2 | inactive (64.04%) | active (630.96nM) | inactive (70%) |
MST3 | inactive (99.66%) | - | inactive (96%) |
MST4 | inactive (95.24%) | - | - |
OSR1 | inactive (91.79%) | - | - |
PAK1 | inactive (95.75%) | inactive (>10000nM) | - |
PAK2 | inactive (66.52%) | - | inactive (108%) |
PAK3 | inactive (95.93%) | - | inactive (107%) |
PAK4 | inactive (72.35%) | inactive (>5011.87nM) | inactive (91%) |
PAK5 | inactive (85.15%) | - | inactive (95%) |
PAK6 | inactive (107.75%) | - | inactive (94%) |
SLK | inactive (88.82%) | inactive (1584.89nM) | - |
YSK1 | inactive (100.74%) | - | - |
STLK3 | inactive (94.86%) | - | - |
TAO1 | inactive (108.57%) | inactive (>10000nM) | inactive (108%) |
TAO2 | inactive (107.41%) | - | inactive (117%) |
TAO3 | inactive (76.7%) | - | inactive (101%) |
MYO3B | inactive (75.76%) | - | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MAP2K1 | inactive (81.94%) | - | active (41%) |
MAP2K2 | inactive (93.18%) | - | - |
MAP2K6 | inactive (102.93%) | - | inactive (60%) |
MAP2K7 | - | - | inactive (81%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
AurA | inactive (77.62%) | active (501.19nM) | active (29%) |
AurB | active (9.65%) | active (39.81nM) | active (6%) |
AurC | active (47.52%) | - | inactive (56%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CaMKK1 | inactive (82.97%) | - | - |
CaMKK2 | inactive (81.6%) | - | - |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Haspin | inactive (95.67%) | - | inactive (100%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
IKKa | inactive (98.28%) | inactive (>3981.07nM) | inactive (93%) |
IKKb | inactive (102.07%) | inactive (>3162.28nM) | inactive (111%) |
IKKe | inactive (72.78%) | - | - |
TBK1 | inactive (67.39%) | - | inactive (70%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
NEK1 | inactive (96.36%) | - | - |
NEK11 | inactive (110.82%) | - | inactive (88%) |
NEK2 | inactive (87.99%) | inactive (>10000nM) | inactive (83%) |
NEK4 | inactive (79.09%) | inactive (>6309.57nM) | - |
NEK6 | inactive (95.14%) | - | inactive (108%) |
NEK7 | inactive (106.5%) | - | inactive (101%) |
NEK9 | inactive (97.3%) | - | - |
NEK3 | inactive (88.81%) | - | inactive (116%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PBK | inactive (88.29%) | inactive (>10000nM) | - |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PLK1 | inactive (104.17%) | inactive (>7943.28nM) | inactive (92%) |
PLK2 | inactive (106.34%) | - | inactive (103%) |
PLK3 | inactive (96.58%) | inactive (>7943.28nM) | inactive (102%) |
PLK4 | - | active (398.11nM) | - |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
SgK496 | inactive (93.89%) | - | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MPSK1 | inactive (94.19%) | - | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TTK | inactive (93.58%) | - | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ULK1 | inactive (75.6%) | - | - |
ULK2 | inactive (120.16%) | - | inactive (100%) |
ULK3 | inactive (60.17%) | - | inactive (53%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Wee1 | inactive (93.3%) | - | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Wnk2 | inactive (105.92%) | - | inactive (111%) |
Wnk3 | inactive (100.05%) | - | inactive (110%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TLK2 | inactive (98.47%) | - | inactive (105%) |
Other - CDC7
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CDC7 | - | inactive (>1258.93nM) | - |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz | Millipore |
---|
CK1 | 7 | 6 | 5 | 4 |
VRK | 3 | 1 | - | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CK1d | active (37.8%) | active (316.23nM) | active (13%) |
CK1g1 | inactive (86.92%) | inactive (>6309.57nM) | inactive (70%) |
CK1g2 | inactive (70.2%) | inactive (1995.26nM) | inactive (51%) |
CK1g3 | inactive (78.52%) | inactive (3981.07nM) | inactive (83%) |
CK1a | inactive (70.96%) | inactive (1995.26nM) | - |
CK1e | active (47.1%) | - | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
VRK1 | inactive (98.95%) | - | - |
VRK2 | - | - | inactive (98%) |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz | Millipore |
---|
CK2 | 3 | 2 | 1 | 2 |
CLK | 4 | 4 | 2 | 2 |
DYRK | 10 | 9 | 6 | 4 |
MAPK | 14 | 10 | 8 | 10 |
GSK | 2 | 2 | 2 | 2 |
SRPK | 3 | 3 | 1 | 3 |
CDK | 20 | - | 7 | - |
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CK2a1 | inactive (73.55%) | inactive (>6309.57nM) | inactive (100%) |
CK2a2 | inactive (98.56%) | - | inactive (120%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CLK1 | inactive (94.07%) | - | - |
CLK2 | inactive (69.21%) | active (398.11nM) | active (49%) |
CLK3 | inactive (91.34%) | - | inactive (80%) |
CLK4 | inactive (80.75%) | active (398.11nM) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DYRK1A | inactive (94.15%) | inactive (>6309.57nM) | - |
DYRK1B | inactive (95.31%) | - | - |
DYRK2 | inactive (101.04%) | - | inactive (91%) |
DYRK3 | inactive (93.48%) | inactive (>6309.57nM) | - |
DYRK4 | inactive (103.92%) | inactive (>7943.28nM) | - |
HIPK1 | inactive (98.19%) | - | inactive (94%) |
HIPK2 | inactive (82.37%) | inactive (>3162.28nM) | inactive (80%) |
HIPK3 | inactive (95.34%) | - | inactive (95%) |
HIPK4 | inactive (99.4%) | inactive (>7943.28nM) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Erk1 | inactive (98.73%) | - | inactive (88%) |
Erk2 | inactive (99.77%) | inactive (>7943.28nM) | inactive (98%) |
JNK3 | inactive (90.63%) | - | inactive (87%) |
NLK | inactive (92.23%) | - | inactive (100%) |
p38a | inactive (104.34%) | - | inactive (79%) |
p38b | inactive (93.74%) | - | inactive (97%) |
p38d | inactive (98.29%) | inactive (>7943.28nM) | inactive (124%) |
p38g | inactive (100.51%) | inactive (>6309.57nM) | inactive (111%) |
JNK1 | inactive (105%) | inactive (>3162.28nM) | inactive (115%) |
JNK2 | inactive (97.67%) | inactive (>3981.07nM) | inactive (102%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
GSK3A | inactive (91.4%) | inactive (>7943.28nM) | inactive (106%) |
GSK3B | inactive (102.11%) | inactive (>6309.57nM) | inactive (93%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MSSK1 | inactive (94.29%) | - | inactive (99%) |
SRPK1 | inactive (99.16%) | inactive (>7943.28nM) | inactive (104%) |
SRPK2 | inactive (91.84%) | - | inactive (93%) |
CMGC - CDK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CDC2 | - | inactive (>7943.28nM) | - |
CDK2 | - | inactive (>7943.28nM) | - |
CDK5 | - | inactive (>10000nM) | - |
CDK8 | - | - | - |
CDK7 | - | - | - |
CDK9 | - | - | - |
CDK11 | - | inactive (>100000nM) | - |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz | Millipore |
---|
PDHK | 5 | 1 | - | - |
Alpha | 6 | - | 1 | 1 |
PIKK | 6 | - | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PDHK1 | inactive (94.21%) | - | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
eEF2K | - | inactive (>3981.07nM) | inactive (92%) |
Atypical - PIKK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FRAP | - | - | inactive (111%) |