Compound Information
Test on : RBC
Compound Name : -
Inchikey : WNWSUJQVZJJGLF-UHFFFAOYSA-N
ChemSpider : 21465179
Pubchem CID : 24906282
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC |
---|
PDK1 | inactive (86.36%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC |
---|
AKT1 | inactive (97.71%) |
AKT2 | inactive (100.6%) |
AKT3 | inactive (89.4%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC |
---|
DMPK1 | inactive (123.61%) |
MRCKa | inactive (93.96%) |
MRCKb | inactive (97.48%) |
ROCK1 | inactive (98.98%) |
ROCK2 | inactive (92.12%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC |
---|
BARK1 | inactive (97.35%) |
BARK2 | inactive (103.72%) |
GPRK4 | inactive (90.09%) |
GPRK5 | inactive (125.29%) |
GPRK6 | inactive (79.92%) |
GPRK7 | inactive (96.68%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC |
---|
MSK1 | inactive (82.58%) |
MSK2 | inactive (56.11%) |
p70S6K | inactive (79.64%) |
p70S6Kb | inactive (100.43%) |
RSK2 | inactive (65.72%) |
RSK4 | active (43.09%) |
RSK1 | active (47.15%) |
RSK3 | active (33.67%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC |
---|
PKACg | - |
PRKX | inactive (92.14%) |
PKACa | inactive (106.35%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC |
---|
PKCa | - |
PKCd | inactive (102.54%) |
PKCe | inactive (92.4%) |
PKCh | inactive (78.61%) |
PKCg | inactive (90.88%) |
PKCi | inactive (97.26%) |
PKCt | inactive (104.61%) |
PKCz | inactive (100.34%) |
PKCb | inactive (107.62%) |
AGC - PKG
Bioactivity |
---|
Kinase | RBC |
---|
PKG2 | inactive (69.14%) |
PKG1 | inactive (89.04%) |
AGC - PKN
Bioactivity |
---|
Kinase | RBC |
---|
PKN1 | inactive (82.16%) |
PKN2 | inactive (85.62%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC |
---|
SGK1 | inactive (60.93%) |
SGK2 | inactive (73.04%) |
SGK3 | inactive (97.19%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC |
---|
NDR1 | active (0%) |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC |
---|
ABL1 | active (19.13%) |
ABL2 | active (8.39%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC |
---|
ACK | active (36.89%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC |
---|
ALK | inactive (88.52%) |
LTK | inactive (89.34%) |
TK - Axl
Bioactivity |
---|
Kinase | RBC |
---|
AXL | inactive (57.7%) |
MER | inactive (79.35%) |
TYRO3 | inactive (81.6%) |
TK - Src
Bioactivity |
---|
Kinase | RBC |
---|
BLK | active (11.28%) |
BRK | inactive (89.32%) |
SRC | active (7.64%) |
FGR | active (2.99%) |
FRK | active (23.19%) |
FYN | active (5.05%) |
HCK | active (13.3%) |
LCK | active (38.99%) |
SRM | inactive (99.64%) |
YES | active (15.81%) |
LYN | active (5.98%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC |
---|
BMX | active (29.2%) |
BTK | active (13.06%) |
ITK | active (46.65%) |
TEC | inactive (104.22%) |
TXK | active (27.74%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC |
---|
KIT | active (42.26%) |
FLT3 | active (4.02%) |
FMS | inactive (74.45%) |
PDGFRb | active (35.2%) |
PDGFRa | inactive (68.38%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC |
---|
CSK | inactive (65.77%) |
CTK | inactive (99.65%) |
TK - DDR
Bioactivity |
---|
Kinase | RBC |
---|
DDR2 | inactive (69.67%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC |
---|
EGFR | inactive (88.98%) |
ErbB2 | inactive (102.04%) |
ErbB4 | inactive (96.8%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC |
---|
EphA1 | inactive (98.47%) |
EphA2 | inactive (70.94%) |
EphA3 | inactive (81.86%) |
EphA4 | inactive (90.23%) |
EphA5 | inactive (70.38%) |
EphA6 | - |
EphA7 | inactive (81.37%) |
EphA8 | inactive (97.61%) |
EphB1 | inactive (72.27%) |
EphB2 | inactive (74.73%) |
EphB3 | inactive (102.8%) |
EphB4 | inactive (78.48%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC |
---|
FAK | inactive (88.98%) |
PYK2 | inactive (56.66%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC |
---|
FER | inactive (69.78%) |
FES | inactive (96.04%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC |
---|
FGFR1 | active (45.1%) |
FGFR2 | inactive (59.24%) |
FGFR3 | inactive (54.64%) |
FGFR4 | inactive (79.61%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC |
---|
FLT1 | inactive (75.06%) |
FLT4 | inactive (50.78%) |
KDR | inactive (64.16%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC |
---|
IGF1R | inactive (103.17%) |
IRR | inactive (80.95%) |
INSR | inactive (92.49%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC |
---|
JAK1 | inactive (76.24%) |
JAK2 | inactive (93.76%) |
JAK3 | inactive (53.33%) |
TYK2 | active (25.6%) |
TK - Musk
Bioactivity |
---|
Kinase | RBC |
---|
MUSK | inactive (84.53%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC |
---|
RET | active (0.06%) |
TK - Met
Bioactivity |
---|
Kinase | RBC |
---|
RON | inactive (98.72%) |
MET | inactive (70.01%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC |
---|
ROS | inactive (82%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC |
---|
SYK | active (45.68%) |
ZAP70 | inactive (106.7%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC |
---|
TIE2 | inactive (96.71%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC |
---|
TRKA | active (34.49%) |
TRKB | active (10.35%) |
TRKC | active (4.98%) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC |
---|
ALK1 | inactive (103.49%) |
ALK2 | inactive (113.62%) |
ALK4 | inactive (100.28%) |
TGFbR1 | inactive (99.75%) |
TGFbR2 | inactive (105.95%) |
TKL - RAF
Bioactivity |
---|
Kinase | RBC |
---|
ARAF | inactive (99.84%) |
BRAF | inactive (98.19%) |
RAF1 | inactive (102.66%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC |
---|
IRAK1 | inactive (103.39%) |
IRAK4 | inactive (90.11%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC |
---|
LIMK1 | inactive (51.69%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC |
---|
LRRK2 | inactive (95.27%) |
TKL - MLK
Bioactivity |
---|
Kinase | RBC |
---|
MLK1 | active (9.21%) |
MLK2 | inactive (92.13%) |
MLK3 | active (16.01%) |
TAK1 | inactive (79.27%) |
ZAK | inactive (68.99%) |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC |
---|
RIPK2 | inactive (75.17%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC |
---|
NuaK1 | active (15.69%) |
BRSK1 | active (14.63%) |
BRSK2 | active (19.39%) |
CHK1 | inactive (57.11%) |
LKB1 | active (42.13%) |
MARK1 | inactive (64.18%) |
MARK3 | inactive (67.03%) |
MARK4 | - |
MELK | active (43.47%) |
PASK | inactive (97.9%) |
QIK | active (31.06%) |
NuaK2 | inactive (73.37%) |
MARK2 | inactive (61.84%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC |
---|
CaMK1a | inactive (96.02%) |
CaMK1b | inactive (105.49%) |
CaMK1d | - |
CaMK1g | inactive (96.04%) |
CaMK4 | inactive (96.27%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC |
---|
CaMK2a | active (13.92%) |
CaMK2b | inactive (65.77%) |
CaMK2d | active (23.02%) |
CaMK2g | active (28.34%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC |
---|
CHK2 | active (48.34%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC |
---|
DAPK1 | inactive (89.99%) |
DAPK2 | inactive (91.02%) |
DRAK1 | active (49.2%) |
DAPK3 | inactive (84.92%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC |
---|
DCLK2 | inactive (99.1%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC |
---|
MAPKAPK2 | inactive (86.86%) |
MAPKAPK3 | inactive (96.13%) |
MAPKAPK5 | inactive (82.66%) |
MNK1 | inactive (102.43%) |
MNK2 | inactive (75.28%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC |
---|
smMLCK | active (44.97%) |
skMLCK | active (17.59%) |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC |
---|
PHKg1 | active (41.75%) |
PHKg2 | inactive (92.45%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC |
---|
PIM1 | inactive (96.14%) |
PIM2 | inactive (95.52%) |
PIM3 | inactive (73.15%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC |
---|
PKD1 | inactive (93.59%) |
PKD3 | inactive (87.75%) |
PKD2 | inactive (94.08%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC |
---|
TSSK1 | inactive (83.03%) |
TSSK2 | inactive (101.45%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC |
---|
STK33 | inactive (69.35%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC |
---|
MAP3K5 | inactive (91.61%) |
MAP3K2 | inactive (90.32%) |
MAP3K3 | inactive (106.79%) |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC |
---|
COT | inactive (101.07%) |
NIK | inactive (89.55%) |
STE - STE20
Bioactivity |
---|
Kinase | RBC |
---|
GCK | inactive (61.47%) |
HGK | active (28.64%) |
KHS1 | active (36.54%) |
LOK | inactive (52.77%) |
MINK | active (47.8%) |
MST1 | active (22.54%) |
MST2 | active (20.54%) |
MST3 | inactive (90.86%) |
MST4 | inactive (121.78%) |
OSR1 | inactive (100.21%) |
PAK1 | inactive (89.76%) |
PAK2 | inactive (90.93%) |
PAK3 | inactive (99.65%) |
PAK4 | inactive (95.28%) |
PAK5 | inactive (103.62%) |
PAK6 | inactive (86.29%) |
SLK | inactive (56.14%) |
YSK1 | inactive (96.32%) |
STLK3 | inactive (103.81%) |
TAO1 | inactive (98.48%) |
TAO2 | inactive (92.11%) |
TAO3 | inactive (56.87%) |
MYO3B | active (0%) |
STE - STE7
Bioactivity |
---|
Kinase | RBC |
---|
MAP2K1 | inactive (103.09%) |
MAP2K2 | inactive (92.42%) |
MAP2K6 | inactive (98.25%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC |
---|
AurA | active (17.14%) |
AurB | active (39.1%) |
AurC | inactive (51.84%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC |
---|
CaMKK1 | inactive (50.51%) |
CaMKK2 | inactive (70.06%) |
Other - Haspin
Bioactivity |
---|
Kinase | RBC |
---|
Haspin | inactive (95.94%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC |
---|
IKKa | inactive (103.52%) |
IKKb | inactive (85.41%) |
IKKe | inactive (66.26%) |
TBK1 | inactive (62.11%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC |
---|
NEK1 | inactive (93.8%) |
NEK11 | inactive (117.56%) |
NEK2 | inactive (95.48%) |
NEK4 | inactive (96.66%) |
NEK6 | inactive (99.85%) |
NEK7 | inactive (102.52%) |
NEK9 | inactive (96.29%) |
NEK3 | inactive (84.4%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC |
---|
PBK | inactive (108.78%) |
Other - PLK
Bioactivity |
---|
Kinase | RBC |
---|
PLK1 | inactive (101.23%) |
PLK2 | inactive (98.91%) |
PLK3 | inactive (95.32%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC |
---|
SgK496 | inactive (101.95%) |
Other - NAK
Bioactivity |
---|
Kinase | RBC |
---|
MPSK1 | inactive (64.02%) |
Other - TTK
Bioactivity |
---|
Kinase | RBC |
---|
TTK | inactive (69.76%) |
Other - ULK
Bioactivity |
---|
Kinase | RBC |
---|
ULK1 | inactive (95.31%) |
ULK2 | inactive (94.04%) |
ULK3 | active (0%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC |
---|
Wee1 | inactive (95.98%) |
Other - WNK
Bioactivity |
---|
Kinase | RBC |
---|
Wnk2 | inactive (104.11%) |
Wnk3 | inactive (93.78%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC |
---|
TLK2 | active (0%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
CK1 | 7 | 6 |
VRK | 3 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC |
---|
CK1d | inactive (85.37%) |
CK1g1 | inactive (87.57%) |
CK1g2 | inactive (105.04%) |
CK1g3 | inactive (78.28%) |
CK1a | inactive (95.11%) |
CK1e | inactive (83.66%) |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC |
---|
VRK1 | inactive (98.03%) |
CMGC
CMGC - CK2
Bioactivity |
---|
Kinase | RBC |
---|
CK2a1 | inactive (82.24%) |
CK2a2 | inactive (63.15%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC |
---|
CLK1 | inactive (93.07%) |
CLK2 | inactive (91.86%) |
CLK3 | inactive (71.17%) |
CLK4 | inactive (96.96%) |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC |
---|
DYRK1A | inactive (101.33%) |
DYRK1B | inactive (80.32%) |
DYRK2 | inactive (90.96%) |
DYRK3 | inactive (103.61%) |
DYRK4 | inactive (99.4%) |
HIPK1 | inactive (103.15%) |
HIPK2 | inactive (96.21%) |
HIPK3 | inactive (64.84%) |
HIPK4 | inactive (105.64%) |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC |
---|
Erk1 | inactive (83.32%) |
Erk2 | inactive (113%) |
JNK3 | inactive (97.89%) |
NLK | inactive (100.73%) |
p38a | inactive (105.34%) |
p38b | inactive (99.56%) |
p38d | inactive (87.46%) |
p38g | inactive (93.82%) |
JNK1 | inactive (98.67%) |
JNK2 | inactive (80.33%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC |
---|
GSK3A | active (3.6%) |
GSK3B | active (3.77%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC |
---|
MSSK1 | inactive (96.36%) |
SRPK1 | inactive (94.9%) |
SRPK2 | inactive (63.92%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
PDHK | 5 | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC |
---|
PDHK1 | inactive (86.36%) |