Compound Information
Test on : DRx, RBC, Metz
Compound Name
DRx, RBC : Sunitinib
Metz : N-(2-(Diethylamino)ethyl)-5-((5-fluoro-2-oxoindolin-3-ylidene)methyl)-2,4-dimethyl-1H-pyrrole-3-carboxamide
Inchikey
Same : WINHZLLDWRZWRT-N
DRx, RBC : WINHZLLDWRZWRT-ATVHPVEESA-N
Metz : WINHZLLDWRZWRT-UHFFFAOYSA-N
ChemSpider
DRx, RBC : 4486264
Metz : 23346185
Pubchem CID
DRx, RBC : 5329102
Metz : 3086686
ChEMBL
DRx, RBC : CHEMBL535
Metz : CHEMBL1990885
DRx, RBC | Metz |
| |
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
Other
Other - NAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AAK1 | active (11nM) | - | - |
BIKE | active (5.5nM) | - | - |
GAK | active (20nM) | - | - |
MPSK1 | active (250nM) | inactive (55.75%) | - |
Other - Aur
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AurA | active (1700nM) | inactive (59.66%) | inactive (>630.96nM) |
AurB | active (380nM) | active (48.72%) | active (630.96nM) |
AurC | active (220nM) | inactive (72.82%) | - |
Other - CAMKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CaMKK1 | active (420nM) | inactive (52.06%) | - |
CaMKK2 | active (1500nM) | inactive (65.25%) | active (630.96nM) |
Other - PEK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
HRI | inactive (10001nM) | - | - |
PKR | active (670nM) | - | - |
Other - IRE
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IRE1 | active (600nM) | - | - |
Other - IKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IKKa | active (520nM) | inactive (92.36%) | inactive (>3981.07nM) |
IKKb | inactive (10001nM) | inactive (80.96%) | inactive (>3162.28nM) |
IKKe | active (620nM) | active (45.57%) | inactive (>2511.89nM) |
TBK1 | active (120nM) | - | inactive (>3162.28nM) |
Other - NEK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
NEK1 | inactive (10001nM) | inactive (72.6%) | - |
NEK11 | inactive (10001nM) | inactive (106.2%) | - |
NEK2 | active (1400nM) | inactive (105.74%) | inactive (>2511.89nM) |
NEK3 | inactive (10001nM) | inactive (91.57%) | - |
NEK4 | inactive (10001nM) | inactive (94.08%) | inactive (>6309.57nM) |
NEK5 | inactive (10001nM) | - | - |
NEK6 | inactive (10001nM) | inactive (89.04%) | - |
NEK7 | inactive (4100nM) | inactive (93.52%) | - |
NEK9 | inactive (10001nM) | inactive (100.15%) | - |
Other - WEE
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MYT1 | inactive (10001nM) | - | - |
Wee1 | active (1100nM) | inactive (91.84%) | - |
Wee1B | inactive (10001nM) | - | - |
Other - PLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PLK1 | inactive (10001nM) | inactive (96.36%) | inactive (>7943.28nM) |
PLK2 | inactive (4700nM) | inactive (99.17%) | - |
PLK3 | inactive (10001nM) | inactive (96.5%) | inactive (>7943.28nM) |
PLK4 | active (190nM) | - | active (316.23nM) |
Other - SgK496
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SgK496 | active (1300nM) | inactive (111.32%) | - |
Other - NKF1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SBK | active (200nM) | - | - |
SgK110 | active (1900nM) | - | - |
Other - NKF4
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CLIK1 | active (1300nM) | - | - |
Other - ULK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Fused | inactive (10001nM) | - | - |
ULK1 | active (23nM) | active (16.28%) | - |
ULK2 | active (13nM) | active (40.31%) | - |
ULK3 | active (42nM) | inactive (57.42%) | - |
Other - TLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TLK1 | active (740nM) | - | - |
TLK2 | active (330nM) | inactive (63.31%) | - |
Other - TTK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TTK | active (63nM) | inactive (68%) | - |
Other - Haspin
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Haspin | - | inactive (53.17%) | - |
Other - TOPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PBK | - | inactive (106.16%) | inactive (>10000nM) |
Other - WNK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Wnk2 | - | inactive (100.21%) | - |
Wnk3 | - | inactive (94.26%) | - |
Other - CDC7
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CDC7 | - | - | inactive (>1258.93nM) |
TK
TK - Abl
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ABL1 | active (270nM) | active (47.24%) | inactive (>316.23nM) |
ABL2 | active (1000nM) | inactive (61.78%) | - |
TK - ALK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ALK | active (170nM) | active (16.62%) | inactive (>1584.89nM) |
LTK | active (1800nM) | active (34.39%) | inactive (>2511.89nM) |
TK - Axl
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AXL | active (9nM) | active (27.41%) | active (15.85nM) |
MER | active (26nM) | active (39.82%) | - |
TYRO3 | active (49nM) | active (28.31%) | inactive (>1000nM) |
TK - Src
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
BLK | active (65nM) | active (28.66%) | active (63.1nM) |
BRK | inactive (4600nM) | inactive (84.49%) | inactive (>2511.89nM) |
FGR | active (270nM) | active (16.44%) | - |
FRK | active (530nM) | inactive (84.45%) | active (125.89nM) |
FYN | active (520nM) | inactive (71.31%) | active (251.19nM) |
HCK | active (880nM) | active (39.95%) | active (199.53nM) |
LCK | active (230nM) | active (13.24%) | active (31.62nM) |
LYN | active (270nM) | active (23%) | active (79.43nM) |
SRC | active (2100nM) | active (39.81%) | active (630.96nM) |
SRM | inactive (10001nM) | inactive (99.6%) | inactive (>1584.89nM) |
YES | active (120nM) | active (5.91%) | - |
TK - Tec
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
BMX | inactive (10001nM) | inactive (99%) | - |
BTK | active (2100nM) | inactive (50.19%) | inactive (>3981.07nM) |
ITK | active (13nM) | inactive (64.35%) | active (25.12nM) |
TEC | inactive (10001nM) | inactive (94.83%) | - |
TXK | inactive (10001nM) | inactive (92.62%) | - |
TK - PDGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FMS | active (2.5nM) | active (7.28%) | active (2.51nM) |
FLT3 | active (0.41nM) | active (2.71%) | active (1.58nM) |
KIT | active (0.37nM) | active (8.74%) | inactive (>3162.28nM) |
PDGFRa | active (0.79nM) | active (10.85%) | inactive (>794.33nM) |
PDGFRb | active (0.08nM) | active (17.64%) | active (1nM) |
TK - Csk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CSK | inactive (10001nM) | inactive (90.17%) | - |
CTK | inactive (7700nM) | inactive (88.84%) | inactive (1584.89nM) |
TK - DDR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DDR1 | active (2000nM) | - | - |
DDR2 | active (2900nM) | inactive (154.16%) | - |
TK - EGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
EGFR | inactive (10001nM) | inactive (89.17%) | inactive (>1995.26nM) |
ErbB2 | inactive (10001nM) | inactive (104.84%) | inactive (>1584.89nM) |
ErbB3 | inactive (10001nM) | - | - |
ErbB4 | inactive (10001nM) | inactive (94.81%) | inactive (>3981.07nM) |
TK - Eph
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
EphA1 | inactive (10001nM) | inactive (95.12%) | - |
EphA2 | inactive (10001nM) | inactive (83.62%) | inactive (>3162.28nM) |
EphA3 | active (2100nM) | inactive (83.96%) | - |
EphA4 | inactive (10001nM) | inactive (84.49%) | - |
EphA5 | active (1200nM) | inactive (87.6%) | - |
EphA6 | active (960nM) | active (29.55%) | - |
EphA7 | active (2400nM) | inactive (50.79%) | - |
EphA8 | inactive (10001nM) | inactive (92.12%) | - |
EphB1 | active (480nM) | inactive (53.59%) | - |
EphB2 | inactive (10001nM) | inactive (72.06%) | - |
EphB3 | inactive (10001nM) | inactive (77.43%) | - |
EphB4 | inactive (3100nM) | inactive (65.53%) | - |
EphB6 | active (1000nM) | - | - |
TK - FAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FAK | active (440nM) | active (27%) | active (316.23nM) |
PYK2 | active (82nM) | active (38.33%) | active (125.89nM) |
TK - Fer
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FER | active (1100nM) | active (31.57%) | active (63.1nM) |
FES | active (960nM) | active (33.67%) | active (125.89nM) |
TK - FGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FGFR1 | active (520nM) | inactive (66.14%) | inactive (>1584.89nM) |
FGFR2 | active (570nM) | inactive (50.48%) | - |
FGFR3 | active (290nM) | active (39.73%) | active (398.11nM) |
FGFR4 | active (2100nM) | inactive (92.51%) | - |
TK - VEGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FLT1 | active (1.8nM) | inactive (58.72%) | inactive (>1258.93nM) |
FLT4 | active (50nM) | active (17.36%) | active (25.12nM) |
KDR | active (1.5nM) | active (28.67%) | active (12.59nM) |
TK - InsR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IGF1R | active (2600nM) | inactive (62.55%) | active (630.96nM) |
INSR | active (500nM) | inactive (51.17%) | active (199.53nM) |
IRR | active (430nM) | active (21.69%) | - |
TK - JakA
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
JAK1 | inactive (6000nM) | inactive (71.88%) | - |
JAK2 | active (410nM) | inactive (88.82%) | inactive (>1995.26nM) |
JAK3 | active (1200nM) | inactive (80.67%) | inactive (>3981.07nM) |
TYK2 | active (1600nM) | inactive (52.6%) | inactive (>1258.93nM) |
TK - Met
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MET | inactive (7200nM) | inactive (90.96%) | inactive (>2511.89nM) |
RON | inactive (10001nM) | inactive (92.01%) | active (25.12nM) |
TK - Musk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MUSK | active (490nM) | inactive (51.26%) | - |
TK - Ret
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
RET | active (13nM) | active (3.43%) | active (2.51nM) |
TK - Sev
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ROS | inactive (10001nM) | inactive (71.58%) | inactive (>2511.89nM) |
TK - Syk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SYK | inactive (10001nM) | inactive (89.19%) | inactive (>1584.89nM) |
ZAP70 | inactive (10001nM) | inactive (97.22%) | - |
TK - Tie
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TIE1 | inactive (3900nM) | - | - |
TIE2 | inactive (10001nM) | inactive (88.57%) | - |
TK - Ack
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TNK1 | active (680nM) | - | - |
ACK | inactive (8900nM) | inactive (64.11%) | inactive (>3162.28nM) |
TK - Trk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TRKA | active (100nM) | active (11.46%) | active (794.33nM) |
TRKB | active (590nM) | active (9.78%) | active (1000nM) |
TRKC | inactive (5100nM) | active (2.37%) | active (794.33nM) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ALK2 | inactive (10001nM) | inactive (120.84%) | inactive (>3981.07nM) |
ALK4 | inactive (10001nM) | inactive (100.56%) | - |
ACTR2 | inactive (10001nM) | - | - |
ACTR2B | inactive (10001nM) | - | - |
ALK1 | inactive (10001nM) | inactive (111.78%) | - |
BMPR1A | inactive (10001nM) | - | - |
BMPR1B | active (2400nM) | - | - |
BMPR2 | active (570nM) | - | - |
TGFbR1 | inactive (10001nM) | inactive (100.85%) | - |
TGFbR2 | inactive (10001nM) | inactive (92.46%) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SgK288 | active (310nM) | - | - |
RIPK1 | active (370nM) | - | - |
RIPK2 | inactive (10001nM) | inactive (104.04%) | - |
ANKRD3 | active (2100nM) | - | - |
TKL - RAF
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
BRAF | inactive (10001nM) | inactive (106.18%) | - |
RAF1 | inactive (10001nM) | inactive (109.94%) | - |
ARAF | - | inactive (124.44%) | - |
TKL - MLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DLK | active (100nM) | - | - |
LZK | active (95nM) | - | - |
MLK1 | inactive (3400nM) | inactive (87.89%) | - |
MLK2 | inactive (10001nM) | inactive (104.25%) | inactive (>3162.28nM) |
MLK3 | active (1300nM) | inactive (68.4%) | - |
TAK1 | active (93nM) | active (18.64%) | - |
HH498 | inactive (10001nM) | - | - |
ZAK | inactive (10001nM) | inactive (97.77%) | inactive (>7943.28nM) |
TKL - IRAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IRAK1 | active (14nM) | active (31.41%) | active (125.89nM) |
IRAK3 | active (940nM) | - | - |
IRAK4 | active (66nM) | active (27.4%) | active (1000nM) |
TKL - LISK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
LIMK1 | inactive (10001nM) | inactive (94.26%) | inactive (2511.89nM) |
LIMK2 | inactive (10001nM) | - | - |
TESK1 | inactive (10001nM) | - | - |
TKL - LRRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
LRRK2 | active (110nM) | active (3.34%) | inactive (>1584.89nM) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz |
---|
ABC1 | 5 | 2 | - | - |
PIKK | 6 | 1 | - | - |
RIO | 3 | 3 | - | - |
Alpha | 6 | 1 | - | 1 |
PDHK | 5 | - | 1 | - |
Atypical - ABC1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ADCK3 | inactive (10001nM) | - | - |
ADCK4 | inactive (10001nM) | - | - |
Atypical - PIKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FRAP | inactive (10001nM) | - | - |
Atypical - RIO
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
RIOK1 | active (35nM) | - | - |
RIOK2 | active (49nM) | - | - |
RIOK3 | inactive (3800nM) | - | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ChaK2 | inactive (10001nM) | - | - |
eEF2K | - | - | inactive (>3981.07nM) |
Atypical - PDHK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PDHK1 | - | inactive (81.56%) | - |
AGC
AGC - Akt
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AKT1 | inactive (10001nM) | inactive (104.83%) | inactive (>5011.87nM) |
AKT2 | active (2700nM) | inactive (87.36%) | inactive (>7943.28nM) |
AKT3 | inactive (10001nM) | inactive (71.68%) | inactive (>6309.57nM) |
AGC - DMPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CRIK | inactive (3900nM) | - | - |
DMPK1 | inactive (10001nM) | inactive (97.74%) | - |
DMPK2 | inactive (10001nM) | - | - |
MRCKa | inactive (10001nM) | inactive (89.52%) | inactive (>10000nM) |
MRCKb | inactive (10001nM) | inactive (100.93%) | - |
ROCK1 | active (460nM) | inactive (99.65%) | inactive (>2511.89nM) |
ROCK2 | active (140nM) | inactive (72.1%) | active (1000nM) |
AGC - GRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
RHOK | active (290nM) | - | - |
GPRK4 | active (140nM) | inactive (75.79%) | - |
GPRK7 | active (180nM) | inactive (71.25%) | - |
BARK1 | - | inactive (94.71%) | - |
BARK2 | - | inactive (94.8%) | - |
GPRK5 | - | inactive (85.3%) | inactive (>3981.07nM) |
GPRK6 | - | inactive (74.68%) | - |
AGC - NDR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
LATS1 | active (630nM) | - | - |
LATS2 | active (460nM) | - | - |
NDR1 | active (410nM) | inactive (93.85%) | - |
NDR2 | active (970nM) | - | - |
AGC - MAST
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAST1 | active (200nM) | - | - |
AGC - PDK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PDK1 | inactive (3500nM) | inactive (81.56%) | active (1000nM) |
AGC - PKA
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKACa | inactive (10001nM) | inactive (89.1%) | inactive (>1995.26nM) |
PKACb | inactive (10001nM) | - | - |
PRKX | inactive (10001nM) | inactive (104.89%) | inactive (>3162.28nM) |
PKACg | - | inactive (109.09%) | - |
AGC - PKN
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKN1 | active (710nM) | inactive (71.42%) | - |
PKN2 | active (1300nM) | inactive (89.13%) | inactive (2511.89nM) |
AGC - PKC
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKCd | inactive (10001nM) | inactive (95.08%) | inactive (5011.87nM) |
PKCe | inactive (10001nM) | inactive (97.95%) | - |
PKCh | inactive (10001nM) | inactive (111.79%) | - |
PKCi | inactive (10001nM) | inactive (102.61%) | inactive (>5011.87nM) |
PKCt | inactive (4300nM) | inactive (63.49%) | inactive (>2511.89nM) |
PKCa | - | inactive (79.88%) | - |
PKCg | - | inactive (83.81%) | inactive (>6309.57nM) |
PKCz | - | inactive (91.71%) | inactive (>7943.28nM) |
PKCb | - | inactive (103.78%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKG1 | inactive (10001nM) | inactive (65.35%) | inactive (>1995.26nM) |
PKG2 | inactive (10001nM) | inactive (96.06%) | inactive (>1584.89nM) |
AGC - RSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
p70S6K | active (48nM) | active (42.32%) | active (398.11nM) |
MSK1 | - | inactive (60.05%) | active (398.11nM) |
MSK2 | - | inactive (50.84%) | active (63.1nM) |
p70S6Kb | - | inactive (113.44%) | - |
RSK2 | - | active (35.46%) | inactive (>1258.93nM) |
RSK4 | - | active (17.51%) | - |
RSK1 | - | active (28.05%) | - |
RSK3 | - | active (17.34%) | - |
AGC - SGK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SGK3 | active (220nM) | inactive (101.31%) | - |
SGK1 | - | inactive (62.78%) | active (316.23nM) |
SGK2 | - | inactive (93.15%) | - |
AGC - YANK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
YANK1 | inactive (10001nM) | - | - |
YANK2 | inactive (10001nM) | - | - |
YANK3 | inactive (10001nM) | - | - |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AMPKa1 | active (19nM) | - | active (63.1nM) |
AMPKa2 | active (89nM) | - | - |
NuaK1 | active (48nM) | active (2.75%) | - |
BRSK1 | inactive (3500nM) | active (45.15%) | active (158.49nM) |
BRSK2 | active (1100nM) | inactive (54.53%) | - |
CHK1 | active (300nM) | active (29.2%) | inactive (>1258.93nM) |
HUNK | active (500nM) | - | - |
LKB1 | active (38nM) | inactive (97.2%) | - |
MARK1 | active (1200nM) | active (40.94%) | - |
MARK2 | active (310nM) | active (40.6%) | active (199.53nM) |
MARK3 | active (410nM) | active (30.35%) | active (199.53nM) |
MARK4 | inactive (3600nM) | active (24.74%) | inactive (>5011.87nM) |
MELK | active (350nM) | active (10.39%) | inactive (>1258.93nM) |
NIM1 | active (850nM) | - | - |
QSK | inactive (10001nM) | - | - |
SIK | inactive (3200nM) | - | - |
QIK | active (580nM) | active (27.84%) | active (316.23nM) |
NuaK2 | active (150nM) | inactive (65.01%) | - |
SNRK | active (640nM) | - | - |
PASK | - | inactive (102.25%) | - |
CAMK - CAMK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CaMK1a | active (970nM) | inactive (75.19%) | inactive (1258.93nM) |
CaMK1d | active (510nM) | inactive (77.9%) | inactive (>1995.26nM) |
CaMK1g | active (440nM) | inactive (67.03%) | - |
CaMK4 | active (890nM) | inactive (88.63%) | - |
CaMK1b | - | inactive (98.47%) | - |
CAMK - CAMK2
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CaMK2a | active (80nM) | active (14.46%) | active (158.49nM) |
CaMK2b | active (1400nM) | active (46.66%) | inactive (1258.93nM) |
CaMK2d | active (420nM) | active (11.56%) | active (25.12nM) |
CaMK2g | active (690nM) | active (25.07%) | active (39.81nM) |
CAMK - CASK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CASK | inactive (10001nM) | - | - |
CAMK - RAD53
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CHK2 | active (10nM) | active (7.13%) | active (31.62nM) |
CAMK - DAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DAPK1 | active (120nM) | inactive (66.85%) | - |
DAPK2 | active (150nM) | - | - |
DAPK3 | active (22nM) | inactive (74.21%) | active (199.53nM) |
DRAK1 | active (1nM) | active (26.74%) | active (794.33nM) |
DRAK2 | active (110nM) | - | - |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DCLK1 | active (370nM) | - | inactive (3981.07nM) |
DCLK2 | active (2700nM) | inactive (85.02%) | - |
DCLK3 | active (110nM) | - | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAPKAPK2 | inactive (10001nM) | inactive (93.22%) | inactive (>7943.28nM) |
MAPKAPK5 | inactive (10001nM) | inactive (82.74%) | inactive (>1584.89nM) |
MNK1 | inactive (3900nM) | inactive (99.35%) | - |
MNK2 | inactive (5700nM) | inactive (99.33%) | inactive (>10000nM) |
MAPKAPK3 | - | inactive (102.23%) | inactive (>10000nM) |
CAMK - MLCK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
caMLCK | active (23nM) | - | - |
smMLCK | active (280nM) | active (25.61%) | - |
skMLCK | active (49nM) | active (7.74%) | - |
SgK085 | active (15nM) | - | - |
CAMK - PHK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PHKg1 | active (5.5nM) | active (5.12%) | - |
PHKg2 | active (5.9nM) | active (20.55%) | active (15.85nM) |
CAMK - PIM
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PIM1 | inactive (10001nM) | inactive (94.44%) | inactive (>6309.57nM) |
PIM2 | inactive (10001nM) | inactive (97.16%) | inactive (>1584.89nM) |
PIM3 | active (2400nM) | inactive (56.81%) | inactive (1584.89nM) |
CAMK - PKD
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKD1 | active (310nM) | active (20.02%) | - |
PKD2 | active (380nM) | active (21.14%) | active (398.11nM) |
PKD3 | active (280nM) | active (16.57%) | inactive (>1584.89nM) |
CAMK - STK33
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
STK33 | active (17nM) | active (31.82%) | - |
CAMK - TSSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TSSK1 | inactive (6300nM) | active (20.67%) | active (199.53nM) |
TSSK2 | - | inactive (72.91%) | active (630.96nM) |
STE
STE - STE11
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAP3K5 | inactive (10001nM) | inactive (100.2%) | - |
MAP3K6 | inactive (10001nM) | - | - |
MAP3K1 | inactive (10001nM) | - | - |
MAP3K7 | active (1300nM) | - | - |
MAP3K2 | active (57nM) | inactive (51.88%) | - |
MAP3K3 | active (220nM) | active (42%) | - |
MAP3K4 | inactive (4800nM) | - | - |
MAP3K8 | active (17nM) | - | - |
STE - STE20
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
HPK1 | active (16nM) | - | - |
LOK | active (19nM) | active (31.22%) | - |
GCK | active (33nM) | active (34.44%) | inactive (>1584.89nM) |
KHS2 | active (180nM) | - | - |
HGK | active (140nM) | active (12.44%) | active (31.62nM) |
KHS1 | active (41nM) | active (4.06%) | active (15.85nM) |
MINK | active (29nM) | active (10.46%) | active (79.43nM) |
MST1 | active (19nM) | active (10.7%) | - |
MST2 | active (56nM) | active (24.8%) | active (100nM) |
MST3 | active (63nM) | active (39.71%) | - |
MST4 | active (340nM) | inactive (110.06%) | - |
MYO3A | inactive (3100nM) | - | - |
MYO3B | inactive (4500nM) | inactive (54.48%) | - |
OSR1 | active (530nM) | inactive (105.18%) | - |
PAK1 | inactive (10001nM) | inactive (118.32%) | inactive (>10000nM) |
PAK2 | inactive (10001nM) | inactive (98.11%) | - |
PAK3 | active (16nM) | inactive (108.98%) | - |
PAK4 | active (2300nM) | inactive (80.93%) | inactive (>3162.28nM) |
PAK6 | active (2400nM) | inactive (107.24%) | - |
PAK5 | active (640nM) | inactive (81.55%) | - |
SLK | active (56nM) | inactive (63.84%) | active (79.43nM) |
STLK3 | active (140nM) | inactive (87.36%) | - |
TAO1 | active (890nM) | inactive (71.46%) | inactive (>3981.07nM) |
TAO2 | inactive (10001nM) | inactive (90.31%) | - |
TAO3 | active (210nM) | inactive (82.92%) | - |
TNIK | active (25nM) | - | - |
YSK1 | active (290nM) | inactive (76.06%) | - |
STE - STE7
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAP2K1 | active (130nM) | inactive (67.8%) | active (39.81nM) |
MAP2K2 | active (110nM) | active (25.41%) | active (50.12nM) |
MAP2K3 | active (1700nM) | - | - |
MAP2K4 | active (700nM) | - | - |
MAP2K5 | active (46nM) | - | - |
MAP2K6 | inactive (5200nM) | inactive (75.85%) | - |
MAP2K7 | inactive (10001nM) | - | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
COT | - | inactive (116.82%) | - |
NIK | - | inactive (127.37%) | - |
CMGC
CMGC - CDK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PITSLRE | inactive (10001nM) | - | - |
CHED | inactive (10001nM) | - | - |
CDK11 | inactive (10001nM) | - | inactive (>100000nM) |
PCTAIRE1 | active (150nM) | - | - |
PCTAIRE2 | active (1200nM) | - | - |
PCTAIRE3 | active (1700nM) | - | - |
PFTAIRE2 | inactive (10001nM) | - | - |
PFTAIRE1 | active (270nM) | - | - |
CDC2 | - | - | inactive (>7943.28nM) |
CDK2 | - | - | inactive (>7943.28nM) |
CDK5 | - | - | inactive (>3162.28nM) |
CDK8 | - | - | inactive (>3981.07nM) |
CDK7 | - | - | active (19.95nM) |
CDK9 | - | - | inactive (>1584.89nM) |
CMGC - CDKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CDKL1 | inactive (10001nM) | - | - |
CDKL2 | active (1100nM) | - | - |
CDKL3 | inactive (10001nM) | - | - |
CDKL5 | inactive (10001nM) | - | - |
CMGC - CLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CLK1 | active (22nM) | active (23.26%) | - |
CLK2 | active (20nM) | active (13.59%) | inactive (>2511.89nM) |
CLK3 | inactive (10001nM) | inactive (105.22%) | - |
CLK4 | active (29nM) | active (26.32%) | inactive (>1000nM) |
CMGC - CK2
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CK2a1 | active (900nM) | inactive (120.61%) | inactive (>5011.87nM) |
CK2a2 | active (160nM) | inactive (92.18%) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DYRK1A | active (200nM) | inactive (56.86%) | inactive (>1995.26nM) |
DYRK1B | active (2300nM) | inactive (59.97%) | inactive (>1995.26nM) |
DYRK2 | active (680nM) | inactive (82.57%) | - |
HIPK1 | active (55nM) | inactive (71.29%) | - |
HIPK2 | active (31nM) | active (41.32%) | active (251.19nM) |
HIPK3 | active (41nM) | active (47.26%) | - |
HIPK4 | active (160nM) | inactive (74.66%) | inactive (1584.89nM) |
PRP4 | active (390nM) | - | - |
DYRK3 | - | inactive (58.21%) | active (1000nM) |
DYRK4 | - | inactive (104.04%) | inactive (>7943.28nM) |
CMGC - MAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Erk1 | inactive (10001nM) | inactive (107.7%) | - |
Erk2 | inactive (10001nM) | inactive (98.48%) | inactive (>7943.28nM) |
Erk3 | inactive (10001nM) | - | - |
Erk4 | inactive (10001nM) | - | - |
Erk5 | inactive (9900nM) | - | - |
Erk7 | inactive (10001nM) | - | - |
JNK1 | inactive (10001nM) | inactive (91.84%) | inactive (>3981.07nM) |
JNK2 | active (2400nM) | inactive (96.74%) | inactive (>3981.07nM) |
JNK3 | inactive (4300nM) | inactive (99.52%) | inactive (>3162.28nM) |
NLK | inactive (10001nM) | inactive (104.58%) | - |
p38a | inactive (10001nM) | inactive (104.88%) | inactive (>3981.07nM) |
p38b | inactive (10001nM) | inactive (99.95%) | - |
p38d | inactive (10001nM) | inactive (92.39%) | inactive (>7943.28nM) |
p38g | inactive (10001nM) | inactive (95.76%) | inactive (>6309.57nM) |
CMGC - GSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
GSK3A | inactive (10001nM) | inactive (85.51%) | inactive (>6309.57nM) |
GSK3B | inactive (10001nM) | inactive (95.78%) | inactive (>2511.89nM) |
CMGC - RCK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ICK | active (470nM) | - | - |
MAK | inactive (10001nM) | - | - |
CMGC - SRPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SRPK1 | active (250nM) | inactive (97.04%) | inactive (>7943.28nM) |
SRPK2 | active (190nM) | inactive (94.98%) | - |
MSSK1 | active (59nM) | inactive (102.34%) | - |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz |
---|
CK1 | 7 | 7 | 6 | 5 |
VRK | 3 | 1 | 1 | - |
CK1 - CK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CK1a | active (99nM) | inactive (53.97%) | inactive (>3162.28nM) |
CK1a2 | active (550nM) | - | - |
CK1d | active (15nM) | active (31.77%) | active (100nM) |
CK1e | active (13nM) | active (46.95%) | - |
CK1g1 | active (930nM) | inactive (55.93%) | active (1000nM) |
CK1g2 | active (110nM) | - | active (630.96nM) |
CK1g3 | active (240nM) | active (30.02%) | active (501.19nM) |
CK1 - VRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
VRK2 | inactive (10001nM) | - | - |
VRK1 | - | inactive (97.28%) | - |