Compound Information
Test on : RBC, Metz, Millipore
Compound Name
RBC, Metz, Millipore : SB220025
Inchikey
Same : VSPFURGQAYMVAN-N
RBC, Metz, Millipore : VSPFURGQAYMVAN-UHFFFAOYSA-N
ChemSpider
RBC, Metz, Millipore : 4980
Pubchem CID
RBC, Metz, Millipore : 5164
ChEMBL
RBC, Metz, Millipore : CHEMBL274064
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PDK1 | inactive (103.15%) | inactive (>3981.07nM) | inactive (109%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
AKT1 | inactive (99.88%) | inactive (>7943.28nM) | inactive (105%) |
AKT2 | inactive (94.79%) | inactive (>7943.28nM) | inactive (103%) |
AKT3 | inactive (92.57%) | inactive (>10000nM) | inactive (87%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DMPK1 | inactive (99.27%) | - | inactive (129%) |
MRCKa | inactive (100.64%) | inactive (>10000nM) | inactive (113%) |
MRCKb | inactive (101.23%) | - | inactive (98%) |
ROCK1 | inactive (102.66%) | inactive (>10000nM) | inactive (128%) |
ROCK2 | inactive (102.5%) | inactive (>7943.28nM) | inactive (99%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
BARK1 | inactive (99.74%) | - | - |
BARK2 | inactive (97.56%) | - | - |
GPRK4 | inactive (96.92%) | - | - |
GPRK5 | inactive (102.69%) | - | inactive (106%) |
GPRK6 | inactive (98.23%) | - | inactive (98%) |
GPRK7 | inactive (105.96%) | - | inactive (107%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MSK1 | inactive (97.9%) | inactive (>1995.26nM) | inactive (106%) |
MSK2 | inactive (98.67%) | - | inactive (97%) |
p70S6K | inactive (98.22%) | inactive (>6309.57nM) | inactive (74%) |
p70S6Kb | inactive (90.87%) | - | - |
RSK2 | inactive (92.25%) | inactive (>7943.28nM) | inactive (54%) |
RSK4 | inactive (109.34%) | - | inactive (89%) |
RSK1 | inactive (96.75%) | - | inactive (83%) |
RSK3 | inactive (99.28%) | - | inactive (105%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKACg | inactive (105.46%) | - | - |
PRKX | inactive (96.75%) | inactive (>1584.89nM) | inactive (110%) |
PKACa | inactive (82.98%) | inactive (1584.89nM) | inactive (95%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKCa | inactive (89.08%) | - | inactive (105%) |
PKCd | inactive (99.76%) | inactive (>7943.28nM) | inactive (105%) |
PKCe | inactive (104.77%) | - | inactive (114%) |
PKCh | inactive (91.94%) | - | inactive (114%) |
PKCg | inactive (87.81%) | inactive (6309.57nM) | inactive (107%) |
PKCi | inactive (98.47%) | - | inactive (113%) |
PKCt | inactive (106.77%) | - | inactive (93%) |
PKCz | inactive (105.77%) | inactive (>7943.28nM) | inactive (111%) |
PKCb | inactive (79.38%) | - | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKG2 | inactive (97.19%) | inactive (>1584.89nM) | - |
PKG1 | inactive (97.69%) | inactive (>1995.26nM) | - |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKN1 | inactive (96.35%) | - | - |
PKN2 | inactive (97.14%) | inactive (>7943.28nM) | inactive (111%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
SGK1 | inactive (97.41%) | inactive (6309.57nM) | inactive (93%) |
SGK2 | inactive (96.93%) | - | inactive (97%) |
SGK3 | inactive (97.48%) | - | inactive (108%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
NDR1 | inactive (99.83%) | - | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ABL1 | inactive (100.65%) | inactive (>630.96nM) | inactive (104%) |
ABL2 | inactive (95.13%) | - | inactive (108%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ACK | inactive (97.95%) | - | inactive (76%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ALK | inactive (102.03%) | inactive (>1258.93nM) | inactive (81%) |
LTK | inactive (97.28%) | - | - |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
AXL | inactive (101.56%) | inactive (>1995.26nM) | inactive (94%) |
MER | inactive (98.01%) | - | inactive (67%) |
TYRO3 | inactive (96.94%) | - | inactive (91%) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
BLK | inactive (102.39%) | inactive (>1584.89nM) | inactive (99%) |
BRK | inactive (73.42%) | inactive (>2511.89nM) | inactive (88%) |
SRC | inactive (94.25%) | inactive (>5011.87nM) | inactive (117%) |
FGR | inactive (95.91%) | - | inactive (81%) |
FRK | inactive (95.42%) | - | inactive (92%) |
FYN | inactive (91.1%) | inactive (>794.33nM) | inactive (75%) |
HCK | inactive (95.54%) | - | inactive (84%) |
LCK | inactive (80.12%) | active (125.89nM) | inactive (58%) |
SRM | inactive (97.49%) | - | - |
YES | inactive (85.25%) | - | inactive (78%) |
LYN | inactive (87.49%) | active (316.23nM) | active (50%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
BMX | inactive (92.85%) | - | inactive (67%) |
BTK | inactive (100.32%) | - | inactive (97%) |
ITK | inactive (90.55%) | inactive (>1584.89nM) | inactive (98%) |
TEC | inactive (110.5%) | - | - |
TXK | inactive (99.07%) | - | inactive (83%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
KIT | inactive (98.39%) | inactive (>1258.93nM) | inactive (121%) |
FLT3 | inactive (90.33%) | inactive (>2511.89nM) | inactive (108%) |
FMS | inactive (100.08%) | inactive (>2511.89nM) | inactive (93%) |
PDGFRb | inactive (98.67%) | - | inactive (114%) |
PDGFRa | inactive (95.79%) | - | inactive (110%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CSK | inactive (90.78%) | - | inactive (114%) |
CTK | inactive (99.49%) | - | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DDR2 | inactive (106.6%) | - | inactive (94%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
EGFR | inactive (94.41%) | inactive (>1258.93nM) | inactive (105%) |
ErbB2 | inactive (93.69%) | inactive (>1584.89nM) | - |
ErbB4 | inactive (86.81%) | inactive (2511.89nM) | inactive (97%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
EphA1 | inactive (98.15%) | - | inactive (119%) |
EphA2 | inactive (102.37%) | inactive (>7943.28nM) | inactive (92%) |
EphA3 | inactive (97.35%) | - | inactive (97%) |
EphA4 | inactive (99.81%) | - | inactive (103%) |
EphA5 | inactive (97.83%) | - | inactive (113%) |
EphA6 | inactive (78.03%) | - | - |
EphA7 | inactive (93.96%) | - | inactive (96%) |
EphA8 | inactive (101.38%) | - | inactive (90%) |
EphB1 | inactive (99.86%) | - | inactive (104%) |
EphB2 | inactive (102.56%) | - | inactive (98%) |
EphB3 | inactive (100.87%) | - | inactive (117%) |
EphB4 | inactive (91.55%) | - | inactive (77%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FAK | inactive (94.06%) | inactive (>1584.89nM) | inactive (103%) |
PYK2 | inactive (94.57%) | inactive (>1584.89nM) | inactive (107%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FER | inactive (98.27%) | - | inactive (103%) |
FES | inactive (103.14%) | - | inactive (106%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FGFR1 | inactive (91.2%) | inactive (>5011.87nM) | inactive (119%) |
FGFR2 | inactive (103.74%) | - | inactive (113%) |
FGFR3 | inactive (100.47%) | inactive (>1995.26nM) | inactive (120%) |
FGFR4 | inactive (85.67%) | - | inactive (116%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FLT1 | inactive (89.27%) | inactive (>398.11nM) | inactive (94%) |
FLT4 | inactive (116.34%) | inactive (6309.57nM) | inactive (69%) |
KDR | inactive (102%) | inactive (5011.87nM) | inactive (104%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
IGF1R | inactive (103.63%) | inactive (>1258.93nM) | inactive (96%) |
IRR | inactive (103.46%) | - | inactive (140%) |
INSR | inactive (94.15%) | inactive (>5011.87nM) | inactive (112%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
JAK1 | inactive (104.17%) | - | - |
JAK2 | inactive (99.57%) | inactive (>1584.89nM) | inactive (106%) |
JAK3 | inactive (96.93%) | inactive (>1584.89nM) | inactive (120%) |
TYK2 | inactive (99.77%) | inactive (>1995.26nM) | - |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MUSK | inactive (86.87%) | - | inactive (99%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
RET | inactive (89.44%) | inactive (1258.93nM) | inactive (97%) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
RON | inactive (100.35%) | - | inactive (100%) |
MET | inactive (103.56%) | inactive (>3162.28nM) | inactive (114%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ROS | inactive (94.09%) | - | inactive (108%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
SYK | inactive (98%) | - | inactive (99%) |
ZAP70 | inactive (92.34%) | - | inactive (130%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TIE2 | inactive (101.43%) | - | inactive (113%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TRKA | inactive (100.39%) | inactive (>2511.89nM) | inactive (100%) |
TRKB | inactive (102.88%) | inactive (>5011.87nM) | inactive (118%) |
TRKC | inactive (97.14%) | - | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ALK1 | inactive (95.62%) | - | - |
ALK2 | inactive (86.49%) | - | - |
ALK4 | inactive (121.3%) | - | inactive (101%) |
TGFbR1 | inactive (101.8%) | - | inactive (81%) |
TGFbR2 | inactive (118.94%) | - | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ARAF | inactive (93.11%) | - | - |
BRAF | inactive (102.62%) | - | - |
RAF1 | inactive (90.85%) | - | inactive (64%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
IRAK1 | inactive (114.45%) | inactive (6309.57nM) | inactive (102%) |
IRAK4 | inactive (123.14%) | inactive (>10000nM) | inactive (92%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
LIMK1 | inactive (89.56%) | active (794.33nM) | inactive (64%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
LRRK2 | inactive (99.91%) | - | - |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MLK1 | inactive (94.51%) | - | inactive (96%) |
MLK2 | inactive (99.79%) | - | - |
MLK3 | inactive (96.26%) | - | - |
TAK1 | inactive (96.86%) | - | inactive (101%) |
ZAK | inactive (98%) | inactive (>7943.28nM) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
RIPK2 | inactive (77.17%) | - | active (43%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
NuaK1 | inactive (98.36%) | - | inactive (111%) |
BRSK1 | inactive (99.71%) | inactive (>10000nM) | inactive (94%) |
BRSK2 | inactive (96.63%) | - | inactive (128%) |
CHK1 | inactive (99.76%) | inactive (>7943.28nM) | inactive (101%) |
LKB1 | inactive (89.14%) | - | inactive (104%) |
MARK1 | inactive (97.93%) | - | inactive (89%) |
MARK3 | inactive (102.83%) | inactive (>6309.57nM) | - |
MARK4 | inactive (97.37%) | - | - |
MELK | inactive (100.04%) | active (794.33nM) | inactive (71%) |
PASK | inactive (98.48%) | - | inactive (129%) |
QIK | inactive (64.69%) | - | - |
NuaK2 | inactive (121.9%) | - | - |
MARK2 | inactive (97.04%) | inactive (>7943.28nM) | inactive (96%) |
AMPKa1 | - | inactive (>6309.57nM) | inactive (102%) |
AMPKa2 | - | - | inactive (96%) |
SIK | - | - | inactive (132%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CaMK1a | inactive (106.88%) | inactive (>3162.28nM) | inactive (92%) |
CaMK1b | inactive (94.31%) | - | - |
CaMK1d | inactive (103.12%) | - | inactive (112%) |
CaMK1g | inactive (99.33%) | - | - |
CaMK4 | inactive (103.44%) | - | inactive (107%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CaMK2a | inactive (100.28%) | - | - |
CaMK2b | inactive (97.71%) | - | inactive (91%) |
CaMK2d | inactive (100.38%) | - | inactive (100%) |
CaMK2g | inactive (93%) | - | inactive (108%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CHK2 | inactive (101.29%) | inactive (>5011.87nM) | inactive (92%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DAPK1 | inactive (88.24%) | - | inactive (86%) |
DAPK2 | inactive (94.09%) | - | inactive (103%) |
DRAK1 | inactive (97.75%) | - | inactive (95%) |
DAPK3 | inactive (96.51%) | inactive (>1258.93nM) | inactive (86%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DCLK2 | inactive (99.91%) | - | inactive (102%) |
DCLK1 | - | inactive (>10000nM) | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MAPKAPK2 | inactive (97.63%) | inactive (>7943.28nM) | inactive (79%) |
MAPKAPK3 | inactive (99.42%) | inactive (>10000nM) | inactive (123%) |
MAPKAPK5 | inactive (94%) | inactive (>1584.89nM) | inactive (118%) |
MNK1 | inactive (98.99%) | - | - |
MNK2 | inactive (92.14%) | inactive (>10000nM) | inactive (101%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
smMLCK | inactive (99.79%) | - | inactive (102%) |
skMLCK | inactive (103.05%) | - | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PHKg1 | inactive (98.25%) | - | - |
PHKg2 | inactive (104.5%) | inactive (>5011.87nM) | inactive (125%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PIM1 | inactive (96.99%) | active (1000nM) | inactive (75%) |
PIM2 | inactive (100.22%) | inactive (>1584.89nM) | inactive (120%) |
PIM3 | inactive (96.03%) | - | inactive (87%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKD1 | inactive (54.62%) | - | active (46%) |
PKD3 | active (37.89%) | active (251.19nM) | - |
PKD2 | inactive (50.37%) | inactive (1258.93nM) | inactive (102%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TSSK1 | inactive (106%) | inactive (>1584.89nM) | inactive (105%) |
TSSK2 | inactive (100.03%) | inactive (>1584.89nM) | inactive (95%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
STK33 | inactive (98.59%) | - | inactive (107%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MAP3K5 | inactive (102.44%) | - | inactive (100%) |
MAP3K2 | inactive (93.96%) | - | - |
MAP3K3 | inactive (100.82%) | - | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
COT | inactive (101.58%) | - | - |
NIK | inactive (107.36%) | - | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
GCK | inactive (101.62%) | inactive (>6309.57nM) | inactive (82%) |
HGK | inactive (76.26%) | active (794.33nM) | - |
KHS1 | inactive (68.14%) | active (501.19nM) | - |
LOK | inactive (90.34%) | - | inactive (99%) |
MINK | inactive (96.13%) | inactive (1258.93nM) | inactive (92%) |
MST1 | inactive (102.85%) | - | inactive (101%) |
MST2 | inactive (103.48%) | inactive (3162.28nM) | inactive (87%) |
MST3 | inactive (98.75%) | - | inactive (82%) |
MST4 | inactive (98.41%) | - | - |
OSR1 | inactive (101.35%) | - | - |
PAK1 | inactive (97.37%) | inactive (>10000nM) | - |
PAK2 | inactive (76.89%) | - | inactive (99%) |
PAK3 | inactive (104.64%) | - | inactive (87%) |
PAK4 | inactive (95.13%) | inactive (>5011.87nM) | inactive (102%) |
PAK5 | inactive (100.63%) | - | inactive (103%) |
PAK6 | inactive (111.42%) | - | inactive (105%) |
SLK | inactive (99.94%) | inactive (>10000nM) | - |
YSK1 | inactive (99.77%) | - | - |
STLK3 | inactive (93.45%) | - | - |
TAO1 | inactive (92.66%) | inactive (>10000nM) | inactive (98%) |
TAO2 | inactive (98.05%) | - | inactive (101%) |
TAO3 | inactive (95.32%) | - | inactive (98%) |
MYO3B | inactive (97.85%) | - | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MAP2K1 | inactive (98.25%) | - | inactive (109%) |
MAP2K2 | inactive (105.22%) | - | - |
MAP2K6 | inactive (105.87%) | - | inactive (80%) |
MAP2K7 | - | - | inactive (92%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
AurA | inactive (100.28%) | inactive (>1995.26nM) | inactive (124%) |
AurB | inactive (103.18%) | inactive (>6309.57nM) | inactive (111%) |
AurC | inactive (97.77%) | - | inactive (103%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CaMKK1 | inactive (102.8%) | - | - |
CaMKK2 | inactive (110.19%) | - | - |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Haspin | inactive (91.37%) | - | inactive (54%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
IKKa | inactive (101.5%) | inactive (>3981.07nM) | inactive (120%) |
IKKb | inactive (104.32%) | inactive (>3162.28nM) | inactive (116%) |
IKKe | inactive (99.51%) | - | - |
TBK1 | inactive (102.32%) | - | inactive (88%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
NEK1 | inactive (100.29%) | - | - |
NEK11 | inactive (104.69%) | - | inactive (68%) |
NEK2 | inactive (102.69%) | inactive (>10000nM) | inactive (97%) |
NEK4 | inactive (99.45%) | inactive (>6309.57nM) | - |
NEK6 | inactive (104.39%) | - | inactive (113%) |
NEK7 | inactive (98.85%) | - | inactive (109%) |
NEK9 | inactive (100.36%) | - | - |
NEK3 | inactive (99%) | - | inactive (82%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PBK | inactive (94.94%) | inactive (>10000nM) | - |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PLK1 | inactive (101.22%) | inactive (>7943.28nM) | inactive (85%) |
PLK2 | inactive (93%) | - | inactive (108%) |
PLK3 | inactive (97.83%) | inactive (>7943.28nM) | inactive (104%) |
PLK4 | - | inactive (>3981.07nM) | - |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
SgK496 | inactive (102.29%) | - | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MPSK1 | inactive (107.79%) | - | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TTK | inactive (107.22%) | - | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ULK1 | inactive (95.26%) | - | - |
ULK2 | inactive (113.28%) | - | inactive (114%) |
ULK3 | inactive (95.53%) | - | inactive (101%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Wee1 | inactive (106.32%) | - | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Wnk2 | inactive (93.06%) | - | inactive (104%) |
Wnk3 | inactive (95.34%) | - | inactive (95%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TLK2 | inactive (95.12%) | - | inactive (104%) |
Other - CDC7
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CDC7 | - | inactive (>1258.93nM) | - |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz | Millipore |
---|
CK1 | 7 | 6 | 5 | 4 |
VRK | 3 | 1 | - | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CK1d | active (1.25%) | active (12.59nM) | active (-2%) |
CK1g1 | inactive (83.08%) | - | inactive (72%) |
CK1g2 | inactive (118.98%) | inactive (3162.28nM) | inactive (89%) |
CK1g3 | inactive (83.87%) | - | inactive (84%) |
CK1a | active (2.82%) | active (12.59nM) | - |
CK1e | active (2.39%) | - | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
VRK1 | inactive (83.43%) | - | - |
VRK2 | - | - | inactive (93%) |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz | Millipore |
---|
CK2 | 3 | 2 | 1 | 2 |
CLK | 4 | 4 | 2 | 2 |
DYRK | 10 | 9 | 6 | 4 |
MAPK | 14 | 10 | 8 | 10 |
GSK | 2 | 2 | 2 | 2 |
SRPK | 3 | 3 | 1 | 3 |
CDK | 20 | - | 7 | - |
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CK2a1 | inactive (94.74%) | active (794.33nM) | inactive (93%) |
CK2a2 | inactive (92.2%) | - | inactive (107%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CLK1 | inactive (98.22%) | - | - |
CLK2 | inactive (99.67%) | inactive (1258.93nM) | inactive (69%) |
CLK3 | inactive (102.49%) | - | inactive (89%) |
CLK4 | inactive (96.94%) | active (1000nM) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DYRK1A | inactive (96.27%) | inactive (>6309.57nM) | - |
DYRK1B | inactive (100.25%) | - | - |
DYRK2 | inactive (95.9%) | - | inactive (83%) |
DYRK3 | inactive (96.05%) | inactive (1995.26nM) | - |
DYRK4 | inactive (99.34%) | - | - |
HIPK1 | inactive (101.05%) | - | inactive (110%) |
HIPK2 | inactive (105.81%) | inactive (>3162.28nM) | inactive (95%) |
HIPK3 | inactive (97.63%) | - | inactive (111%) |
HIPK4 | inactive (96.57%) | inactive (>7943.28nM) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Erk1 | inactive (100.45%) | - | inactive (88%) |
Erk2 | inactive (96.62%) | inactive (3162.28nM) | inactive (111%) |
JNK3 | inactive (104.9%) | - | inactive (69%) |
NLK | active (12.1%) | - | active (34%) |
p38a | active (13.08%) | - | active (2%) |
p38b | inactive (101.33%) | - | inactive (58%) |
p38d | inactive (102%) | inactive (>7943.28nM) | inactive (105%) |
p38g | inactive (102.16%) | inactive (>6309.57nM) | inactive (104%) |
JNK1 | inactive (94.84%) | inactive (>3162.28nM) | inactive (108%) |
JNK2 | inactive (105.46%) | inactive (2511.89nM) | inactive (76%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
GSK3A | inactive (97.54%) | inactive (2511.89nM) | inactive (92%) |
GSK3B | inactive (101.23%) | inactive (>6309.57nM) | inactive (111%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MSSK1 | inactive (99.29%) | - | inactive (101%) |
SRPK1 | inactive (103.26%) | inactive (>7943.28nM) | inactive (108%) |
SRPK2 | inactive (96.39%) | - | inactive (101%) |
CMGC - CDK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CDC2 | - | inactive (>7943.28nM) | - |
CDK2 | - | inactive (>7943.28nM) | - |
CDK5 | - | inactive (>10000nM) | - |
CDK8 | - | - | - |
CDK7 | - | - | - |
CDK9 | - | - | - |
CDK11 | - | - | - |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz | Millipore |
---|
PDHK | 5 | 1 | - | - |
Alpha | 6 | - | 1 | 1 |
PIKK | 6 | - | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PDHK1 | inactive (103.15%) | - | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
eEF2K | - | inactive (>3981.07nM) | inactive (117%) |
Atypical - PIKK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FRAP | - | - | inactive (109%) |