Compound Information
Test on : RBC, Metz, Millipore
Compound Name
RBC, Metz, Millipore : Pyridone 6
Inchikey
Same : VNDWQCSOSCCWIP-N
RBC, Metz, Millipore : VNDWQCSOSCCWIP-UHFFFAOYSA-N
ChemSpider
RBC, Metz, Millipore : 4591874
Pubchem CID
RBC, Metz, Millipore : 5494425
ChEMBL
RBC, Metz, Millipore : CHEMBL21156
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PDK1 | active (26.99%) | - | active (3%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
AKT1 | inactive (86.83%) | - | inactive (98%) |
AKT2 | inactive (89.83%) | - | inactive (146%) |
AKT3 | inactive (76.4%) | - | inactive (60%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DMPK1 | inactive (104.64%) | - | inactive (116%) |
MRCKa | inactive (95.71%) | - | inactive (86%) |
MRCKb | inactive (96.82%) | - | inactive (78%) |
ROCK1 | inactive (74.94%) | active (501.19nM) | inactive (91%) |
ROCK2 | inactive (70.72%) | - | inactive (57%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
BARK1 | inactive (98.48%) | - | - |
BARK2 | inactive (104.22%) | - | - |
GPRK4 | inactive (74.16%) | - | - |
GPRK5 | inactive (72.94%) | active (398.11nM) | inactive (72%) |
GPRK6 | active (48.16%) | - | inactive (59%) |
GPRK7 | inactive (60.47%) | - | active (42%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MSK1 | inactive (57.97%) | - | inactive (80%) |
MSK2 | active (44.71%) | - | active (36%) |
p70S6K | inactive (74.09%) | - | active (47%) |
p70S6Kb | inactive (101.62%) | - | - |
RSK2 | active (44.83%) | active (398.11nM) | active (43%) |
RSK4 | active (33.89%) | - | active (42%) |
RSK1 | active (38.57%) | - | active (25%) |
RSK3 | active (34.6%) | - | inactive (65%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKACg | - | - | - |
PRKX | inactive (79.18%) | inactive (>3162.28nM) | inactive (86%) |
PKACa | inactive (97.95%) | active (501.19nM) | inactive (89%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKCa | inactive (65.62%) | - | inactive (65%) |
PKCd | active (43.64%) | - | inactive (54%) |
PKCe | inactive (51.38%) | - | inactive (70%) |
PKCh | inactive (81.46%) | - | inactive (82%) |
PKCg | inactive (79.93%) | - | active (40%) |
PKCi | inactive (95.98%) | - | inactive (90%) |
PKCt | inactive (66.8%) | active (794.33nM) | active (45%) |
PKCz | inactive (93.16%) | - | inactive (103%) |
PKCb | inactive (90.57%) | - | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKG2 | active (14.27%) | - | - |
PKG1 | active (40.16%) | - | - |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKN1 | active (28.26%) | - | - |
PKN2 | inactive (67.14%) | - | active (29%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
SGK1 | inactive (50.91%) | - | inactive (63%) |
SGK2 | inactive (84.44%) | - | inactive (63%) |
SGK3 | inactive (96.64%) | - | inactive (80%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
NDR1 | active (0%) | - | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ABL1 | inactive (98.37%) | inactive (>2511.89nM) | inactive (86%) |
ABL2 | inactive (90.28%) | - | inactive (128%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ACK | active (4.36%) | active (125.89nM) | active (10%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ALK | active (19.98%) | active (158.49nM) | active (30%) |
LTK | active (20.64%) | active (25.12nM) | - |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
AXL | inactive (81.87%) | - | active (40%) |
MER | inactive (79.39%) | - | active (29%) |
TYRO3 | inactive (90.28%) | inactive (>3162.28nM) | inactive (75%) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
BLK | inactive (93.53%) | - | inactive (76%) |
BRK | inactive (88.05%) | - | inactive (93%) |
SRC | inactive (93.45%) | - | inactive (72%) |
FGR | inactive (76.85%) | - | inactive (69%) |
FRK | inactive (103.98%) | - | inactive (74%) |
FYN | inactive (52.34%) | inactive (>6309.57nM) | inactive (77%) |
HCK | inactive (84.79%) | - | active (49%) |
LCK | inactive (93.01%) | inactive (>6309.57nM) | inactive (115%) |
SRM | inactive (98.68%) | - | - |
YES | inactive (76.12%) | - | inactive (87%) |
LYN | inactive (101.37%) | - | inactive (65%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
BMX | inactive (71.87%) | - | active (28%) |
BTK | inactive (80.46%) | inactive (>6309.57nM) | inactive (71%) |
ITK | inactive (86.03%) | - | inactive (84%) |
TEC | inactive (106.35%) | - | - |
TXK | inactive (77.14%) | - | inactive (63%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
KIT | inactive (96.11%) | - | inactive (119%) |
FLT3 | active (13.58%) | inactive (>3162.28nM) | active (45%) |
FMS | inactive (93%) | inactive (>2511.89nM) | inactive (54%) |
PDGFRb | inactive (74.83%) | inactive (>1995.26nM) | inactive (107%) |
PDGFRa | inactive (92.14%) | inactive (>2511.89nM) | inactive (102%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CSK | inactive (114.02%) | - | inactive (93%) |
CTK | inactive (101.51%) | - | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DDR2 | inactive (107.06%) | - | inactive (110%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
EGFR | inactive (94.84%) | - | inactive (121%) |
ErbB2 | inactive (108.6%) | - | - |
ErbB4 | inactive (99.91%) | - | inactive (90%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
EphA1 | inactive (80.5%) | - | inactive (74%) |
EphA2 | inactive (98.48%) | - | inactive (103%) |
EphA3 | inactive (89.2%) | - | inactive (99%) |
EphA4 | inactive (100.92%) | - | inactive (105%) |
EphA5 | inactive (99.99%) | - | inactive (95%) |
EphA6 | - | - | - |
EphA7 | inactive (96.05%) | - | inactive (89%) |
EphA8 | inactive (104.94%) | - | inactive (103%) |
EphB1 | inactive (94.91%) | - | inactive (84%) |
EphB2 | inactive (92.84%) | - | inactive (115%) |
EphB3 | inactive (87.06%) | - | inactive (105%) |
EphB4 | inactive (88.23%) | - | inactive (90%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FAK | active (35.31%) | active (794.33nM) | inactive (51%) |
PYK2 | active (48.38%) | - | active (17%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FER | active (34.04%) | - | inactive (67%) |
FES | inactive (78.01%) | - | inactive (76%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FGFR1 | inactive (75.78%) | inactive (>3981.07nM) | active (43%) |
FGFR2 | inactive (99.11%) | - | inactive (79%) |
FGFR3 | inactive (93.02%) | - | inactive (94%) |
FGFR4 | inactive (96.49%) | - | inactive (119%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FLT1 | inactive (92.28%) | inactive (>3981.07nM) | inactive (52%) |
FLT4 | inactive (71.19%) | - | active (28%) |
KDR | inactive (102.99%) | inactive (1584.89nM) | inactive (65%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
IGF1R | inactive (91.27%) | inactive (>2511.89nM) | inactive (119%) |
IRR | inactive (75.21%) | - | inactive (101%) |
INSR | inactive (80.6%) | - | inactive (101%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
JAK1 | active (2.54%) | - | - |
JAK2 | active (1.37%) | active (2.51nM) | active (-1%) |
JAK3 | active (0.44%) | active (39.81nM) | active (1%) |
TYK2 | active (1.48%) | - | - |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MUSK | inactive (81.74%) | - | inactive (86%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
RET | active (18.33%) | active (199.53nM) | active (18%) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
RON | inactive (102.83%) | active (31.62nM) | inactive (87%) |
MET | inactive (91.03%) | inactive (>2511.89nM) | inactive (91%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ROS | active (31.17%) | - | inactive (90%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
SYK | inactive (79.04%) | - | inactive (110%) |
ZAP70 | inactive (88.9%) | - | inactive (91%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TIE2 | inactive (101.01%) | - | inactive (78%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TRKA | active (48.68%) | inactive (>3162.28nM) | active (3%) |
TRKB | active (16.09%) | active (1000nM) | inactive (71%) |
TRKC | active (6.81%) | inactive (3162.28nM) | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ALK1 | inactive (105.26%) | - | - |
ALK2 | inactive (134.71%) | inactive (>3981.07nM) | - |
ALK4 | inactive (109.56%) | - | inactive (110%) |
TGFbR1 | inactive (102.13%) | - | inactive (75%) |
TGFbR2 | inactive (58.17%) | - | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ARAF | inactive (122.34%) | - | - |
BRAF | inactive (116.94%) | - | - |
RAF1 | inactive (134.07%) | - | inactive (82%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
IRAK1 | inactive (76.31%) | - | inactive (55%) |
IRAK4 | inactive (96.34%) | - | inactive (61%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
LIMK1 | inactive (73.73%) | inactive (>3162.28nM) | inactive (98%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
LRRK2 | active (47.53%) | active (25.12nM) | - |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MLK1 | active (20.38%) | - | active (9%) |
MLK2 | inactive (89.75%) | - | - |
MLK3 | inactive (56.98%) | - | - |
TAK1 | active (46.58%) | - | active (44%) |
ZAK | inactive (78.1%) | - | - |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
RIPK2 | active (34.6%) | - | active (18%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
NuaK1 | active (3.04%) | - | active (8%) |
BRSK1 | active (15.37%) | - | active (32%) |
BRSK2 | active (21.35%) | - | active (13%) |
CHK1 | active (22.86%) | inactive (3162.28nM) | active (37%) |
LKB1 | inactive (58.44%) | - | inactive (99%) |
MARK1 | active (40.15%) | - | active (29%) |
MARK3 | inactive (55.86%) | - | - |
MARK4 | active (44.46%) | - | - |
MELK | active (5.23%) | - | active (2%) |
PASK | inactive (83.15%) | - | inactive (87%) |
QIK | inactive (60.19%) | - | - |
NuaK2 | inactive (66.02%) | - | - |
MARK2 | active (41.5%) | - | active (40%) |
AMPKa1 | - | active (158.49nM) | active (33%) |
AMPKa2 | - | - | active (20%) |
SIK | - | - | active (31%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CaMK1a | inactive (79.28%) | - | inactive (60%) |
CaMK1b | inactive (112.17%) | - | - |
CaMK1d | inactive (81.58%) | inactive (>2511.89nM) | inactive (60%) |
CaMK1g | inactive (95.34%) | - | - |
CaMK4 | inactive (81.8%) | - | active (1%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CaMK2a | active (35.1%) | inactive (>3981.07nM) | - |
CaMK2b | inactive (73.41%) | - | active (43%) |
CaMK2d | inactive (59.43%) | - | active (24%) |
CaMK2g | inactive (72.82%) | - | active (21%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CHK2 | active (0.72%) | - | active (2%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DAPK1 | active (3.03%) | - | active (8%) |
DAPK2 | active (18.04%) | - | active (11%) |
DRAK1 | active (6.42%) | - | active (0%) |
DAPK3 | active (2.18%) | active (1nM) | active (0%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DCLK2 | inactive (65.79%) | - | active (38%) |
DCLK1 | - | - | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MAPKAPK2 | inactive (99.56%) | - | inactive (79%) |
MAPKAPK3 | inactive (94.38%) | - | inactive (89%) |
MAPKAPK5 | inactive (88.1%) | - | active (47%) |
MNK1 | inactive (100.6%) | - | - |
MNK2 | inactive (61.97%) | - | inactive (66%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
smMLCK | active (9.03%) | - | active (2%) |
skMLCK | inactive (67.2%) | - | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PHKg1 | active (34.53%) | - | - |
PHKg2 | inactive (57.34%) | - | active (41%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PIM1 | active (38.6%) | active (630.96nM) | active (43%) |
PIM2 | inactive (90.83%) | - | active (43%) |
PIM3 | active (33.91%) | - | inactive (88%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKD1 | active (8.19%) | - | active (8%) |
PKD3 | active (10.81%) | active (79.43nM) | - |
PKD2 | active (6.13%) | - | active (40%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TSSK1 | active (37.33%) | - | active (42%) |
TSSK2 | inactive (92.52%) | - | inactive (81%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
STK33 | inactive (53.81%) | - | active (34%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MAP3K5 | inactive (84.35%) | - | inactive (81%) |
MAP3K2 | active (33.88%) | - | - |
MAP3K3 | inactive (61.13%) | - | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
COT | inactive (128%) | - | - |
NIK | inactive (71.26%) | - | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
GCK | inactive (66.15%) | inactive (2511.89nM) | active (19%) |
HGK | active (38.41%) | inactive (>5011.87nM) | - |
KHS1 | inactive (65.77%) | - | - |
LOK | inactive (72.55%) | - | inactive (72%) |
MINK | inactive (52%) | - | inactive (81%) |
MST1 | active (6.84%) | - | active (8%) |
MST2 | active (5.45%) | - | active (14%) |
MST3 | inactive (82.38%) | - | active (41%) |
MST4 | inactive (70.9%) | - | - |
OSR1 | inactive (100.27%) | - | - |
PAK1 | inactive (82.05%) | - | - |
PAK2 | inactive (88.81%) | - | inactive (93%) |
PAK3 | inactive (90.07%) | - | inactive (59%) |
PAK4 | inactive (105.06%) | inactive (>5011.87nM) | inactive (70%) |
PAK5 | inactive (90.55%) | - | inactive (78%) |
PAK6 | inactive (90.9%) | - | inactive (96%) |
SLK | inactive (91.38%) | - | - |
YSK1 | inactive (86.88%) | - | - |
STLK3 | inactive (93.85%) | - | - |
TAO1 | inactive (86.89%) | inactive (>6309.57nM) | inactive (56%) |
TAO2 | inactive (87.76%) | - | inactive (88%) |
TAO3 | inactive (50.29%) | - | inactive (68%) |
MYO3B | active (0%) | - | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MAP2K1 | inactive (94.94%) | active (100nM) | inactive (66%) |
MAP2K2 | inactive (82.13%) | active (398.11nM) | - |
MAP2K6 | inactive (89%) | - | active (39%) |
MAP2K7 | - | - | inactive (69%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
AurA | active (22.34%) | inactive (>1584.89nM) | active (13%) |
AurB | active (11.19%) | active (50.12nM) | active (1%) |
AurC | active (29.25%) | - | active (11%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CaMKK1 | inactive (81.35%) | - | - |
CaMKK2 | inactive (69.37%) | - | - |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Haspin | inactive (67.15%) | - | inactive (74%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
IKKa | inactive (101.66%) | - | inactive (52%) |
IKKb | inactive (52.14%) | - | active (42%) |
IKKe | active (25.4%) | active (100nM) | - |
TBK1 | active (24.02%) | active (199.53nM) | active (15%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
NEK1 | active (49%) | - | - |
NEK11 | inactive (92.41%) | - | inactive (98%) |
NEK2 | inactive (101.95%) | inactive (>3162.28nM) | inactive (72%) |
NEK4 | inactive (65.56%) | - | - |
NEK6 | inactive (82.52%) | - | inactive (85%) |
NEK7 | inactive (76.51%) | - | inactive (87%) |
NEK9 | inactive (71.68%) | - | - |
NEK3 | inactive (74.36%) | - | inactive (92%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PBK | active (39.06%) | - | - |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PLK1 | active (10.48%) | - | active (14%) |
PLK2 | inactive (92.61%) | - | active (49%) |
PLK3 | active (10.99%) | - | inactive (55%) |
PLK4 | - | - | - |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
SgK496 | inactive (62.01%) | - | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MPSK1 | inactive (90.08%) | - | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TTK | inactive (65.28%) | - | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ULK1 | active (12.78%) | - | - |
ULK2 | active (41.5%) | - | active (26%) |
ULK3 | active (0%) | - | inactive (56%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Wee1 | inactive (87.42%) | - | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Wnk2 | inactive (104.5%) | - | inactive (96%) |
Wnk3 | inactive (90.01%) | - | inactive (101%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TLK2 | active (0%) | - | inactive (54%) |
Other - CDC7
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CDC7 | - | - | - |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz | Millipore |
---|
CK1 | 7 | 6 | 5 | 4 |
VRK | 3 | 1 | - | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CK1d | inactive (89.13%) | - | inactive (82%) |
CK1g1 | inactive (96.52%) | - | inactive (78%) |
CK1g2 | inactive (100.31%) | - | inactive (86%) |
CK1g3 | inactive (105.3%) | - | inactive (111%) |
CK1a | inactive (94.63%) | inactive (>3981.07nM) | - |
CK1e | inactive (85.61%) | - | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
VRK1 | inactive (82.21%) | - | - |
VRK2 | - | - | inactive (89%) |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz | Millipore |
---|
CK2 | 3 | 2 | 1 | 2 |
CLK | 4 | 4 | 2 | 2 |
DYRK | 10 | 9 | 6 | 4 |
MAPK | 14 | 10 | 8 | 10 |
GSK | 2 | 2 | 2 | 2 |
SRPK | 3 | 3 | 1 | 3 |
CDK | 20 | - | 7 | - |
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CK2a1 | inactive (82.91%) | - | inactive (56%) |
CK2a2 | inactive (91.5%) | - | inactive (100%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CLK1 | inactive (81.58%) | - | - |
CLK2 | inactive (93.9%) | inactive (>3981.07nM) | active (34%) |
CLK3 | inactive (50.48%) | - | inactive (68%) |
CLK4 | inactive (70.71%) | active (79.43nM) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DYRK1A | inactive (101.7%) | inactive (>1995.26nM) | - |
DYRK1B | inactive (88.22%) | inactive (>2511.89nM) | - |
DYRK2 | inactive (62.54%) | - | inactive (76%) |
DYRK3 | inactive (104.65%) | - | - |
DYRK4 | inactive (104.11%) | - | - |
HIPK1 | inactive (88.72%) | - | inactive (84%) |
HIPK2 | inactive (98.69%) | - | inactive (65%) |
HIPK3 | inactive (78.56%) | - | inactive (79%) |
HIPK4 | inactive (106.89%) | - | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Erk1 | inactive (85.7%) | - | active (47%) |
Erk2 | inactive (96.11%) | - | inactive (92%) |
JNK3 | inactive (107.42%) | - | active (-2%) |
NLK | active (26.05%) | - | active (34%) |
p38a | inactive (93.48%) | inactive (>3981.07nM) | inactive (73%) |
p38b | inactive (83.43%) | - | inactive (62%) |
p38d | inactive (103.86%) | - | inactive (83%) |
p38g | inactive (97.88%) | - | inactive (81%) |
JNK1 | inactive (73.73%) | active (15.85nM) | active (32%) |
JNK2 | active (31.11%) | active (79.43nM) | inactive (64%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
GSK3A | inactive (121.43%) | inactive (>3981.07nM) | inactive (109%) |
GSK3B | inactive (95.12%) | inactive (>3981.07nM) | inactive (90%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MSSK1 | inactive (58.64%) | - | inactive (79%) |
SRPK1 | inactive (114.78%) | - | inactive (99%) |
SRPK2 | inactive (70.53%) | - | inactive (84%) |
CMGC - CDK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CDC2 | - | - | - |
CDK2 | - | - | - |
CDK5 | - | inactive (>3162.28nM) | - |
CDK8 | - | inactive (>3981.07nM) | - |
CDK7 | - | inactive (>3981.07nM) | - |
CDK9 | - | inactive (>1584.89nM) | - |
CDK11 | - | - | - |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz | Millipore |
---|
PDHK | 5 | 1 | - | - |
Alpha | 6 | - | 1 | 1 |
PIKK | 6 | - | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PDHK1 | active (26.99%) | - | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
eEF2K | - | - | inactive (81%) |
Atypical - PIKK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FRAP | - | - | inactive (91%) |