Compound Information
Test on : RBC, Millipore
Compound Name
RBC, Millipore : Tyrphostin A1
Inchikey
Same : UOHFCPXBKJPCAD-N
RBC, Millipore : UOHFCPXBKJPCAD-UHFFFAOYSA-N
ChemSpider
RBC, Millipore : 1979
Pubchem CID
RBC, Millipore : 2063
ChEMBL
RBC, Millipore : CHEMBL77456
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDK1 | inactive (72.61%) | inactive (113%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AKT1 | inactive (95.95%) | inactive (101%) |
AKT2 | inactive (98.1%) | inactive (133%) |
AKT3 | inactive (90.62%) | inactive (93%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DMPK1 | inactive (103%) | inactive (101%) |
MRCKa | inactive (110.88%) | inactive (97%) |
MRCKb | inactive (120.66%) | inactive (92%) |
ROCK1 | inactive (103.34%) | inactive (125%) |
ROCK2 | inactive (101.04%) | inactive (98%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BARK1 | inactive (107.36%) | - |
BARK2 | inactive (93.61%) | - |
GPRK4 | inactive (108.1%) | - |
GPRK5 | inactive (107.32%) | inactive (104%) |
GPRK6 | inactive (95.48%) | inactive (95%) |
GPRK7 | inactive (104.28%) | inactive (96%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSK1 | inactive (99.61%) | inactive (128%) |
MSK2 | inactive (98.61%) | inactive (94%) |
p70S6K | inactive (95.28%) | inactive (86%) |
p70S6Kb | inactive (91.21%) | - |
RSK2 | inactive (90.39%) | inactive (75%) |
RSK4 | inactive (113.37%) | inactive (102%) |
RSK1 | inactive (98.26%) | inactive (116%) |
RSK3 | inactive (105.26%) | inactive (135%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKACg | inactive (107.1%) | - |
PRKX | inactive (95.71%) | inactive (95%) |
PKACa | inactive (102.24%) | inactive (95%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKCa | inactive (91.95%) | inactive (102%) |
PKCd | inactive (102.13%) | inactive (102%) |
PKCe | inactive (98.14%) | inactive (81%) |
PKCh | inactive (92.1%) | inactive (103%) |
PKCg | inactive (85.31%) | inactive (115%) |
PKCi | inactive (102.34%) | inactive (78%) |
PKCt | inactive (101.68%) | inactive (95%) |
PKCz | inactive (109.8%) | inactive (110%) |
PKCb | inactive (95.85%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKG2 | inactive (96.63%) | - |
PKG1 | inactive (105.45%) | - |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKN1 | inactive (92.87%) | - |
PKN2 | inactive (91.6%) | inactive (106%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SGK1 | inactive (103.84%) | inactive (107%) |
SGK2 | inactive (106.3%) | inactive (89%) |
SGK3 | inactive (98.54%) | inactive (101%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NDR1 | inactive (93.96%) | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ABL1 | inactive (102.26%) | inactive (98%) |
ABL2 | inactive (98.45%) | inactive (106%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ACK | inactive (100.03%) | inactive (83%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK | inactive (110.29%) | inactive (84%) |
LTK | inactive (96.48%) | - |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AXL | inactive (99.85%) | inactive (91%) |
MER | inactive (86.61%) | inactive (108%) |
TYRO3 | inactive (106.22%) | inactive (105%) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BLK | inactive (100.82%) | inactive (115%) |
BRK | inactive (87.31%) | inactive (108%) |
SRC | inactive (99.94%) | inactive (89%) |
FGR | inactive (93.39%) | inactive (107%) |
FRK | inactive (98.79%) | inactive (106%) |
FYN | inactive (86.55%) | inactive (95%) |
HCK | inactive (92.6%) | inactive (79%) |
LCK | inactive (94.47%) | inactive (106%) |
SRM | inactive (111.36%) | - |
YES | inactive (100.48%) | inactive (108%) |
LYN | inactive (93.47%) | inactive (93%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BMX | inactive (83.79%) | inactive (95%) |
BTK | inactive (90.95%) | inactive (110%) |
ITK | inactive (100.93%) | inactive (103%) |
TEC | inactive (100.12%) | - |
TXK | inactive (101.5%) | inactive (100%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
KIT | inactive (92.21%) | inactive (107%) |
FLT3 | inactive (91.51%) | inactive (105%) |
FMS | inactive (100.43%) | inactive (73%) |
PDGFRb | inactive (103.88%) | inactive (114%) |
PDGFRa | inactive (94.93%) | inactive (115%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CSK | inactive (104.88%) | inactive (107%) |
CTK | inactive (95.44%) | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DDR2 | inactive (98.67%) | inactive (111%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EGFR | inactive (85.13%) | inactive (119%) |
ErbB2 | inactive (96.76%) | - |
ErbB4 | inactive (93.94%) | inactive (103%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EphA1 | inactive (102.39%) | inactive (92%) |
EphA2 | inactive (101.16%) | inactive (110%) |
EphA3 | inactive (105.04%) | inactive (103%) |
EphA4 | inactive (99.19%) | inactive (114%) |
EphA5 | inactive (94.59%) | inactive (113%) |
EphA6 | inactive (99.83%) | - |
EphA7 | inactive (89.05%) | inactive (95%) |
EphA8 | inactive (99.32%) | inactive (93%) |
EphB1 | inactive (94.34%) | inactive (108%) |
EphB2 | inactive (100.6%) | inactive (122%) |
EphB3 | inactive (97.55%) | inactive (102%) |
EphB4 | inactive (90.62%) | inactive (105%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FAK | inactive (92.52%) | inactive (124%) |
PYK2 | inactive (78.76%) | inactive (133%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FER | inactive (90.05%) | inactive (113%) |
FES | inactive (102.71%) | inactive (115%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FGFR1 | inactive (92.62%) | inactive (131%) |
FGFR2 | inactive (85.33%) | inactive (112%) |
FGFR3 | inactive (97.55%) | inactive (114%) |
FGFR4 | inactive (74.53%) | inactive (112%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FLT1 | inactive (89.38%) | inactive (97%) |
FLT4 | inactive (98.68%) | inactive (99%) |
KDR | inactive (106.36%) | inactive (105%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IGF1R | inactive (89.43%) | inactive (134%) |
IRR | inactive (98.14%) | inactive (89%) |
INSR | inactive (84.91%) | inactive (111%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
JAK1 | inactive (106.5%) | - |
JAK2 | inactive (106.29%) | inactive (101%) |
JAK3 | inactive (91.03%) | inactive (110%) |
TYK2 | inactive (103.78%) | - |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MUSK | inactive (109.86%) | inactive (98%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RET | inactive (96.54%) | inactive (96%) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RON | inactive (101.65%) | inactive (104%) |
MET | inactive (97.49%) | inactive (89%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ROS | inactive (104.1%) | inactive (89%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SYK | inactive (90.6%) | inactive (125%) |
ZAP70 | inactive (100.45%) | inactive (126%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TIE2 | inactive (94.57%) | inactive (95%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TRKA | inactive (100.18%) | inactive (79%) |
TRKB | inactive (103.08%) | inactive (122%) |
TRKC | inactive (96.03%) | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK1 | inactive (97.62%) | - |
ALK2 | inactive (96.73%) | - |
ALK4 | inactive (97.86%) | inactive (126%) |
TGFbR1 | inactive (97.78%) | inactive (90%) |
TGFbR2 | inactive (99.36%) | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ARAF | inactive (96.14%) | - |
BRAF | inactive (94.21%) | - |
RAF1 | inactive (89.56%) | inactive (76%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IRAK1 | inactive (118%) | inactive (97%) |
IRAK4 | inactive (89.15%) | inactive (113%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LIMK1 | inactive (93.99%) | inactive (104%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LRRK2 | inactive (97.74%) | - |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MLK1 | inactive (93.55%) | inactive (99%) |
MLK2 | inactive (98.28%) | - |
MLK3 | inactive (96.19%) | - |
TAK1 | inactive (104.5%) | inactive (91%) |
ZAK | inactive (103.73%) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RIPK2 | inactive (100.45%) | inactive (101%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NuaK1 | inactive (95.55%) | inactive (114%) |
BRSK1 | inactive (106.63%) | inactive (100%) |
BRSK2 | inactive (97.88%) | inactive (127%) |
CHK1 | inactive (95.84%) | inactive (89%) |
LKB1 | inactive (92.22%) | inactive (105%) |
MARK1 | inactive (95.28%) | inactive (85%) |
MARK3 | inactive (72.49%) | - |
MARK4 | inactive (104.43%) | - |
MELK | inactive (98.58%) | inactive (98%) |
PASK | inactive (85.98%) | inactive (132%) |
QIK | inactive (95.93%) | - |
NuaK2 | inactive (136.62%) | - |
MARK2 | inactive (97.94%) | inactive (99%) |
AMPKa1 | - | inactive (90%) |
AMPKa2 | - | inactive (115%) |
SIK | - | inactive (110%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK1a | inactive (95.41%) | inactive (104%) |
CaMK1b | inactive (97.25%) | - |
CaMK1d | inactive (97.65%) | inactive (110%) |
CaMK1g | inactive (97.97%) | - |
CaMK4 | inactive (98.07%) | inactive (118%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK2a | inactive (104.02%) | - |
CaMK2b | inactive (99.34%) | inactive (94%) |
CaMK2d | inactive (96.7%) | inactive (106%) |
CaMK2g | inactive (84.44%) | inactive (116%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CHK2 | inactive (96.79%) | inactive (81%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DAPK1 | inactive (126.48%) | inactive (87%) |
DAPK2 | inactive (97.25%) | inactive (103%) |
DRAK1 | inactive (113.53%) | inactive (85%) |
DAPK3 | inactive (94.17%) | inactive (97%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DCLK2 | inactive (95.72%) | inactive (108%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAPKAPK2 | inactive (100.37%) | inactive (80%) |
MAPKAPK3 | inactive (98.02%) | inactive (111%) |
MAPKAPK5 | inactive (93.9%) | inactive (84%) |
MNK1 | inactive (84.04%) | - |
MNK2 | inactive (80.77%) | inactive (111%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
smMLCK | inactive (101.34%) | inactive (93%) |
skMLCK | inactive (100.7%) | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PHKg1 | inactive (92.19%) | - |
PHKg2 | inactive (94.78%) | inactive (106%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PIM1 | inactive (106.38%) | inactive (87%) |
PIM2 | inactive (97.31%) | inactive (125%) |
PIM3 | inactive (102.36%) | inactive (100%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKD1 | inactive (98.67%) | inactive (102%) |
PKD3 | inactive (95.42%) | - |
PKD2 | inactive (100.12%) | inactive (94%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TSSK1 | inactive (84.19%) | inactive (95%) |
TSSK2 | inactive (99.17%) | inactive (93%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
STK33 | inactive (96.04%) | inactive (92%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP3K5 | inactive (105.6%) | inactive (91%) |
MAP3K2 | inactive (82.69%) | - |
MAP3K3 | inactive (99.46%) | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
COT | inactive (93.96%) | - |
NIK | inactive (105.26%) | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GCK | inactive (93.92%) | inactive (89%) |
HGK | inactive (94.96%) | - |
KHS1 | inactive (102.39%) | - |
LOK | inactive (93.96%) | inactive (101%) |
MINK | inactive (103.79%) | inactive (104%) |
MST1 | inactive (100.96%) | inactive (98%) |
MST2 | inactive (89.35%) | inactive (110%) |
MST3 | inactive (100.68%) | inactive (78%) |
MST4 | inactive (98.27%) | - |
OSR1 | inactive (100.55%) | - |
PAK1 | inactive (98.95%) | - |
PAK2 | inactive (58.06%) | inactive (106%) |
PAK3 | inactive (121.17%) | inactive (78%) |
PAK4 | inactive (87.91%) | inactive (97%) |
PAK5 | inactive (92%) | inactive (85%) |
PAK6 | inactive (88.97%) | inactive (100%) |
SLK | inactive (96.42%) | - |
YSK1 | inactive (92.96%) | - |
STLK3 | inactive (89.13%) | - |
TAO1 | inactive (95.94%) | inactive (108%) |
TAO2 | inactive (89.62%) | inactive (115%) |
TAO3 | inactive (93.6%) | inactive (106%) |
MYO3B | inactive (91.26%) | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP2K1 | inactive (96.96%) | inactive (103%) |
MAP2K2 | inactive (105.42%) | - |
MAP2K6 | inactive (102.91%) | inactive (84%) |
MAP2K7 | - | inactive (88%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AurA | inactive (96.51%) | inactive (98%) |
AurB | inactive (95.54%) | inactive (105%) |
AurC | inactive (97.2%) | inactive (98%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMKK1 | inactive (102.43%) | - |
CaMKK2 | inactive (94.61%) | - |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Haspin | inactive (96.68%) | inactive (100%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IKKa | inactive (95.97%) | inactive (92%) |
IKKb | inactive (104.87%) | inactive (108%) |
IKKe | inactive (102.82%) | - |
TBK1 | inactive (90.73%) | inactive (84%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NEK1 | inactive (98.89%) | - |
NEK11 | inactive (100.16%) | inactive (75%) |
NEK2 | inactive (94.71%) | inactive (82%) |
NEK4 | inactive (92.43%) | - |
NEK6 | inactive (98.74%) | inactive (112%) |
NEK7 | inactive (103.84%) | inactive (97%) |
NEK9 | inactive (97.01%) | - |
NEK3 | inactive (96.53%) | inactive (115%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PBK | inactive (90.69%) | - |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PLK1 | inactive (97.79%) | inactive (88%) |
PLK2 | inactive (103.63%) | inactive (99%) |
PLK3 | inactive (97.63%) | inactive (84%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SgK496 | inactive (89.58%) | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MPSK1 | inactive (102.54%) | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TTK | inactive (104.17%) | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ULK1 | inactive (89.48%) | - |
ULK2 | inactive (103.24%) | inactive (110%) |
ULK3 | inactive (79.58%) | inactive (103%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wee1 | inactive (83.85%) | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wnk2 | inactive (103.52%) | inactive (103%) |
Wnk3 | inactive (96.23%) | inactive (102%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TLK2 | inactive (105.57%) | inactive (95%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK1 | 7 | 6 | 4 |
VRK | 3 | 1 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK1d | inactive (104.04%) | inactive (86%) |
CK1g1 | inactive (90.95%) | inactive (93%) |
CK1g2 | inactive (93.04%) | inactive (102%) |
CK1g3 | inactive (102.03%) | inactive (116%) |
CK1a | inactive (94.91%) | - |
CK1e | inactive (116.82%) | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
VRK1 | inactive (110.04%) | - |
VRK2 | - | inactive (105%) |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK2 | 3 | 2 | 2 |
CLK | 4 | 4 | 2 |
DYRK | 10 | 9 | 4 |
MAPK | 14 | 10 | 10 |
GSK | 2 | 2 | 2 |
SRPK | 3 | 3 | 3 |
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK2a1 | inactive (87.09%) | inactive (97%) |
CK2a2 | inactive (106.79%) | inactive (128%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CLK1 | inactive (100.24%) | - |
CLK2 | inactive (87.38%) | inactive (112%) |
CLK3 | inactive (102.37%) | inactive (89%) |
CLK4 | inactive (102.52%) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DYRK1A | inactive (95.72%) | - |
DYRK1B | inactive (107.67%) | - |
DYRK2 | inactive (101.62%) | inactive (96%) |
DYRK3 | inactive (97.26%) | - |
DYRK4 | inactive (93.07%) | - |
HIPK1 | inactive (95.17%) | inactive (93%) |
HIPK2 | inactive (99.64%) | inactive (94%) |
HIPK3 | inactive (97.35%) | inactive (102%) |
HIPK4 | inactive (82.65%) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Erk1 | inactive (97.82%) | inactive (80%) |
Erk2 | inactive (116.78%) | inactive (105%) |
JNK3 | inactive (97.15%) | inactive (105%) |
NLK | inactive (77%) | inactive (95%) |
p38a | inactive (120.45%) | inactive (80%) |
p38b | inactive (93.62%) | inactive (102%) |
p38d | inactive (101.53%) | inactive (105%) |
p38g | inactive (90.79%) | inactive (107%) |
JNK1 | inactive (107.38%) | inactive (121%) |
JNK2 | inactive (84.26%) | inactive (108%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GSK3A | inactive (99.68%) | inactive (113%) |
GSK3B | inactive (109.62%) | inactive (98%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSSK1 | inactive (98.34%) | inactive (118%) |
SRPK1 | inactive (101.8%) | inactive (108%) |
SRPK2 | inactive (94.07%) | inactive (94%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
PDHK | 5 | 1 | - |
Alpha | 6 | - | 1 |
PIKK | 6 | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDHK1 | inactive (72.61%) | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
eEF2K | - | inactive (94%) |
Atypical - PIKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FRAP | - | inactive (114%) |