Compound Information
Test on : DRx, RBC, Metz
Compound Name
DRx : (3S,4R)-Tofacitinib
RBC : (3R,4S)-Tofacitinib
Metz : racemic-Tasocitinib
Inchikey
Same : UJLAWZDWDVHWOW-N
DRx : UJLAWZDWDVHWOW-DGCLKSJQSA-N
RBC : UJLAWZDWDVHWOW-AAEUAGOBSA-N
Metz : UJLAWZDWDVHWOW-UHFFFAOYSA-N
ChemSpider
DRx : 8142130
RBC : 24691638
Metz : 7993981
Pubchem CID
DRx : 9966538
RBC : 25180101
Metz : 9818231
ChEMBL
DRx : CHEMBL459977
RBC : CHEMBL457871
Metz : CHEMBL234085
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
Other
Other - NAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AAK1 | inactive (10001nM) | - | - |
BIKE | inactive (7100nM) | - | - |
GAK | inactive (10001nM) | - | - |
MPSK1 | inactive (10001nM) | inactive (94.69%) | - |
Other - Aur
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AurA | inactive (10001nM) | inactive (84.13%) | inactive (>1584.89nM) |
AurB | inactive (10001nM) | inactive (99.25%) | inactive (>3981.07nM) |
AurC | inactive (10001nM) | inactive (85.31%) | - |
Other - CAMKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CaMKK1 | inactive (10001nM) | inactive (100.53%) | - |
CaMKK2 | inactive (10001nM) | inactive (97.66%) | inactive (>2511.89nM) |
Other - PEK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
HRI | inactive (10001nM) | - | - |
PKR | inactive (10001nM) | - | - |
Other - IRE
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IRE1 | inactive (10001nM) | - | - |
Other - IKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IKKa | inactive (10001nM) | inactive (94.96%) | - |
IKKb | inactive (10001nM) | inactive (88.18%) | - |
IKKe | inactive (10001nM) | inactive (94.77%) | inactive (>3162.28nM) |
TBK1 | inactive (10001nM) | inactive (92.53%) | inactive (>3162.28nM) |
Other - NEK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
NEK1 | inactive (10001nM) | inactive (84.64%) | - |
NEK11 | inactive (10001nM) | inactive (91.69%) | - |
NEK2 | inactive (10001nM) | inactive (103.32%) | inactive (>3981.07nM) |
NEK3 | inactive (10001nM) | inactive (94.48%) | - |
NEK4 | inactive (10001nM) | inactive (96.04%) | inactive (>6309.57nM) |
NEK5 | inactive (10001nM) | - | - |
NEK6 | inactive (10001nM) | inactive (83.19%) | - |
NEK7 | inactive (10001nM) | inactive (93.99%) | - |
NEK9 | inactive (10001nM) | inactive (96.2%) | - |
Other - WEE
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MYT1 | inactive (10001nM) | - | - |
Wee1 | inactive (10001nM) | inactive (97.72%) | - |
Wee1B | inactive (10001nM) | - | - |
Other - PLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PLK1 | inactive (10001nM) | inactive (100.93%) | inactive (>7943.28nM) |
PLK2 | inactive (10001nM) | inactive (102.27%) | - |
PLK3 | inactive (10001nM) | inactive (99.08%) | inactive (>7943.28nM) |
PLK4 | inactive (10001nM) | - | inactive (>3981.07nM) |
Other - SgK496
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SgK496 | inactive (10001nM) | inactive (98.41%) | - |
Other - NKF1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SBK | inactive (10001nM) | - | - |
SgK110 | inactive (10001nM) | - | - |
Other - NKF4
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CLIK1 | inactive (10001nM) | - | - |
Other - ULK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Fused | inactive (10001nM) | - | - |
ULK1 | inactive (10001nM) | inactive (83.05%) | - |
ULK2 | inactive (10001nM) | inactive (92.04%) | - |
ULK3 | inactive (6400nM) | inactive (101.31%) | - |
Other - TLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TLK1 | inactive (10001nM) | - | - |
TLK2 | inactive (10001nM) | inactive (94.41%) | - |
Other - TTK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TTK | inactive (10001nM) | inactive (107.75%) | - |
Other - Haspin
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Haspin | - | inactive (77.94%) | - |
Other - TOPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PBK | - | inactive (101.6%) | inactive (>7943.28nM) |
Other - WNK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Wnk2 | - | inactive (100.52%) | - |
Wnk3 | - | inactive (103.88%) | - |
Other - CDC7
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CDC7 | - | - | inactive (>1258.93nM) |
TK
TK - Abl
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ABL1 | inactive (10001nM) | inactive (100.92%) | inactive (>3981.07nM) |
ABL2 | inactive (10001nM) | inactive (90.51%) | - |
TK - ALK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ALK | inactive (10001nM) | inactive (106.54%) | inactive (>6309.57nM) |
LTK | inactive (10001nM) | inactive (96.02%) | inactive (>1000nM) |
TK - Axl
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AXL | inactive (10001nM) | inactive (97.7%) | inactive (>1995.26nM) |
MER | inactive (10001nM) | inactive (113.67%) | - |
TYRO3 | inactive (10001nM) | inactive (102.8%) | inactive (>3162.28nM) |
TK - Src
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
BLK | inactive (10001nM) | inactive (92.53%) | inactive (>1584.89nM) |
BRK | inactive (10001nM) | inactive (100.89%) | inactive (>2511.89nM) |
FGR | inactive (10001nM) | inactive (91.09%) | - |
FRK | inactive (10001nM) | inactive (105.98%) | inactive (>2511.89nM) |
FYN | active (1100nM) | inactive (93.96%) | inactive (>5011.87nM) |
HCK | inactive (10001nM) | inactive (88.3%) | inactive (>3162.28nM) |
LCK | active (460nM) | inactive (80.24%) | inactive (>6309.57nM) |
LYN | inactive (10001nM) | inactive (96.35%) | inactive (>1584.89nM) |
SRC | inactive (10001nM) | inactive (99.77%) | inactive (>1995.26nM) |
SRM | inactive (10001nM) | inactive (95.82%) | inactive (>1584.89nM) |
YES | inactive (10001nM) | inactive (87.06%) | - |
TK - Tec
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
BMX | inactive (10001nM) | inactive (110.76%) | - |
BTK | inactive (10001nM) | inactive (98.72%) | inactive (>6309.57nM) |
ITK | inactive (10001nM) | inactive (99.14%) | inactive (>5011.87nM) |
TEC | inactive (10001nM) | inactive (95.44%) | - |
TXK | inactive (10001nM) | inactive (98.42%) | - |
TK - PDGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FMS | inactive (10001nM) | inactive (100.56%) | inactive (>2511.89nM) |
FLT3 | inactive (10001nM) | inactive (77.86%) | inactive (>1995.26nM) |
KIT | inactive (10001nM) | inactive (98.86%) | inactive (>5011.87nM) |
PDGFRa | inactive (10001nM) | inactive (104.11%) | inactive (>3162.28nM) |
PDGFRb | inactive (10001nM) | inactive (95.1%) | inactive (>1995.26nM) |
TK - Csk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CSK | inactive (10001nM) | inactive (100.63%) | - |
CTK | inactive (10001nM) | inactive (66.89%) | inactive (>1995.26nM) |
TK - DDR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DDR1 | inactive (10001nM) | - | - |
DDR2 | inactive (10001nM) | inactive (104.4%) | - |
TK - EGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
EGFR | inactive (10001nM) | inactive (95.96%) | inactive (>1995.26nM) |
ErbB2 | inactive (10001nM) | inactive (108.75%) | inactive (>1584.89nM) |
ErbB3 | inactive (10001nM) | - | - |
ErbB4 | inactive (10001nM) | inactive (100.25%) | inactive (>3981.07nM) |
TK - Eph
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
EphA1 | inactive (10001nM) | inactive (97.97%) | - |
EphA2 | inactive (10001nM) | inactive (95.75%) | inactive (>3162.28nM) |
EphA3 | inactive (10001nM) | inactive (94.09%) | - |
EphA4 | inactive (10001nM) | inactive (99.06%) | - |
EphA5 | inactive (10001nM) | inactive (99.94%) | - |
EphA6 | inactive (10001nM) | inactive (98.98%) | - |
EphA7 | inactive (10001nM) | inactive (89.04%) | - |
EphA8 | inactive (10001nM) | inactive (108.81%) | - |
EphB1 | inactive (10001nM) | inactive (105.59%) | - |
EphB2 | inactive (10001nM) | inactive (100.21%) | - |
EphB3 | inactive (10001nM) | inactive (54.86%) | - |
EphB4 | inactive (10001nM) | inactive (89.83%) | - |
EphB6 | inactive (10001nM) | - | - |
TK - FAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FAK | inactive (10001nM) | inactive (103.35%) | inactive (>6309.57nM) |
PYK2 | inactive (10001nM) | inactive (100.12%) | inactive (>1584.89nM) |
TK - Fer
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FER | inactive (10001nM) | inactive (104.16%) | inactive (>1584.89nM) |
FES | inactive (10001nM) | inactive (103.64%) | inactive (>1995.26nM) |
TK - FGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FGFR1 | inactive (10001nM) | inactive (101.08%) | inactive (>3981.07nM) |
FGFR2 | inactive (10001nM) | inactive (91.68%) | - |
FGFR3 | inactive (10001nM) | inactive (95.27%) | inactive (>1995.26nM) |
FGFR4 | inactive (10001nM) | inactive (94.28%) | - |
TK - VEGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FLT1 | inactive (10001nM) | inactive (100.56%) | inactive (>3981.07nM) |
FLT4 | inactive (10001nM) | inactive (97.52%) | inactive (>6309.57nM) |
KDR | inactive (10001nM) | inactive (105.92%) | inactive (>1000nM) |
TK - InsR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IGF1R | inactive (10001nM) | inactive (93.1%) | inactive (>2511.89nM) |
INSR | inactive (10001nM) | inactive (101.25%) | inactive (>5011.87nM) |
IRR | inactive (10001nM) | inactive (97.47%) | - |
TK - JakA
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
JAK1 | active (1.6nM) | active (2.3%) | - |
JAK2 | active (0.58nM) | active (5.14%) | active (3.98nM) |
JAK3 | active (0.16nM) | active (1.93%) | active (5.01nM) |
TYK2 | active (4.8nM) | active (12.04%) | active (50.12nM) |
TK - Met
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MET | inactive (10001nM) | inactive (86.66%) | inactive (>2511.89nM) |
RON | inactive (10001nM) | inactive (102%) | inactive (>3981.07nM) |
TK - Musk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MUSK | inactive (10001nM) | inactive (103.43%) | - |
TK - Ret
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
RET | inactive (10001nM) | inactive (92.43%) | inactive (>3981.07nM) |
TK - Sev
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ROS | inactive (10001nM) | inactive (94.09%) | inactive (>3162.28nM) |
TK - Syk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SYK | inactive (10001nM) | inactive (107.39%) | inactive (>1584.89nM) |
ZAP70 | inactive (10001nM) | inactive (104.83%) | - |
TK - Tie
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TIE1 | inactive (10001nM) | - | - |
TIE2 | inactive (10001nM) | inactive (96.58%) | - |
TK - Ack
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TNK1 | active (120nM) | - | - |
ACK | inactive (10001nM) | inactive (87.07%) | inactive (>3981.07nM) |
TK - Trk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TRKA | inactive (10001nM) | inactive (94.13%) | inactive (>3162.28nM) |
TRKB | inactive (10001nM) | inactive (97.08%) | inactive (>3981.07nM) |
TRKC | inactive (10001nM) | inactive (90.04%) | inactive (>3162.28nM) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ALK2 | inactive (10001nM) | inactive (104.12%) | inactive (>3981.07nM) |
ALK4 | inactive (10001nM) | inactive (99.76%) | - |
ACTR2 | inactive (10001nM) | - | - |
ACTR2B | inactive (10001nM) | - | - |
ALK1 | inactive (10001nM) | inactive (100.43%) | - |
BMPR1A | inactive (10001nM) | - | - |
BMPR1B | inactive (10001nM) | - | - |
BMPR2 | inactive (10001nM) | - | - |
TGFbR1 | inactive (10001nM) | inactive (98.83%) | - |
TGFbR2 | inactive (10001nM) | inactive (98.76%) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SgK288 | inactive (10001nM) | - | - |
RIPK1 | inactive (10001nM) | - | - |
RIPK2 | inactive (10001nM) | inactive (112.68%) | - |
ANKRD3 | inactive (10001nM) | - | - |
TKL - RAF
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
BRAF | inactive (10001nM) | inactive (93.69%) | - |
RAF1 | inactive (10001nM) | inactive (95.46%) | - |
ARAF | - | inactive (102.24%) | - |
TKL - MLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DLK | inactive (10001nM) | - | - |
LZK | inactive (10001nM) | - | - |
MLK1 | inactive (10001nM) | inactive (113.25%) | - |
MLK2 | inactive (10001nM) | inactive (105.13%) | inactive (>3162.28nM) |
MLK3 | inactive (10001nM) | inactive (104.31%) | - |
TAK1 | inactive (10001nM) | inactive (87.46%) | - |
HH498 | inactive (10001nM) | - | - |
ZAK | inactive (10001nM) | inactive (98.18%) | inactive (>7943.28nM) |
TKL - IRAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IRAK1 | inactive (10001nM) | inactive (93.93%) | inactive (>7943.28nM) |
IRAK3 | inactive (10001nM) | - | - |
IRAK4 | inactive (10001nM) | inactive (88.48%) | inactive (>10000nM) |
TKL - LISK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
LIMK1 | inactive (10001nM) | inactive (81.96%) | inactive (>3162.28nM) |
LIMK2 | inactive (10001nM) | - | - |
TESK1 | inactive (10001nM) | - | - |
TKL - LRRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
LRRK2 | active (1300nM) | inactive (51.35%) | active (199.53nM) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz |
---|
ABC1 | 5 | 2 | - | - |
PIKK | 6 | 1 | - | - |
RIO | 3 | 3 | - | - |
Alpha | 6 | 1 | - | 1 |
PDHK | 5 | - | 1 | - |
Atypical - ABC1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ADCK3 | inactive (10001nM) | - | - |
ADCK4 | inactive (10001nM) | - | - |
Atypical - PIKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FRAP | inactive (10001nM) | - | - |
Atypical - RIO
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
RIOK1 | inactive (10001nM) | - | - |
RIOK2 | inactive (10001nM) | - | - |
RIOK3 | inactive (10001nM) | - | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ChaK2 | inactive (10001nM) | - | - |
eEF2K | - | - | inactive (>3981.07nM) |
Atypical - PDHK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PDHK1 | - | inactive (94.07%) | - |
AGC
AGC - Akt
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AKT1 | inactive (10001nM) | inactive (90.27%) | inactive (>7943.28nM) |
AKT2 | inactive (10001nM) | inactive (98.03%) | inactive (>7943.28nM) |
AKT3 | inactive (10001nM) | inactive (85.83%) | inactive (>7943.28nM) |
AGC - DMPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CRIK | inactive (10001nM) | - | - |
DMPK1 | active (1200nM) | inactive (108.48%) | - |
DMPK2 | inactive (10001nM) | - | - |
MRCKa | inactive (10001nM) | inactive (110.03%) | inactive (>10000nM) |
MRCKb | inactive (10001nM) | inactive (95.41%) | - |
ROCK1 | active (470nM) | inactive (90.13%) | active (251.19nM) |
ROCK2 | active (420nM) | inactive (69.86%) | active (398.11nM) |
AGC - GRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
RHOK | inactive (10001nM) | - | - |
GPRK4 | inactive (10001nM) | inactive (93.47%) | - |
GPRK7 | inactive (4300nM) | inactive (101.65%) | - |
BARK1 | - | inactive (95.26%) | - |
BARK2 | - | inactive (99.23%) | - |
GPRK5 | - | inactive (107.02%) | inactive (>3981.07nM) |
GPRK6 | - | inactive (100.81%) | - |
AGC - NDR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
LATS1 | inactive (10001nM) | - | - |
LATS2 | inactive (10001nM) | - | - |
NDR1 | inactive (10001nM) | inactive (95.68%) | - |
NDR2 | inactive (10001nM) | - | - |
AGC - MAST
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAST1 | inactive (10001nM) | - | - |
AGC - PDK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PDK1 | inactive (10001nM) | inactive (94.07%) | inactive (>3981.07nM) |
AGC - PKA
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKACa | inactive (10001nM) | inactive (96.54%) | inactive (>3162.28nM) |
PKACb | inactive (10001nM) | - | - |
PRKX | inactive (10001nM) | inactive (109.77%) | inactive (>3162.28nM) |
PKACg | - | inactive (110.73%) | - |
AGC - PKN
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKN1 | active (170nM) | active (16.5%) | - |
PKN2 | active (1200nM) | inactive (85.55%) | active (251.19nM) |
AGC - PKC
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKCd | active (2000nM) | inactive (75.29%) | inactive (6309.57nM) |
PKCe | inactive (10001nM) | inactive (98.51%) | - |
PKCh | inactive (10001nM) | inactive (100.23%) | - |
PKCi | inactive (10001nM) | inactive (103.42%) | inactive (>5011.87nM) |
PKCt | inactive (10001nM) | inactive (89.03%) | inactive (>1995.26nM) |
PKCa | - | inactive (78.73%) | - |
PKCg | - | inactive (90.56%) | inactive (3981.07nM) |
PKCz | - | inactive (91.72%) | inactive (>7943.28nM) |
PKCb | - | inactive (88.11%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKG1 | inactive (10001nM) | inactive (82.05%) | inactive (>1995.26nM) |
PKG2 | inactive (10001nM) | inactive (106.03%) | inactive (>1584.89nM) |
AGC - RSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
p70S6K | inactive (10001nM) | inactive (102.86%) | inactive (>3981.07nM) |
MSK1 | - | inactive (94.83%) | inactive (>1995.26nM) |
MSK2 | - | inactive (104.64%) | - |
p70S6Kb | - | inactive (100.47%) | - |
RSK2 | - | inactive (96.99%) | inactive (>3981.07nM) |
RSK4 | - | inactive (98.15%) | - |
RSK1 | - | inactive (90.91%) | - |
RSK3 | - | inactive (89.66%) | - |
AGC - SGK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SGK3 | inactive (10001nM) | inactive (98.06%) | - |
SGK1 | - | inactive (122.84%) | inactive (>6309.57nM) |
SGK2 | - | inactive (103.65%) | - |
AGC - YANK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
YANK1 | inactive (10001nM) | - | - |
YANK2 | inactive (10001nM) | - | - |
YANK3 | inactive (10001nM) | - | - |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AMPKa1 | inactive (10001nM) | - | inactive (>3162.28nM) |
AMPKa2 | inactive (10001nM) | - | - |
NuaK1 | inactive (10001nM) | inactive (71.18%) | - |
BRSK1 | inactive (10001nM) | inactive (101.71%) | inactive (>10000nM) |
BRSK2 | inactive (10001nM) | inactive (86.94%) | - |
CHK1 | inactive (10001nM) | inactive (94.12%) | inactive (>3981.07nM) |
HUNK | inactive (10001nM) | - | - |
LKB1 | inactive (10001nM) | inactive (103.67%) | - |
MARK1 | inactive (10001nM) | inactive (118.55%) | - |
MARK2 | inactive (10001nM) | inactive (91.83%) | active (630.96nM) |
MARK3 | inactive (10001nM) | inactive (78.64%) | active (630.96nM) |
MARK4 | inactive (10001nM) | inactive (81.68%) | active (630.96nM) |
MELK | inactive (10001nM) | inactive (79.44%) | inactive (>630.96nM) |
NIM1 | inactive (10001nM) | - | - |
QSK | inactive (10001nM) | - | - |
SIK | inactive (10001nM) | - | - |
QIK | inactive (10001nM) | inactive (89.23%) | inactive (1258.93nM) |
NuaK2 | active (240nM) | inactive (80.25%) | - |
SNRK | inactive (10001nM) | - | - |
PASK | - | inactive (105.23%) | - |
CAMK - CAMK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CaMK1a | active (1200nM) | inactive (99.27%) | inactive (>7943.28nM) |
CaMK1d | active (1600nM) | inactive (111.35%) | inactive (>1584.89nM) |
CaMK1g | inactive (10001nM) | inactive (97.81%) | - |
CaMK4 | inactive (10001nM) | inactive (96.25%) | - |
CaMK1b | - | inactive (104.03%) | - |
CAMK - CAMK2
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CaMK2a | inactive (3500nM) | inactive (99.64%) | inactive (>3981.07nM) |
CaMK2b | inactive (10001nM) | inactive (96.61%) | inactive (>7943.28nM) |
CaMK2d | active (2700nM) | inactive (98.17%) | inactive (1258.93nM) |
CaMK2g | inactive (10001nM) | inactive (126.64%) | inactive (>3981.07nM) |
CAMK - CASK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CASK | inactive (10001nM) | - | - |
CAMK - RAD53
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CHK2 | inactive (10001nM) | inactive (104%) | inactive (>1584.89nM) |
CAMK - DAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DAPK1 | inactive (10001nM) | inactive (108.52%) | - |
DAPK2 | inactive (10001nM) | inactive (89.5%) | - |
DAPK3 | inactive (10001nM) | inactive (105.7%) | inactive (>5011.87nM) |
DRAK1 | inactive (10001nM) | inactive (105.93%) | inactive (>3981.07nM) |
DRAK2 | inactive (10001nM) | - | - |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DCLK1 | inactive (6700nM) | - | inactive (>10000nM) |
DCLK2 | inactive (10001nM) | inactive (96.63%) | - |
DCLK3 | active (12nM) | - | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAPKAPK2 | inactive (10001nM) | inactive (96.63%) | inactive (>7943.28nM) |
MAPKAPK5 | inactive (10001nM) | inactive (97.32%) | inactive (>1584.89nM) |
MNK1 | inactive (10001nM) | inactive (89.94%) | - |
MNK2 | active (1600nM) | inactive (97.38%) | inactive (>10000nM) |
MAPKAPK3 | - | inactive (100.22%) | inactive (>10000nM) |
CAMK - MLCK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
caMLCK | inactive (10001nM) | - | - |
smMLCK | inactive (10001nM) | inactive (89.95%) | - |
skMLCK | inactive (10001nM) | inactive (98.97%) | - |
SgK085 | inactive (10001nM) | - | - |
CAMK - PHK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PHKg1 | inactive (10001nM) | inactive (90%) | - |
PHKg2 | inactive (10001nM) | inactive (98.64%) | inactive (>5011.87nM) |
CAMK - PIM
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PIM1 | inactive (10001nM) | inactive (101.99%) | inactive (>6309.57nM) |
PIM2 | inactive (10001nM) | inactive (115.85%) | inactive (>1584.89nM) |
PIM3 | inactive (10001nM) | inactive (96.47%) | inactive (>7943.28nM) |
CAMK - PKD
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKD1 | inactive (10001nM) | inactive (97.32%) | - |
PKD2 | inactive (10001nM) | inactive (92.61%) | inactive (>10000nM) |
PKD3 | inactive (10001nM) | inactive (89.78%) | inactive (>3981.07nM) |
CAMK - STK33
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
STK33 | inactive (10001nM) | inactive (97.78%) | - |
CAMK - TSSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TSSK1 | inactive (10001nM) | inactive (85.05%) | inactive (>1584.89nM) |
TSSK2 | - | inactive (87.91%) | inactive (>1584.89nM) |
STE
STE - STE11
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAP3K5 | inactive (10001nM) | inactive (97.83%) | - |
MAP3K6 | inactive (10001nM) | - | - |
MAP3K1 | inactive (10001nM) | - | - |
MAP3K7 | inactive (10001nM) | - | - |
MAP3K2 | inactive (10001nM) | inactive (122.78%) | - |
MAP3K3 | inactive (10001nM) | inactive (114.8%) | - |
MAP3K4 | inactive (10001nM) | - | - |
MAP3K8 | inactive (10001nM) | - | - |
STE - STE20
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
HPK1 | inactive (10001nM) | - | - |
LOK | inactive (10001nM) | inactive (92.9%) | - |
GCK | inactive (4800nM) | inactive (101.97%) | inactive (>3162.28nM) |
KHS2 | inactive (10001nM) | - | - |
HGK | inactive (10001nM) | inactive (101.16%) | inactive (>5011.87nM) |
KHS1 | inactive (10001nM) | inactive (112.09%) | inactive (>7943.28nM) |
MINK | inactive (10001nM) | inactive (100.25%) | inactive (>7943.28nM) |
MST1 | inactive (10001nM) | inactive (95.49%) | - |
MST2 | inactive (10001nM) | inactive (85.77%) | inactive (>3162.28nM) |
MST3 | inactive (10001nM) | inactive (96.15%) | - |
MST4 | inactive (10001nM) | inactive (104.52%) | - |
MYO3A | inactive (10001nM) | - | - |
MYO3B | inactive (10001nM) | inactive (89.31%) | - |
OSR1 | inactive (10001nM) | inactive (98.25%) | - |
PAK1 | inactive (10001nM) | inactive (108.21%) | inactive (>10000nM) |
PAK2 | inactive (10001nM) | inactive (111.02%) | - |
PAK3 | inactive (10001nM) | inactive (105.36%) | - |
PAK4 | inactive (10001nM) | inactive (99.17%) | inactive (>5011.87nM) |
PAK6 | inactive (10001nM) | inactive (102.39%) | - |
PAK5 | inactive (10001nM) | inactive (93.64%) | - |
SLK | inactive (10001nM) | inactive (89.23%) | inactive (5011.87nM) |
STLK3 | inactive (10001nM) | inactive (95.14%) | - |
TAO1 | inactive (10001nM) | inactive (99.93%) | inactive (>6309.57nM) |
TAO2 | inactive (10001nM) | inactive (100.09%) | - |
TAO3 | inactive (10001nM) | inactive (94.87%) | - |
TNIK | inactive (10001nM) | - | - |
YSK1 | inactive (10001nM) | inactive (97.18%) | - |
STE - STE7
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAP2K1 | inactive (10001nM) | inactive (111.98%) | inactive (>3162.28nM) |
MAP2K2 | inactive (10001nM) | inactive (117.38%) | inactive (>3981.07nM) |
MAP2K3 | inactive (10001nM) | - | - |
MAP2K4 | inactive (10001nM) | - | - |
MAP2K5 | inactive (10001nM) | - | - |
MAP2K6 | inactive (10001nM) | inactive (99.42%) | - |
MAP2K7 | inactive (10001nM) | - | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
COT | - | inactive (93.5%) | - |
NIK | - | inactive (106.82%) | - |
CMGC
CMGC - CDK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PITSLRE | inactive (10001nM) | - | - |
CHED | inactive (10001nM) | - | - |
CDK11 | inactive (10001nM) | - | - |
PCTAIRE1 | inactive (10001nM) | - | - |
PCTAIRE2 | inactive (10001nM) | - | - |
PCTAIRE3 | inactive (10001nM) | - | - |
PFTAIRE2 | inactive (10001nM) | - | - |
PFTAIRE1 | inactive (10001nM) | - | - |
CDC2 | - | - | inactive (>7943.28nM) |
CDK2 | - | - | inactive (>7943.28nM) |
CDK5 | - | - | inactive (>3981.07nM) |
CDK8 | - | - | inactive (1584.89nM) |
CDK7 | - | - | inactive (>3981.07nM) |
CDK9 | - | - | inactive (>1584.89nM) |
CMGC - CDKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CDKL1 | inactive (10001nM) | - | - |
CDKL2 | inactive (10001nM) | - | - |
CDKL3 | inactive (10001nM) | - | - |
CDKL5 | inactive (10001nM) | - | - |
CMGC - CLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CLK1 | inactive (10001nM) | inactive (99.5%) | - |
CLK2 | inactive (10001nM) | inactive (85.77%) | inactive (>1995.26nM) |
CLK3 | inactive (10001nM) | inactive (105.54%) | - |
CLK4 | inactive (10001nM) | inactive (111.22%) | inactive (>3162.28nM) |
CMGC - CK2
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CK2a1 | inactive (10001nM) | inactive (103.65%) | inactive (>6309.57nM) |
CK2a2 | inactive (10001nM) | inactive (96.58%) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DYRK1A | inactive (10001nM) | inactive (101.97%) | inactive (>1995.26nM) |
DYRK1B | inactive (10001nM) | inactive (96.97%) | inactive (>2511.89nM) |
DYRK2 | inactive (10001nM) | inactive (111.71%) | - |
HIPK1 | inactive (10001nM) | inactive (98.07%) | - |
HIPK2 | inactive (10001nM) | inactive (96.9%) | inactive (>3162.28nM) |
HIPK3 | inactive (10001nM) | inactive (99.99%) | - |
HIPK4 | inactive (10001nM) | inactive (96.24%) | inactive (>7943.28nM) |
PRP4 | inactive (10001nM) | - | - |
DYRK3 | - | inactive (106.27%) | inactive (>6309.57nM) |
DYRK4 | - | inactive (97.22%) | inactive (>7943.28nM) |
CMGC - MAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Erk1 | inactive (10001nM) | inactive (98.62%) | - |
Erk2 | inactive (10001nM) | inactive (88.63%) | - |
Erk3 | inactive (10001nM) | - | - |
Erk4 | inactive (10001nM) | - | - |
Erk5 | inactive (10001nM) | - | - |
Erk7 | inactive (10001nM) | - | - |
JNK1 | inactive (10001nM) | inactive (108.13%) | inactive (>5011.87nM) |
JNK2 | inactive (10001nM) | inactive (112.1%) | inactive (>3981.07nM) |
JNK3 | inactive (10001nM) | inactive (100.43%) | inactive (>3162.28nM) |
NLK | inactive (10001nM) | inactive (109.53%) | - |
p38a | inactive (10001nM) | inactive (93.36%) | inactive (>3981.07nM) |
p38b | inactive (10001nM) | inactive (103.31%) | - |
p38d | inactive (10001nM) | inactive (93.77%) | inactive (>7943.28nM) |
p38g | inactive (10001nM) | inactive (96.73%) | inactive (>6309.57nM) |
CMGC - GSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
GSK3A | inactive (10001nM) | inactive (102.73%) | inactive (>3981.07nM) |
GSK3B | inactive (10001nM) | inactive (99.58%) | inactive (>3981.07nM) |
CMGC - RCK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ICK | inactive (10001nM) | - | - |
MAK | inactive (10001nM) | - | - |
CMGC - SRPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SRPK1 | inactive (10001nM) | inactive (99.77%) | inactive (>7943.28nM) |
SRPK2 | inactive (10001nM) | inactive (90.66%) | - |
MSSK1 | inactive (10001nM) | inactive (103.04%) | - |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz |
---|
CK1 | 7 | 7 | 6 | 5 |
VRK | 3 | 1 | 1 | - |
CK1 - CK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CK1a | inactive (10001nM) | inactive (99.74%) | inactive (>3981.07nM) |
CK1a2 | inactive (10001nM) | - | - |
CK1d | inactive (10001nM) | inactive (86.02%) | inactive (>7943.28nM) |
CK1e | inactive (10001nM) | inactive (101.07%) | - |
CK1g1 | inactive (10001nM) | inactive (101%) | - |
CK1g2 | inactive (10001nM) | inactive (95.4%) | inactive (>7943.28nM) |
CK1g3 | inactive (10001nM) | inactive (100.67%) | - |
CK1 - VRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
VRK2 | inactive (10001nM) | - | - |
VRK1 | - | inactive (100.09%) | - |