Compound Information
Test on : RBC, Millipore
Compound Name
RBC, Millipore : Alsterpaullone, 2-Cyanoethyl
Inchikey
Same : UBLFSMURWWWWMH-N
RBC, Millipore : UBLFSMURWWWWMH-UHFFFAOYSA-N
ChemSpider
RBC, Millipore : 21396098
Pubchem CID
RBC, Millipore : 16760286
ChEMBL
RBC, Millipore : CHEMBL260138
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDK1 | inactive (79.75%) | active (17%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AKT1 | inactive (111.3%) | inactive (108%) |
AKT2 | inactive (100.39%) | inactive (98%) |
AKT3 | inactive (95.52%) | inactive (102%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DMPK1 | inactive (89.76%) | inactive (109%) |
MRCKa | inactive (73.1%) | active (35%) |
MRCKb | inactive (54.06%) | active (9%) |
ROCK1 | active (38.92%) | inactive (52%) |
ROCK2 | active (28.59%) | active (8%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BARK1 | inactive (96.37%) | - |
BARK2 | inactive (97.07%) | - |
GPRK4 | inactive (100.51%) | - |
GPRK5 | inactive (103.02%) | inactive (96%) |
GPRK6 | inactive (91.53%) | inactive (105%) |
GPRK7 | inactive (97.72%) | inactive (85%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSK1 | inactive (94.19%) | inactive (108%) |
MSK2 | inactive (85.82%) | inactive (88%) |
p70S6K | inactive (97.98%) | inactive (97%) |
p70S6Kb | inactive (96.11%) | - |
RSK2 | active (28.62%) | active (9%) |
RSK4 | active (13.37%) | active (16%) |
RSK1 | inactive (59.89%) | active (8%) |
RSK3 | active (24.4%) | active (45%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKACg | - | - |
PRKX | inactive (78.37%) | inactive (72%) |
PKACa | inactive (87.57%) | inactive (85%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKCa | inactive (80.91%) | inactive (92%) |
PKCd | inactive (74.86%) | inactive (68%) |
PKCe | inactive (95.44%) | inactive (81%) |
PKCh | inactive (99.43%) | inactive (100%) |
PKCg | inactive (93.33%) | inactive (91%) |
PKCi | inactive (65.29%) | inactive (102%) |
PKCt | inactive (111.01%) | inactive (83%) |
PKCz | inactive (83.43%) | inactive (69%) |
PKCb | inactive (76.26%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKG2 | inactive (93.93%) | - |
PKG1 | inactive (99.28%) | - |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKN1 | inactive (77.98%) | - |
PKN2 | inactive (77.88%) | inactive (57%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SGK1 | inactive (87.86%) | inactive (89%) |
SGK2 | inactive (113.59%) | inactive (86%) |
SGK3 | inactive (99.23%) | inactive (113%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NDR1 | active (0%) | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ABL1 | active (47.8%) | active (31%) |
ABL2 | active (49.81%) | active (48%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ACK | inactive (75.44%) | active (32%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK | inactive (78.84%) | inactive (73%) |
LTK | inactive (79.97%) | - |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AXL | inactive (95.54%) | inactive (57%) |
MER | inactive (77.54%) | inactive (84%) |
TYRO3 | inactive (94.84%) | inactive (75%) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BLK | inactive (78.84%) | active (24%) |
BRK | inactive (94.55%) | inactive (105%) |
SRC | active (30.77%) | active (46%) |
FGR | active (31.01%) | active (15%) |
FRK | inactive (92.68%) | inactive (54%) |
FYN | inactive (52.23%) | active (17%) |
HCK | inactive (63.81%) | active (30%) |
LCK | inactive (78.2%) | active (14%) |
SRM | inactive (78.63%) | - |
YES | active (35.83%) | active (9%) |
LYN | active (22.97%) | active (5%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BMX | inactive (99.45%) | inactive (75%) |
BTK | inactive (94.58%) | inactive (79%) |
ITK | inactive (99.89%) | inactive (81%) |
TEC | inactive (119.51%) | - |
TXK | inactive (67.64%) | active (26%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
KIT | inactive (76.57%) | inactive (102%) |
FLT3 | active (15.08%) | active (19%) |
FMS | active (43.41%) | active (24%) |
PDGFRb | inactive (83.89%) | inactive (115%) |
PDGFRa | inactive (87.41%) | inactive (108%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CSK | inactive (96.31%) | inactive (104%) |
CTK | inactive (100.71%) | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DDR2 | inactive (104.61%) | inactive (98%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EGFR | inactive (94.44%) | inactive (100%) |
ErbB2 | inactive (98.57%) | - |
ErbB4 | inactive (91.76%) | inactive (97%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EphA1 | inactive (91.74%) | inactive (99%) |
EphA2 | inactive (93.6%) | inactive (100%) |
EphA3 | inactive (93.9%) | inactive (77%) |
EphA4 | inactive (85.19%) | inactive (107%) |
EphA5 | inactive (88.47%) | inactive (93%) |
EphA6 | - | - |
EphA7 | inactive (95.29%) | inactive (79%) |
EphA8 | inactive (104.53%) | inactive (77%) |
EphB1 | inactive (99.08%) | inactive (87%) |
EphB2 | inactive (98.47%) | inactive (104%) |
EphB3 | inactive (102.48%) | inactive (106%) |
EphB4 | inactive (82.16%) | inactive (86%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FAK | inactive (82.19%) | active (50%) |
PYK2 | inactive (62.94%) | active (19%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FER | inactive (72.72%) | inactive (90%) |
FES | active (37.94%) | active (16%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FGFR1 | inactive (91.9%) | active (47%) |
FGFR2 | inactive (93.2%) | inactive (104%) |
FGFR3 | inactive (90.27%) | inactive (108%) |
FGFR4 | inactive (89.11%) | inactive (101%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FLT1 | inactive (99.66%) | active (24%) |
FLT4 | inactive (66.49%) | active (10%) |
KDR | inactive (75.49%) | active (30%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IGF1R | inactive (92.18%) | inactive (117%) |
IRR | inactive (99.2%) | inactive (100%) |
INSR | inactive (94.08%) | inactive (118%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
JAK1 | inactive (91.94%) | - |
JAK2 | inactive (93.01%) | inactive (101%) |
JAK3 | inactive (101.07%) | inactive (104%) |
TYK2 | active (48.15%) | - |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MUSK | inactive (62.95%) | inactive (68%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RET | inactive (80.78%) | inactive (80%) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RON | inactive (106.89%) | inactive (87%) |
MET | inactive (119.09%) | inactive (90%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ROS | inactive (70.96%) | inactive (102%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SYK | inactive (58.02%) | inactive (56%) |
ZAP70 | inactive (106.44%) | inactive (107%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TIE2 | inactive (97.64%) | inactive (94%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TRKA | inactive (115.26%) | inactive (54%) |
TRKB | inactive (86.39%) | inactive (71%) |
TRKC | inactive (61.23%) | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK1 | inactive (53.56%) | - |
ALK2 | inactive (58.78%) | - |
ALK4 | inactive (109.92%) | inactive (67%) |
TGFbR1 | inactive (102.58%) | inactive (73%) |
TGFbR2 | active (10.12%) | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ARAF | inactive (94.46%) | - |
BRAF | inactive (99.29%) | - |
RAF1 | inactive (103.71%) | inactive (88%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IRAK1 | inactive (74.92%) | active (45%) |
IRAK4 | inactive (154.56%) | inactive (62%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LIMK1 | inactive (99.94%) | inactive (99%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LRRK2 | inactive (73.85%) | - |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MLK1 | active (18.22%) | active (7%) |
MLK2 | active (29.99%) | - |
MLK3 | active (18.43%) | - |
TAK1 | active (38.14%) | inactive (57%) |
ZAK | inactive (88.64%) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RIPK2 | active (21.54%) | active (18%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NuaK1 | active (14.12%) | active (10%) |
BRSK1 | active (46.8%) | inactive (84%) |
BRSK2 | active (42%) | active (39%) |
CHK1 | active (45.15%) | active (39%) |
LKB1 | inactive (96.33%) | inactive (96%) |
MARK1 | inactive (67.37%) | active (30%) |
MARK3 | inactive (67.28%) | - |
MARK4 | inactive (62.54%) | - |
MELK | inactive (88.6%) | inactive (69%) |
PASK | inactive (96.9%) | inactive (103%) |
QIK | active (44.19%) | - |
NuaK2 | inactive (67.63%) | - |
MARK2 | inactive (65.49%) | active (38%) |
AMPKa1 | - | inactive (57%) |
AMPKa2 | - | active (27%) |
SIK | - | inactive (96%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK1a | inactive (96.02%) | inactive (97%) |
CaMK1b | inactive (107.27%) | - |
CaMK1d | inactive (91.84%) | inactive (110%) |
CaMK1g | inactive (102.95%) | - |
CaMK4 | inactive (98.41%) | inactive (109%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK2a | inactive (69.14%) | - |
CaMK2b | inactive (99.26%) | inactive (54%) |
CaMK2d | inactive (57.84%) | active (10%) |
CaMK2g | inactive (66.03%) | active (6%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CHK2 | active (12.59%) | active (4%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DAPK1 | inactive (96.52%) | inactive (105%) |
DAPK2 | inactive (96.49%) | inactive (93%) |
DRAK1 | active (46.76%) | active (11%) |
DAPK3 | inactive (99.29%) | inactive (107%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DCLK2 | inactive (104.16%) | inactive (83%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAPKAPK2 | inactive (83.43%) | inactive (57%) |
MAPKAPK3 | inactive (96.75%) | inactive (100%) |
MAPKAPK5 | inactive (94.28%) | inactive (68%) |
MNK1 | inactive (66.67%) | - |
MNK2 | inactive (87.73%) | inactive (72%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
smMLCK | inactive (95.21%) | inactive (92%) |
skMLCK | inactive (93.85%) | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PHKg1 | active (7.72%) | - |
PHKg2 | inactive (99.06%) | inactive (93%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PIM1 | inactive (93.57%) | inactive (101%) |
PIM2 | inactive (104.49%) | inactive (120%) |
PIM3 | inactive (70.91%) | inactive (96%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKD1 | inactive (87.49%) | inactive (89%) |
PKD3 | inactive (84.02%) | - |
PKD2 | inactive (94.17%) | inactive (99%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TSSK1 | inactive (59.19%) | active (39%) |
TSSK2 | inactive (78.74%) | inactive (91%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
STK33 | inactive (78.8%) | inactive (100%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP3K5 | inactive (100.66%) | inactive (91%) |
MAP3K2 | inactive (61.55%) | - |
MAP3K3 | inactive (83.35%) | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
COT | inactive (87.49%) | - |
NIK | inactive (160.83%) | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GCK | active (13.97%) | active (2%) |
HGK | active (6.82%) | - |
KHS1 | active (7.61%) | - |
LOK | inactive (74.08%) | inactive (57%) |
MINK | active (29.86%) | active (38%) |
MST1 | active (30.92%) | active (10%) |
MST2 | active (40.89%) | active (27%) |
MST3 | inactive (57.7%) | active (37%) |
MST4 | inactive (65.1%) | - |
OSR1 | inactive (94.59%) | - |
PAK1 | inactive (52.1%) | - |
PAK2 | inactive (55.59%) | inactive (62%) |
PAK3 | inactive (97.08%) | inactive (69%) |
PAK4 | inactive (86.36%) | active (13%) |
PAK5 | inactive (60.27%) | active (16%) |
PAK6 | inactive (104.02%) | inactive (55%) |
SLK | inactive (87.23%) | - |
YSK1 | inactive (91.07%) | - |
STLK3 | inactive (96.42%) | - |
TAO1 | inactive (73.12%) | inactive (58%) |
TAO2 | inactive (86.45%) | inactive (64%) |
TAO3 | inactive (66.01%) | inactive (56%) |
MYO3B | active (0%) | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP2K1 | inactive (97.06%) | inactive (114%) |
MAP2K2 | inactive (90.3%) | - |
MAP2K6 | inactive (97.22%) | inactive (86%) |
MAP2K7 | - | inactive (91%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AurA | inactive (78.71%) | inactive (61%) |
AurB | inactive (79.96%) | active (8%) |
AurC | inactive (83.56%) | inactive (63%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMKK1 | inactive (86.67%) | - |
CaMKK2 | inactive (86.84%) | - |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Haspin | inactive (110.25%) | inactive (103%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IKKa | inactive (105.01%) | inactive (99%) |
IKKb | inactive (96.28%) | inactive (92%) |
IKKe | inactive (89.24%) | - |
TBK1 | inactive (83.73%) | active (38%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NEK1 | inactive (131.68%) | - |
NEK11 | inactive (100.52%) | inactive (86%) |
NEK2 | inactive (92.74%) | inactive (99%) |
NEK4 | inactive (103.85%) | - |
NEK6 | inactive (100.57%) | inactive (113%) |
NEK7 | inactive (87.39%) | inactive (112%) |
NEK9 | inactive (102.67%) | - |
NEK3 | inactive (103.67%) | inactive (79%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PBK | inactive (95.36%) | - |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PLK1 | inactive (100.69%) | inactive (86%) |
PLK2 | inactive (99%) | inactive (82%) |
PLK3 | inactive (99.72%) | inactive (100%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SgK496 | inactive (67.09%) | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MPSK1 | inactive (87.02%) | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TTK | inactive (71.66%) | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ULK1 | inactive (94.23%) | - |
ULK2 | inactive (73.09%) | active (47%) |
ULK3 | active (0%) | active (33%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wee1 | inactive (100.26%) | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wnk2 | inactive (112.27%) | inactive (102%) |
Wnk3 | inactive (96.52%) | inactive (101%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TLK2 | active (0%) | inactive (92%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK1 | 7 | 6 | 4 |
VRK | 3 | 1 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK1d | inactive (97.37%) | inactive (84%) |
CK1g1 | inactive (81.6%) | inactive (93%) |
CK1g2 | inactive (84.76%) | inactive (66%) |
CK1g3 | inactive (89.68%) | inactive (102%) |
CK1a | inactive (95.11%) | - |
CK1e | inactive (91.4%) | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
VRK1 | inactive (97.51%) | - |
VRK2 | - | inactive (100%) |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK2 | 3 | 2 | 2 |
CLK | 4 | 4 | 2 |
DYRK | 10 | 9 | 4 |
MAPK | 14 | 10 | 10 |
GSK | 2 | 2 | 2 |
SRPK | 3 | 3 | 3 |
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK2a1 | inactive (91.22%) | inactive (104%) |
CK2a2 | inactive (92.93%) | inactive (107%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CLK1 | inactive (99.55%) | - |
CLK2 | inactive (103.64%) | inactive (94%) |
CLK3 | inactive (107.67%) | inactive (84%) |
CLK4 | inactive (77.09%) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DYRK1A | inactive (85.86%) | - |
DYRK1B | inactive (76.83%) | - |
DYRK2 | active (46.84%) | active (28%) |
DYRK3 | inactive (97.56%) | - |
DYRK4 | inactive (100.14%) | - |
HIPK1 | inactive (97.86%) | inactive (96%) |
HIPK2 | inactive (105.91%) | inactive (64%) |
HIPK3 | inactive (103.64%) | inactive (97%) |
HIPK4 | inactive (112.65%) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Erk1 | inactive (95.05%) | inactive (58%) |
Erk2 | inactive (118.68%) | inactive (87%) |
JNK3 | inactive (93.3%) | inactive (67%) |
NLK | inactive (89.69%) | inactive (82%) |
p38a | inactive (91.82%) | inactive (100%) |
p38b | inactive (101.36%) | inactive (90%) |
p38d | inactive (98.2%) | inactive (89%) |
p38g | inactive (98.93%) | inactive (97%) |
JNK1 | inactive (93.07%) | inactive (112%) |
JNK2 | inactive (97.07%) | inactive (91%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GSK3A | active (0.8%) | active (1%) |
GSK3B | active (2.71%) | active (-3%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSSK1 | inactive (94.63%) | inactive (103%) |
SRPK1 | inactive (106.76%) | inactive (98%) |
SRPK2 | inactive (109.47%) | inactive (103%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
PDHK | 5 | 1 | - |
Alpha | 6 | - | 1 |
PIKK | 6 | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDHK1 | inactive (79.75%) | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
eEF2K | - | inactive (109%) |
Atypical - PIKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FRAP | - | inactive (116%) |