Compound Information
Test on : DRx, RBC, Metz, Millipore
Compound Name
DRx, RBC, Metz, Millipore : PI-103
Inchikey
Same : TUVCWJQQGGETHL-N
DRx, RBC, Metz, Millipore : TUVCWJQQGGETHL-UHFFFAOYSA-N
ChemSpider
DRx, RBC, Metz, Millipore : 8060359
Pubchem CID
DRx, RBC, Metz, Millipore : 9884685
ChEMBL
DRx, RBC, Metz, Millipore : CHEMBL573339
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
Other
Other - NAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
AAK1 | inactive (10001nM) | - | - | - |
BIKE | inactive (10001nM) | - | - | - |
GAK | inactive (10001nM) | - | - | - |
MPSK1 | inactive (10001nM) | inactive (91.72%) | - | - |
Other - Aur
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
AurA | inactive (10001nM) | inactive (91.94%) | - | inactive (104%) |
AurB | inactive (10001nM) | inactive (99.38%) | - | inactive (98%) |
AurC | inactive (10001nM) | inactive (98.13%) | - | inactive (102%) |
Other - CAMKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CaMKK1 | inactive (10001nM) | inactive (84.63%) | - | - |
CaMKK2 | inactive (10001nM) | inactive (79.77%) | - | - |
Other - PEK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
HRI | inactive (10001nM) | - | - | - |
PKR | inactive (10001nM) | - | - | - |
Other - IRE
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
IRE1 | inactive (10001nM) | - | - | - |
Other - IKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
IKKa | active (1700nM) | inactive (94.82%) | - | inactive (108%) |
IKKb | inactive (10001nM) | inactive (98.34%) | - | inactive (113%) |
IKKe | inactive (10001nM) | inactive (98.77%) | - | - |
TBK1 | inactive (10001nM) | inactive (93.03%) | - | inactive (82%) |
Other - NEK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
NEK1 | inactive (10001nM) | inactive (77.83%) | - | - |
NEK11 | inactive (10001nM) | inactive (109.33%) | - | inactive (98%) |
NEK2 | inactive (10001nM) | inactive (88.58%) | - | inactive (83%) |
NEK3 | inactive (10001nM) | inactive (92.89%) | - | inactive (117%) |
NEK4 | inactive (10001nM) | inactive (90.43%) | - | - |
NEK5 | inactive (10001nM) | - | - | - |
NEK6 | inactive (10001nM) | inactive (105.59%) | - | inactive (102%) |
NEK7 | inactive (10001nM) | inactive (97.29%) | - | inactive (100%) |
NEK9 | inactive (10001nM) | inactive (99.3%) | - | - |
Other - WEE
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
MYT1 | inactive (10001nM) | - | - | - |
Wee1 | inactive (10001nM) | inactive (81.62%) | - | - |
Wee1B | inactive (10001nM) | - | - | - |
Other - PLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PLK1 | inactive (10001nM) | inactive (97.88%) | inactive (>7943.28nM) | inactive (102%) |
PLK2 | inactive (10001nM) | inactive (94.72%) | - | inactive (111%) |
PLK3 | inactive (10001nM) | inactive (94.62%) | inactive (>7943.28nM) | inactive (102%) |
PLK4 | inactive (10001nM) | - | - | - |
Other - SgK496
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
SgK496 | inactive (10001nM) | inactive (96.14%) | - | - |
Other - NKF1
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
SBK | inactive (10001nM) | - | - | - |
SgK110 | inactive (10001nM) | - | - | - |
Other - NKF4
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CLIK1 | inactive (10001nM) | - | - | - |
Other - ULK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
Fused | inactive (10001nM) | - | - | - |
ULK1 | inactive (10001nM) | inactive (113.44%) | - | - |
ULK2 | inactive (10001nM) | inactive (105.68%) | - | inactive (108%) |
ULK3 | inactive (10001nM) | inactive (99.68%) | - | inactive (111%) |
Other - TLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
TLK1 | inactive (10001nM) | - | - | - |
TLK2 | inactive (10001nM) | inactive (102.44%) | - | inactive (109%) |
Other - TTK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
TTK | inactive (10001nM) | inactive (93.29%) | - | - |
Other - Haspin
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
Haspin | - | inactive (90.28%) | - | inactive (76%) |
Other - TOPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PBK | - | inactive (88.65%) | inactive (>10000nM) | - |
Other - WNK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
Wnk2 | - | inactive (118.77%) | - | inactive (112%) |
Wnk3 | - | inactive (93.94%) | - | inactive (119%) |
Other - CDC7
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CDC7 | - | - | - | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
ABL1 | inactive (10001nM) | inactive (94.36%) | - | inactive (102%) |
ABL2 | inactive (10001nM) | inactive (94.91%) | - | inactive (99%) |
TK - ALK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
ALK | inactive (10001nM) | inactive (90.45%) | - | inactive (100%) |
LTK | inactive (10001nM) | inactive (97.64%) | - | - |
TK - Axl
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
AXL | inactive (10001nM) | inactive (105.4%) | - | inactive (111%) |
MER | inactive (10001nM) | inactive (87.76%) | - | inactive (110%) |
TYRO3 | inactive (10001nM) | inactive (101.63%) | - | inactive (82%) |
TK - Src
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
BLK | inactive (10001nM) | inactive (101%) | - | inactive (112%) |
BRK | inactive (10001nM) | inactive (80.81%) | - | inactive (113%) |
FGR | inactive (10001nM) | inactive (94.84%) | - | inactive (118%) |
FRK | inactive (10001nM) | inactive (91.34%) | - | inactive (101%) |
FYN | inactive (10001nM) | inactive (91.68%) | - | inactive (82%) |
HCK | inactive (10001nM) | inactive (91.87%) | - | inactive (83%) |
LCK | inactive (10001nM) | inactive (97.99%) | - | inactive (133%) |
LYN | inactive (10001nM) | inactive (101.9%) | - | inactive (99%) |
SRC | inactive (10001nM) | inactive (97.23%) | - | inactive (91%) |
SRM | inactive (10001nM) | inactive (96.19%) | - | - |
YES | inactive (10001nM) | inactive (94.32%) | - | inactive (110%) |
TK - Tec
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
BMX | inactive (10001nM) | inactive (101.04%) | - | inactive (92%) |
BTK | inactive (10001nM) | inactive (95.22%) | - | inactive (101%) |
ITK | inactive (10001nM) | inactive (93.1%) | - | inactive (102%) |
TEC | inactive (10001nM) | inactive (113.23%) | - | - |
TXK | inactive (10001nM) | inactive (94.78%) | - | inactive (93%) |
TK - PDGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
FMS | inactive (10001nM) | inactive (108.04%) | - | inactive (78%) |
FLT3 | active (2500nM) | inactive (87.1%) | - | inactive (89%) |
KIT | inactive (10001nM) | inactive (88.92%) | - | inactive (118%) |
PDGFRa | inactive (10001nM) | inactive (99.39%) | - | inactive (127%) |
PDGFRb | inactive (10001nM) | inactive (99.24%) | - | inactive (112%) |
TK - Csk
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CSK | inactive (10001nM) | inactive (88.32%) | - | inactive (127%) |
CTK | inactive (10001nM) | inactive (86.67%) | - | - |
TK - DDR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
DDR1 | inactive (10001nM) | - | - | - |
DDR2 | inactive (10001nM) | inactive (94.64%) | - | inactive (107%) |
TK - EGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
EGFR | inactive (10001nM) | inactive (83.82%) | - | inactive (119%) |
ErbB2 | inactive (10001nM) | inactive (105.36%) | - | - |
ErbB3 | inactive (10001nM) | - | - | - |
ErbB4 | inactive (10001nM) | inactive (97.65%) | - | inactive (104%) |
TK - Eph
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
EphA1 | inactive (10001nM) | inactive (87.81%) | - | inactive (91%) |
EphA2 | inactive (10001nM) | inactive (99.91%) | - | inactive (113%) |
EphA3 | inactive (10001nM) | inactive (93.69%) | - | inactive (114%) |
EphA4 | inactive (10001nM) | inactive (96.36%) | - | inactive (119%) |
EphA5 | inactive (10001nM) | inactive (101.8%) | - | inactive (98%) |
EphA6 | inactive (10001nM) | inactive (78.99%) | - | - |
EphA7 | inactive (10001nM) | inactive (93.86%) | - | inactive (103%) |
EphA8 | inactive (10001nM) | inactive (93.88%) | - | inactive (107%) |
EphB1 | inactive (10001nM) | inactive (89.58%) | - | inactive (95%) |
EphB2 | inactive (10001nM) | inactive (88.61%) | - | inactive (130%) |
EphB3 | inactive (10001nM) | inactive (92.96%) | - | inactive (116%) |
EphB4 | inactive (10001nM) | inactive (104.49%) | - | inactive (106%) |
EphB6 | inactive (10001nM) | - | - | - |
TK - FAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
FAK | inactive (10001nM) | inactive (93.47%) | - | inactive (144%) |
PYK2 | inactive (10001nM) | inactive (102.84%) | - | inactive (142%) |
TK - Fer
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
FER | inactive (10001nM) | inactive (97.78%) | - | inactive (119%) |
FES | inactive (10001nM) | inactive (98.82%) | - | inactive (137%) |
TK - FGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
FGFR1 | inactive (10001nM) | inactive (91.72%) | - | inactive (97%) |
FGFR2 | inactive (10001nM) | inactive (95.75%) | - | inactive (122%) |
FGFR3 | inactive (10001nM) | inactive (100.59%) | - | inactive (112%) |
FGFR4 | inactive (10001nM) | inactive (101.99%) | - | inactive (112%) |
TK - VEGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
FLT1 | inactive (10001nM) | inactive (83.59%) | - | inactive (91%) |
FLT4 | inactive (10001nM) | inactive (104.05%) | - | inactive (79%) |
KDR | inactive (10001nM) | inactive (85.89%) | - | inactive (109%) |
TK - InsR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
IGF1R | inactive (10001nM) | inactive (97.13%) | - | inactive (131%) |
INSR | inactive (10001nM) | inactive (98.59%) | - | inactive (98%) |
IRR | inactive (10001nM) | inactive (113.55%) | - | inactive (128%) |
TK - JakA
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
JAK1 | inactive (10001nM) | inactive (103.69%) | - | - |
JAK2 | inactive (10001nM) | inactive (92.6%) | - | inactive (107%) |
JAK3 | inactive (10001nM) | inactive (99%) | - | inactive (103%) |
TYK2 | inactive (10001nM) | inactive (73.63%) | - | - |
TK - Met
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
MET | inactive (10001nM) | inactive (97.79%) | - | inactive (121%) |
RON | inactive (10001nM) | inactive (94.31%) | - | inactive (102%) |
TK - Musk
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
MUSK | inactive (10001nM) | inactive (87.81%) | - | inactive (114%) |
TK - Ret
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
RET | inactive (10001nM) | inactive (99.79%) | - | inactive (101%) |
TK - Sev
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
ROS | inactive (10001nM) | inactive (93.13%) | - | inactive (96%) |
TK - Syk
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
SYK | inactive (10001nM) | inactive (94.15%) | - | inactive (131%) |
ZAP70 | inactive (10001nM) | inactive (91.43%) | - | inactive (110%) |
TK - Tie
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
TIE1 | inactive (10001nM) | - | - | - |
TIE2 | inactive (10001nM) | inactive (87.7%) | - | inactive (80%) |
TK - Ack
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
TNK1 | inactive (10001nM) | - | - | - |
ACK | inactive (10001nM) | inactive (89.56%) | - | inactive (78%) |
TK - Trk
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
TRKA | inactive (10001nM) | inactive (94.95%) | - | inactive (93%) |
TRKB | inactive (10001nM) | inactive (90.16%) | - | inactive (113%) |
TRKC | inactive (10001nM) | inactive (91.1%) | - | - |
TKL
TKL
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz | Millipore |
---|
STKR | 12 | 10 | 5 | 1 | 2 |
RIPK | 5 | 4 | 1 | - | 1 |
RAF | 5 | 2 | 3 | 1 | 1 |
MLK | 10 | 8 | 5 | 2 | 2 |
IRAK | 4 | 3 | 2 | 2 | 2 |
LISK | 4 | 3 | 1 | 1 | 1 |
LRRK | 2 | 1 | 1 | 1 | - |
TKL - STKR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
ALK2 | inactive (10001nM) | inactive (104.87%) | - | - |
ALK4 | inactive (10001nM) | inactive (98.03%) | - | inactive (148%) |
ACTR2 | inactive (10001nM) | - | - | - |
ACTR2B | inactive (10001nM) | - | - | - |
ALK1 | inactive (10001nM) | inactive (105.37%) | - | - |
BMPR1A | inactive (10001nM) | - | - | - |
BMPR1B | inactive (10001nM) | - | - | - |
BMPR2 | inactive (10001nM) | - | - | - |
TGFbR1 | inactive (10001nM) | inactive (94.96%) | - | inactive (82%) |
TGFbR2 | inactive (10001nM) | inactive (101.62%) | - | - |
TKL - RIPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
SgK288 | inactive (10001nM) | - | - | - |
RIPK1 | inactive (10001nM) | - | - | - |
RIPK2 | inactive (10001nM) | inactive (87.41%) | - | inactive (89%) |
ANKRD3 | inactive (10001nM) | - | - | - |
TKL - RAF
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
BRAF | active (2900nM) | inactive (94%) | - | - |
RAF1 | inactive (3700nM) | inactive (79.1%) | - | inactive (81%) |
ARAF | - | inactive (92.04%) | - | - |
TKL - MLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
DLK | inactive (10001nM) | - | - | - |
LZK | inactive (10001nM) | - | - | - |
MLK1 | inactive (10001nM) | inactive (103.36%) | - | inactive (90%) |
MLK2 | inactive (10001nM) | inactive (91.96%) | - | - |
MLK3 | inactive (10001nM) | inactive (96.53%) | - | - |
TAK1 | inactive (10001nM) | inactive (97.36%) | - | inactive (99%) |
HH498 | inactive (10001nM) | - | - | - |
ZAK | inactive (10001nM) | inactive (96.18%) | inactive (>7943.28nM) | - |
TKL - IRAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
IRAK1 | inactive (10001nM) | inactive (84.2%) | inactive (>7943.28nM) | inactive (101%) |
IRAK3 | inactive (10001nM) | - | - | - |
IRAK4 | inactive (10001nM) | inactive (104.48%) | inactive (>10000nM) | inactive (99%) |
TKL - LISK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
LIMK1 | inactive (10001nM) | inactive (93.7%) | - | inactive (113%) |
LIMK2 | inactive (3500nM) | - | - | - |
TESK1 | inactive (10001nM) | - | - | - |
TKL - LRRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
LRRK2 | inactive (10001nM) | inactive (100.52%) | - | - |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz | Millipore |
---|
ABC1 | 5 | 2 | - | - | - |
PIKK | 6 | 1 | - | - | 1 |
RIO | 3 | 3 | - | - | - |
Alpha | 6 | 1 | - | 1 | 1 |
PDHK | 5 | - | 1 | - | - |
Atypical - ABC1
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
ADCK3 | inactive (10001nM) | - | - | - |
ADCK4 | inactive (10001nM) | - | - | - |
Atypical - PIKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
FRAP | active (12nM) | - | - | active (49%) |
Atypical - RIO
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
RIOK1 | inactive (10001nM) | - | - | - |
RIOK2 | active (770nM) | - | - | - |
RIOK3 | inactive (10001nM) | - | - | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
ChaK2 | inactive (10001nM) | - | - | - |
eEF2K | - | - | - | inactive (102%) |
Atypical - PDHK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PDHK1 | - | inactive (102.92%) | - | - |
AGC
AGC - Akt
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
AKT1 | inactive (10001nM) | inactive (95.26%) | inactive (>7943.28nM) | inactive (104%) |
AKT2 | inactive (10001nM) | inactive (99.13%) | inactive (>7943.28nM) | inactive (130%) |
AKT3 | inactive (10001nM) | inactive (99.03%) | inactive (>10000nM) | inactive (95%) |
AGC - DMPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CRIK | inactive (10001nM) | - | - | - |
DMPK1 | inactive (10001nM) | inactive (99.51%) | - | inactive (101%) |
DMPK2 | inactive (10001nM) | - | - | - |
MRCKa | active (1800nM) | inactive (94.5%) | inactive (>10000nM) | inactive (97%) |
MRCKb | inactive (10001nM) | inactive (99.36%) | - | inactive (91%) |
ROCK1 | inactive (10001nM) | inactive (94.9%) | - | inactive (123%) |
ROCK2 | inactive (10001nM) | inactive (94.5%) | - | inactive (103%) |
AGC - GRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
RHOK | inactive (10001nM) | - | - | - |
GPRK4 | inactive (10001nM) | inactive (101.95%) | - | - |
GPRK7 | inactive (10001nM) | inactive (99.98%) | - | inactive (93%) |
BARK1 | - | inactive (107.47%) | - | - |
BARK2 | - | inactive (109.79%) | - | - |
GPRK5 | - | inactive (103.5%) | - | inactive (104%) |
GPRK6 | - | inactive (98.15%) | - | inactive (103%) |
AGC - NDR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
LATS1 | inactive (10001nM) | - | - | - |
LATS2 | inactive (10001nM) | - | - | - |
NDR1 | inactive (10001nM) | inactive (98.99%) | - | - |
NDR2 | inactive (10001nM) | - | - | - |
AGC - MAST
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
MAST1 | inactive (10001nM) | - | - | - |
AGC - PDK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PDK1 | inactive (10001nM) | inactive (102.92%) | - | inactive (116%) |
AGC - PKA
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PKACa | inactive (10001nM) | inactive (99.53%) | - | inactive (95%) |
PKACb | inactive (10001nM) | - | - | - |
PRKX | inactive (10001nM) | inactive (96.15%) | - | inactive (96%) |
PKACg | - | inactive (101.32%) | - | - |
AGC - PKN
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PKN1 | inactive (10001nM) | inactive (101.14%) | - | - |
PKN2 | inactive (10001nM) | inactive (87.56%) | - | inactive (101%) |
AGC - PKC
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PKCd | inactive (10001nM) | inactive (95.95%) | inactive (>7943.28nM) | inactive (94%) |
PKCe | inactive (10001nM) | inactive (100.44%) | - | inactive (91%) |
PKCh | inactive (10001nM) | inactive (89.75%) | - | inactive (107%) |
PKCi | inactive (10001nM) | inactive (94.9%) | - | inactive (89%) |
PKCt | inactive (10001nM) | inactive (104.89%) | - | inactive (84%) |
PKCa | - | inactive (102.91%) | - | inactive (106%) |
PKCg | - | inactive (101.72%) | inactive (>7943.28nM) | inactive (114%) |
PKCz | - | inactive (99.07%) | inactive (>7943.28nM) | inactive (104%) |
PKCb | - | inactive (102.48%) | - | - |
AGC - PKG
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PKG1 | inactive (10001nM) | inactive (96.3%) | - | - |
PKG2 | inactive (10001nM) | inactive (89.24%) | - | - |
AGC - RSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
p70S6K | inactive (10001nM) | inactive (105.51%) | - | inactive (68%) |
MSK1 | - | inactive (86.47%) | - | inactive (130%) |
MSK2 | - | inactive (104.45%) | - | inactive (98%) |
p70S6Kb | - | inactive (95.79%) | - | - |
RSK2 | - | inactive (101.09%) | - | inactive (70%) |
RSK4 | - | inactive (98.2%) | - | inactive (115%) |
RSK1 | - | inactive (79.48%) | - | inactive (108%) |
RSK3 | - | inactive (88.09%) | - | inactive (141%) |
AGC - SGK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
SGK3 | inactive (10001nM) | inactive (95.79%) | - | inactive (102%) |
SGK1 | - | inactive (100.35%) | inactive (>7943.28nM) | inactive (105%) |
SGK2 | - | inactive (96.68%) | - | inactive (112%) |
AGC - YANK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
YANK1 | inactive (10001nM) | - | - | - |
YANK2 | inactive (10001nM) | - | - | - |
YANK3 | inactive (10001nM) | - | - | - |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
AMPKa1 | inactive (10001nM) | - | - | inactive (114%) |
AMPKa2 | inactive (10001nM) | - | - | inactive (113%) |
NuaK1 | inactive (10001nM) | inactive (86.63%) | - | inactive (98%) |
BRSK1 | inactive (10001nM) | inactive (91.08%) | inactive (>10000nM) | inactive (95%) |
BRSK2 | inactive (10001nM) | inactive (97.12%) | - | inactive (96%) |
CHK1 | inactive (10001nM) | inactive (93.96%) | - | inactive (93%) |
HUNK | inactive (10001nM) | - | - | - |
LKB1 | inactive (10001nM) | inactive (86.38%) | - | inactive (104%) |
MARK1 | inactive (10001nM) | inactive (97.63%) | - | inactive (104%) |
MARK2 | inactive (10001nM) | inactive (92.94%) | inactive (>7943.28nM) | inactive (91%) |
MARK3 | inactive (10001nM) | inactive (97.41%) | - | - |
MARK4 | inactive (10001nM) | inactive (93.36%) | - | - |
MELK | inactive (10001nM) | inactive (75.49%) | - | inactive (74%) |
NIM1 | inactive (10001nM) | - | - | - |
QSK | inactive (10001nM) | - | - | - |
SIK | inactive (10001nM) | - | - | inactive (91%) |
QIK | inactive (10001nM) | inactive (98.95%) | - | - |
NuaK2 | inactive (10001nM) | inactive (75.29%) | - | - |
SNRK | inactive (10001nM) | - | - | - |
PASK | - | inactive (83.82%) | - | inactive (107%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CaMK1a | inactive (10001nM) | inactive (100.64%) | - | inactive (103%) |
CaMK1d | inactive (10001nM) | inactive (120.58%) | - | inactive (102%) |
CaMK1g | inactive (10001nM) | inactive (99.24%) | - | - |
CaMK4 | inactive (10001nM) | inactive (103.33%) | - | inactive (108%) |
CaMK1b | - | inactive (96.67%) | - | - |
CAMK - CAMK2
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CaMK2a | inactive (10001nM) | inactive (93.74%) | - | - |
CaMK2b | inactive (10001nM) | inactive (98.24%) | inactive (>7943.28nM) | inactive (98%) |
CaMK2d | inactive (10001nM) | inactive (96.18%) | - | inactive (104%) |
CaMK2g | inactive (10001nM) | inactive (100.02%) | - | inactive (98%) |
CAMK - CASK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CASK | inactive (10001nM) | - | - | - |
CAMK - RAD53
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CHK2 | inactive (10001nM) | inactive (90.42%) | - | inactive (100%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
DAPK1 | active (2400nM) | inactive (77.96%) | - | inactive (99%) |
DAPK2 | active (2700nM) | inactive (116.67%) | - | inactive (93%) |
DAPK3 | active (840nM) | inactive (93.13%) | active (794.33nM) | inactive (85%) |
DRAK1 | inactive (10001nM) | inactive (93.79%) | - | inactive (116%) |
DRAK2 | inactive (10001nM) | - | - | - |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
DCLK1 | inactive (10001nM) | - | inactive (>10000nM) | - |
DCLK2 | inactive (10001nM) | inactive (101.53%) | - | inactive (94%) |
DCLK3 | inactive (10001nM) | - | - | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
MAPKAPK2 | inactive (10001nM) | inactive (97.81%) | inactive (>7943.28nM) | inactive (81%) |
MAPKAPK5 | inactive (10001nM) | inactive (85.66%) | - | inactive (98%) |
MNK1 | inactive (10001nM) | inactive (102.44%) | - | - |
MNK2 | inactive (10001nM) | inactive (92.6%) | inactive (>10000nM) | inactive (109%) |
MAPKAPK3 | - | inactive (93.92%) | inactive (>10000nM) | inactive (92%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
caMLCK | inactive (10001nM) | - | - | - |
smMLCK | active (1500nM) | inactive (77.15%) | - | inactive (71%) |
skMLCK | inactive (10001nM) | inactive (98.98%) | - | - |
SgK085 | inactive (10001nM) | - | - | - |
CAMK - PHK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PHKg1 | inactive (10001nM) | inactive (93.34%) | - | - |
PHKg2 | inactive (10001nM) | inactive (99.1%) | - | inactive (105%) |
CAMK - PIM
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PIM1 | inactive (10001nM) | inactive (91.23%) | - | inactive (88%) |
PIM2 | inactive (10001nM) | inactive (96.93%) | - | inactive (102%) |
PIM3 | inactive (10001nM) | inactive (104.04%) | inactive (5011.87nM) | inactive (98%) |
CAMK - PKD
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PKD1 | inactive (10001nM) | inactive (98.33%) | - | inactive (97%) |
PKD2 | inactive (10001nM) | inactive (93.83%) | inactive (>10000nM) | inactive (99%) |
PKD3 | inactive (10001nM) | inactive (92.93%) | - | - |
CAMK - STK33
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
STK33 | inactive (10001nM) | inactive (101.23%) | - | inactive (101%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
TSSK1 | inactive (10001nM) | inactive (93.39%) | - | inactive (104%) |
TSSK2 | - | inactive (101.57%) | - | inactive (93%) |
STE
STE
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz | Millipore |
---|
STE11 | 8 | 8 | 3 | - | 1 |
STE20 | 31 | 27 | 23 | 9 | 14 |
STE7 | 7 | 7 | 3 | 2 | 3 |
STE-Unique | 2 | - | 2 | - | - |
STE - STE11
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
MAP3K5 | inactive (10001nM) | inactive (101.41%) | - | inactive (109%) |
MAP3K6 | inactive (10001nM) | - | - | - |
MAP3K1 | inactive (10001nM) | - | - | - |
MAP3K7 | inactive (10001nM) | - | - | - |
MAP3K2 | inactive (10001nM) | inactive (103.2%) | - | - |
MAP3K3 | inactive (10001nM) | inactive (96.04%) | - | - |
MAP3K4 | inactive (10001nM) | - | - | - |
MAP3K8 | active (930nM) | - | - | - |
STE - STE20
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
HPK1 | inactive (10001nM) | - | - | - |
LOK | inactive (10001nM) | inactive (92.13%) | - | inactive (96%) |
GCK | inactive (10001nM) | inactive (93.01%) | - | inactive (101%) |
KHS2 | inactive (10001nM) | - | - | - |
HGK | inactive (10001nM) | inactive (91.37%) | - | - |
KHS1 | inactive (10001nM) | inactive (82.41%) | - | - |
MINK | inactive (10001nM) | inactive (96%) | inactive (>7943.28nM) | inactive (110%) |
MST1 | inactive (10001nM) | inactive (93.34%) | - | inactive (97%) |
MST2 | inactive (10001nM) | inactive (105.2%) | - | inactive (120%) |
MST3 | inactive (10001nM) | inactive (100.02%) | - | inactive (75%) |
MST4 | inactive (10001nM) | inactive (98.65%) | - | - |
MYO3A | inactive (10001nM) | - | - | - |
MYO3B | inactive (10001nM) | inactive (81.27%) | - | - |
OSR1 | inactive (10001nM) | inactive (93.23%) | - | - |
PAK1 | inactive (10001nM) | inactive (97.59%) | inactive (>10000nM) | - |
PAK2 | inactive (10001nM) | inactive (97.49%) | - | inactive (105%) |
PAK3 | inactive (10001nM) | inactive (97.51%) | - | inactive (60%) |
PAK4 | inactive (10001nM) | inactive (90.69%) | - | inactive (100%) |
PAK6 | inactive (10001nM) | inactive (104.61%) | - | inactive (100%) |
PAK5 | inactive (10001nM) | inactive (92.83%) | - | inactive (84%) |
SLK | inactive (10001nM) | inactive (101.43%) | inactive (>10000nM) | - |
STLK3 | inactive (10001nM) | inactive (104.72%) | - | - |
TAO1 | inactive (10001nM) | inactive (91.57%) | - | inactive (93%) |
TAO2 | inactive (10001nM) | inactive (92.21%) | - | inactive (104%) |
TAO3 | inactive (10001nM) | inactive (86.75%) | - | inactive (109%) |
TNIK | inactive (10001nM) | - | - | - |
YSK1 | inactive (10001nM) | inactive (93.39%) | - | - |
STE - STE7
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
MAP2K1 | inactive (10001nM) | inactive (97.66%) | - | inactive (102%) |
MAP2K2 | inactive (10001nM) | inactive (85.03%) | - | - |
MAP2K3 | inactive (10001nM) | - | - | - |
MAP2K4 | inactive (10001nM) | - | - | - |
MAP2K5 | inactive (10001nM) | - | - | - |
MAP2K6 | inactive (10001nM) | inactive (86.57%) | - | inactive (91%) |
MAP2K7 | inactive (10001nM) | - | - | inactive (101%) |
STE - STE-Unique
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
COT | - | inactive (99.19%) | - | - |
NIK | - | - | - | - |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz | Millipore |
---|
CDK | 20 | 8 | - | 7 | - |
CDKL | 5 | 4 | - | - | - |
CLK | 4 | 4 | 4 | 2 | 2 |
CK2 | 3 | 2 | 2 | 1 | 2 |
DYRK | 10 | 8 | 9 | 6 | 4 |
MAPK | 14 | 14 | 10 | 8 | 10 |
GSK | 2 | 2 | 2 | 2 | 2 |
RCK | 3 | 2 | - | - | - |
SRPK | 3 | 3 | 3 | 1 | 3 |
CMGC - CDK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PITSLRE | inactive (10001nM) | - | - | - |
CHED | inactive (10001nM) | - | - | - |
CDK11 | inactive (10001nM) | - | - | - |
PCTAIRE1 | inactive (10001nM) | - | - | - |
PCTAIRE2 | inactive (10001nM) | - | - | - |
PCTAIRE3 | inactive (10001nM) | - | - | - |
PFTAIRE2 | inactive (10001nM) | - | - | - |
PFTAIRE1 | inactive (10001nM) | - | - | - |
CDC2 | - | - | inactive (>7943.28nM) | - |
CDK2 | - | - | inactive (>7943.28nM) | - |
CDK5 | - | - | - | - |
CDK8 | - | - | - | - |
CDK7 | - | - | - | - |
CDK9 | - | - | - | - |
CMGC - CDKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CDKL1 | inactive (10001nM) | - | - | - |
CDKL2 | inactive (10001nM) | - | - | - |
CDKL3 | inactive (10001nM) | - | - | - |
CDKL5 | inactive (10001nM) | - | - | - |
CMGC - CLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CLK1 | inactive (3900nM) | inactive (85.18%) | - | - |
CLK2 | inactive (5500nM) | inactive (87.96%) | - | inactive (118%) |
CLK3 | inactive (5900nM) | inactive (93.1%) | - | inactive (79%) |
CLK4 | inactive (10001nM) | inactive (81.51%) | active (794.33nM) | - |
CMGC - CK2
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CK2a1 | inactive (5400nM) | inactive (94.66%) | - | inactive (89%) |
CK2a2 | active (2900nM) | inactive (56.22%) | - | inactive (140%) |
CMGC - DYRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
DYRK1A | inactive (10001nM) | inactive (94.31%) | - | - |
DYRK1B | inactive (5700nM) | inactive (98.91%) | - | - |
DYRK2 | inactive (4100nM) | inactive (97.64%) | - | inactive (94%) |
HIPK1 | inactive (3300nM) | inactive (101.2%) | - | inactive (85%) |
HIPK2 | active (290nM) | inactive (102.05%) | inactive (2511.89nM) | inactive (84%) |
HIPK3 | active (310nM) | inactive (93.82%) | - | inactive (93%) |
HIPK4 | inactive (10001nM) | inactive (106.74%) | inactive (>7943.28nM) | - |
PRP4 | inactive (10001nM) | - | - | - |
DYRK3 | - | inactive (94.86%) | - | - |
DYRK4 | - | inactive (96.63%) | - | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
Erk1 | inactive (10001nM) | inactive (94.12%) | - | inactive (83%) |
Erk2 | inactive (10001nM) | inactive (88.98%) | - | inactive (122%) |
Erk3 | inactive (10001nM) | - | - | - |
Erk4 | inactive (10001nM) | - | - | - |
Erk5 | inactive (10001nM) | - | - | - |
Erk7 | inactive (10001nM) | - | - | - |
JNK1 | inactive (10001nM) | inactive (89.83%) | - | inactive (109%) |
JNK2 | inactive (10001nM) | inactive (89.43%) | - | inactive (107%) |
JNK3 | inactive (10001nM) | inactive (101.88%) | - | inactive (91%) |
NLK | inactive (10001nM) | inactive (97.37%) | - | inactive (102%) |
p38a | inactive (10001nM) | inactive (101.07%) | - | inactive (109%) |
p38b | inactive (10001nM) | inactive (102.62%) | - | inactive (102%) |
p38d | inactive (10001nM) | inactive (97.41%) | inactive (>7943.28nM) | inactive (106%) |
p38g | inactive (10001nM) | inactive (93.4%) | - | inactive (112%) |
CMGC - GSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
GSK3A | inactive (10001nM) | inactive (90.21%) | - | inactive (111%) |
GSK3B | inactive (10001nM) | inactive (94.8%) | - | inactive (101%) |
CMGC - RCK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
ICK | inactive (10001nM) | - | - | - |
MAK | inactive (10001nM) | - | - | - |
CMGC - SRPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
SRPK1 | inactive (10001nM) | inactive (104.96%) | inactive (>7943.28nM) | inactive (97%) |
SRPK2 | inactive (10001nM) | inactive (97.31%) | - | inactive (103%) |
MSSK1 | inactive (10001nM) | inactive (95.04%) | - | inactive (110%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz | Millipore |
---|
CK1 | 7 | 7 | 6 | 5 | 4 |
VRK | 3 | 1 | 1 | - | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CK1a | inactive (10001nM) | inactive (87.88%) | - | - |
CK1a2 | inactive (10001nM) | - | - | - |
CK1d | inactive (10001nM) | inactive (91.33%) | inactive (>7943.28nM) | inactive (83%) |
CK1e | inactive (10001nM) | inactive (87.09%) | - | - |
CK1g1 | inactive (10001nM) | inactive (89.41%) | - | inactive (90%) |
CK1g2 | inactive (10001nM) | inactive (88.13%) | - | inactive (108%) |
CK1g3 | inactive (10001nM) | inactive (99.94%) | - | inactive (115%) |
CK1 - VRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
VRK2 | inactive (10001nM) | - | - | inactive (111%) |
VRK1 | - | inactive (98.35%) | - | - |