Compound Information
Test on : RBC
Compound Name : -
Inchikey : RKUMZEVCWKZXFV-YOCZKUTFSA-N
ChemSpider : 25057868
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC |
---|
PDK1 | inactive (83.33%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC |
---|
AKT1 | inactive (95.55%) |
AKT2 | inactive (90.1%) |
AKT3 | inactive (92.95%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC |
---|
DMPK1 | inactive (99.47%) |
MRCKa | inactive (88.59%) |
MRCKb | inactive (96.58%) |
ROCK1 | inactive (100.82%) |
ROCK2 | inactive (90.96%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC |
---|
BARK1 | inactive (100.55%) |
BARK2 | inactive (99.98%) |
GPRK4 | inactive (74.71%) |
GPRK5 | inactive (84.64%) |
GPRK6 | inactive (53.06%) |
GPRK7 | inactive (70.25%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC |
---|
MSK1 | active (37.45%) |
MSK2 | active (21.7%) |
p70S6K | active (47.82%) |
p70S6Kb | inactive (105.58%) |
RSK2 | active (18.29%) |
RSK4 | active (16.4%) |
RSK1 | active (8.85%) |
RSK3 | active (12.14%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC |
---|
PKACg | - |
PRKX | inactive (84.17%) |
PKACa | inactive (89.06%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC |
---|
PKCa | inactive (100.93%) |
PKCd | inactive (80.59%) |
PKCe | inactive (92.21%) |
PKCh | inactive (82.16%) |
PKCg | inactive (92.04%) |
PKCi | inactive (100.22%) |
PKCt | inactive (92.9%) |
PKCz | inactive (98.49%) |
PKCb | inactive (87.98%) |
AGC - PKG
Bioactivity |
---|
Kinase | RBC |
---|
PKG2 | active (28.07%) |
PKG1 | active (45.15%) |
AGC - PKN
Bioactivity |
---|
Kinase | RBC |
---|
PKN1 | active (49.9%) |
PKN2 | inactive (90.06%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC |
---|
SGK1 | inactive (51.04%) |
SGK2 | inactive (75.85%) |
SGK3 | inactive (100.24%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC |
---|
NDR1 | active (0%) |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC |
---|
ABL1 | inactive (71.92%) |
ABL2 | active (38.52%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC |
---|
ACK | active (4.93%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC |
---|
ALK | active (38.1%) |
LTK | active (34.75%) |
TK - Axl
Bioactivity |
---|
Kinase | RBC |
---|
AXL | active (42.68%) |
MER | active (49.36%) |
TYRO3 | inactive (71.52%) |
TK - Src
Bioactivity |
---|
Kinase | RBC |
---|
BLK | active (39.06%) |
BRK | inactive (73.29%) |
SRC | active (22.59%) |
FGR | active (11.63%) |
FRK | active (49.68%) |
FYN | active (12.97%) |
HCK | active (23.02%) |
LCK | active (29.71%) |
SRM | inactive (101.81%) |
YES | active (13.38%) |
LYN | active (25.41%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC |
---|
BMX | active (40.23%) |
BTK | active (24.08%) |
ITK | active (34.8%) |
TEC | inactive (101.13%) |
TXK | active (25.57%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC |
---|
KIT | active (44.84%) |
FLT3 | active (1.07%) |
FMS | active (21.14%) |
PDGFRb | active (42.84%) |
PDGFRa | inactive (76.67%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC |
---|
CSK | inactive (86.27%) |
CTK | inactive (100.86%) |
TK - DDR
Bioactivity |
---|
Kinase | RBC |
---|
DDR2 | inactive (86.1%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC |
---|
EGFR | inactive (88.11%) |
ErbB2 | inactive (95.25%) |
ErbB4 | inactive (97.48%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC |
---|
EphA1 | inactive (82.25%) |
EphA2 | inactive (65.31%) |
EphA3 | inactive (69.01%) |
EphA4 | inactive (77.94%) |
EphA5 | inactive (67.97%) |
EphA6 | - |
EphA7 | inactive (71.45%) |
EphA8 | inactive (91.92%) |
EphB1 | inactive (65.89%) |
EphB2 | inactive (74.98%) |
EphB3 | - |
EphB4 | inactive (72.17%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC |
---|
FAK | active (34.96%) |
PYK2 | active (30.5%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC |
---|
FER | active (28.78%) |
FES | inactive (81.66%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC |
---|
FGFR1 | active (27.88%) |
FGFR2 | inactive (75.97%) |
FGFR3 | active (45.83%) |
FGFR4 | inactive (65.67%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC |
---|
FLT1 | inactive (51.03%) |
FLT4 | active (22.26%) |
KDR | inactive (56.4%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC |
---|
IGF1R | active (39.12%) |
IRR | active (2.77%) |
INSR | active (44.92%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC |
---|
JAK1 | active (25.86%) |
JAK2 | active (43.1%) |
JAK3 | active (16.93%) |
TYK2 | active (9.42%) |
TK - Musk
Bioactivity |
---|
Kinase | RBC |
---|
MUSK | inactive (58.02%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC |
---|
RET | active (1.22%) |
TK - Met
Bioactivity |
---|
Kinase | RBC |
---|
RON | inactive (100.7%) |
MET | inactive (122.95%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC |
---|
ROS | active (26.97%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC |
---|
SYK | active (38.56%) |
ZAP70 | inactive (97.76%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC |
---|
TIE2 | inactive (100.82%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC |
---|
TRKA | active (3.84%) |
TRKB | active (1.62%) |
TRKC | active (1.01%) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC |
---|
ALK1 | inactive (102.55%) |
ALK2 | inactive (199.37%) |
ALK4 | inactive (110.43%) |
TGFbR1 | inactive (102.36%) |
TGFbR2 | inactive (118.64%) |
TKL - RAF
Bioactivity |
---|
Kinase | RBC |
---|
ARAF | inactive (106.61%) |
BRAF | inactive (102.98%) |
RAF1 | inactive (100.28%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC |
---|
IRAK1 | active (34.48%) |
IRAK4 | inactive (60.26%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC |
---|
LIMK1 | active (39.53%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC |
---|
LRRK2 | inactive (81.2%) |
TKL - MLK
Bioactivity |
---|
Kinase | RBC |
---|
MLK1 | active (7.06%) |
MLK2 | inactive (86.88%) |
MLK3 | active (10.48%) |
TAK1 | inactive (50.49%) |
ZAK | inactive (76.37%) |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC |
---|
RIPK2 | inactive (62.75%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC |
---|
NuaK1 | active (2.81%) |
BRSK1 | active (39.54%) |
BRSK2 | active (33.35%) |
CHK1 | inactive (67.03%) |
LKB1 | active (5.77%) |
MARK1 | inactive (60.54%) |
MARK3 | inactive (75.23%) |
MARK4 | active (43.52%) |
MELK | active (13.12%) |
PASK | inactive (89.79%) |
QIK | inactive (75.06%) |
NuaK2 | inactive (55.11%) |
MARK2 | inactive (57.43%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC |
---|
CaMK1a | inactive (75.96%) |
CaMK1b | inactive (101.37%) |
CaMK1d | inactive (80.35%) |
CaMK1g | inactive (101.8%) |
CaMK4 | inactive (93.58%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC |
---|
CaMK2a | active (12.24%) |
CaMK2b | inactive (57.86%) |
CaMK2d | active (29.13%) |
CaMK2g | active (35.32%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC |
---|
CHK2 | active (26.95%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC |
---|
DAPK1 | inactive (80.9%) |
DAPK2 | inactive (103.69%) |
DRAK1 | active (22.48%) |
DAPK3 | inactive (66.55%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC |
---|
DCLK2 | inactive (86.36%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC |
---|
MAPKAPK2 | inactive (98.37%) |
MAPKAPK3 | inactive (98.86%) |
MAPKAPK5 | inactive (86.77%) |
MNK1 | inactive (95.32%) |
MNK2 | inactive (72.37%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC |
---|
smMLCK | active (32.26%) |
skMLCK | active (27.32%) |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC |
---|
PHKg1 | active (8.06%) |
PHKg2 | active (34.88%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC |
---|
PIM1 | inactive (59.73%) |
PIM2 | inactive (99.48%) |
PIM3 | inactive (58.5%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC |
---|
PKD1 | inactive (72.65%) |
PKD3 | inactive (68.14%) |
PKD2 | inactive (74.26%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC |
---|
TSSK1 | inactive (76.62%) |
TSSK2 | inactive (96.16%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC |
---|
STK33 | active (22.3%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC |
---|
MAP3K5 | inactive (91.16%) |
MAP3K2 | inactive (60.65%) |
MAP3K3 | inactive (87.79%) |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC |
---|
COT | inactive (123.2%) |
NIK | inactive (88.98%) |
STE - STE20
Bioactivity |
---|
Kinase | RBC |
---|
GCK | inactive (51.72%) |
HGK | active (11.58%) |
KHS1 | active (15.46%) |
LOK | inactive (52.09%) |
MINK | active (20.99%) |
MST1 | active (8.29%) |
MST2 | active (4.81%) |
MST3 | inactive (51.86%) |
MST4 | inactive (73.1%) |
OSR1 | inactive (98.58%) |
PAK1 | inactive (71.31%) |
PAK2 | inactive (82.06%) |
PAK3 | inactive (73.84%) |
PAK4 | inactive (84.48%) |
PAK5 | inactive (81%) |
PAK6 | inactive (93.5%) |
SLK | inactive (59.86%) |
YSK1 | inactive (73.98%) |
STLK3 | inactive (79.25%) |
TAO1 | inactive (98.17%) |
TAO2 | inactive (83.38%) |
TAO3 | inactive (55.38%) |
MYO3B | active (0%) |
STE - STE7
Bioactivity |
---|
Kinase | RBC |
---|
MAP2K1 | inactive (99.66%) |
MAP2K2 | inactive (86.53%) |
MAP2K6 | inactive (79.66%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC |
---|
AurA | active (9.78%) |
AurB | active (27.36%) |
AurC | active (43.19%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC |
---|
CaMKK1 | active (26.18%) |
CaMKK2 | active (25.96%) |
Other - Haspin
Bioactivity |
---|
Kinase | RBC |
---|
Haspin | active (32.81%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC |
---|
IKKa | inactive (96.62%) |
IKKb | inactive (90.54%) |
IKKe | active (45.67%) |
TBK1 | active (29.85%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC |
---|
NEK1 | inactive (92.85%) |
NEK11 | inactive (92.25%) |
NEK2 | inactive (113.62%) |
NEK4 | inactive (83.94%) |
NEK6 | inactive (96.26%) |
NEK7 | inactive (98.88%) |
NEK9 | inactive (73.61%) |
NEK3 | inactive (101.91%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC |
---|
PBK | inactive (80.58%) |
Other - PLK
Bioactivity |
---|
Kinase | RBC |
---|
PLK1 | inactive (103.16%) |
PLK2 | inactive (104.75%) |
PLK3 | inactive (102.29%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC |
---|
SgK496 | inactive (104.37%) |
Other - NAK
Bioactivity |
---|
Kinase | RBC |
---|
MPSK1 | active (12.72%) |
Other - TTK
Bioactivity |
---|
Kinase | RBC |
---|
TTK | active (46.11%) |
Other - ULK
Bioactivity |
---|
Kinase | RBC |
---|
ULK1 | inactive (98.35%) |
ULK2 | inactive (102.32%) |
ULK3 | active (0%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC |
---|
Wee1 | inactive (82.04%) |
Other - WNK
Bioactivity |
---|
Kinase | RBC |
---|
Wnk2 | inactive (85.35%) |
Wnk3 | inactive (79.7%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC |
---|
TLK2 | active (0%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
CK1 | 7 | 6 |
VRK | 3 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC |
---|
CK1d | inactive (52.93%) |
CK1g1 | inactive (89.22%) |
CK1g2 | inactive (85.19%) |
CK1g3 | inactive (90.69%) |
CK1a | inactive (84.83%) |
CK1e | active (43.16%) |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC |
---|
VRK1 | inactive (88.35%) |
CMGC
CMGC - CK2
Bioactivity |
---|
Kinase | RBC |
---|
CK2a1 | inactive (57.6%) |
CK2a2 | active (28.25%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC |
---|
CLK1 | active (36.65%) |
CLK2 | inactive (92.01%) |
CLK3 | active (16.08%) |
CLK4 | active (6.19%) |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC |
---|
DYRK1A | inactive (82.76%) |
DYRK1B | inactive (65.12%) |
DYRK2 | inactive (61.4%) |
DYRK3 | inactive (105.04%) |
DYRK4 | inactive (100.35%) |
HIPK1 | inactive (95.98%) |
HIPK2 | inactive (97.61%) |
HIPK3 | inactive (66.22%) |
HIPK4 | inactive (108.1%) |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC |
---|
Erk1 | inactive (98.66%) |
Erk2 | inactive (89.78%) |
JNK3 | inactive (103.04%) |
NLK | inactive (100.57%) |
p38a | inactive (101.04%) |
p38b | inactive (95.22%) |
p38d | inactive (94.8%) |
p38g | inactive (89.87%) |
JNK1 | inactive (101.07%) |
JNK2 | active (44.34%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC |
---|
GSK3A | active (7.31%) |
GSK3B | active (12.58%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC |
---|
MSSK1 | inactive (59.51%) |
SRPK1 | inactive (71.33%) |
SRPK2 | inactive (86.55%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
PDHK | 5 | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC |
---|
PDHK1 | inactive (83.33%) |