Compound Information
Test on : RBC, Millipore
Compound Name
RBC : CTK5I7912
Millipore : VEGF Receptor 2 Kinase Inhibitor II
Inchikey
Same : RFHPWPWVGFSLOP-N
RBC : RFHPWPWVGFSLOP-UHFFFAOYSA-N
Millipore : RFHPWPWVGFSLOP-ZROIWOOFSA-N
ChemSpider
RBC : 5453
Millipore : 4486317
Pubchem CID
RBC : 5655
Millipore : 5329155
ChEMBL
RBC : -
Millipore : CHEMBL88606
RBC | Millipore |
| |
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDK1 | inactive (95.27%) | inactive (109%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AKT1 | inactive (99.82%) | inactive (95%) |
AKT2 | inactive (90.3%) | inactive (112%) |
AKT3 | inactive (96.61%) | inactive (105%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DMPK1 | inactive (101.07%) | inactive (115%) |
MRCKa | inactive (81.85%) | inactive (108%) |
MRCKb | inactive (113.52%) | inactive (98%) |
ROCK1 | inactive (98.77%) | inactive (119%) |
ROCK2 | inactive (92.79%) | inactive (101%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BARK1 | inactive (105.14%) | - |
BARK2 | inactive (89.86%) | - |
GPRK4 | inactive (100.86%) | - |
GPRK5 | inactive (105.93%) | inactive (104%) |
GPRK6 | inactive (95.79%) | inactive (102%) |
GPRK7 | inactive (85.17%) | inactive (98%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSK1 | inactive (90.35%) | inactive (111%) |
MSK2 | inactive (94.21%) | inactive (88%) |
p70S6K | inactive (91.92%) | inactive (84%) |
p70S6Kb | inactive (102.37%) | - |
RSK2 | inactive (80.87%) | active (45%) |
RSK4 | inactive (78.64%) | inactive (79%) |
RSK1 | inactive (70.43%) | inactive (79%) |
RSK3 | inactive (71.96%) | inactive (84%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKACg | inactive (98.09%) | - |
PRKX | inactive (97.21%) | inactive (113%) |
PKACa | inactive (96.53%) | inactive (108%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKCa | inactive (101.97%) | inactive (104%) |
PKCd | inactive (95.62%) | inactive (100%) |
PKCe | inactive (99.08%) | inactive (84%) |
PKCh | inactive (97.43%) | inactive (102%) |
PKCg | inactive (100.1%) | inactive (109%) |
PKCi | inactive (91.95%) | inactive (84%) |
PKCt | inactive (98.4%) | inactive (100%) |
PKCz | inactive (104.03%) | inactive (103%) |
PKCb | inactive (85.48%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKG2 | inactive (92.38%) | - |
PKG1 | inactive (77.01%) | - |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKN1 | inactive (91.66%) | - |
PKN2 | inactive (91.33%) | inactive (95%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SGK1 | inactive (93.4%) | inactive (104%) |
SGK2 | inactive (101.18%) | inactive (111%) |
SGK3 | inactive (97.57%) | inactive (96%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NDR1 | inactive (80.12%) | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ABL1 | inactive (91.77%) | inactive (105%) |
ABL2 | inactive (82.57%) | inactive (94%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ACK | inactive (92.85%) | inactive (54%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK | inactive (88.48%) | inactive (76%) |
LTK | inactive (70.57%) | - |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AXL | inactive (90.01%) | inactive (72%) |
MER | inactive (81.2%) | inactive (68%) |
TYRO3 | inactive (103.62%) | inactive (93%) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BLK | inactive (74.42%) | inactive (82%) |
BRK | inactive (82.28%) | inactive (107%) |
SRC | inactive (88.76%) | inactive (73%) |
FGR | inactive (67.67%) | inactive (81%) |
FRK | inactive (91.03%) | inactive (102%) |
FYN | inactive (87.54%) | inactive (74%) |
HCK | inactive (88.49%) | inactive (59%) |
LCK | inactive (84.5%) | inactive (123%) |
SRM | inactive (104.07%) | - |
YES | inactive (67.17%) | inactive (79%) |
LYN | inactive (70.81%) | active (21%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BMX | inactive (89.94%) | inactive (96%) |
BTK | inactive (90.54%) | inactive (93%) |
ITK | inactive (87.48%) | inactive (87%) |
TEC | inactive (128.82%) | - |
TXK | inactive (97.26%) | inactive (107%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
KIT | active (30.49%) | inactive (66%) |
FLT3 | active (3.86%) | active (3%) |
FMS | active (49.69%) | active (11%) |
PDGFRb | inactive (58.77%) | inactive (74%) |
PDGFRa | inactive (76.16%) | active (34%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CSK | inactive (98.5%) | inactive (118%) |
CTK | inactive (94.21%) | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DDR2 | inactive (101.47%) | inactive (110%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EGFR | inactive (87.38%) | inactive (103%) |
ErbB2 | inactive (115.1%) | - |
ErbB4 | inactive (84.61%) | inactive (109%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EphA1 | inactive (93.12%) | inactive (91%) |
EphA2 | inactive (110.13%) | inactive (112%) |
EphA3 | inactive (94.62%) | inactive (108%) |
EphA4 | inactive (94.84%) | inactive (106%) |
EphA5 | inactive (91.31%) | inactive (110%) |
EphA6 | inactive (89.15%) | - |
EphA7 | inactive (85.29%) | inactive (94%) |
EphA8 | inactive (94.45%) | inactive (93%) |
EphB1 | inactive (85.48%) | inactive (101%) |
EphB2 | inactive (85.38%) | inactive (111%) |
EphB3 | inactive (99.69%) | inactive (114%) |
EphB4 | inactive (88.59%) | inactive (118%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FAK | inactive (81.92%) | inactive (78%) |
PYK2 | inactive (82.4%) | inactive (75%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FER | inactive (74.67%) | inactive (119%) |
FES | inactive (83.82%) | inactive (107%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FGFR1 | inactive (76.66%) | inactive (81%) |
FGFR2 | inactive (87.38%) | inactive (63%) |
FGFR3 | inactive (55.84%) | inactive (86%) |
FGFR4 | inactive (77.02%) | inactive (116%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FLT1 | inactive (73.44%) | active (17%) |
FLT4 | inactive (56.12%) | active (1%) |
KDR | inactive (70.92%) | active (12%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IGF1R | inactive (74.28%) | inactive (120%) |
IRR | inactive (94.78%) | inactive (114%) |
INSR | inactive (85.84%) | inactive (96%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
JAK1 | inactive (99.35%) | - |
JAK2 | inactive (95.22%) | inactive (105%) |
JAK3 | inactive (89.34%) | inactive (108%) |
TYK2 | inactive (86.03%) | - |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MUSK | inactive (88.6%) | inactive (61%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RET | active (42.87%) | inactive (74%) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RON | inactive (88.31%) | inactive (116%) |
MET | inactive (81.57%) | inactive (104%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ROS | inactive (98.61%) | inactive (94%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SYK | inactive (90.49%) | inactive (123%) |
ZAP70 | inactive (93.86%) | inactive (112%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TIE2 | inactive (98.18%) | inactive (110%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TRKA | inactive (51.76%) | active (19%) |
TRKB | active (43.58%) | active (48%) |
TRKC | active (11.87%) | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK1 | inactive (102.88%) | - |
ALK2 | inactive (96.96%) | - |
ALK4 | inactive (99.01%) | inactive (112%) |
TGFbR1 | inactive (100.44%) | inactive (98%) |
TGFbR2 | inactive (101.18%) | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ARAF | inactive (106.31%) | - |
BRAF | inactive (92.47%) | - |
RAF1 | inactive (88.25%) | inactive (99%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IRAK1 | inactive (97.02%) | inactive (92%) |
IRAK4 | inactive (67.23%) | inactive (82%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LIMK1 | inactive (82.95%) | inactive (99%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LRRK2 | active (7.03%) | - |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MLK1 | inactive (53.42%) | inactive (63%) |
MLK2 | inactive (99.82%) | - |
MLK3 | active (16.75%) | - |
TAK1 | inactive (60.94%) | inactive (94%) |
ZAK | inactive (87.69%) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RIPK2 | inactive (87.15%) | inactive (100%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NuaK1 | active (27.73%) | inactive (70%) |
BRSK1 | inactive (80.78%) | inactive (90%) |
BRSK2 | inactive (93.84%) | inactive (107%) |
CHK1 | inactive (81.76%) | inactive (78%) |
LKB1 | inactive (88.74%) | inactive (97%) |
MARK1 | inactive (69.05%) | inactive (72%) |
MARK3 | inactive (84.87%) | - |
MARK4 | inactive (82.86%) | - |
MELK | inactive (75.62%) | inactive (78%) |
PASK | inactive (98.86%) | inactive (129%) |
QIK | inactive (92.73%) | - |
NuaK2 | inactive (133.13%) | - |
MARK2 | inactive (77%) | inactive (81%) |
AMPKa1 | - | inactive (76%) |
AMPKa2 | - | inactive (87%) |
SIK | - | inactive (97%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK1a | inactive (98.41%) | inactive (105%) |
CaMK1b | inactive (98.59%) | - |
CaMK1d | inactive (96.76%) | inactive (114%) |
CaMK1g | inactive (103.45%) | - |
CaMK4 | inactive (97.49%) | inactive (135%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK2a | inactive (93.32%) | - |
CaMK2b | inactive (85.78%) | inactive (72%) |
CaMK2d | inactive (84.21%) | active (18%) |
CaMK2g | inactive (92.38%) | active (20%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CHK2 | inactive (68.23%) | active (44%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DAPK1 | inactive (110.94%) | inactive (98%) |
DAPK2 | inactive (102.44%) | inactive (95%) |
DRAK1 | inactive (72.86%) | active (48%) |
DAPK3 | inactive (92.79%) | inactive (96%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DCLK2 | inactive (98.16%) | inactive (94%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAPKAPK2 | inactive (97.45%) | inactive (108%) |
MAPKAPK3 | inactive (95.07%) | inactive (126%) |
MAPKAPK5 | inactive (90.64%) | inactive (82%) |
MNK1 | inactive (106.37%) | - |
MNK2 | inactive (87.13%) | inactive (108%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
smMLCK | inactive (95.68%) | inactive (83%) |
skMLCK | inactive (78.2%) | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PHKg1 | inactive (60.17%) | - |
PHKg2 | inactive (90.5%) | inactive (77%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PIM1 | inactive (100.64%) | inactive (96%) |
PIM2 | inactive (100.15%) | inactive (129%) |
PIM3 | inactive (87.52%) | inactive (105%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKD1 | inactive (93.82%) | inactive (91%) |
PKD3 | inactive (90.3%) | - |
PKD2 | inactive (95.84%) | inactive (96%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TSSK1 | active (36.09%) | inactive (98%) |
TSSK2 | inactive (89.85%) | inactive (90%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
STK33 | inactive (77.26%) | inactive (89%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP3K5 | inactive (100.88%) | inactive (83%) |
MAP3K2 | inactive (93.61%) | - |
MAP3K3 | inactive (88.55%) | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
COT | inactive (105.06%) | - |
NIK | inactive (111.64%) | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GCK | inactive (58.08%) | active (24%) |
HGK | active (6.84%) | - |
KHS1 | active (17.7%) | - |
LOK | inactive (65.53%) | inactive (74%) |
MINK | active (26.38%) | inactive (87%) |
MST1 | active (44.08%) | inactive (60%) |
MST2 | inactive (60.67%) | active (46%) |
MST3 | inactive (94.2%) | inactive (88%) |
MST4 | inactive (87.9%) | - |
OSR1 | inactive (96.74%) | - |
PAK1 | inactive (95.67%) | - |
PAK2 | inactive (90.02%) | inactive (113%) |
PAK3 | inactive (96.42%) | inactive (114%) |
PAK4 | inactive (76.76%) | inactive (84%) |
PAK5 | inactive (85.39%) | inactive (93%) |
PAK6 | inactive (89.82%) | inactive (85%) |
SLK | inactive (73.45%) | - |
YSK1 | inactive (101.6%) | - |
STLK3 | inactive (85.98%) | - |
TAO1 | inactive (92.32%) | inactive (104%) |
TAO2 | inactive (89.4%) | inactive (111%) |
TAO3 | inactive (75.3%) | inactive (100%) |
MYO3B | inactive (55.14%) | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP2K1 | inactive (84.82%) | inactive (87%) |
MAP2K2 | inactive (92.1%) | - |
MAP2K6 | inactive (109.87%) | inactive (76%) |
MAP2K7 | - | inactive (87%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AurA | inactive (87.45%) | inactive (85%) |
AurB | inactive (56.68%) | active (18%) |
AurC | inactive (86.27%) | inactive (82%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMKK1 | inactive (69.65%) | - |
CaMKK2 | inactive (68.09%) | - |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Haspin | inactive (88.01%) | inactive (87%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IKKa | inactive (99.09%) | inactive (102%) |
IKKb | inactive (102.15%) | inactive (101%) |
IKKe | inactive (89.53%) | - |
TBK1 | inactive (66.88%) | inactive (59%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NEK1 | inactive (94.64%) | - |
NEK11 | inactive (110.69%) | inactive (87%) |
NEK2 | inactive (87.89%) | inactive (91%) |
NEK4 | inactive (80.52%) | - |
NEK6 | inactive (102.57%) | inactive (104%) |
NEK7 | inactive (103.17%) | inactive (101%) |
NEK9 | inactive (85.62%) | - |
NEK3 | inactive (86.73%) | inactive (102%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PBK | inactive (87.83%) | - |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PLK1 | inactive (102.17%) | inactive (82%) |
PLK2 | inactive (101.79%) | inactive (105%) |
PLK3 | inactive (97.85%) | inactive (87%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SgK496 | inactive (93.05%) | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MPSK1 | inactive (94.27%) | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TTK | inactive (95.08%) | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ULK1 | inactive (69.42%) | - |
ULK2 | inactive (113.58%) | inactive (100%) |
ULK3 | inactive (55.47%) | inactive (52%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wee1 | inactive (95.89%) | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wnk2 | inactive (100.82%) | inactive (110%) |
Wnk3 | inactive (93.77%) | inactive (118%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TLK2 | inactive (100.56%) | inactive (107%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK1 | 7 | 6 | 4 |
VRK | 3 | 1 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK1d | inactive (72.41%) | inactive (86%) |
CK1g1 | inactive (101.73%) | inactive (100%) |
CK1g2 | inactive (96.83%) | inactive (95%) |
CK1g3 | inactive (102.91%) | inactive (118%) |
CK1a | inactive (100.49%) | - |
CK1e | inactive (84.26%) | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
VRK1 | inactive (107.82%) | - |
VRK2 | - | inactive (98%) |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK2 | 3 | 2 | 2 |
CLK | 4 | 4 | 2 |
DYRK | 10 | 9 | 4 |
MAPK | 14 | 10 | 10 |
GSK | 2 | 2 | 2 |
SRPK | 3 | 3 | 3 |
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK2a1 | inactive (96.05%) | inactive (77%) |
CK2a2 | - | inactive (120%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CLK1 | inactive (97.21%) | - |
CLK2 | inactive (88.58%) | inactive (106%) |
CLK3 | inactive (101.23%) | inactive (91%) |
CLK4 | inactive (84.45%) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DYRK1A | inactive (87.15%) | - |
DYRK1B | inactive (93.86%) | - |
DYRK2 | inactive (90.83%) | inactive (97%) |
DYRK3 | inactive (94.03%) | - |
DYRK4 | inactive (101.72%) | - |
HIPK1 | inactive (97.21%) | inactive (98%) |
HIPK2 | inactive (90.96%) | inactive (82%) |
HIPK3 | inactive (96.73%) | inactive (97%) |
HIPK4 | inactive (103.93%) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Erk1 | inactive (95.02%) | inactive (89%) |
Erk2 | inactive (103.47%) | inactive (104%) |
JNK3 | inactive (98.68%) | inactive (115%) |
NLK | - | inactive (97%) |
p38a | - | inactive (86%) |
p38b | inactive (96.78%) | inactive (98%) |
p38d | inactive (100.2%) | inactive (111%) |
p38g | inactive (93.04%) | inactive (115%) |
JNK1 | inactive (106.63%) | inactive (114%) |
JNK2 | inactive (99.43%) | inactive (101%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GSK3A | inactive (88.47%) | inactive (113%) |
GSK3B | inactive (94.12%) | inactive (86%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSSK1 | inactive (77.82%) | inactive (101%) |
SRPK1 | inactive (98.32%) | inactive (111%) |
SRPK2 | inactive (90.59%) | inactive (88%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
PDHK | 5 | 1 | - |
Alpha | 6 | - | 1 |
PIKK | 6 | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDHK1 | inactive (95.27%) | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
eEF2K | - | inactive (91%) |
Atypical - PIKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FRAP | - | inactive (116%) |