Compound Information
Test on : RBC, Metz, Millipore
Compound Name
RBC, Metz, Millipore : kenpaullone
Inchikey
Same : QQUXFYAWXPMDOE-N
RBC, Metz, Millipore : QQUXFYAWXPMDOE-UHFFFAOYSA-N
ChemSpider
RBC, Metz, Millipore : 3688
Pubchem CID
RBC, Metz, Millipore : 3820
ChEMBL
RBC, Metz, Millipore : CHEMBL296586
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PDK1 | inactive (94.88%) | inactive (1258.93nM) | inactive (85%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
AKT1 | inactive (99.92%) | inactive (>7943.28nM) | inactive (107%) |
AKT2 | inactive (103.58%) | inactive (>7943.28nM) | inactive (89%) |
AKT3 | inactive (105.46%) | inactive (>10000nM) | inactive (101%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DMPK1 | inactive (109.51%) | - | inactive (97%) |
MRCKa | inactive (98.98%) | inactive (5011.87nM) | inactive (103%) |
MRCKb | inactive (95.93%) | - | inactive (72%) |
ROCK1 | inactive (96.09%) | inactive (1995.26nM) | inactive (117%) |
ROCK2 | inactive (84.61%) | inactive (2511.89nM) | inactive (73%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
BARK1 | inactive (102.54%) | - | - |
BARK2 | inactive (108.68%) | - | - |
GPRK4 | inactive (97.88%) | - | - |
GPRK5 | inactive (96.96%) | - | inactive (95%) |
GPRK6 | inactive (104.51%) | - | inactive (92%) |
GPRK7 | inactive (100.16%) | - | inactive (89%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MSK1 | inactive (99.63%) | - | inactive (99%) |
MSK2 | inactive (108.12%) | - | inactive (82%) |
p70S6K | inactive (102.94%) | inactive (>6309.57nM) | inactive (66%) |
p70S6Kb | inactive (99.4%) | - | - |
RSK2 | inactive (94.26%) | inactive (>7943.28nM) | active (33%) |
RSK4 | inactive (95.89%) | - | inactive (85%) |
RSK1 | inactive (90.79%) | - | active (12%) |
RSK3 | inactive (94.87%) | - | inactive (78%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKACg | inactive (105.21%) | - | - |
PRKX | inactive (100.2%) | - | inactive (85%) |
PKACa | inactive (102.02%) | inactive (>7943.28nM) | inactive (89%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKCa | inactive (98.57%) | - | inactive (90%) |
PKCd | inactive (92.74%) | inactive (>7943.28nM) | inactive (99%) |
PKCe | inactive (96.89%) | - | inactive (103%) |
PKCh | inactive (95.26%) | - | inactive (72%) |
PKCg | inactive (93.79%) | inactive (>7943.28nM) | inactive (104%) |
PKCi | inactive (89.07%) | - | inactive (103%) |
PKCt | inactive (114.32%) | - | active (49%) |
PKCz | inactive (98.3%) | inactive (>7943.28nM) | inactive (107%) |
PKCb | inactive (102.33%) | - | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKG2 | inactive (100.6%) | - | - |
PKG1 | inactive (95.88%) | - | - |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKN1 | inactive (101.44%) | - | - |
PKN2 | inactive (96.77%) | - | inactive (60%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
SGK1 | inactive (106.58%) | inactive (>10000nM) | inactive (95%) |
SGK2 | inactive (98.95%) | - | inactive (99%) |
SGK3 | inactive (106.58%) | - | inactive (91%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
NDR1 | inactive (98.61%) | - | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ABL1 | inactive (82.59%) | active (158.49nM) | inactive (64%) |
ABL2 | inactive (84.89%) | - | inactive (76%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ACK | active (38.76%) | - | active (24%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ALK | inactive (90.82%) | - | inactive (88%) |
LTK | inactive (91.82%) | - | - |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
AXL | inactive (101.42%) | - | inactive (85%) |
MER | inactive (89.46%) | - | inactive (78%) |
TYRO3 | inactive (97.74%) | - | inactive (92%) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
BLK | inactive (92.74%) | inactive (>1584.89nM) | active (48%) |
BRK | inactive (87.72%) | - | inactive (95%) |
SRC | inactive (71.35%) | active (1000nM) | inactive (73%) |
FGR | inactive (74.42%) | - | active (48%) |
FRK | inactive (97.43%) | - | inactive (68%) |
FYN | inactive (73.44%) | active (63.1nM) | active (31%) |
HCK | inactive (85.46%) | - | active (48%) |
LCK | inactive (81.93%) | inactive (1584.89nM) | active (18%) |
SRM | inactive (105.02%) | - | - |
YES | inactive (59.11%) | - | active (42%) |
LYN | inactive (67.18%) | active (125.89nM) | active (10%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
BMX | inactive (99.62%) | - | inactive (72%) |
BTK | inactive (97.95%) | - | inactive (85%) |
ITK | inactive (101.58%) | inactive (>1584.89nM) | inactive (83%) |
TEC | inactive (96.37%) | - | - |
TXK | inactive (82.63%) | - | inactive (73%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
KIT | inactive (90.31%) | inactive (>1258.93nM) | inactive (116%) |
FLT3 | active (47.73%) | inactive (1584.89nM) | inactive (65%) |
FMS | inactive (92.57%) | inactive (1995.26nM) | active (49%) |
PDGFRb | inactive (93.22%) | - | inactive (112%) |
PDGFRa | inactive (102.61%) | - | inactive (117%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CSK | inactive (88.04%) | - | inactive (104%) |
CTK | inactive (93.57%) | - | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DDR2 | inactive (98.41%) | - | inactive (89%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
EGFR | inactive (103.57%) | inactive (>1995.26nM) | inactive (113%) |
ErbB2 | inactive (103.31%) | inactive (>1584.89nM) | - |
ErbB4 | inactive (100.86%) | inactive (>3981.07nM) | inactive (111%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
EphA1 | inactive (100.1%) | - | inactive (91%) |
EphA2 | inactive (98.34%) | inactive (>3162.28nM) | inactive (91%) |
EphA3 | inactive (95.98%) | - | inactive (83%) |
EphA4 | inactive (96.12%) | - | inactive (103%) |
EphA5 | inactive (96.61%) | - | inactive (114%) |
EphA6 | inactive (93.66%) | - | - |
EphA7 | inactive (100.98%) | - | inactive (98%) |
EphA8 | inactive (101.39%) | - | inactive (95%) |
EphB1 | inactive (93.55%) | - | inactive (98%) |
EphB2 | inactive (95.55%) | - | inactive (121%) |
EphB3 | inactive (92.31%) | - | inactive (114%) |
EphB4 | inactive (100.12%) | - | inactive (89%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FAK | inactive (94.28%) | - | inactive (82%) |
PYK2 | inactive (101.61%) | - | inactive (89%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FER | inactive (89.75%) | - | inactive (86%) |
FES | inactive (87.83%) | - | inactive (63%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FGFR1 | inactive (99.37%) | inactive (>5011.87nM) | inactive (87%) |
FGFR2 | inactive (100.39%) | - | inactive (106%) |
FGFR3 | inactive (100.55%) | inactive (>1995.26nM) | inactive (127%) |
FGFR4 | inactive (112.73%) | - | inactive (118%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FLT1 | inactive (78.92%) | active (398.11nM) | inactive (77%) |
FLT4 | inactive (78.7%) | active (398.11nM) | inactive (56%) |
KDR | inactive (98.1%) | inactive (1995.26nM) | inactive (74%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
IGF1R | inactive (102.8%) | inactive (>1995.26nM) | inactive (113%) |
IRR | inactive (95.81%) | - | inactive (107%) |
INSR | inactive (101.03%) | inactive (>5011.87nM) | inactive (95%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
JAK1 | inactive (102.5%) | - | - |
JAK2 | inactive (101.67%) | inactive (>1584.89nM) | inactive (100%) |
JAK3 | inactive (102.8%) | inactive (>1584.89nM) | inactive (104%) |
TYK2 | inactive (81.69%) | inactive (>1995.26nM) | - |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MUSK | inactive (87.65%) | - | active (42%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
RET | inactive (102.32%) | - | inactive (93%) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
RON | inactive (93.59%) | - | inactive (72%) |
MET | inactive (101.88%) | inactive (>3162.28nM) | inactive (123%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ROS | inactive (83.59%) | - | inactive (100%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
SYK | inactive (81.51%) | - | inactive (72%) |
ZAP70 | inactive (93.62%) | - | inactive (110%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TIE2 | inactive (105.64%) | - | inactive (98%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TRKA | inactive (111.59%) | inactive (>2511.89nM) | inactive (59%) |
TRKB | inactive (95.04%) | inactive (>5011.87nM) | inactive (103%) |
TRKC | inactive (70.66%) | - | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ALK1 | inactive (99.04%) | - | - |
ALK2 | inactive (162.08%) | - | - |
ALK4 | inactive (99.77%) | - | inactive (105%) |
TGFbR1 | inactive (97.67%) | - | inactive (85%) |
TGFbR2 | inactive (74.25%) | - | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ARAF | inactive (103.94%) | - | - |
BRAF | inactive (97.66%) | - | - |
RAF1 | inactive (91.53%) | - | inactive (75%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
IRAK1 | inactive (98.6%) | - | inactive (94%) |
IRAK4 | inactive (88.25%) | inactive (>10000nM) | inactive (81%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
LIMK1 | inactive (99.18%) | inactive (7943.28nM) | inactive (89%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
LRRK2 | inactive (78.66%) | - | - |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MLK1 | inactive (64.56%) | - | active (22%) |
MLK2 | inactive (79.29%) | - | - |
MLK3 | active (49.38%) | - | - |
TAK1 | inactive (84.16%) | - | inactive (81%) |
ZAK | inactive (88.49%) | - | - |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
RIPK2 | inactive (75.94%) | - | active (49%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
NuaK1 | active (14.59%) | - | active (13%) |
BRSK1 | inactive (60.51%) | - | inactive (64%) |
BRSK2 | inactive (62.66%) | - | inactive (60%) |
CHK1 | inactive (89.01%) | inactive (3981.07nM) | inactive (77%) |
LKB1 | inactive (95.66%) | - | inactive (97%) |
MARK1 | inactive (88.29%) | - | inactive (51%) |
MARK3 | inactive (76.82%) | active (630.96nM) | - |
MARK4 | inactive (60.19%) | - | - |
MELK | inactive (74.77%) | - | inactive (89%) |
PASK | inactive (98.02%) | - | inactive (118%) |
QIK | inactive (63.46%) | - | - |
NuaK2 | inactive (71.06%) | - | - |
MARK2 | inactive (74.32%) | active (1000nM) | inactive (62%) |
AMPKa1 | - | inactive (>10000nM) | inactive (75%) |
AMPKa2 | - | - | inactive (61%) |
SIK | - | - | inactive (91%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CaMK1a | inactive (105.73%) | inactive (>7943.28nM) | inactive (94%) |
CaMK1b | inactive (99.65%) | - | - |
CaMK1d | inactive (112.44%) | - | inactive (93%) |
CaMK1g | inactive (97.38%) | - | - |
CaMK4 | inactive (98.06%) | - | inactive (101%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CaMK2a | inactive (105.22%) | - | - |
CaMK2b | inactive (97.81%) | - | inactive (81%) |
CaMK2d | inactive (91.07%) | - | inactive (58%) |
CaMK2g | inactive (116.13%) | - | active (50%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CHK2 | inactive (59.03%) | active (630.96nM) | active (37%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DAPK1 | inactive (101.06%) | - | inactive (84%) |
DAPK2 | inactive (100.49%) | - | inactive (101%) |
DRAK1 | inactive (101.65%) | - | inactive (76%) |
DAPK3 | inactive (110.54%) | inactive (>1258.93nM) | inactive (94%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DCLK2 | inactive (94.6%) | - | inactive (108%) |
DCLK1 | - | - | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MAPKAPK2 | inactive (101.49%) | inactive (>7943.28nM) | inactive (73%) |
MAPKAPK3 | inactive (100.29%) | inactive (>10000nM) | inactive (106%) |
MAPKAPK5 | inactive (94.59%) | - | inactive (97%) |
MNK1 | inactive (98.44%) | - | - |
MNK2 | inactive (101.83%) | - | inactive (90%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
smMLCK | inactive (96.34%) | - | inactive (89%) |
skMLCK | inactive (96.82%) | - | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PHKg1 | active (49.73%) | - | - |
PHKg2 | inactive (98.89%) | - | inactive (120%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PIM1 | inactive (96.8%) | inactive (2511.89nM) | inactive (75%) |
PIM2 | inactive (104.2%) | inactive (>1584.89nM) | inactive (100%) |
PIM3 | inactive (84.59%) | - | inactive (83%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKD1 | inactive (100.82%) | - | inactive (99%) |
PKD3 | inactive (95.53%) | - | - |
PKD2 | inactive (100.12%) | inactive (>10000nM) | inactive (104%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TSSK1 | inactive (80.44%) | - | inactive (87%) |
TSSK2 | inactive (99.3%) | - | inactive (96%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
STK33 | inactive (102.61%) | - | inactive (97%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MAP3K5 | inactive (99.19%) | - | inactive (84%) |
MAP3K2 | inactive (94.2%) | - | - |
MAP3K3 | inactive (93.19%) | - | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
COT | inactive (98.63%) | - | - |
NIK | inactive (106.07%) | - | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
GCK | active (20.06%) | - | active (6%) |
HGK | active (6.61%) | - | - |
KHS1 | active (30.06%) | - | - |
LOK | inactive (89.85%) | - | inactive (96%) |
MINK | active (29.57%) | - | active (27%) |
MST1 | inactive (81.79%) | - | active (44%) |
MST2 | inactive (83.2%) | active (630.96nM) | inactive (87%) |
MST3 | inactive (84.78%) | - | inactive (65%) |
MST4 | inactive (107.77%) | - | - |
OSR1 | inactive (107.32%) | - | - |
PAK1 | inactive (85.04%) | inactive (>10000nM) | - |
PAK2 | inactive (95.54%) | - | inactive (91%) |
PAK3 | inactive (96.64%) | - | inactive (94%) |
PAK4 | inactive (92.2%) | inactive (>5011.87nM) | active (25%) |
PAK5 | inactive (85.12%) | - | active (35%) |
PAK6 | inactive (97.84%) | - | inactive (73%) |
SLK | inactive (95.68%) | - | - |
YSK1 | inactive (98.8%) | - | - |
STLK3 | inactive (90.08%) | - | - |
TAO1 | inactive (99.36%) | - | inactive (76%) |
TAO2 | inactive (93.97%) | - | inactive (84%) |
TAO3 | inactive (82.77%) | - | inactive (78%) |
MYO3B | inactive (97.39%) | - | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MAP2K1 | inactive (84.31%) | - | inactive (107%) |
MAP2K2 | inactive (115.56%) | - | - |
MAP2K6 | inactive (95.29%) | - | inactive (100%) |
MAP2K7 | - | - | inactive (95%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
AurA | inactive (99.71%) | inactive (1258.93nM) | inactive (97%) |
AurB | inactive (84.25%) | inactive (6309.57nM) | inactive (69%) |
AurC | inactive (90.91%) | - | inactive (76%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CaMKK1 | inactive (99.85%) | - | - |
CaMKK2 | inactive (77.82%) | - | - |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Haspin | inactive (89.05%) | - | inactive (60%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
IKKa | inactive (98.59%) | inactive (>3981.07nM) | inactive (124%) |
IKKb | inactive (100.96%) | inactive (>3162.28nM) | inactive (115%) |
IKKe | inactive (89.81%) | - | - |
TBK1 | inactive (92.95%) | - | inactive (53%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
NEK1 | inactive (95.36%) | - | - |
NEK11 | inactive (106.71%) | - | active (38%) |
NEK2 | inactive (87.11%) | inactive (>10000nM) | inactive (95%) |
NEK4 | inactive (98.92%) | - | - |
NEK6 | inactive (100.22%) | - | inactive (113%) |
NEK7 | inactive (94.29%) | - | inactive (100%) |
NEK9 | inactive (94.03%) | - | - |
NEK3 | inactive (96.2%) | - | inactive (81%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PBK | inactive (99.28%) | - | - |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PLK1 | inactive (94.86%) | inactive (>7943.28nM) | inactive (76%) |
PLK2 | inactive (99.14%) | - | inactive (99%) |
PLK3 | inactive (95.98%) | inactive (>7943.28nM) | inactive (95%) |
PLK4 | - | active (398.11nM) | - |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
SgK496 | inactive (98.62%) | - | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MPSK1 | inactive (98.87%) | - | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TTK | inactive (80.87%) | - | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ULK1 | inactive (93.83%) | - | - |
ULK2 | inactive (90.06%) | - | inactive (79%) |
ULK3 | inactive (83.18%) | - | inactive (74%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Wee1 | inactive (87.69%) | - | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Wnk2 | inactive (112.21%) | - | inactive (93%) |
Wnk3 | inactive (95.51%) | - | inactive (88%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TLK2 | inactive (99.39%) | - | inactive (89%) |
Other - CDC7
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CDC7 | - | active (100nM) | - |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz | Millipore |
---|
CK1 | 7 | 6 | 5 | 4 |
VRK | 3 | 1 | - | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CK1d | inactive (103.59%) | inactive (>7943.28nM) | inactive (80%) |
CK1g1 | inactive (101.78%) | - | inactive (106%) |
CK1g2 | inactive (101.59%) | - | inactive (114%) |
CK1g3 | inactive (102.99%) | - | inactive (101%) |
CK1a | inactive (95.15%) | - | - |
CK1e | inactive (103.27%) | - | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
VRK1 | inactive (87.27%) | - | - |
VRK2 | - | - | inactive (99%) |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz | Millipore |
---|
CK2 | 3 | 2 | 1 | 2 |
CLK | 4 | 4 | 2 | 2 |
DYRK | 10 | 9 | 6 | 4 |
MAPK | 14 | 10 | 8 | 10 |
GSK | 2 | 2 | 2 | 2 |
SRPK | 3 | 3 | 1 | 3 |
CDK | 20 | - | 7 | - |
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CK2a1 | inactive (79.07%) | active (398.11nM) | inactive (79%) |
CK2a2 | inactive (74.58%) | - | inactive (112%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CLK1 | inactive (96.72%) | - | - |
CLK2 | inactive (95.69%) | - | inactive (80%) |
CLK3 | inactive (99.27%) | - | inactive (78%) |
CLK4 | inactive (91.13%) | - | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DYRK1A | inactive (98.84%) | inactive (5011.87nM) | - |
DYRK1B | inactive (101.93%) | - | - |
DYRK2 | inactive (106.83%) | - | inactive (92%) |
DYRK3 | inactive (112.62%) | - | - |
DYRK4 | inactive (97.16%) | - | - |
HIPK1 | inactive (102.91%) | - | inactive (103%) |
HIPK2 | inactive (106.86%) | - | inactive (98%) |
HIPK3 | inactive (109.29%) | - | inactive (102%) |
HIPK4 | inactive (104.94%) | - | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Erk1 | inactive (100.3%) | - | inactive (85%) |
Erk2 | inactive (90.48%) | inactive (>7943.28nM) | inactive (114%) |
JNK3 | inactive (89.57%) | - | inactive (67%) |
NLK | inactive (98.7%) | - | inactive (83%) |
p38a | inactive (92.98%) | - | inactive (90%) |
p38b | inactive (103.63%) | - | inactive (98%) |
p38d | inactive (102.75%) | inactive (>7943.28nM) | inactive (98%) |
p38g | inactive (101.45%) | inactive (>6309.57nM) | inactive (101%) |
JNK1 | inactive (87.45%) | inactive (>3162.28nM) | inactive (95%) |
JNK2 | inactive (93.85%) | inactive (>3981.07nM) | inactive (87%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
GSK3A | active (5.87%) | active (7.94nM) | active (5%) |
GSK3B | active (19.67%) | active (19.95nM) | active (8%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MSSK1 | inactive (100.45%) | - | inactive (98%) |
SRPK1 | inactive (99.57%) | - | inactive (105%) |
SRPK2 | inactive (98.94%) | - | inactive (105%) |
CMGC - CDK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CDC2 | - | - | - |
CDK2 | - | active (100nM) | - |
CDK5 | - | inactive (1584.89nM) | - |
CDK8 | - | - | - |
CDK7 | - | - | - |
CDK9 | - | - | - |
CDK11 | - | - | - |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz | Millipore |
---|
PDHK | 5 | 1 | - | - |
Alpha | 6 | - | 1 | 1 |
PIKK | 6 | - | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PDHK1 | inactive (94.88%) | - | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
eEF2K | - | - | inactive (106%) |
Atypical - PIKK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FRAP | - | - | inactive (114%) |