Compound Information
Test on : RBC, Millipore
Compound Name
RBC : 3-[(2-chloro-1H-indol-3-yl)methylidene]-1H-indol-2-one
Millipore : cdk1 inhibitor
Inchikey
Same : QJKBRWSJWQVKLY-N
RBC : QJKBRWSJWQVKLY-UHFFFAOYSA-N
Millipore : QJKBRWSJWQVKLY-UKTHLTGXSA-N
ChemSpider
RBC : 2508
Millipore : 4582471
Pubchem CID
RBC : 2607
Millipore : 5472558
ChEMBL
RBC : -
Millipore : CHEMBL261425
RBC | Millipore |
| |
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDK1 | inactive (94.29%) | inactive (109%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AKT1 | inactive (93.96%) | inactive (113%) |
AKT2 | inactive (96.77%) | inactive (92%) |
AKT3 | inactive (93.6%) | inactive (104%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DMPK1 | inactive (101.3%) | inactive (119%) |
MRCKa | inactive (95.69%) | inactive (106%) |
MRCKb | inactive (101.52%) | inactive (89%) |
ROCK1 | inactive (100.93%) | inactive (121%) |
ROCK2 | inactive (90.22%) | inactive (98%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BARK1 | inactive (98.92%) | - |
BARK2 | inactive (90.13%) | - |
GPRK4 | inactive (102.2%) | - |
GPRK5 | inactive (108.9%) | inactive (96%) |
GPRK6 | inactive (106.66%) | inactive (89%) |
GPRK7 | inactive (105.69%) | inactive (99%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSK1 | inactive (85.45%) | inactive (100%) |
MSK2 | inactive (93.61%) | inactive (92%) |
p70S6K | inactive (99.65%) | inactive (87%) |
p70S6Kb | inactive (99.41%) | - |
RSK2 | inactive (82.87%) | inactive (60%) |
RSK4 | inactive (91.24%) | inactive (51%) |
RSK1 | inactive (105.21%) | inactive (91%) |
RSK3 | inactive (81.07%) | inactive (106%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKACg | - | - |
PRKX | inactive (106%) | inactive (125%) |
PKACa | inactive (102.1%) | inactive (105%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKCa | inactive (63.2%) | inactive (106%) |
PKCd | inactive (88.43%) | inactive (91%) |
PKCe | inactive (95.11%) | inactive (93%) |
PKCh | inactive (73.56%) | inactive (89%) |
PKCg | inactive (89.22%) | inactive (92%) |
PKCi | inactive (99.24%) | inactive (112%) |
PKCt | inactive (91.74%) | inactive (81%) |
PKCz | inactive (103.07%) | inactive (101%) |
PKCb | inactive (92.61%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKG2 | inactive (71.71%) | - |
PKG1 | inactive (92.49%) | - |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKN1 | inactive (94.56%) | - |
PKN2 | inactive (96.26%) | inactive (106%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SGK1 | inactive (116.3%) | inactive (101%) |
SGK2 | inactive (103.19%) | inactive (98%) |
SGK3 | inactive (101.84%) | inactive (111%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NDR1 | active (0%) | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ABL1 | inactive (95.15%) | inactive (110%) |
ABL2 | inactive (91.4%) | inactive (116%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ACK | inactive (98.4%) | inactive (84%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK | inactive (97.87%) | inactive (81%) |
LTK | inactive (95.1%) | - |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AXL | inactive (97.81%) | inactive (111%) |
MER | inactive (88.21%) | inactive (77%) |
TYRO3 | inactive (99.36%) | inactive (98%) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BLK | inactive (95.41%) | inactive (108%) |
BRK | inactive (76.95%) | inactive (97%) |
SRC | inactive (78.48%) | inactive (115%) |
FGR | inactive (90.47%) | inactive (97%) |
FRK | inactive (100.01%) | inactive (83%) |
FYN | inactive (100.8%) | inactive (81%) |
HCK | inactive (98.48%) | inactive (79%) |
LCK | inactive (95.52%) | inactive (83%) |
SRM | inactive (84.24%) | - |
YES | inactive (93.87%) | inactive (102%) |
LYN | inactive (99.69%) | inactive (89%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BMX | inactive (99.81%) | inactive (86%) |
BTK | inactive (94.63%) | inactive (98%) |
ITK | inactive (103.98%) | inactive (102%) |
TEC | inactive (124.31%) | - |
TXK | inactive (99.64%) | inactive (83%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
KIT | inactive (90.16%) | inactive (109%) |
FLT3 | inactive (80.49%) | inactive (88%) |
FMS | inactive (97.24%) | inactive (79%) |
PDGFRb | inactive (101.78%) | inactive (108%) |
PDGFRa | inactive (88.72%) | inactive (102%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CSK | inactive (100.56%) | inactive (110%) |
CTK | inactive (89.49%) | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DDR2 | inactive (92.74%) | inactive (94%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EGFR | inactive (97.55%) | inactive (106%) |
ErbB2 | inactive (97.26%) | - |
ErbB4 | inactive (102.92%) | inactive (107%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EphA1 | inactive (98.49%) | inactive (87%) |
EphA2 | inactive (97.35%) | inactive (100%) |
EphA3 | inactive (95.05%) | inactive (100%) |
EphA4 | inactive (93.42%) | inactive (117%) |
EphA5 | inactive (83.39%) | inactive (118%) |
EphA6 | - | - |
EphA7 | inactive (95.29%) | inactive (95%) |
EphA8 | inactive (102.81%) | inactive (100%) |
EphB1 | inactive (90.85%) | inactive (101%) |
EphB2 | inactive (94.19%) | inactive (115%) |
EphB3 | inactive (91.35%) | inactive (107%) |
EphB4 | inactive (90.2%) | inactive (117%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FAK | inactive (101.23%) | inactive (98%) |
PYK2 | inactive (95.49%) | inactive (96%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FER | inactive (91.82%) | inactive (95%) |
FES | inactive (96.62%) | inactive (99%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FGFR1 | inactive (91.95%) | inactive (107%) |
FGFR2 | inactive (102.4%) | inactive (119%) |
FGFR3 | inactive (101.13%) | inactive (105%) |
FGFR4 | inactive (96.9%) | inactive (104%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FLT1 | inactive (88.61%) | inactive (88%) |
FLT4 | inactive (107.51%) | inactive (64%) |
KDR | inactive (96.34%) | inactive (96%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IGF1R | inactive (105.17%) | inactive (111%) |
IRR | inactive (93.66%) | inactive (108%) |
INSR | inactive (91.22%) | inactive (104%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
JAK1 | inactive (96.63%) | - |
JAK2 | inactive (102.97%) | inactive (96%) |
JAK3 | inactive (102.35%) | inactive (109%) |
TYK2 | inactive (110.31%) | - |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MUSK | inactive (96.38%) | inactive (78%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RET | inactive (93.01%) | inactive (108%) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RON | inactive (97.51%) | inactive (86%) |
MET | inactive (108.96%) | inactive (121%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ROS | inactive (109.49%) | inactive (93%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SYK | inactive (101.83%) | inactive (105%) |
ZAP70 | inactive (105.64%) | inactive (90%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TIE2 | inactive (97.09%) | inactive (97%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TRKA | inactive (90.68%) | inactive (85%) |
TRKB | inactive (94.99%) | inactive (87%) |
TRKC | inactive (92.9%) | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK1 | inactive (99.83%) | - |
ALK2 | inactive (100.16%) | - |
ALK4 | inactive (105.15%) | inactive (106%) |
TGFbR1 | inactive (94.4%) | inactive (98%) |
TGFbR2 | inactive (95.59%) | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ARAF | inactive (125.31%) | - |
BRAF | inactive (94.53%) | - |
RAF1 | inactive (89.9%) | inactive (85%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IRAK1 | inactive (89.5%) | inactive (100%) |
IRAK4 | inactive (102.06%) | inactive (92%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LIMK1 | inactive (109.34%) | inactive (91%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LRRK2 | inactive (102.29%) | - |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MLK1 | inactive (97.9%) | inactive (95%) |
MLK2 | inactive (94.73%) | - |
MLK3 | inactive (100.31%) | - |
TAK1 | inactive (99.17%) | inactive (99%) |
ZAK | inactive (99.19%) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RIPK2 | inactive (85.37%) | inactive (84%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NuaK1 | inactive (86.04%) | inactive (91%) |
BRSK1 | inactive (91.92%) | inactive (94%) |
BRSK2 | inactive (96.2%) | inactive (106%) |
CHK1 | inactive (93.72%) | inactive (97%) |
LKB1 | inactive (83.41%) | inactive (100%) |
MARK1 | inactive (96.03%) | inactive (92%) |
MARK3 | inactive (104.25%) | - |
MARK4 | inactive (105.99%) | - |
MELK | inactive (85.66%) | inactive (77%) |
PASK | inactive (89.29%) | inactive (99%) |
QIK | inactive (102.53%) | - |
NuaK2 | inactive (105.82%) | - |
MARK2 | inactive (94.66%) | inactive (113%) |
AMPKa1 | - | inactive (104%) |
AMPKa2 | - | inactive (93%) |
SIK | - | inactive (120%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK1a | inactive (106.4%) | inactive (93%) |
CaMK1b | inactive (92.9%) | - |
CaMK1d | inactive (101.58%) | inactive (117%) |
CaMK1g | - | - |
CaMK4 | inactive (101.77%) | inactive (116%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK2a | inactive (102.97%) | - |
CaMK2b | inactive (107.68%) | inactive (95%) |
CaMK2d | inactive (86.73%) | inactive (87%) |
CaMK2g | inactive (102.88%) | inactive (97%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CHK2 | inactive (99.35%) | inactive (75%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DAPK1 | inactive (88.11%) | inactive (95%) |
DAPK2 | inactive (96.82%) | inactive (103%) |
DRAK1 | inactive (95.17%) | inactive (83%) |
DAPK3 | inactive (91.21%) | inactive (98%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DCLK2 | inactive (93.47%) | inactive (107%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAPKAPK2 | inactive (101.17%) | inactive (88%) |
MAPKAPK3 | inactive (91.34%) | inactive (110%) |
MAPKAPK5 | inactive (121.43%) | inactive (104%) |
MNK1 | inactive (105.43%) | - |
MNK2 | inactive (93.51%) | inactive (98%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
smMLCK | inactive (90.38%) | inactive (91%) |
skMLCK | inactive (94.58%) | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PHKg1 | inactive (85.36%) | - |
PHKg2 | inactive (84.16%) | inactive (87%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PIM1 | inactive (88.53%) | inactive (92%) |
PIM2 | inactive (106.27%) | inactive (73%) |
PIM3 | inactive (99.99%) | inactive (88%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKD1 | inactive (89.5%) | inactive (99%) |
PKD3 | inactive (87.74%) | - |
PKD2 | inactive (90.21%) | inactive (106%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TSSK1 | inactive (101.32%) | inactive (81%) |
TSSK2 | inactive (113.43%) | inactive (91%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
STK33 | inactive (105.34%) | inactive (99%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP3K5 | inactive (107.21%) | inactive (88%) |
MAP3K2 | inactive (94.03%) | - |
MAP3K3 | inactive (111.56%) | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
COT | inactive (94.31%) | - |
NIK | inactive (92.59%) | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GCK | inactive (97.87%) | inactive (88%) |
HGK | inactive (75.71%) | - |
KHS1 | inactive (95%) | - |
LOK | inactive (90.95%) | inactive (84%) |
MINK | inactive (94.91%) | inactive (101%) |
MST1 | inactive (91.04%) | inactive (51%) |
MST2 | inactive (89.07%) | inactive (101%) |
MST3 | inactive (81.48%) | inactive (83%) |
MST4 | - | - |
OSR1 | inactive (89.1%) | - |
PAK1 | inactive (92.81%) | - |
PAK2 | inactive (101%) | inactive (101%) |
PAK3 | inactive (98.79%) | inactive (89%) |
PAK4 | inactive (103.89%) | inactive (96%) |
PAK5 | inactive (105.86%) | inactive (106%) |
PAK6 | inactive (100.69%) | inactive (109%) |
SLK | inactive (93.53%) | - |
YSK1 | inactive (97.74%) | - |
STLK3 | inactive (103.56%) | - |
TAO1 | inactive (100.21%) | inactive (92%) |
TAO2 | inactive (103.95%) | inactive (94%) |
TAO3 | inactive (93.92%) | inactive (85%) |
MYO3B | active (0%) | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP2K1 | inactive (84.82%) | inactive (101%) |
MAP2K2 | inactive (98.66%) | - |
MAP2K6 | inactive (93.39%) | inactive (88%) |
MAP2K7 | - | inactive (88%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AurA | inactive (107.93%) | inactive (99%) |
AurB | inactive (97.86%) | inactive (94%) |
AurC | inactive (89.45%) | inactive (89%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMKK1 | inactive (115.97%) | - |
CaMKK2 | inactive (97.82%) | - |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Haspin | inactive (90.99%) | inactive (85%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IKKa | inactive (94.17%) | inactive (106%) |
IKKb | inactive (105.86%) | inactive (111%) |
IKKe | inactive (97.95%) | - |
TBK1 | inactive (95.88%) | inactive (72%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NEK1 | inactive (96.72%) | - |
NEK11 | inactive (98.52%) | inactive (64%) |
NEK2 | inactive (99.05%) | inactive (88%) |
NEK4 | inactive (97.72%) | - |
NEK6 | inactive (96.5%) | inactive (108%) |
NEK7 | inactive (97.59%) | inactive (112%) |
NEK9 | inactive (94.23%) | - |
NEK3 | inactive (91.17%) | inactive (82%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PBK | inactive (101.55%) | - |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PLK1 | inactive (95.36%) | inactive (86%) |
PLK2 | inactive (98.18%) | inactive (99%) |
PLK3 | inactive (100.77%) | inactive (98%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SgK496 | inactive (95.7%) | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MPSK1 | inactive (101.77%) | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TTK | inactive (101.3%) | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ULK1 | inactive (105.53%) | - |
ULK2 | inactive (99.71%) | inactive (104%) |
ULK3 | active (0%) | inactive (93%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wee1 | inactive (107.33%) | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wnk2 | inactive (93.4%) | inactive (96%) |
Wnk3 | inactive (101.34%) | inactive (95%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TLK2 | active (0%) | inactive (90%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK1 | 7 | 6 | 4 |
VRK | 3 | 1 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK1d | inactive (90.5%) | inactive (85%) |
CK1g1 | inactive (99.25%) | inactive (103%) |
CK1g2 | inactive (96.35%) | inactive (96%) |
CK1g3 | inactive (92.78%) | inactive (85%) |
CK1a | inactive (101.53%) | - |
CK1e | inactive (87.77%) | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
VRK1 | inactive (104.35%) | - |
VRK2 | - | inactive (76%) |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK2 | 3 | 2 | 2 |
CLK | 4 | 4 | 2 |
DYRK | 10 | 9 | 4 |
MAPK | 14 | 10 | 10 |
GSK | 2 | 2 | 2 |
SRPK | 3 | 3 | 3 |
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK2a1 | inactive (89.4%) | inactive (99%) |
CK2a2 | inactive (94.26%) | inactive (106%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CLK1 | inactive (103.2%) | - |
CLK2 | inactive (92.66%) | inactive (105%) |
CLK3 | inactive (102.04%) | inactive (94%) |
CLK4 | inactive (105.05%) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DYRK1A | inactive (106.68%) | - |
DYRK1B | inactive (99.31%) | - |
DYRK2 | inactive (102.9%) | inactive (97%) |
DYRK3 | inactive (101.45%) | - |
DYRK4 | inactive (97.36%) | - |
HIPK1 | inactive (100%) | inactive (114%) |
HIPK2 | inactive (96.55%) | inactive (102%) |
HIPK3 | inactive (99.98%) | inactive (101%) |
HIPK4 | inactive (98.84%) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Erk1 | inactive (109.14%) | inactive (92%) |
Erk2 | inactive (96.39%) | inactive (121%) |
JNK3 | inactive (102.94%) | inactive (83%) |
NLK | inactive (107.4%) | inactive (95%) |
p38a | inactive (101.11%) | inactive (88%) |
p38b | inactive (94.45%) | inactive (99%) |
p38d | inactive (98.94%) | inactive (102%) |
p38g | inactive (93.01%) | inactive (88%) |
JNK1 | inactive (93.47%) | inactive (102%) |
JNK2 | inactive (101%) | inactive (94%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GSK3A | inactive (99.29%) | inactive (105%) |
GSK3B | inactive (105.34%) | inactive (141%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSSK1 | inactive (97.13%) | inactive (109%) |
SRPK1 | inactive (94.18%) | inactive (104%) |
SRPK2 | inactive (94.4%) | inactive (100%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
PDHK | 5 | 1 | - |
Alpha | 6 | - | 1 |
PIKK | 6 | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDHK1 | inactive (94.29%) | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
eEF2K | - | inactive (103%) |
Atypical - PIKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FRAP | - | inactive (118%) |