Compound Information
Test on : RBC
Compound Name : -
Inchikey : QDLHCMPXEPAAMD-BLNDMVMCSA-N
CANNOT FIND
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC |
---|
PDK1 | inactive (96.53%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC |
---|
AKT1 | inactive (95.43%) |
AKT2 | inactive (94.17%) |
AKT3 | inactive (94.59%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC |
---|
DMPK1 | inactive (98.68%) |
MRCKa | inactive (89.2%) |
MRCKb | inactive (111.86%) |
ROCK1 | inactive (90.74%) |
ROCK2 | inactive (88.17%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC |
---|
BARK1 | inactive (98.29%) |
BARK2 | inactive (92.78%) |
GPRK4 | inactive (95.35%) |
GPRK5 | inactive (106.99%) |
GPRK6 | inactive (101.29%) |
GPRK7 | inactive (90.4%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC |
---|
MSK1 | inactive (92.2%) |
MSK2 | inactive (96.74%) |
p70S6K | inactive (89.02%) |
p70S6Kb | inactive (100.44%) |
RSK2 | inactive (87.47%) |
RSK4 | inactive (96.73%) |
RSK1 | inactive (91.34%) |
RSK3 | inactive (94.8%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC |
---|
PKACg | inactive (96.11%) |
PRKX | inactive (91.68%) |
PKACa | inactive (93.02%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC |
---|
PKCa | inactive (96.3%) |
PKCd | inactive (96.1%) |
PKCe | inactive (86.47%) |
PKCh | inactive (100.2%) |
PKCg | inactive (113.77%) |
PKCi | inactive (89.99%) |
PKCt | inactive (94.69%) |
PKCz | inactive (99.2%) |
PKCb | inactive (117.13%) |
AGC - PKG
Bioactivity |
---|
Kinase | RBC |
---|
PKG2 | inactive (100.94%) |
PKG1 | inactive (97.41%) |
AGC - PKN
Bioactivity |
---|
Kinase | RBC |
---|
PKN1 | inactive (94.23%) |
PKN2 | inactive (98.53%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC |
---|
SGK1 | inactive (100.56%) |
SGK2 | inactive (98.99%) |
SGK3 | inactive (101.94%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC |
---|
NDR1 | inactive (110.69%) |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC |
---|
ABL1 | inactive (101.37%) |
ABL2 | inactive (94.89%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC |
---|
ACK | inactive (102.42%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC |
---|
ALK | inactive (102.75%) |
LTK | inactive (100.4%) |
TK - Axl
Bioactivity |
---|
Kinase | RBC |
---|
AXL | inactive (98.98%) |
MER | inactive (88.72%) |
TYRO3 | inactive (106.65%) |
TK - Src
Bioactivity |
---|
Kinase | RBC |
---|
BLK | inactive (87.76%) |
BRK | inactive (81.73%) |
SRC | inactive (99.48%) |
FGR | inactive (87.89%) |
FRK | inactive (94.26%) |
FYN | inactive (92.28%) |
HCK | inactive (91.33%) |
LCK | inactive (92.73%) |
SRM | inactive (103.2%) |
YES | inactive (98.33%) |
LYN | inactive (103.01%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC |
---|
BMX | inactive (92.26%) |
BTK | inactive (103.86%) |
ITK | inactive (90.04%) |
TEC | inactive (117.97%) |
TXK | inactive (98.95%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC |
---|
KIT | inactive (91.29%) |
FLT3 | inactive (93.38%) |
FMS | inactive (93.6%) |
PDGFRb | inactive (98.05%) |
PDGFRa | inactive (97.39%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC |
---|
CSK | inactive (101.03%) |
CTK | inactive (98.75%) |
TK - DDR
Bioactivity |
---|
Kinase | RBC |
---|
DDR2 | inactive (95.7%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC |
---|
EGFR | inactive (97.02%) |
ErbB2 | inactive (94.5%) |
ErbB4 | inactive (83.88%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC |
---|
EphA1 | inactive (98.34%) |
EphA2 | inactive (100.05%) |
EphA3 | inactive (98.05%) |
EphA4 | inactive (96.02%) |
EphA5 | inactive (86.53%) |
EphA6 | inactive (89.74%) |
EphA7 | inactive (89.38%) |
EphA8 | inactive (96.36%) |
EphB1 | inactive (89.93%) |
EphB2 | inactive (101.83%) |
EphB3 | inactive (96.85%) |
EphB4 | inactive (96.84%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC |
---|
FAK | inactive (98.2%) |
PYK2 | inactive (86.26%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC |
---|
FER | inactive (81.68%) |
FES | inactive (98.2%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC |
---|
FGFR1 | inactive (89.59%) |
FGFR2 | inactive (95.39%) |
FGFR3 | inactive (96.45%) |
FGFR4 | inactive (88.86%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC |
---|
FLT1 | inactive (85.88%) |
FLT4 | inactive (112.89%) |
KDR | inactive (88.4%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC |
---|
IGF1R | inactive (81.89%) |
IRR | inactive (100.01%) |
INSR | inactive (87.68%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC |
---|
JAK1 | inactive (90.91%) |
JAK2 | inactive (102.27%) |
JAK3 | inactive (95.47%) |
TYK2 | inactive (92.11%) |
TK - Musk
Bioactivity |
---|
Kinase | RBC |
---|
MUSK | inactive (94.78%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC |
---|
RET | inactive (96.93%) |
TK - Met
Bioactivity |
---|
Kinase | RBC |
---|
RON | inactive (92.71%) |
MET | inactive (100.36%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC |
---|
ROS | inactive (100.32%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC |
---|
SYK | inactive (106.68%) |
ZAP70 | inactive (91.64%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC |
---|
TIE2 | inactive (90.87%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC |
---|
TRKA | inactive (97.9%) |
TRKB | inactive (99.92%) |
TRKC | inactive (87.78%) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC |
---|
ALK1 | inactive (98.79%) |
ALK2 | inactive (92.95%) |
ALK4 | inactive (97.71%) |
TGFbR1 | inactive (93.85%) |
TGFbR2 | inactive (103.52%) |
TKL - RAF
Bioactivity |
---|
Kinase | RBC |
---|
ARAF | inactive (82.47%) |
BRAF | inactive (96.39%) |
RAF1 | inactive (95.97%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC |
---|
IRAK1 | inactive (118.88%) |
IRAK4 | inactive (86.27%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC |
---|
LIMK1 | inactive (86.69%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC |
---|
LRRK2 | inactive (97.57%) |
TKL - MLK
Bioactivity |
---|
Kinase | RBC |
---|
MLK1 | inactive (91.56%) |
MLK2 | inactive (102.18%) |
MLK3 | inactive (97.06%) |
TAK1 | inactive (97.18%) |
ZAK | inactive (94.32%) |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC |
---|
RIPK2 | inactive (99.7%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC |
---|
NuaK1 | inactive (94.95%) |
BRSK1 | inactive (91.24%) |
BRSK2 | inactive (95.26%) |
CHK1 | inactive (102.47%) |
LKB1 | inactive (83.49%) |
MARK1 | inactive (98.14%) |
MARK3 | inactive (112.09%) |
MARK4 | inactive (101.75%) |
MELK | inactive (92.43%) |
PASK | inactive (87.88%) |
QIK | inactive (96.83%) |
NuaK2 | inactive (130.67%) |
MARK2 | inactive (92.96%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC |
---|
CaMK1a | inactive (104.18%) |
CaMK1b | inactive (98.15%) |
CaMK1d | inactive (95.91%) |
CaMK1g | inactive (96.67%) |
CaMK4 | inactive (98.54%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC |
---|
CaMK2a | inactive (97.08%) |
CaMK2b | inactive (95.73%) |
CaMK2d | inactive (98.09%) |
CaMK2g | inactive (86.4%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC |
---|
CHK2 | inactive (95.58%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC |
---|
DAPK1 | inactive (105.53%) |
DAPK2 | inactive (87.07%) |
DRAK1 | inactive (96.17%) |
DAPK3 | inactive (87.55%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC |
---|
DCLK2 | inactive (96.66%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC |
---|
MAPKAPK2 | inactive (96.86%) |
MAPKAPK3 | inactive (96.51%) |
MAPKAPK5 | inactive (88.35%) |
MNK1 | inactive (107.3%) |
MNK2 | inactive (80.23%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC |
---|
smMLCK | active (29.52%) |
skMLCK | inactive (95.86%) |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC |
---|
PHKg1 | inactive (92.55%) |
PHKg2 | inactive (88.2%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC |
---|
PIM1 | inactive (72.42%) |
PIM2 | inactive (60.57%) |
PIM3 | inactive (92.99%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC |
---|
PKD1 | inactive (97.31%) |
PKD3 | inactive (94.23%) |
PKD2 | inactive (96.59%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC |
---|
TSSK1 | - |
TSSK2 | inactive (96.95%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC |
---|
STK33 | inactive (88.25%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC |
---|
MAP3K5 | inactive (104.51%) |
MAP3K2 | inactive (98.42%) |
MAP3K3 | inactive (107.54%) |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC |
---|
COT | inactive (108.32%) |
NIK | inactive (106.02%) |
STE - STE20
Bioactivity |
---|
Kinase | RBC |
---|
GCK | inactive (97.67%) |
HGK | inactive (93.04%) |
KHS1 | inactive (95.62%) |
LOK | inactive (87.29%) |
MINK | inactive (91.24%) |
MST1 | inactive (89.6%) |
MST2 | inactive (79.45%) |
MST3 | inactive (93.12%) |
MST4 | inactive (95.8%) |
OSR1 | inactive (99.56%) |
PAK1 | inactive (95.26%) |
PAK2 | inactive (86.5%) |
PAK3 | inactive (91.43%) |
PAK4 | inactive (91.04%) |
PAK5 | inactive (95.76%) |
PAK6 | inactive (95.42%) |
SLK | inactive (94.06%) |
YSK1 | inactive (90.34%) |
STLK3 | inactive (96.48%) |
TAO1 | inactive (112.9%) |
TAO2 | inactive (97.61%) |
TAO3 | inactive (96.94%) |
MYO3B | inactive (86.41%) |
STE - STE7
Bioactivity |
---|
Kinase | RBC |
---|
MAP2K1 | inactive (97.32%) |
MAP2K2 | inactive (93.78%) |
MAP2K6 | inactive (101.04%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC |
---|
AurA | inactive (93.91%) |
AurB | inactive (94.21%) |
AurC | inactive (99.59%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC |
---|
CaMKK1 | inactive (92.1%) |
CaMKK2 | inactive (79.3%) |
Other - Haspin
Bioactivity |
---|
Kinase | RBC |
---|
Haspin | inactive (88.29%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC |
---|
IKKa | inactive (106.14%) |
IKKb | inactive (96.86%) |
IKKe | inactive (97.96%) |
TBK1 | inactive (92.6%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC |
---|
NEK1 | inactive (83.33%) |
NEK11 | inactive (95.1%) |
NEK2 | inactive (89.15%) |
NEK4 | inactive (74.74%) |
NEK6 | inactive (102.54%) |
NEK7 | inactive (108.33%) |
NEK9 | inactive (92.28%) |
NEK3 | inactive (97.93%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC |
---|
PBK | inactive (103.52%) |
Other - PLK
Bioactivity |
---|
Kinase | RBC |
---|
PLK1 | active (2.36%) |
PLK2 | inactive (51.56%) |
PLK3 | active (14.41%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC |
---|
SgK496 | inactive (95.41%) |
Other - NAK
Bioactivity |
---|
Kinase | RBC |
---|
MPSK1 | inactive (88.77%) |
Other - TTK
Bioactivity |
---|
Kinase | RBC |
---|
TTK | inactive (98.2%) |
Other - ULK
Bioactivity |
---|
Kinase | RBC |
---|
ULK1 | inactive (87.49%) |
ULK2 | inactive (100.66%) |
ULK3 | inactive (84.42%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC |
---|
Wee1 | inactive (96.92%) |
Other - WNK
Bioactivity |
---|
Kinase | RBC |
---|
Wnk2 | inactive (93.04%) |
Wnk3 | inactive (99.49%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC |
---|
TLK2 | inactive (99.5%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
CK1 | 7 | 6 |
VRK | 3 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC |
---|
CK1d | inactive (96.62%) |
CK1g1 | inactive (94.63%) |
CK1g2 | inactive (85.83%) |
CK1g3 | inactive (96.2%) |
CK1a | inactive (91.7%) |
CK1e | inactive (95.53%) |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC |
---|
VRK1 | inactive (101.49%) |
CMGC
CMGC - CK2
Bioactivity |
---|
Kinase | RBC |
---|
CK2a1 | inactive (94.85%) |
CK2a2 | inactive (98.32%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC |
---|
CLK1 | inactive (90.74%) |
CLK2 | inactive (88.01%) |
CLK3 | inactive (97.51%) |
CLK4 | inactive (85.41%) |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC |
---|
DYRK1A | inactive (97.34%) |
DYRK1B | inactive (99.97%) |
DYRK2 | inactive (110.84%) |
DYRK3 | inactive (92.58%) |
DYRK4 | inactive (101.55%) |
HIPK1 | inactive (108.19%) |
HIPK2 | inactive (99.63%) |
HIPK3 | inactive (103.48%) |
HIPK4 | inactive (99.27%) |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC |
---|
Erk1 | inactive (94.66%) |
Erk2 | inactive (101.4%) |
JNK3 | inactive (96.78%) |
NLK | inactive (93.79%) |
p38a | inactive (119.92%) |
p38b | inactive (91.6%) |
p38d | inactive (105.45%) |
p38g | inactive (97.74%) |
JNK1 | inactive (98.73%) |
JNK2 | inactive (100.13%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC |
---|
GSK3A | inactive (92.84%) |
GSK3B | inactive (80.53%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC |
---|
MSSK1 | inactive (95.26%) |
SRPK1 | inactive (94.4%) |
SRPK2 | inactive (85.4%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
PDHK | 5 | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC |
---|
PDHK1 | inactive (96.53%) |