Compound Information
Test on : RBC, Millipore
Compound Name
RBC : CHEMBL80611
Millipore : PURVALANOLA
Inchikey
Same : PMXCMJLOPOFPBT-N
RBC : PMXCMJLOPOFPBT-OAHLLOKOSA-N
Millipore : PMXCMJLOPOFPBT-UHFFFAOYSA-N
ChemSpider
RBC : 23168357
Millipore : 4813
Pubchem CID
RBC : 12084804
Millipore : 4987
ChEMBL
RBC : CHEMBL80611
Millipore : -
RBC | Millipore |
| |
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDK1 | inactive (91.6%) | inactive (111%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AKT1 | inactive (101.66%) | inactive (113%) |
AKT2 | inactive (90.02%) | inactive (105%) |
AKT3 | inactive (102.15%) | inactive (106%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DMPK1 | inactive (107.76%) | inactive (98%) |
MRCKa | inactive (92.32%) | inactive (112%) |
MRCKb | inactive (108%) | inactive (98%) |
ROCK1 | inactive (99.98%) | inactive (115%) |
ROCK2 | inactive (100.47%) | inactive (95%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BARK1 | inactive (102.68%) | - |
BARK2 | inactive (99.12%) | - |
GPRK4 | inactive (91.14%) | - |
GPRK5 | inactive (101.41%) | inactive (97%) |
GPRK6 | inactive (98.27%) | inactive (103%) |
GPRK7 | inactive (88.8%) | inactive (95%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSK1 | inactive (100.26%) | inactive (111%) |
MSK2 | inactive (90.06%) | inactive (95%) |
p70S6K | inactive (90.84%) | inactive (88%) |
p70S6Kb | inactive (101.32%) | - |
RSK2 | inactive (86.27%) | inactive (62%) |
RSK4 | inactive (96.79%) | active (40%) |
RSK1 | inactive (77.32%) | inactive (75%) |
RSK3 | inactive (69.39%) | inactive (77%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKACg | inactive (113.34%) | - |
PRKX | inactive (97.36%) | inactive (81%) |
PKACa | inactive (101.57%) | inactive (106%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKCa | inactive (115.28%) | inactive (104%) |
PKCd | inactive (103.89%) | inactive (107%) |
PKCe | inactive (115.31%) | inactive (112%) |
PKCh | inactive (92.75%) | inactive (100%) |
PKCg | inactive (98.2%) | inactive (102%) |
PKCi | inactive (96.57%) | inactive (115%) |
PKCt | inactive (126.83%) | inactive (70%) |
PKCz | inactive (102.48%) | inactive (101%) |
PKCb | inactive (88.65%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKG2 | inactive (89.3%) | - |
PKG1 | inactive (71.4%) | - |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKN1 | inactive (100.2%) | - |
PKN2 | inactive (103.67%) | inactive (104%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SGK1 | inactive (99.11%) | inactive (112%) |
SGK2 | inactive (102.84%) | inactive (99%) |
SGK3 | inactive (97.62%) | inactive (107%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NDR1 | inactive (90.51%) | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ABL1 | inactive (75.56%) | inactive (62%) |
ABL2 | active (32.16%) | active (22%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ACK | inactive (55.62%) | active (45%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK | inactive (100.46%) | inactive (71%) |
LTK | inactive (100.1%) | - |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AXL | inactive (94.75%) | inactive (90%) |
MER | inactive (84.67%) | active (26%) |
TYRO3 | inactive (98.94%) | inactive (85%) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BLK | inactive (68.83%) | active (38%) |
BRK | inactive (89.23%) | inactive (109%) |
SRC | active (24.57%) | active (23%) |
FGR | active (44.33%) | active (23%) |
FRK | inactive (90.18%) | inactive (59%) |
FYN | active (48.85%) | active (4%) |
HCK | inactive (55.65%) | active (20%) |
LCK | inactive (86.89%) | active (28%) |
SRM | inactive (104.29%) | - |
YES | active (21.19%) | active (4%) |
LYN | inactive (60.16%) | active (11%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BMX | inactive (84.29%) | active (34%) |
BTK | inactive (75.6%) | inactive (56%) |
ITK | inactive (86.89%) | inactive (68%) |
TEC | inactive (126.6%) | - |
TXK | inactive (54.14%) | inactive (66%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
KIT | inactive (91.02%) | inactive (117%) |
FLT3 | active (16.39%) | active (17%) |
FMS | inactive (96.85%) | inactive (70%) |
PDGFRb | inactive (105.76%) | inactive (107%) |
PDGFRa | inactive (96.91%) | inactive (109%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CSK | inactive (98.11%) | inactive (107%) |
CTK | inactive (93.12%) | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DDR2 | inactive (99.06%) | inactive (91%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EGFR | inactive (94.15%) | inactive (109%) |
ErbB2 | inactive (97.09%) | - |
ErbB4 | inactive (78.38%) | inactive (105%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EphA1 | inactive (98.3%) | inactive (69%) |
EphA2 | inactive (89.54%) | inactive (69%) |
EphA3 | inactive (104.86%) | inactive (86%) |
EphA4 | inactive (102.46%) | inactive (95%) |
EphA5 | inactive (87.9%) | inactive (83%) |
EphA6 | inactive (93.8%) | - |
EphA7 | inactive (86.79%) | inactive (76%) |
EphA8 | inactive (101.92%) | inactive (85%) |
EphB1 | inactive (83.54%) | inactive (63%) |
EphB2 | inactive (99.27%) | inactive (71%) |
EphB3 | inactive (102.34%) | inactive (77%) |
EphB4 | inactive (71.67%) | active (37%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FAK | inactive (85.87%) | inactive (65%) |
PYK2 | inactive (66.48%) | active (35%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FER | inactive (62.93%) | inactive (90%) |
FES | inactive (95.94%) | inactive (79%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FGFR1 | inactive (80.62%) | inactive (98%) |
FGFR2 | inactive (104.79%) | inactive (104%) |
FGFR3 | inactive (99.15%) | inactive (98%) |
FGFR4 | inactive (78.96%) | inactive (118%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FLT1 | inactive (101.98%) | inactive (88%) |
FLT4 | inactive (110.3%) | active (42%) |
KDR | inactive (95%) | inactive (105%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IGF1R | inactive (100.35%) | inactive (98%) |
IRR | inactive (88.23%) | inactive (83%) |
INSR | inactive (83.02%) | inactive (81%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
JAK1 | inactive (107.54%) | - |
JAK2 | inactive (97.73%) | inactive (106%) |
JAK3 | inactive (92.49%) | inactive (114%) |
TYK2 | inactive (95.19%) | - |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MUSK | inactive (56.76%) | active (48%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RET | inactive (81.36%) | inactive (91%) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RON | inactive (90.64%) | inactive (92%) |
MET | inactive (96.2%) | inactive (83%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ROS | inactive (88.11%) | inactive (106%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SYK | inactive (88.9%) | inactive (102%) |
ZAP70 | inactive (99.74%) | inactive (118%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TIE2 | inactive (93.83%) | inactive (99%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TRKA | inactive (67.31%) | active (3%) |
TRKB | active (33.4%) | active (8%) |
TRKC | active (15.04%) | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK1 | inactive (96.67%) | - |
ALK2 | inactive (92.63%) | - |
ALK4 | inactive (99.83%) | inactive (115%) |
TGFbR1 | inactive (102.55%) | inactive (95%) |
TGFbR2 | inactive (98.07%) | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ARAF | inactive (96.48%) | - |
BRAF | inactive (92.68%) | - |
RAF1 | inactive (98.86%) | inactive (73%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IRAK1 | inactive (109.44%) | inactive (81%) |
IRAK4 | inactive (88.56%) | active (45%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LIMK1 | inactive (86.27%) | inactive (98%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LRRK2 | inactive (77.65%) | - |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MLK1 | active (37.76%) | active (10%) |
MLK2 | inactive (98.01%) | - |
MLK3 | active (40.19%) | - |
TAK1 | inactive (71.06%) | inactive (73%) |
ZAK | inactive (107.72%) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RIPK2 | inactive (88.09%) | inactive (91%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NuaK1 | inactive (71.07%) | inactive (84%) |
BRSK1 | inactive (100.31%) | inactive (95%) |
BRSK2 | inactive (97.78%) | inactive (122%) |
CHK1 | inactive (97.9%) | inactive (99%) |
LKB1 | inactive (84.44%) | inactive (99%) |
MARK1 | inactive (94.48%) | inactive (78%) |
MARK3 | inactive (96.55%) | - |
MARK4 | inactive (89.81%) | - |
MELK | inactive (69.45%) | inactive (66%) |
PASK | inactive (93.06%) | inactive (135%) |
QIK | inactive (92.21%) | - |
NuaK2 | inactive (133.94%) | - |
MARK2 | inactive (95.75%) | inactive (95%) |
AMPKa1 | - | inactive (92%) |
AMPKa2 | - | inactive (95%) |
SIK | - | inactive (85%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK1a | inactive (109.55%) | inactive (93%) |
CaMK1b | inactive (97.78%) | - |
CaMK1d | inactive (103.17%) | inactive (121%) |
CaMK1g | inactive (94.86%) | - |
CaMK4 | inactive (95.32%) | inactive (107%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK2a | inactive (101.38%) | - |
CaMK2b | inactive (94.32%) | inactive (95%) |
CaMK2d | inactive (101.75%) | inactive (99%) |
CaMK2g | inactive (96.85%) | inactive (100%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CHK2 | inactive (88.07%) | inactive (96%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DAPK1 | inactive (99.75%) | inactive (87%) |
DAPK2 | inactive (110.72%) | inactive (104%) |
DRAK1 | inactive (94.99%) | inactive (116%) |
DAPK3 | inactive (104.05%) | inactive (96%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DCLK2 | inactive (100.41%) | inactive (128%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAPKAPK2 | inactive (102.12%) | inactive (81%) |
MAPKAPK3 | inactive (85.4%) | inactive (124%) |
MAPKAPK5 | inactive (97.56%) | inactive (102%) |
MNK1 | inactive (79.82%) | - |
MNK2 | inactive (87.52%) | inactive (111%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
smMLCK | inactive (95.06%) | inactive (106%) |
skMLCK | inactive (97.05%) | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PHKg1 | inactive (89.87%) | - |
PHKg2 | inactive (116.71%) | inactive (122%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PIM1 | inactive (103.5%) | inactive (100%) |
PIM2 | inactive (104.82%) | inactive (116%) |
PIM3 | inactive (84.86%) | inactive (87%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKD1 | inactive (96.92%) | inactive (81%) |
PKD3 | inactive (95.48%) | - |
PKD2 | inactive (99.67%) | inactive (105%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TSSK1 | inactive (102.31%) | inactive (97%) |
TSSK2 | inactive (97.51%) | inactive (94%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
STK33 | inactive (74.37%) | inactive (89%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP3K5 | inactive (107.94%) | inactive (102%) |
MAP3K2 | inactive (97.77%) | - |
MAP3K3 | inactive (102.5%) | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
COT | inactive (101.26%) | - |
NIK | inactive (112.27%) | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GCK | inactive (97.59%) | inactive (75%) |
HGK | inactive (84.86%) | - |
KHS1 | inactive (97.51%) | - |
LOK | inactive (81.75%) | inactive (91%) |
MINK | inactive (98.64%) | inactive (103%) |
MST1 | inactive (87.69%) | inactive (63%) |
MST2 | inactive (90.77%) | inactive (104%) |
MST3 | inactive (80.79%) | inactive (58%) |
MST4 | inactive (100.13%) | - |
OSR1 | inactive (94.45%) | - |
PAK1 | inactive (92.77%) | - |
PAK2 | inactive (102.87%) | inactive (99%) |
PAK3 | inactive (94.17%) | inactive (100%) |
PAK4 | inactive (99.49%) | active (31%) |
PAK5 | inactive (76.8%) | active (50%) |
PAK6 | inactive (110.57%) | inactive (57%) |
SLK | inactive (73.1%) | - |
YSK1 | inactive (116.21%) | - |
STLK3 | inactive (99.21%) | - |
TAO1 | inactive (95.44%) | inactive (82%) |
TAO2 | inactive (91.29%) | inactive (98%) |
TAO3 | inactive (91.12%) | inactive (82%) |
MYO3B | inactive (94.2%) | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP2K1 | inactive (95.96%) | inactive (111%) |
MAP2K2 | inactive (103.67%) | - |
MAP2K6 | inactive (104.87%) | inactive (97%) |
MAP2K7 | - | inactive (75%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AurA | inactive (80.61%) | inactive (111%) |
AurB | inactive (96.98%) | inactive (72%) |
AurC | inactive (93.19%) | inactive (96%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMKK1 | inactive (101.26%) | - |
CaMKK2 | inactive (70.91%) | - |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Haspin | inactive (93.59%) | inactive (100%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IKKa | inactive (105.98%) | inactive (114%) |
IKKb | inactive (106.93%) | inactive (116%) |
IKKe | inactive (99.24%) | - |
TBK1 | inactive (93.03%) | inactive (90%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NEK1 | inactive (107.36%) | - |
NEK11 | inactive (67.12%) | inactive (59%) |
NEK2 | inactive (101.76%) | inactive (90%) |
NEK4 | inactive (94.35%) | - |
NEK6 | inactive (91.25%) | inactive (117%) |
NEK7 | inactive (100.57%) | inactive (102%) |
NEK9 | inactive (93.07%) | - |
NEK3 | inactive (94.24%) | inactive (84%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PBK | inactive (101.79%) | - |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PLK1 | inactive (89.21%) | inactive (75%) |
PLK2 | inactive (101.82%) | inactive (101%) |
PLK3 | inactive (86.39%) | inactive (99%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SgK496 | inactive (104.54%) | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MPSK1 | inactive (102.26%) | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TTK | inactive (115.51%) | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ULK1 | inactive (67.46%) | - |
ULK2 | inactive (97.68%) | inactive (83%) |
ULK3 | inactive (59.62%) | active (39%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wee1 | inactive (82.56%) | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wnk2 | inactive (92.38%) | inactive (91%) |
Wnk3 | inactive (89.13%) | inactive (82%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TLK2 | inactive (94.66%) | inactive (100%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK1 | 7 | 6 | 4 |
VRK | 3 | 1 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK1d | inactive (92.15%) | inactive (74%) |
CK1g1 | active (28.02%) | active (10%) |
CK1g2 | active (32.37%) | active (22%) |
CK1g3 | active (17.33%) | inactive (72%) |
CK1a | inactive (91.76%) | - |
CK1e | inactive (87.34%) | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
VRK1 | inactive (99.48%) | - |
VRK2 | - | inactive (85%) |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK2 | 3 | 2 | 2 |
CLK | 4 | 4 | 2 |
DYRK | 10 | 9 | 4 |
MAPK | 14 | 10 | 10 |
GSK | 2 | 2 | 2 |
SRPK | 3 | 3 | 3 |
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK2a1 | inactive (100.59%) | inactive (99%) |
CK2a2 | inactive (93.2%) | inactive (110%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CLK1 | inactive (67.54%) | - |
CLK2 | active (21.89%) | active (8%) |
CLK3 | inactive (89.75%) | inactive (55%) |
CLK4 | inactive (50.89%) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DYRK1A | inactive (65.36%) | - |
DYRK1B | active (49.92%) | - |
DYRK2 | inactive (98.38%) | inactive (99%) |
DYRK3 | inactive (104.82%) | - |
DYRK4 | inactive (91.2%) | - |
HIPK1 | inactive (103.13%) | inactive (97%) |
HIPK2 | inactive (86.29%) | inactive (88%) |
HIPK3 | inactive (102.2%) | inactive (101%) |
HIPK4 | inactive (88.69%) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Erk1 | inactive (103.85%) | inactive (98%) |
Erk2 | inactive (86.74%) | inactive (102%) |
JNK3 | inactive (96.68%) | inactive (102%) |
NLK | inactive (99.23%) | inactive (100%) |
p38a | inactive (99.44%) | inactive (88%) |
p38b | inactive (109.17%) | inactive (101%) |
p38d | inactive (122.11%) | inactive (108%) |
p38g | inactive (105.89%) | inactive (109%) |
JNK1 | inactive (98.97%) | inactive (103%) |
JNK2 | inactive (101.74%) | inactive (90%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GSK3A | inactive (108.29%) | inactive (104%) |
GSK3B | inactive (103.03%) | inactive (134%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSSK1 | inactive (70.4%) | inactive (73%) |
SRPK1 | inactive (77.02%) | inactive (52%) |
SRPK2 | inactive (53.56%) | active (32%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
PDHK | 5 | 1 | - |
Alpha | 6 | - | 1 |
PIKK | 6 | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDHK1 | inactive (91.6%) | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
eEF2K | - | inactive (109%) |
Atypical - PIKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FRAP | - | inactive (101%) |