Compound Information
Test on : RBC, Metz
Compound Name
RBC, Metz : Dovitinib
Inchikey
Same : PIQCTGMSNWUMAF-N
RBC, Metz : PIQCTGMSNWUMAF-UHFFFAOYSA-N
ChemSpider
RBC, Metz : 11530944
Pubchem CID
RBC, Metz : 135398510
ChEMBL
RBC, Metz : CHEMBL522892
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Metz |
---|
PDK1 | inactive (87.98%) | active (1000nM) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Metz |
---|
AKT1 | inactive (98.49%) | inactive (>7943.28nM) |
AKT2 | inactive (108.64%) | inactive (>7943.28nM) |
AKT3 | inactive (88.04%) | - |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
DMPK1 | inactive (107.34%) | - |
MRCKa | inactive (97.02%) | inactive (>10000nM) |
MRCKb | inactive (99.16%) | - |
ROCK1 | inactive (100.36%) | inactive (>1584.89nM) |
ROCK2 | inactive (79.34%) | inactive (3981.07nM) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
BARK1 | inactive (98.13%) | - |
BARK2 | inactive (97.48%) | - |
GPRK4 | inactive (94.16%) | - |
GPRK5 | inactive (106.94%) | inactive (>3981.07nM) |
GPRK6 | inactive (103.22%) | - |
GPRK7 | inactive (95.24%) | - |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
MSK1 | inactive (81.08%) | active (1000nM) |
MSK2 | inactive (72.07%) | - |
p70S6K | inactive (77.32%) | active (100nM) |
p70S6Kb | inactive (100.2%) | - |
RSK2 | active (34.34%) | active (316.23nM) |
RSK4 | active (16.12%) | - |
RSK1 | active (22.25%) | - |
RSK3 | active (13.05%) | - |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Metz |
---|
PKACg | inactive (118.71%) | - |
PRKX | inactive (103.97%) | inactive (1584.89nM) |
PKACa | inactive (101.03%) | inactive (>3162.28nM) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Metz |
---|
PKCa | inactive (83.83%) | - |
PKCd | inactive (90.91%) | inactive (1995.26nM) |
PKCe | inactive (101.04%) | - |
PKCh | inactive (103.06%) | - |
PKCg | inactive (86.91%) | inactive (>7943.28nM) |
PKCi | inactive (104.62%) | - |
PKCt | inactive (97.57%) | inactive (>2511.89nM) |
PKCz | inactive (80.99%) | inactive (>7943.28nM) |
PKCb | inactive (92.02%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Metz |
---|
PKG2 | inactive (99.03%) | inactive (>1584.89nM) |
PKG1 | inactive (81.18%) | inactive (>1995.26nM) |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Metz |
---|
PKN1 | active (15.54%) | - |
PKN2 | inactive (98.53%) | active (630.96nM) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
SGK1 | inactive (88.24%) | inactive (1258.93nM) |
SGK2 | inactive (89.84%) | - |
SGK3 | inactive (98.42%) | - |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Metz |
---|
NDR1 | inactive (97.05%) | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Metz |
---|
ABL1 | active (24.01%) | active (100nM) |
ABL2 | active (24.26%) | - |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Metz |
---|
ACK | inactive (83.12%) | inactive (>3981.07nM) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
ALK | inactive (80.51%) | active (630.96nM) |
LTK | inactive (92.48%) | inactive (>1995.26nM) |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Metz |
---|
AXL | active (44.35%) | active (251.19nM) |
MER | inactive (91.95%) | - |
TYRO3 | active (23.77%) | active (50.12nM) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Metz |
---|
BLK | active (12.26%) | active (12.59nM) |
BRK | inactive (96.39%) | - |
SRC | active (15.98%) | active (63.1nM) |
FGR | active (6.34%) | - |
FRK | inactive (56.05%) | - |
FYN | active (22.51%) | active (63.1nM) |
HCK | active (29.94%) | active (158.49nM) |
LCK | active (4.75%) | active (19.95nM) |
SRM | inactive (94.42%) | - |
YES | active (6.3%) | - |
LYN | active (9.15%) | active (63.1nM) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Metz |
---|
BMX | inactive (70.11%) | - |
BTK | active (37.34%) | inactive (1995.26nM) |
ITK | inactive (70.9%) | active (50.12nM) |
TEC | inactive (91.01%) | - |
TXK | inactive (75.1%) | - |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Metz |
---|
KIT | active (9.89%) | active (19.95nM) |
FLT3 | active (2.97%) | active (3.16nM) |
FMS | active (21.46%) | active (39.81nM) |
PDGFRb | active (17.23%) | active (6.31nM) |
PDGFRa | active (12.61%) | active (251.19nM) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Metz |
---|
CSK | inactive (88.36%) | - |
CTK | inactive (74.92%) | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Metz |
---|
DDR2 | inactive (195.15%) | - |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Metz |
---|
EGFR | inactive (97.24%) | inactive (>1995.26nM) |
ErbB2 | inactive (105.94%) | inactive (>1584.89nM) |
ErbB4 | inactive (95.22%) | inactive (>3981.07nM) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Metz |
---|
EphA1 | inactive (90.56%) | - |
EphA2 | inactive (76.87%) | inactive (>3162.28nM) |
EphA3 | inactive (88.05%) | - |
EphA4 | inactive (93.36%) | - |
EphA5 | inactive (99.11%) | - |
EphA6 | active (44.62%) | - |
EphA7 | inactive (76.54%) | - |
EphA8 | inactive (105.29%) | - |
EphB1 | inactive (58.15%) | - |
EphB2 | inactive (86.06%) | - |
EphB3 | inactive (51.93%) | - |
EphB4 | inactive (73.45%) | - |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
FAK | inactive (95.3%) | inactive (>3981.07nM) |
PYK2 | inactive (84.31%) | inactive (>1584.89nM) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Metz |
---|
FER | inactive (94.57%) | - |
FES | inactive (91.86%) | - |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Metz |
---|
FGFR1 | active (18.21%) | active (25.12nM) |
FGFR2 | active (21.99%) | - |
FGFR3 | active (12.39%) | active (39.81nM) |
FGFR4 | inactive (59.62%) | - |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Metz |
---|
FLT1 | active (26.24%) | active (39.81nM) |
FLT4 | active (11.3%) | active (100nM) |
KDR | active (31.47%) | active (19.95nM) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Metz |
---|
IGF1R | inactive (89.77%) | inactive (>1258.93nM) |
IRR | inactive (67.12%) | - |
INSR | inactive (84%) | inactive (1584.89nM) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Metz |
---|
JAK1 | inactive (92.06%) | - |
JAK2 | inactive (92.02%) | active (1000nM) |
JAK3 | inactive (83.88%) | inactive (>3162.28nM) |
TYK2 | inactive (59.4%) | active (199.53nM) |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Metz |
---|
MUSK | inactive (63.16%) | - |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Metz |
---|
RET | active (2.45%) | active (5.01nM) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Metz |
---|
RON | inactive (95.36%) | active (25.12nM) |
MET | inactive (84.4%) | inactive (>2511.89nM) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Metz |
---|
ROS | inactive (95.46%) | inactive (>3162.28nM) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Metz |
---|
SYK | inactive (65.37%) | - |
ZAP70 | inactive (107.35%) | - |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Metz |
---|
TIE2 | inactive (81.32%) | - |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Metz |
---|
TRKA | active (4.57%) | active (251.19nM) |
TRKB | active (5.72%) | active (100nM) |
TRKC | active (1.45%) | active (199.53nM) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Metz |
---|
ALK1 | inactive (125.16%) | - |
ALK2 | inactive (154.7%) | inactive (1258.93nM) |
ALK4 | inactive (98.78%) | - |
TGFbR1 | inactive (99.28%) | - |
TGFbR2 | inactive (108.68%) | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Metz |
---|
ARAF | inactive (122.99%) | - |
BRAF | inactive (104.9%) | - |
RAF1 | inactive (114.76%) | - |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
IRAK1 | inactive (65.08%) | inactive (1258.93nM) |
IRAK4 | active (31.76%) | inactive (>10000nM) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
LIMK1 | inactive (88.28%) | inactive (1995.26nM) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
LRRK2 | active (24.5%) | active (316.23nM) |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
MLK1 | inactive (52.42%) | - |
MLK2 | inactive (91.44%) | inactive (1584.89nM) |
MLK3 | active (26.36%) | - |
TAK1 | active (19.34%) | - |
ZAK | inactive (91.52%) | inactive (7943.28nM) |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
RIPK2 | inactive (92.98%) | - |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Metz |
---|
NuaK1 | active (3.13%) | - |
BRSK1 | inactive (59.8%) | active (398.11nM) |
BRSK2 | inactive (59.42%) | - |
CHK1 | active (30.81%) | active (158.49nM) |
LKB1 | inactive (103.58%) | - |
MARK1 | active (34.76%) | - |
MARK3 | active (36.5%) | active (125.89nM) |
MARK4 | active (25.51%) | active (100nM) |
MELK | active (7.72%) | active (31.62nM) |
PASK | inactive (104.74%) | inactive (>1584.89nM) |
QIK | active (25.46%) | active (100nM) |
NuaK2 | inactive (60.22%) | - |
MARK2 | active (47.44%) | active (125.89nM) |
AMPKa1 | - | active (79.43nM) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Metz |
---|
CaMK1a | inactive (85.77%) | inactive (>6309.57nM) |
CaMK1b | inactive (103.78%) | - |
CaMK1d | inactive (103.26%) | inactive (>1995.26nM) |
CaMK1g | inactive (100.36%) | - |
CaMK4 | inactive (91.72%) | - |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Metz |
---|
CaMK2a | inactive (53.95%) | inactive (>3162.28nM) |
CaMK2b | inactive (85.6%) | inactive (>7943.28nM) |
CaMK2d | inactive (56.88%) | active (316.23nM) |
CaMK2g | inactive (97.57%) | active (794.33nM) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Metz |
---|
CHK2 | inactive (84.45%) | inactive (1584.89nM) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
DAPK1 | inactive (107.67%) | - |
DAPK2 | inactive (82.29%) | - |
DRAK1 | inactive (67.98%) | - |
DAPK3 | inactive (108.71%) | inactive (>2511.89nM) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Metz |
---|
DCLK2 | inactive (94.11%) | - |
DCLK1 | - | inactive (>10000nM) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
MAPKAPK2 | inactive (96.89%) | inactive (>7943.28nM) |
MAPKAPK3 | inactive (99.31%) | inactive (>10000nM) |
MAPKAPK5 | inactive (93.86%) | inactive (>1584.89nM) |
MNK1 | inactive (88.74%) | - |
MNK2 | inactive (89.62%) | inactive (>10000nM) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
smMLCK | inactive (76.57%) | - |
skMLCK | active (5.92%) | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
PHKg1 | active (30.38%) | - |
PHKg2 | inactive (87.64%) | active (1000nM) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Metz |
---|
PIM1 | inactive (99.19%) | inactive (>6309.57nM) |
PIM2 | inactive (114.1%) | inactive (1258.93nM) |
PIM3 | inactive (95.63%) | - |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Metz |
---|
PKD1 | inactive (69%) | - |
PKD3 | inactive (60.22%) | inactive (1258.93nM) |
PKD2 | inactive (66.2%) | inactive (1995.26nM) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
TSSK1 | inactive (54.43%) | active (501.19nM) |
TSSK2 | inactive (80.57%) | inactive (>1584.89nM) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Metz |
---|
STK33 | inactive (60.75%) | - |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Metz |
---|
MAP3K5 | inactive (98.45%) | - |
MAP3K2 | inactive (66.17%) | - |
MAP3K3 | active (46.49%) | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Metz |
---|
COT | inactive (106.9%) | - |
NIK | inactive (110.1%) | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Metz |
---|
GCK | active (49.39%) | active (630.96nM) |
HGK | active (2.96%) | active (25.12nM) |
KHS1 | active (3.26%) | active (31.62nM) |
LOK | active (41.57%) | - |
MINK | active (1.65%) | active (10nM) |
MST1 | active (10.01%) | - |
MST2 | active (34.36%) | active (199.53nM) |
MST3 | active (44.46%) | - |
MST4 | inactive (105.06%) | - |
OSR1 | inactive (98.72%) | - |
PAK1 | inactive (111.43%) | inactive (>10000nM) |
PAK2 | inactive (96.94%) | - |
PAK3 | inactive (103.38%) | - |
PAK4 | inactive (92.96%) | inactive (1995.26nM) |
PAK5 | inactive (82.71%) | - |
PAK6 | inactive (102.88%) | - |
SLK | inactive (68.06%) | active (199.53nM) |
YSK1 | inactive (86.03%) | - |
STLK3 | inactive (92.32%) | - |
TAO1 | inactive (98.35%) | inactive (>5011.87nM) |
TAO2 | inactive (97.4%) | - |
TAO3 | inactive (84.17%) | - |
MYO3B | inactive (79.68%) | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Metz |
---|
MAP2K1 | inactive (88.71%) | active (125.89nM) |
MAP2K2 | active (43.05%) | active (158.49nM) |
MAP2K6 | inactive (82.58%) | - |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Metz |
---|
AurA | inactive (60.63%) | inactive (>1000nM) |
AurB | active (26.95%) | active (79.43nM) |
AurC | inactive (82.35%) | - |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
CaMKK1 | active (48.51%) | - |
CaMKK2 | inactive (85.92%) | active (158.49nM) |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Metz |
---|
Haspin | inactive (75%) | - |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
IKKa | inactive (88.1%) | inactive (>3981.07nM) |
IKKb | inactive (87.77%) | inactive (>3162.28nM) |
IKKe | active (42.88%) | active (794.33nM) |
TBK1 | active (38.5%) | inactive (>1000nM) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
NEK1 | inactive (64.34%) | - |
NEK11 | inactive (93.59%) | - |
NEK2 | inactive (104.22%) | active (501.19nM) |
NEK4 | inactive (83.55%) | inactive (5011.87nM) |
NEK6 | inactive (84.47%) | - |
NEK7 | inactive (91.08%) | - |
NEK9 | inactive (58.87%) | - |
NEK3 | inactive (88.15%) | - |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
PBK | inactive (101.36%) | inactive (>10000nM) |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
PLK1 | inactive (96.87%) | inactive (>7943.28nM) |
PLK2 | inactive (101.84%) | - |
PLK3 | inactive (100.99%) | inactive (>7943.28nM) |
PLK4 | - | inactive (1258.93nM) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Metz |
---|
SgK496 | inactive (98.38%) | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
MPSK1 | active (46.26%) | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
TTK | inactive (101.89%) | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
ULK1 | active (20.43%) | - |
ULK2 | active (45.68%) | - |
ULK3 | inactive (65.97%) | - |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Metz |
---|
Wee1 | inactive (92.02%) | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
Wnk2 | inactive (99.88%) | - |
Wnk3 | inactive (96.07%) | - |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
TLK2 | inactive (89.33%) | - |
Other - CDC7
Bioactivity |
---|
Kinase | RBC | Metz |
---|
CDC7 | - | inactive (>1258.93nM) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz |
---|
CK1 | 7 | 6 | 5 |
VRK | 3 | 1 | - |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Metz |
---|
CK1d | inactive (79.3%) | inactive (1584.89nM) |
CK1g1 | inactive (96.43%) | inactive (>6309.57nM) |
CK1g2 | inactive (91.36%) | inactive (>7943.28nM) |
CK1g3 | inactive (94.63%) | - |
CK1a | inactive (95.11%) | inactive (>5011.87nM) |
CK1e | inactive (94.09%) | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
VRK1 | inactive (98.51%) | - |
CMGC
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Metz |
---|
CK2a1 | inactive (113.54%) | inactive (>6309.57nM) |
CK2a2 | inactive (85.55%) | - |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
CLK1 | inactive (67.82%) | - |
CLK2 | active (38.61%) | active (794.33nM) |
CLK3 | inactive (103.88%) | - |
CLK4 | inactive (52.16%) | active (100nM) |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
DYRK1A | inactive (96.52%) | inactive (>2511.89nM) |
DYRK1B | inactive (87.95%) | inactive (>2511.89nM) |
DYRK2 | inactive (104.6%) | - |
DYRK3 | inactive (103.37%) | inactive (>6309.57nM) |
DYRK4 | inactive (98.15%) | - |
HIPK1 | inactive (95.71%) | - |
HIPK2 | inactive (81.48%) | inactive (>3162.28nM) |
HIPK3 | inactive (95.61%) | - |
HIPK4 | inactive (96.29%) | inactive (>7943.28nM) |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
Erk1 | inactive (99.62%) | - |
Erk2 | inactive (82.39%) | inactive (>7943.28nM) |
JNK3 | inactive (107.94%) | active (630.96nM) |
NLK | inactive (110.18%) | - |
p38a | inactive (94%) | inactive (>3981.07nM) |
p38b | inactive (103.75%) | - |
p38d | inactive (90.42%) | inactive (>7943.28nM) |
p38g | inactive (100.84%) | inactive (>6309.57nM) |
JNK1 | inactive (105.64%) | inactive (3162.28nM) |
JNK2 | inactive (108.97%) | inactive (>3981.07nM) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
GSK3A | inactive (100.04%) | inactive (>5011.87nM) |
GSK3B | inactive (98.56%) | inactive (>3162.28nM) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
MSSK1 | inactive (103.81%) | - |
SRPK1 | inactive (97.54%) | inactive (5011.87nM) |
SRPK2 | inactive (99.93%) | - |
CMGC - CDK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
CDC2 | - | inactive (>7943.28nM) |
CDK2 | - | inactive (>7943.28nM) |
CDK5 | - | inactive (>3981.07nM) |
CDK8 | - | inactive (>3981.07nM) |
CDK7 | - | active (251.19nM) |
CDK9 | - | inactive (>1584.89nM) |
CDK11 | - | - |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz |
---|
PDHK | 5 | 1 | - |
Alpha | 6 | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Metz |
---|
PDHK1 | inactive (87.98%) | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Metz |
---|
eEF2K | - | inactive (>3981.07nM) |