Compound Information
Test on : RBC
Compound Name : JNK Inhibitor II, Negative Control
Inchikey : ODZGYELAMAOARP-UHFFFAOYSA-N
ChemSpider : 9840563
Pubchem CID : 11665831
ChEMBL : CHEMBL1802485
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC |
---|
PDK1 | inactive (94.54%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC |
---|
AKT1 | inactive (99.08%) |
AKT2 | inactive (98.92%) |
AKT3 | inactive (102.1%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC |
---|
DMPK1 | inactive (107.03%) |
MRCKa | inactive (106.27%) |
MRCKb | inactive (97.97%) |
ROCK1 | inactive (98.43%) |
ROCK2 | inactive (92.33%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC |
---|
BARK1 | inactive (102.94%) |
BARK2 | inactive (93.57%) |
GPRK4 | inactive (104.58%) |
GPRK5 | inactive (93.8%) |
GPRK6 | inactive (89.22%) |
GPRK7 | inactive (113.04%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC |
---|
MSK1 | inactive (100.29%) |
MSK2 | inactive (104.51%) |
p70S6K | inactive (96.32%) |
p70S6Kb | inactive (94.71%) |
RSK2 | inactive (97.31%) |
RSK4 | inactive (90.42%) |
RSK1 | inactive (93.71%) |
RSK3 | inactive (93.51%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC |
---|
PKACg | inactive (107.5%) |
PRKX | inactive (100.55%) |
PKACa | inactive (103.63%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC |
---|
PKCa | inactive (96.08%) |
PKCd | inactive (92.33%) |
PKCe | inactive (95.67%) |
PKCh | inactive (94.34%) |
PKCg | inactive (90.6%) |
PKCi | inactive (98.49%) |
PKCt | inactive (105.66%) |
PKCz | inactive (97.94%) |
PKCb | inactive (97.75%) |
AGC - PKG
Bioactivity |
---|
Kinase | RBC |
---|
PKG2 | inactive (105.39%) |
PKG1 | inactive (95.98%) |
AGC - PKN
Bioactivity |
---|
Kinase | RBC |
---|
PKN1 | inactive (100.85%) |
PKN2 | inactive (97.27%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC |
---|
SGK1 | inactive (94.85%) |
SGK2 | inactive (98.93%) |
SGK3 | inactive (107.17%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC |
---|
NDR1 | inactive (98.55%) |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC |
---|
ABL1 | inactive (99.09%) |
ABL2 | inactive (97.83%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC |
---|
ACK | inactive (83.32%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC |
---|
ALK | inactive (87.44%) |
LTK | inactive (86.69%) |
TK - Axl
Bioactivity |
---|
Kinase | RBC |
---|
AXL | inactive (104.18%) |
MER | inactive (95.85%) |
TYRO3 | inactive (99.76%) |
TK - Src
Bioactivity |
---|
Kinase | RBC |
---|
BLK | inactive (106.26%) |
BRK | inactive (91.82%) |
SRC | inactive (90.66%) |
FGR | inactive (93.42%) |
FRK | inactive (94.26%) |
FYN | inactive (93.83%) |
HCK | inactive (94.57%) |
LCK | inactive (99.22%) |
SRM | inactive (104.29%) |
YES | inactive (94.45%) |
LYN | inactive (96.1%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC |
---|
BMX | inactive (101.14%) |
BTK | inactive (89.49%) |
ITK | inactive (88.26%) |
TEC | inactive (101.94%) |
TXK | inactive (91.98%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC |
---|
KIT | inactive (86.44%) |
FLT3 | inactive (59.28%) |
FMS | inactive (96.96%) |
PDGFRb | inactive (100.5%) |
PDGFRa | inactive (97.58%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC |
---|
CSK | inactive (88.72%) |
CTK | inactive (87.98%) |
TK - DDR
Bioactivity |
---|
Kinase | RBC |
---|
DDR2 | inactive (95.1%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC |
---|
EGFR | inactive (104.98%) |
ErbB2 | inactive (96.9%) |
ErbB4 | inactive (94.29%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC |
---|
EphA1 | inactive (94.79%) |
EphA2 | inactive (104.14%) |
EphA3 | inactive (93.48%) |
EphA4 | inactive (103.71%) |
EphA5 | inactive (126.4%) |
EphA6 | inactive (87.61%) |
EphA7 | inactive (104.01%) |
EphA8 | inactive (99.37%) |
EphB1 | inactive (94.61%) |
EphB2 | inactive (103.66%) |
EphB3 | inactive (85.51%) |
EphB4 | inactive (99.95%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC |
---|
FAK | inactive (92.75%) |
PYK2 | inactive (101.82%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC |
---|
FER | inactive (99.25%) |
FES | inactive (94.4%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC |
---|
FGFR1 | inactive (99.48%) |
FGFR2 | inactive (105.09%) |
FGFR3 | inactive (95.9%) |
FGFR4 | inactive (108.36%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC |
---|
FLT1 | inactive (84.32%) |
FLT4 | inactive (86.83%) |
KDR | inactive (101.05%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC |
---|
IGF1R | inactive (95.94%) |
IRR | inactive (82.71%) |
INSR | inactive (99.5%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC |
---|
JAK1 | inactive (109.85%) |
JAK2 | inactive (95.93%) |
JAK3 | inactive (107.42%) |
TYK2 | inactive (89.36%) |
TK - Musk
Bioactivity |
---|
Kinase | RBC |
---|
MUSK | inactive (88.35%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC |
---|
RET | inactive (83.83%) |
TK - Met
Bioactivity |
---|
Kinase | RBC |
---|
RON | inactive (96.73%) |
MET | inactive (106.84%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC |
---|
ROS | inactive (104.47%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC |
---|
SYK | inactive (94.78%) |
ZAP70 | inactive (95.11%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC |
---|
TIE2 | inactive (98.22%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC |
---|
TRKA | inactive (95.05%) |
TRKB | inactive (84.02%) |
TRKC | inactive (71.58%) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC |
---|
ALK1 | inactive (102.33%) |
ALK2 | inactive (110.08%) |
ALK4 | inactive (101.53%) |
TGFbR1 | inactive (93.67%) |
TGFbR2 | inactive (94.87%) |
TKL - RAF
Bioactivity |
---|
Kinase | RBC |
---|
ARAF | inactive (105.69%) |
BRAF | inactive (96.07%) |
RAF1 | inactive (87.03%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC |
---|
IRAK1 | inactive (99.57%) |
IRAK4 | inactive (97.26%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC |
---|
LIMK1 | inactive (97.06%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC |
---|
LRRK2 | inactive (55.86%) |
TKL - MLK
Bioactivity |
---|
Kinase | RBC |
---|
MLK1 | inactive (99.41%) |
MLK2 | inactive (91.41%) |
MLK3 | inactive (97.23%) |
TAK1 | inactive (83.95%) |
ZAK | inactive (83.1%) |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC |
---|
RIPK2 | inactive (75.74%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC |
---|
NuaK1 | active (46.21%) |
BRSK1 | inactive (92.51%) |
BRSK2 | inactive (96.4%) |
CHK1 | inactive (93.74%) |
LKB1 | inactive (87.71%) |
MARK1 | inactive (95.75%) |
MARK3 | inactive (96.56%) |
MARK4 | inactive (91.08%) |
MELK | inactive (83.57%) |
PASK | inactive (94.58%) |
QIK | inactive (100.2%) |
NuaK2 | inactive (85.74%) |
MARK2 | inactive (94.06%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC |
---|
CaMK1a | inactive (103.97%) |
CaMK1b | inactive (100.98%) |
CaMK1d | inactive (70.34%) |
CaMK1g | inactive (95.52%) |
CaMK4 | inactive (100.43%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC |
---|
CaMK2a | inactive (105.74%) |
CaMK2b | inactive (95.26%) |
CaMK2d | inactive (90.03%) |
CaMK2g | inactive (109.12%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC |
---|
CHK2 | inactive (89.79%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC |
---|
DAPK1 | inactive (86.38%) |
DAPK2 | inactive (104.35%) |
DRAK1 | inactive (83.68%) |
DAPK3 | inactive (101.97%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC |
---|
DCLK2 | inactive (94.22%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC |
---|
MAPKAPK2 | inactive (101.64%) |
MAPKAPK3 | inactive (103.75%) |
MAPKAPK5 | inactive (94.54%) |
MNK1 | inactive (105.34%) |
MNK2 | inactive (94.07%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC |
---|
smMLCK | inactive (77.39%) |
skMLCK | inactive (78.84%) |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC |
---|
PHKg1 | inactive (86.44%) |
PHKg2 | inactive (95.42%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC |
---|
PIM1 | inactive (80.34%) |
PIM2 | inactive (105.06%) |
PIM3 | inactive (76.78%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC |
---|
PKD1 | inactive (69.26%) |
PKD3 | inactive (65.48%) |
PKD2 | inactive (76.96%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC |
---|
TSSK1 | inactive (98.38%) |
TSSK2 | inactive (95.39%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC |
---|
STK33 | inactive (81.27%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC |
---|
MAP3K5 | inactive (93.05%) |
MAP3K2 | inactive (102.61%) |
MAP3K3 | inactive (94.4%) |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC |
---|
COT | inactive (94.34%) |
NIK | inactive (107.16%) |
STE - STE20
Bioactivity |
---|
Kinase | RBC |
---|
GCK | inactive (75.38%) |
HGK | inactive (85.08%) |
KHS1 | inactive (86.03%) |
LOK | inactive (94.54%) |
MINK | inactive (92.32%) |
MST1 | inactive (78.86%) |
MST2 | inactive (88.37%) |
MST3 | inactive (98.58%) |
MST4 | inactive (107.89%) |
OSR1 | inactive (101.8%) |
PAK1 | inactive (98.54%) |
PAK2 | inactive (102.2%) |
PAK3 | inactive (101.03%) |
PAK4 | inactive (90.43%) |
PAK5 | inactive (102.17%) |
PAK6 | inactive (98.63%) |
SLK | inactive (103.29%) |
YSK1 | inactive (96.49%) |
STLK3 | inactive (101.13%) |
TAO1 | inactive (100.13%) |
TAO2 | inactive (104.17%) |
TAO3 | inactive (87.62%) |
MYO3B | inactive (97.74%) |
STE - STE7
Bioactivity |
---|
Kinase | RBC |
---|
MAP2K1 | inactive (86.29%) |
MAP2K2 | inactive (102.15%) |
MAP2K6 | inactive (96.36%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC |
---|
AurA | inactive (89.4%) |
AurB | inactive (83.55%) |
AurC | inactive (89.3%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC |
---|
CaMKK1 | inactive (102.41%) |
CaMKK2 | inactive (74.92%) |
Other - Haspin
Bioactivity |
---|
Kinase | RBC |
---|
Haspin | inactive (53.11%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC |
---|
IKKa | inactive (96.98%) |
IKKb | inactive (102.99%) |
IKKe | inactive (92.34%) |
TBK1 | inactive (88.76%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC |
---|
NEK1 | inactive (78.3%) |
NEK11 | inactive (104.7%) |
NEK2 | inactive (88.24%) |
NEK4 | inactive (89.8%) |
NEK6 | inactive (108.39%) |
NEK7 | inactive (93.11%) |
NEK9 | inactive (96.64%) |
NEK3 | inactive (96.66%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC |
---|
PBK | inactive (107.83%) |
Other - PLK
Bioactivity |
---|
Kinase | RBC |
---|
PLK1 | inactive (96.98%) |
PLK2 | inactive (93.48%) |
PLK3 | inactive (96.16%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC |
---|
SgK496 | inactive (101.23%) |
Other - NAK
Bioactivity |
---|
Kinase | RBC |
---|
MPSK1 | inactive (83.28%) |
Other - TTK
Bioactivity |
---|
Kinase | RBC |
---|
TTK | inactive (77.69%) |
Other - ULK
Bioactivity |
---|
Kinase | RBC |
---|
ULK1 | inactive (101.46%) |
ULK2 | inactive (108.89%) |
ULK3 | inactive (94.9%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC |
---|
Wee1 | inactive (92.35%) |
Other - WNK
Bioactivity |
---|
Kinase | RBC |
---|
Wnk2 | inactive (103.95%) |
Wnk3 | inactive (91.97%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC |
---|
TLK2 | inactive (100.78%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
CK1 | 7 | 6 |
VRK | 3 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC |
---|
CK1d | active (20.78%) |
CK1g1 | inactive (102.3%) |
CK1g2 | inactive (91.55%) |
CK1g3 | inactive (81.44%) |
CK1a | active (47.78%) |
CK1e | active (34.34%) |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC |
---|
VRK1 | inactive (84.12%) |
CMGC
CMGC - CK2
Bioactivity |
---|
Kinase | RBC |
---|
CK2a1 | inactive (90.25%) |
CK2a2 | inactive (86.63%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC |
---|
CLK1 | inactive (92.71%) |
CLK2 | inactive (94.45%) |
CLK3 | inactive (98.54%) |
CLK4 | inactive (69.82%) |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC |
---|
DYRK1A | inactive (94.13%) |
DYRK1B | inactive (93.06%) |
DYRK2 | inactive (99.45%) |
DYRK3 | inactive (128.7%) |
DYRK4 | inactive (91.2%) |
HIPK1 | inactive (111.81%) |
HIPK2 | inactive (104.84%) |
HIPK3 | inactive (113.03%) |
HIPK4 | inactive (102.34%) |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC |
---|
Erk1 | inactive (98.93%) |
Erk2 | inactive (91.75%) |
JNK3 | inactive (97.31%) |
NLK | inactive (100.5%) |
p38a | inactive (93.64%) |
p38b | inactive (108.79%) |
p38d | inactive (106.26%) |
p38g | inactive (93.77%) |
JNK1 | inactive (87.23%) |
JNK2 | inactive (85.25%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC |
---|
GSK3A | inactive (91.11%) |
GSK3B | inactive (94.01%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC |
---|
MSSK1 | inactive (96.27%) |
SRPK1 | inactive (99.68%) |
SRPK2 | inactive (97.23%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
PDHK | 5 | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC |
---|
PDHK1 | inactive (94.54%) |