Compound Information
Test on : DRx, RBC, Metz, Millipore, GPCR
Compound Name
DRx, RBC, Metz, Millipore, GPCR : GW2580
Inchikey
Same : MYQAUKPBNJWPIE-N
DRx, RBC, Metz, Millipore, GPCR : MYQAUKPBNJWPIE-UHFFFAOYSA-N
ChemSpider
DRx, RBC, Metz, Millipore, GPCR : 9792308
Pubchem CID
DRx, RBC, Metz, Millipore, GPCR : 11617559
ChEMBL
DRx, RBC, Metz, Millipore, GPCR : CHEMBL261849
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
Other
Other - NAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
AAK1 | inactive (10001nM) | - | - | - | - |
BIKE | inactive (10001nM) | - | - | - | - |
GAK | inactive (10001nM) | - | - | - | - |
MPSK1 | inactive (10001nM) | inactive (106.22%) | - | - | - |
Other - Aur
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
AurA | inactive (10001nM) | inactive (104.91%) | inactive (>1584.89nM) | inactive (108%) | inactive (2.3%) |
AurB | inactive (10001nM) | inactive (103.66%) | inactive (>3981.07nM) | inactive (110%) | inactive (4.95%) |
AurC | inactive (10001nM) | inactive (97.55%) | - | inactive (90%) | inactive (16.16%) |
Other - CAMKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
CaMKK1 | inactive (10001nM) | inactive (115.36%) | - | - | - |
CaMKK2 | inactive (10001nM) | inactive (102.6%) | - | - | - |
Other - PEK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
HRI | inactive (10001nM) | - | - | - | - |
PKR | inactive (10001nM) | - | - | - | - |
Other - IRE
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
IRE1 | inactive (10001nM) | - | - | - | - |
Other - IKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
IKKa | inactive (10001nM) | inactive (94.72%) | - | inactive (114%) | inactive (-7.71%) |
IKKb | inactive (10001nM) | inactive (99.87%) | - | inactive (109%) | inactive (-1.34%) |
IKKe | inactive (10001nM) | inactive (96.75%) | inactive (>3162.28nM) | - | inactive (-2.21%) |
TBK1 | inactive (10001nM) | inactive (102.72%) | inactive (>3162.28nM) | inactive (61%) | inactive (2.86%) |
Other - NEK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
NEK1 | inactive (10001nM) | inactive (95.61%) | - | - | inactive (1.56%) |
NEK11 | inactive (10001nM) | inactive (102.92%) | - | inactive (110%) | - |
NEK2 | inactive (10001nM) | inactive (99.2%) | - | inactive (77%) | inactive (-1.4%) |
NEK3 | inactive (10001nM) | inactive (98.07%) | - | inactive (105%) | - |
NEK4 | inactive (10001nM) | inactive (92.24%) | - | - | - |
NEK5 | inactive (10001nM) | - | - | - | - |
NEK6 | inactive (10001nM) | inactive (99.42%) | - | inactive (97%) | inactive (-3.71%) |
NEK7 | inactive (10001nM) | inactive (100.37%) | - | inactive (96%) | inactive (1.75%) |
NEK9 | inactive (10001nM) | inactive (93.33%) | - | - | inactive (-4.1%) |
Other - WEE
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
MYT1 | inactive (10001nM) | - | - | - | - |
Wee1 | inactive (10001nM) | inactive (90.33%) | - | - | - |
Wee1B | inactive (10001nM) | - | - | - | - |
Other - PLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
PLK1 | inactive (10001nM) | inactive (97.1%) | - | inactive (80%) | inactive (3.71%) |
PLK2 | inactive (10001nM) | inactive (115.91%) | - | inactive (98%) | - |
PLK3 | inactive (10001nM) | inactive (95.91%) | - | inactive (83%) | - |
PLK4 | inactive (10001nM) | - | - | - | - |
Other - SgK496
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
SgK496 | inactive (10001nM) | inactive (94.96%) | - | - | - |
Other - NKF1
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
SBK | inactive (10001nM) | - | - | - | - |
SgK110 | inactive (10001nM) | - | - | - | - |
Other - NKF4
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
CLIK1 | inactive (10001nM) | - | - | - | - |
Other - ULK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
Fused | inactive (10001nM) | - | - | - | - |
ULK1 | inactive (10001nM) | inactive (99.68%) | - | - | - |
ULK2 | inactive (10001nM) | inactive (105.43%) | - | inactive (99%) | - |
ULK3 | inactive (10001nM) | active (0%) | - | inactive (99%) | - |
Other - TLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
TLK1 | inactive (10001nM) | - | - | - | - |
TLK2 | inactive (10001nM) | active (0%) | - | inactive (96%) | - |
Other - TTK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
TTK | inactive (10001nM) | inactive (105.27%) | - | - | inactive (3.14%) |
Other - Haspin
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
Haspin | - | inactive (97.75%) | - | inactive (92%) | - |
Other - TOPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
PBK | - | inactive (99.39%) | - | - | - |
Other - WNK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
Wnk2 | - | inactive (94.6%) | - | inactive (106%) | - |
Wnk3 | - | inactive (100.44%) | - | inactive (108%) | - |
Other - CDC7
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
CDC7 | - | - | - | - | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
ABL1 | inactive (10001nM) | inactive (101.84%) | inactive (>3981.07nM) | inactive (93%) | inactive (7.34%) |
ABL2 | inactive (10001nM) | inactive (106.95%) | - | inactive (113%) | inactive (5.98%) |
TK - ALK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
ALK | inactive (10001nM) | inactive (97.36%) | inactive (>6309.57nM) | inactive (74%) | inactive (0.01%) |
LTK | inactive (10001nM) | inactive (100.44%) | inactive (>2511.89nM) | - | inactive (-0.41%) |
TK - Axl
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
AXL | inactive (10001nM) | inactive (96.45%) | - | inactive (80%) | inactive (8.25%) |
MER | inactive (10001nM) | inactive (90.25%) | - | inactive (108%) | inactive (3.48%) |
TYRO3 | inactive (10001nM) | inactive (109.93%) | inactive (>3162.28nM) | inactive (86%) | inactive (0.77%) |
TK - Src
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
BLK | inactive (10001nM) | inactive (98.61%) | - | inactive (107%) | inactive (0.47%) |
BRK | inactive (10001nM) | inactive (96.13%) | - | inactive (109%) | inactive (-1.6%) |
FGR | inactive (10001nM) | inactive (92.3%) | - | inactive (101%) | inactive (4.25%) |
FRK | inactive (10001nM) | inactive (101.56%) | - | inactive (102%) | inactive (2.07%) |
FYN | inactive (10001nM) | inactive (102.15%) | inactive (>6309.57nM) | inactive (92%) | inactive (1.28%) |
HCK | inactive (10001nM) | inactive (101.72%) | - | inactive (88%) | inactive (3.12%) |
LCK | inactive (10001nM) | inactive (96.31%) | inactive (>6309.57nM) | inactive (110%) | inactive (2.78%) |
LYN | inactive (10001nM) | inactive (99.94%) | - | inactive (104%) | - |
SRC | inactive (10001nM) | inactive (97.85%) | - | inactive (84%) | inactive (1.97%) |
SRM | inactive (10001nM) | inactive (95.94%) | - | - | inactive (1.88%) |
YES | inactive (10001nM) | inactive (94.8%) | - | inactive (104%) | inactive (-3.3%) |
TK - Tec
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
BMX | inactive (10001nM) | inactive (93.42%) | - | inactive (86%) | inactive (2.06%) |
BTK | inactive (10001nM) | inactive (104.37%) | inactive (>6309.57nM) | inactive (103%) | inactive (3.61%) |
ITK | inactive (10001nM) | inactive (98.14%) | - | inactive (100%) | inactive (2.31%) |
TEC | inactive (10001nM) | inactive (113.91%) | - | - | inactive (2.91%) |
TXK | inactive (10001nM) | inactive (101%) | - | inactive (83%) | inactive (4.97%) |
TK - PDGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
FMS | active (2.2nM) | active (19.3%) | active (39.81nM) | active (1%) | active (95.81%) |
FLT3 | inactive (10001nM) | inactive (102.71%) | inactive (>3162.28nM) | inactive (96%) | inactive (1.13%) |
KIT | inactive (10001nM) | inactive (105.76%) | - | inactive (107%) | inactive (7.39%) |
PDGFRa | inactive (10001nM) | inactive (99.43%) | inactive (>2511.89nM) | inactive (107%) | inactive (15.65%) |
PDGFRb | inactive (10001nM) | inactive (98.2%) | inactive (>1995.26nM) | inactive (106%) | inactive (10.01%) |
TK - Csk
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
CSK | inactive (10001nM) | inactive (101.18%) | - | inactive (105%) | inactive (-3.17%) |
CTK | inactive (10001nM) | inactive (94.84%) | - | - | - |
TK - DDR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
DDR1 | inactive (10001nM) | - | - | - | - |
DDR2 | inactive (10001nM) | inactive (99.57%) | - | inactive (112%) | inactive (8.13%) |
TK - EGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
EGFR | inactive (10001nM) | inactive (96.86%) | - | inactive (112%) | inactive (5.41%) |
ErbB2 | inactive (10001nM) | inactive (105.63%) | - | - | inactive (-2.79%) |
ErbB3 | inactive (10001nM) | - | - | - | - |
ErbB4 | inactive (10001nM) | inactive (109.79%) | - | inactive (99%) | inactive (3.43%) |
TK - Eph
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
EphA1 | inactive (10001nM) | inactive (85.75%) | - | inactive (96%) | - |
EphA2 | inactive (10001nM) | inactive (107.42%) | - | inactive (110%) | inactive (2.74%) |
EphA3 | inactive (10001nM) | inactive (109.36%) | - | inactive (108%) | inactive (0.08%) |
EphA4 | inactive (10001nM) | inactive (104.75%) | - | inactive (108%) | inactive (-0.14%) |
EphA5 | inactive (10001nM) | inactive (110.75%) | - | inactive (111%) | - |
EphA6 | inactive (10001nM) | - | - | - | - |
EphA7 | inactive (10001nM) | inactive (100.59%) | - | inactive (91%) | - |
EphA8 | inactive (10001nM) | inactive (98.05%) | - | inactive (93%) | - |
EphB1 | inactive (10001nM) | inactive (102.56%) | - | inactive (97%) | - |
EphB2 | inactive (10001nM) | inactive (87.4%) | - | inactive (108%) | inactive (8.3%) |
EphB3 | inactive (10001nM) | inactive (91.84%) | - | inactive (114%) | inactive (-4.82%) |
EphB4 | inactive (10001nM) | inactive (90.52%) | - | inactive (99%) | inactive (3.27%) |
EphB6 | inactive (10001nM) | - | - | - | - |
TK - FAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
FAK | inactive (10001nM) | inactive (95.46%) | inactive (>6309.57nM) | inactive (115%) | - |
PYK2 | inactive (10001nM) | inactive (86.06%) | - | inactive (103%) | inactive (-2.43%) |
TK - Fer
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
FER | inactive (10001nM) | inactive (93.36%) | - | inactive (107%) | inactive (2.33%) |
FES | inactive (10001nM) | - | - | inactive (94%) | inactive (2.24%) |
TK - FGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
FGFR1 | inactive (10001nM) | inactive (107.65%) | inactive (>3981.07nM) | inactive (112%) | inactive (2.1%) |
FGFR2 | inactive (10001nM) | inactive (101.66%) | - | inactive (112%) | inactive (6.83%) |
FGFR3 | inactive (10001nM) | inactive (105.01%) | - | inactive (108%) | inactive (0.98%) |
FGFR4 | inactive (10001nM) | inactive (99.66%) | - | inactive (131%) | inactive (3.16%) |
TK - VEGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
FLT1 | inactive (10001nM) | inactive (99.66%) | inactive (>3981.07nM) | inactive (94%) | inactive (2.11%) |
FLT4 | inactive (10001nM) | inactive (105.08%) | - | inactive (95%) | inactive (-0.86%) |
KDR | inactive (10001nM) | inactive (109.1%) | inactive (>2511.89nM) | inactive (97%) | inactive (9.65%) |
TK - InsR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
IGF1R | inactive (10001nM) | inactive (122.76%) | inactive (>2511.89nM) | inactive (128%) | inactive (-0.91%) |
INSR | inactive (10001nM) | inactive (97.04%) | - | inactive (102%) | inactive (-1%) |
IRR | inactive (10001nM) | inactive (99.37%) | - | inactive (137%) | inactive (-0.57%) |
TK - JakA
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
JAK1 | inactive (10001nM) | inactive (105.07%) | - | - | inactive (-0.05%) |
JAK2 | inactive (10001nM) | inactive (89.19%) | inactive (>2511.89nM) | inactive (101%) | inactive (4.19%) |
JAK3 | inactive (10001nM) | inactive (95.93%) | inactive (>5011.87nM) | inactive (105%) | inactive (3.61%) |
TYK2 | inactive (10001nM) | inactive (97.62%) | - | - | inactive (0.26%) |
TK - Met
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
MET | inactive (10001nM) | inactive (76.12%) | inactive (>2511.89nM) | inactive (109%) | inactive (5.98%) |
RON | inactive (10001nM) | inactive (103.86%) | inactive (>3981.07nM) | inactive (87%) | inactive (5.55%) |
TK - Musk
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
MUSK | inactive (10001nM) | inactive (102.07%) | - | inactive (92%) | inactive (9.52%) |
TK - Ret
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
RET | inactive (10001nM) | inactive (107.79%) | inactive (>3162.28nM) | inactive (92%) | inactive (9.77%) |
TK - Sev
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
ROS | inactive (10001nM) | inactive (99.85%) | - | inactive (81%) | inactive (4.98%) |
TK - Syk
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
SYK | inactive (10001nM) | inactive (88.99%) | - | inactive (118%) | inactive (0.65%) |
ZAP70 | inactive (10001nM) | inactive (94.33%) | - | inactive (93%) | inactive (4.05%) |
TK - Tie
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
TIE1 | inactive (10001nM) | - | - | - | - |
TIE2 | inactive (10001nM) | inactive (101.07%) | - | inactive (90%) | inactive (8.78%) |
TK - Ack
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
TNK1 | inactive (10001nM) | - | - | - | inactive (-8.3%) |
ACK | inactive (10001nM) | inactive (105.22%) | inactive (>3981.07nM) | inactive (79%) | inactive (3.64%) |
TK - Trk
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
TRKA | active (630nM) | inactive (51.33%) | inactive (1584.89nM) | active (49%) | inactive (49.99%) |
TRKB | active (36nM) | active (31.23%) | active (158.49nM) | inactive (55%) | active (75.4%) |
TRKC | active (120nM) | active (17.7%) | active (316.23nM) | - | active (72.72%) |
TKL
TKL
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
STKR | 12 | 10 | 5 | 1 | 2 | - |
RIPK | 5 | 4 | 1 | - | 1 | - |
RAF | 5 | 2 | 3 | 1 | 1 | 1 |
MLK | 10 | 8 | 5 | 2 | 2 | - |
IRAK | 4 | 3 | 2 | 2 | 2 | 1 |
LISK | 4 | 3 | 1 | 1 | 1 | - |
LRRK | 2 | 1 | 1 | 1 | - | - |
TKL - STKR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
ALK2 | inactive (10001nM) | inactive (100.04%) | inactive (>3981.07nM) | - | - |
ALK4 | inactive (10001nM) | inactive (97.82%) | - | inactive (120%) | - |
ACTR2 | inactive (10001nM) | - | - | - | - |
ACTR2B | inactive (10001nM) | - | - | - | - |
ALK1 | inactive (10001nM) | inactive (100.56%) | - | - | - |
BMPR1A | inactive (10001nM) | - | - | - | - |
BMPR1B | inactive (10001nM) | - | - | - | - |
BMPR2 | inactive (10001nM) | - | - | - | - |
TGFbR1 | inactive (10001nM) | inactive (97.03%) | - | inactive (79%) | - |
TGFbR2 | inactive (10001nM) | inactive (126.76%) | - | - | - |
TKL - RIPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
SgK288 | inactive (10001nM) | - | - | - | - |
RIPK1 | inactive (10001nM) | - | - | - | - |
RIPK2 | inactive (10001nM) | inactive (81.95%) | - | inactive (83%) | - |
ANKRD3 | inactive (10001nM) | - | - | - | - |
TKL - RAF
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
BRAF | inactive (10001nM) | inactive (98.96%) | - | - | inactive (-0.42%) |
RAF1 | inactive (10001nM) | inactive (97.03%) | - | inactive (86%) | - |
ARAF | - | inactive (96.55%) | - | - | - |
TKL - MLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
DLK | inactive (10001nM) | - | - | - | - |
LZK | inactive (10001nM) | - | - | - | - |
MLK1 | inactive (10001nM) | inactive (104.62%) | - | inactive (91%) | - |
MLK2 | inactive (10001nM) | inactive (96.37%) | - | - | - |
MLK3 | inactive (10001nM) | inactive (100.55%) | - | - | - |
TAK1 | inactive (10001nM) | inactive (97.94%) | - | inactive (88%) | - |
HH498 | inactive (10001nM) | - | - | - | - |
ZAK | inactive (10001nM) | inactive (97.41%) | - | - | - |
TKL - IRAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
IRAK1 | inactive (10001nM) | inactive (122.69%) | - | inactive (76%) | - |
IRAK3 | inactive (10001nM) | - | - | - | - |
IRAK4 | inactive (10001nM) | inactive (109.57%) | - | inactive (106%) | inactive (0.89%) |
TKL - LISK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
LIMK1 | inactive (10001nM) | inactive (94.49%) | - | inactive (93%) | - |
LIMK2 | inactive (10001nM) | - | - | - | - |
TESK1 | inactive (10001nM) | - | - | - | - |
TKL - LRRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
LRRK2 | inactive (10001nM) | inactive (92.62%) | inactive (>2511.89nM) | - | - |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
ABC1 | 5 | 2 | - | - | - | - |
PIKK | 6 | 1 | - | - | 1 | - |
RIO | 3 | 3 | - | - | - | - |
Alpha | 6 | 1 | - | 1 | 1 | - |
PDHK | 5 | - | 1 | - | - | - |
Atypical - ABC1
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
ADCK3 | inactive (10001nM) | - | - | - | - |
ADCK4 | inactive (10001nM) | - | - | - | - |
Atypical - PIKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
FRAP | inactive (10001nM) | - | - | inactive (116%) | - |
Atypical - RIO
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
RIOK1 | inactive (10001nM) | - | - | - | - |
RIOK2 | inactive (10001nM) | - | - | - | - |
RIOK3 | inactive (10001nM) | - | - | - | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
ChaK2 | inactive (10001nM) | - | - | - | - |
eEF2K | - | - | - | inactive (92%) | - |
Atypical - PDHK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
PDHK1 | - | inactive (89.44%) | - | - | - |
AGC
AGC - Akt
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
AKT1 | inactive (10001nM) | inactive (97.39%) | - | inactive (106%) | inactive (-0.15%) |
AKT2 | inactive (10001nM) | inactive (102.47%) | - | inactive (88%) | inactive (-0.17%) |
AKT3 | inactive (10001nM) | inactive (96.52%) | - | inactive (98%) | inactive (0.93%) |
AGC - DMPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
CRIK | inactive (10001nM) | - | - | - | - |
DMPK1 | inactive (10001nM) | inactive (101.27%) | - | inactive (115%) | - |
DMPK2 | inactive (10001nM) | - | - | - | - |
MRCKa | inactive (10001nM) | inactive (94.45%) | - | inactive (102%) | inactive (-0.63%) |
MRCKb | inactive (10001nM) | inactive (96.93%) | - | inactive (91%) | inactive (3.93%) |
ROCK1 | inactive (10001nM) | inactive (100.07%) | inactive (>3981.07nM) | inactive (112%) | inactive (2.94%) |
ROCK2 | inactive (10001nM) | inactive (84.13%) | - | inactive (88%) | inactive (-1.22%) |
AGC - GRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
RHOK | inactive (10001nM) | - | - | - | - |
GPRK4 | inactive (10001nM) | inactive (106%) | - | - | - |
GPRK7 | inactive (10001nM) | inactive (103.77%) | - | inactive (88%) | inactive (-7.03%) |
BARK1 | - | inactive (96.08%) | - | - | - |
BARK2 | - | inactive (103.15%) | - | - | - |
GPRK5 | - | inactive (108.55%) | inactive (>3981.07nM) | inactive (83%) | - |
GPRK6 | - | inactive (99.76%) | - | inactive (95%) | inactive (-5.27%) |
AGC - NDR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
LATS1 | inactive (10001nM) | - | - | - | - |
LATS2 | inactive (10001nM) | - | - | - | - |
NDR1 | inactive (10001nM) | active (0%) | - | - | - |
NDR2 | inactive (10001nM) | - | - | - | - |
AGC - MAST
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
MAST1 | inactive (10001nM) | - | - | - | - |
AGC - PDK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
PDK1 | inactive (10001nM) | inactive (89.44%) | - | inactive (104%) | inactive (2.38%) |
AGC - PKA
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
PKACa | inactive (10001nM) | inactive (104.38%) | inactive (>1258.93nM) | inactive (108%) | - |
PKACb | inactive (10001nM) | - | - | - | - |
PRKX | inactive (10001nM) | inactive (104.5%) | inactive (>3162.28nM) | inactive (98%) | inactive (1.07%) |
PKACg | - | - | - | - | - |
AGC - PKN
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
PKN1 | inactive (10001nM) | inactive (101.02%) | - | - | - |
PKN2 | inactive (10001nM) | inactive (90.9%) | - | inactive (99%) | - |
AGC - PKC
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
PKCd | inactive (10001nM) | inactive (87.82%) | - | inactive (98%) | - |
PKCe | inactive (10001nM) | inactive (95.66%) | - | inactive (89%) | - |
PKCh | inactive (10001nM) | inactive (88.56%) | - | inactive (96%) | inactive (-0.03%) |
PKCi | inactive (10001nM) | inactive (91.58%) | - | inactive (97%) | inactive (2.56%) |
PKCt | inactive (10001nM) | inactive (97.97%) | inactive (>2511.89nM) | inactive (88%) | inactive (-0.58%) |
PKCa | - | inactive (95.9%) | - | inactive (103%) | inactive (1.13%) |
PKCg | - | inactive (101.71%) | - | inactive (103%) | inactive (0.23%) |
PKCz | - | inactive (93.37%) | - | inactive (101%) | - |
PKCb | - | inactive (109.6%) | - | - | - |
AGC - PKG
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
PKG1 | inactive (10001nM) | inactive (98.33%) | - | - | inactive (3.2%) |
PKG2 | inactive (10001nM) | inactive (103.91%) | - | - | inactive (3.2%) |
AGC - RSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
p70S6K | inactive (10001nM) | inactive (89.46%) | - | inactive (80%) | inactive (0.73%) |
MSK1 | - | inactive (103.15%) | - | inactive (131%) | inactive (5.97%) |
MSK2 | - | inactive (107.09%) | - | inactive (91%) | inactive (1.84%) |
p70S6Kb | - | inactive (100.3%) | - | - | - |
RSK2 | - | inactive (104.9%) | inactive (>3981.07nM) | inactive (64%) | inactive (-0.8%) |
RSK4 | - | inactive (100.52%) | - | inactive (110%) | inactive (-0.61%) |
RSK1 | - | inactive (92.69%) | - | inactive (94%) | inactive (-1.81%) |
RSK3 | - | inactive (104.93%) | - | inactive (131%) | inactive (-1%) |
AGC - SGK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
SGK3 | inactive (10001nM) | inactive (105.06%) | - | inactive (87%) | inactive (1.28%) |
SGK1 | - | inactive (97.88%) | - | inactive (105%) | inactive (1.31%) |
SGK2 | - | inactive (97.54%) | - | inactive (108%) | inactive (3%) |
AGC - YANK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
YANK1 | inactive (10001nM) | - | - | - | - |
YANK2 | inactive (10001nM) | - | - | - | - |
YANK3 | inactive (10001nM) | - | - | - | - |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
AMPKa1 | inactive (10001nM) | - | inactive (>3162.28nM) | inactive (90%) | inactive (-0.28%) |
AMPKa2 | inactive (10001nM) | - | - | inactive (94%) | inactive (2.37%) |
NuaK1 | inactive (10001nM) | inactive (106.25%) | - | inactive (91%) | inactive (3.71%) |
BRSK1 | inactive (10001nM) | inactive (95.59%) | - | inactive (89%) | inactive (3.19%) |
BRSK2 | inactive (10001nM) | inactive (96.78%) | - | inactive (99%) | inactive (2.49%) |
CHK1 | inactive (10001nM) | inactive (106.75%) | - | inactive (91%) | inactive (7.23%) |
HUNK | inactive (10001nM) | - | - | - | - |
LKB1 | inactive (10001nM) | inactive (103.19%) | - | inactive (106%) | - |
MARK1 | inactive (10001nM) | inactive (103.3%) | - | inactive (80%) | inactive (0.09%) |
MARK2 | inactive (10001nM) | inactive (105.58%) | - | inactive (106%) | - |
MARK3 | inactive (10001nM) | inactive (103.12%) | - | - | inactive (2.06%) |
MARK4 | inactive (10001nM) | inactive (89.74%) | - | - | inactive (1.47%) |
MELK | inactive (10001nM) | inactive (101.85%) | - | inactive (89%) | inactive (-1.43%) |
NIM1 | inactive (10001nM) | - | - | - | - |
QSK | inactive (10001nM) | - | - | - | - |
SIK | inactive (10001nM) | - | - | inactive (86%) | inactive (2.92%) |
QIK | inactive (10001nM) | inactive (98.58%) | - | - | inactive (-1.07%) |
NuaK2 | inactive (10001nM) | inactive (98.12%) | - | - | - |
SNRK | inactive (10001nM) | - | - | - | - |
PASK | - | inactive (102.98%) | - | inactive (79%) | inactive (0.54%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
CaMK1a | inactive (10001nM) | inactive (102.78%) | - | inactive (105%) | - |
CaMK1d | inactive (10001nM) | inactive (93.02%) | inactive (>2511.89nM) | inactive (103%) | inactive (5.51%) |
CaMK1g | inactive (10001nM) | inactive (98.28%) | - | - | - |
CaMK4 | inactive (10001nM) | inactive (94.66%) | - | inactive (130%) | inactive (3.54%) |
CaMK1b | - | inactive (98.44%) | - | - | - |
CAMK - CAMK2
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
CaMK2a | inactive (10001nM) | inactive (104.73%) | inactive (>7943.28nM) | - | inactive (5.8%) |
CaMK2b | inactive (10001nM) | inactive (100.21%) | - | inactive (91%) | - |
CaMK2d | inactive (10001nM) | inactive (109.11%) | - | inactive (101%) | inactive (2.5%) |
CaMK2g | inactive (10001nM) | inactive (94.36%) | - | inactive (97%) | - |
CAMK - CASK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
CASK | inactive (10001nM) | - | - | - | - |
CAMK - RAD53
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
CHK2 | inactive (10001nM) | inactive (106.71%) | - | inactive (97%) | inactive (4.77%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
DAPK1 | inactive (10001nM) | inactive (101.52%) | - | inactive (94%) | inactive (9.42%) |
DAPK2 | inactive (10001nM) | inactive (95.26%) | - | inactive (106%) | - |
DAPK3 | inactive (10001nM) | inactive (104.3%) | inactive (>5011.87nM) | inactive (96%) | - |
DRAK1 | inactive (10001nM) | inactive (102.41%) | - | inactive (112%) | - |
DRAK2 | inactive (10001nM) | - | - | - | - |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
DCLK1 | inactive (10001nM) | - | - | - | - |
DCLK2 | inactive (10001nM) | inactive (101.19%) | - | inactive (105%) | inactive (8.82%) |
DCLK3 | inactive (10001nM) | - | - | - | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
MAPKAPK2 | inactive (10001nM) | inactive (102.73%) | - | inactive (84%) | inactive (3.22%) |
MAPKAPK5 | inactive (10001nM) | inactive (87.52%) | - | inactive (81%) | inactive (-1.74%) |
MNK1 | inactive (10001nM) | inactive (113.09%) | - | - | inactive (0.82%) |
MNK2 | inactive (10001nM) | inactive (90.59%) | - | inactive (108%) | inactive (0.25%) |
MAPKAPK3 | - | inactive (95.97%) | - | inactive (125%) | inactive (7.43%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
caMLCK | inactive (10001nM) | - | - | - | - |
smMLCK | inactive (10001nM) | inactive (95.68%) | - | inactive (83%) | - |
skMLCK | inactive (10001nM) | inactive (104.21%) | - | - | - |
SgK085 | inactive (10001nM) | - | - | - | - |
CAMK - PHK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
PHKg1 | inactive (10001nM) | inactive (95.29%) | - | - | inactive (1.56%) |
PHKg2 | inactive (10001nM) | inactive (105.6%) | - | inactive (91%) | inactive (-1.66%) |
CAMK - PIM
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
PIM1 | inactive (10001nM) | inactive (103.56%) | inactive (>6309.57nM) | inactive (97%) | inactive (0.49%) |
PIM2 | inactive (10001nM) | inactive (107.01%) | - | inactive (96%) | inactive (3.29%) |
PIM3 | inactive (10001nM) | inactive (95.86%) | - | inactive (90%) | inactive (0.23%) |
CAMK - PKD
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
PKD1 | inactive (10001nM) | inactive (95.21%) | - | inactive (81%) | inactive (2.03%) |
PKD2 | inactive (10001nM) | inactive (99.4%) | - | inactive (101%) | inactive (4.2%) |
PKD3 | inactive (10001nM) | inactive (97.11%) | inactive (>3981.07nM) | - | inactive (2.56%) |
CAMK - STK33
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
STK33 | inactive (10001nM) | inactive (96.37%) | - | inactive (108%) | - |
CAMK - TSSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
TSSK1 | inactive (10001nM) | inactive (95.22%) | - | inactive (91%) | inactive (-1.27%) |
TSSK2 | - | inactive (109.38%) | - | inactive (93%) | inactive (-0.65%) |
STE
STE
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
STE11 | 8 | 8 | 3 | - | 1 | - |
STE20 | 31 | 27 | 23 | 9 | 14 | 12 |
STE7 | 7 | 7 | 3 | 2 | 3 | 1 |
STE-Unique | 2 | - | 2 | - | - | - |
STE - STE11
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
MAP3K5 | inactive (10001nM) | inactive (89%) | - | inactive (85%) | - |
MAP3K6 | inactive (10001nM) | - | - | - | - |
MAP3K1 | inactive (10001nM) | - | - | - | - |
MAP3K7 | inactive (10001nM) | - | - | - | - |
MAP3K2 | inactive (10001nM) | inactive (108.43%) | - | - | - |
MAP3K3 | inactive (10001nM) | inactive (97.78%) | - | - | - |
MAP3K4 | inactive (10001nM) | - | - | - | - |
MAP3K8 | inactive (10001nM) | - | - | - | - |
STE - STE20
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
HPK1 | inactive (10001nM) | - | - | - | - |
LOK | inactive (10001nM) | inactive (100.03%) | - | inactive (88%) | inactive (7.31%) |
GCK | inactive (10001nM) | inactive (119.84%) | inactive (>2511.89nM) | inactive (83%) | inactive (3.99%) |
KHS2 | inactive (10001nM) | - | - | - | - |
HGK | inactive (10001nM) | inactive (98.97%) | inactive (>5011.87nM) | - | inactive (6.03%) |
KHS1 | inactive (10001nM) | inactive (97.43%) | - | - | - |
MINK | inactive (10001nM) | inactive (86.53%) | - | inactive (84%) | inactive (4.81%) |
MST1 | inactive (10001nM) | inactive (106.11%) | - | inactive (93%) | inactive (4.23%) |
MST2 | inactive (10001nM) | inactive (98.38%) | - | inactive (105%) | inactive (3.04%) |
MST3 | inactive (10001nM) | inactive (93.55%) | - | inactive (61%) | - |
MST4 | inactive (10001nM) | inactive (95.52%) | - | - | inactive (0.63%) |
MYO3A | inactive (10001nM) | - | - | - | - |
MYO3B | inactive (10001nM) | active (0%) | - | - | - |
OSR1 | inactive (10001nM) | inactive (103.2%) | - | - | - |
PAK1 | inactive (10001nM) | inactive (93.36%) | - | - | inactive (5.79%) |
PAK2 | inactive (10001nM) | inactive (95.27%) | - | inactive (98%) | inactive (0.32%) |
PAK3 | inactive (10001nM) | inactive (101.66%) | - | inactive (73%) | inactive (1.06%) |
PAK4 | inactive (10001nM) | inactive (101.39%) | inactive (>5011.87nM) | inactive (99%) | - |
PAK6 | inactive (10001nM) | inactive (94.86%) | - | inactive (112%) | inactive (-2.29%) |
PAK5 | inactive (10001nM) | inactive (102.83%) | - | inactive (86%) | inactive (7.84%) |
SLK | inactive (10001nM) | inactive (97.74%) | - | - | - |
STLK3 | inactive (10001nM) | inactive (87.58%) | - | - | - |
TAO1 | inactive (10001nM) | inactive (109.59%) | inactive (>6309.57nM) | inactive (95%) | - |
TAO2 | inactive (10001nM) | inactive (94.74%) | - | inactive (100%) | - |
TAO3 | inactive (10001nM) | inactive (102.2%) | - | inactive (95%) | - |
TNIK | inactive (10001nM) | - | - | - | - |
YSK1 | inactive (10001nM) | inactive (96.95%) | - | - | - |
STE - STE7
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
MAP2K1 | inactive (10001nM) | inactive (98.64%) | inactive (>3162.28nM) | inactive (100%) | inactive (0.97%) |
MAP2K2 | inactive (10001nM) | inactive (101.23%) | inactive (>3981.07nM) | - | - |
MAP2K3 | inactive (10001nM) | - | - | - | - |
MAP2K4 | inactive (10001nM) | - | - | - | - |
MAP2K5 | inactive (10001nM) | - | - | - | - |
MAP2K6 | inactive (10001nM) | inactive (87.4%) | - | inactive (78%) | - |
MAP2K7 | inactive (10001nM) | - | - | inactive (113%) | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
COT | - | inactive (98.35%) | - | - | - |
NIK | - | inactive (81.77%) | - | - | - |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
CDK | 20 | 8 | - | 7 | - | - |
CDKL | 5 | 4 | - | - | - | - |
CLK | 4 | 4 | 4 | 2 | 2 | 2 |
CK2 | 3 | 2 | 2 | 1 | 2 | 1 |
DYRK | 10 | 8 | 9 | 6 | 4 | 5 |
MAPK | 14 | 14 | 10 | 8 | 10 | 6 |
GSK | 2 | 2 | 2 | 2 | 2 | 2 |
RCK | 3 | 2 | - | - | - | - |
SRPK | 3 | 3 | 3 | 1 | 3 | 2 |
CMGC - CDK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
PITSLRE | inactive (10001nM) | - | - | - | - |
CHED | inactive (10001nM) | - | - | - | - |
CDK11 | inactive (10001nM) | - | - | - | - |
PCTAIRE1 | inactive (10001nM) | - | - | - | - |
PCTAIRE2 | inactive (10001nM) | - | - | - | - |
PCTAIRE3 | inactive (10001nM) | - | - | - | - |
PFTAIRE2 | inactive (10001nM) | - | - | - | - |
PFTAIRE1 | inactive (10001nM) | - | - | - | - |
CDC2 | - | - | - | - | - |
CDK2 | - | - | - | - | - |
CDK5 | - | - | inactive (>3162.28nM) | - | - |
CDK8 | - | - | inactive (>3981.07nM) | - | - |
CDK7 | - | - | inactive (>3981.07nM) | - | - |
CDK9 | - | - | inactive (>1584.89nM) | - | - |
CMGC - CDKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
CDKL1 | inactive (10001nM) | - | - | - | - |
CDKL2 | inactive (10001nM) | - | - | - | - |
CDKL3 | inactive (10001nM) | - | - | - | - |
CDKL5 | inactive (10001nM) | - | - | - | - |
CMGC - CLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
CLK1 | inactive (10001nM) | inactive (102.63%) | - | - | - |
CLK2 | inactive (10001nM) | inactive (94.33%) | inactive (>3981.07nM) | inactive (108%) | inactive (1.66%) |
CLK3 | inactive (10001nM) | inactive (98.34%) | - | inactive (86%) | inactive (-0.53%) |
CLK4 | inactive (10001nM) | inactive (86.5%) | inactive (>2511.89nM) | - | - |
CMGC - CK2
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
CK2a1 | inactive (10001nM) | inactive (104.85%) | - | inactive (86%) | inactive (-8.59%) |
CK2a2 | inactive (10001nM) | inactive (97.35%) | - | inactive (110%) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
DYRK1A | inactive (10001nM) | inactive (88.12%) | inactive (>1995.26nM) | - | inactive (0.52%) |
DYRK1B | inactive (10001nM) | inactive (104.29%) | inactive (>2511.89nM) | - | inactive (2.57%) |
DYRK2 | inactive (10001nM) | inactive (104.62%) | - | inactive (97%) | inactive (0.42%) |
HIPK1 | inactive (10001nM) | inactive (109.76%) | - | inactive (107%) | inactive (0.13%) |
HIPK2 | inactive (10001nM) | inactive (102.6%) | - | inactive (100%) | - |
HIPK3 | inactive (10001nM) | inactive (102.19%) | - | inactive (92%) | - |
HIPK4 | inactive (10001nM) | inactive (97.69%) | - | - | inactive (4.49%) |
PRP4 | inactive (10001nM) | - | - | - | - |
DYRK3 | - | inactive (108.33%) | - | - | - |
DYRK4 | - | inactive (101.36%) | - | - | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
Erk1 | inactive (10001nM) | inactive (99.11%) | - | inactive (100%) | inactive (0.29%) |
Erk2 | inactive (10001nM) | inactive (109.54%) | - | inactive (102%) | inactive (-0.13%) |
Erk3 | inactive (10001nM) | - | - | - | - |
Erk4 | inactive (10001nM) | - | - | - | - |
Erk5 | inactive (10001nM) | - | - | - | - |
Erk7 | inactive (10001nM) | - | - | - | - |
JNK1 | inactive (10001nM) | inactive (91.91%) | inactive (>5011.87nM) | inactive (101%) | - |
JNK2 | inactive (10001nM) | inactive (106.24%) | inactive (>3981.07nM) | inactive (105%) | inactive (0.51%) |
JNK3 | inactive (10001nM) | inactive (84.42%) | - | inactive (89%) | - |
NLK | inactive (10001nM) | inactive (105.31%) | - | inactive (97%) | - |
p38a | inactive (10001nM) | inactive (106.22%) | inactive (>3981.07nM) | inactive (84%) | inactive (4.45%) |
p38b | inactive (10001nM) | inactive (98.68%) | - | inactive (95%) | inactive (1%) |
p38d | inactive (10001nM) | inactive (96.04%) | - | inactive (111%) | inactive (0.37%) |
p38g | inactive (10001nM) | inactive (101.82%) | - | inactive (88%) | - |
CMGC - GSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
GSK3A | inactive (10001nM) | inactive (108.17%) | inactive (>3981.07nM) | inactive (120%) | inactive (0.34%) |
GSK3B | inactive (10001nM) | inactive (97.76%) | inactive (>3981.07nM) | inactive (106%) | inactive (0.94%) |
CMGC - RCK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
ICK | inactive (10001nM) | - | - | - | - |
MAK | inactive (10001nM) | - | - | - | - |
CMGC - SRPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
SRPK1 | inactive (10001nM) | inactive (90.37%) | - | inactive (99%) | inactive (-2.52%) |
SRPK2 | inactive (10001nM) | inactive (87.44%) | - | inactive (91%) | - |
MSSK1 | inactive (10001nM) | inactive (102.33%) | - | inactive (111%) | inactive (0.79%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
CK1 | 7 | 7 | 6 | 5 | 4 | 4 |
VRK | 3 | 1 | 1 | - | 1 | - |
CK1 - CK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
CK1a | inactive (10001nM) | inactive (97.93%) | inactive (>3981.07nM) | - | inactive (0.48%) |
CK1a2 | inactive (10001nM) | - | - | - | - |
CK1d | inactive (10001nM) | inactive (98.52%) | - | inactive (88%) | - |
CK1e | inactive (10001nM) | inactive (97.08%) | - | - | - |
CK1g1 | inactive (10001nM) | inactive (92.7%) | - | inactive (103%) | inactive (-0.45%) |
CK1g2 | inactive (10001nM) | inactive (100.57%) | - | inactive (89%) | inactive (0.05%) |
CK1g3 | inactive (10001nM) | inactive (102.62%) | - | inactive (103%) | inactive (0.85%) |
CK1 - VRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore | GPCR |
---|
VRK2 | inactive (10001nM) | - | - | inactive (92%) | - |
VRK1 | - | inactive (91.39%) | - | - | - |