Compound Information
Test on : RBC, Millipore
Compound Name
RBC, Millipore : 3-(4-Pyridyl)indole
Inchikey
Same : LLJRXVHJOJRCSM-N
RBC, Millipore : LLJRXVHJOJRCSM-UHFFFAOYSA-N
ChemSpider
RBC, Millipore : 559358
Pubchem CID
RBC, Millipore : 644354
ChEMBL
RBC, Millipore : CHEMBL380071
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDK1 | inactive (96.57%) | inactive (111%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AKT1 | inactive (100.35%) | inactive (103%) |
AKT2 | inactive (96.36%) | inactive (121%) |
AKT3 | inactive (101.18%) | inactive (89%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DMPK1 | inactive (108.53%) | inactive (147%) |
MRCKa | inactive (99.88%) | inactive (113%) |
MRCKb | inactive (103.84%) | inactive (94%) |
ROCK1 | inactive (84.16%) | inactive (114%) |
ROCK2 | inactive (71.86%) | active (37%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BARK1 | inactive (97.73%) | - |
BARK2 | inactive (95.37%) | - |
GPRK4 | inactive (94.9%) | - |
GPRK5 | inactive (99.24%) | inactive (98%) |
GPRK6 | inactive (103.35%) | inactive (87%) |
GPRK7 | inactive (98.37%) | inactive (96%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSK1 | inactive (96.73%) | inactive (115%) |
MSK2 | inactive (90.99%) | inactive (80%) |
p70S6K | inactive (79.94%) | inactive (53%) |
p70S6Kb | inactive (97.81%) | - |
RSK2 | inactive (97.35%) | inactive (72%) |
RSK4 | inactive (111.79%) | inactive (89%) |
RSK1 | inactive (93.82%) | inactive (98%) |
RSK3 | inactive (88.96%) | inactive (117%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKACg | inactive (107.09%) | - |
PRKX | inactive (54.25%) | active (48%) |
PKACa | inactive (91.61%) | inactive (93%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKCa | inactive (97.4%) | inactive (98%) |
PKCd | inactive (83.22%) | inactive (63%) |
PKCe | inactive (81.5%) | inactive (73%) |
PKCh | inactive (84.89%) | inactive (64%) |
PKCg | inactive (99.37%) | inactive (106%) |
PKCi | inactive (82.38%) | inactive (89%) |
PKCt | inactive (125.25%) | inactive (88%) |
PKCz | inactive (98.26%) | inactive (94%) |
PKCb | inactive (89.49%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKG2 | active (38.27%) | - |
PKG1 | inactive (64.81%) | - |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKN1 | inactive (66.4%) | - |
PKN2 | inactive (80.81%) | active (30%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SGK1 | inactive (93.77%) | inactive (102%) |
SGK2 | inactive (91.02%) | inactive (92%) |
SGK3 | inactive (92.82%) | inactive (101%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NDR1 | inactive (109.32%) | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ABL1 | inactive (98.8%) | inactive (98%) |
ABL2 | inactive (91.86%) | inactive (110%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ACK | inactive (96.15%) | inactive (80%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK | inactive (105.9%) | inactive (76%) |
LTK | inactive (102.77%) | - |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AXL | inactive (99.81%) | inactive (81%) |
MER | inactive (92.99%) | inactive (100%) |
TYRO3 | inactive (98.14%) | inactive (91%) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BLK | inactive (99.59%) | inactive (125%) |
BRK | inactive (85.51%) | inactive (95%) |
SRC | inactive (99.97%) | inactive (80%) |
FGR | inactive (94.53%) | inactive (117%) |
FRK | inactive (105.56%) | inactive (88%) |
FYN | inactive (98.69%) | inactive (89%) |
HCK | inactive (99.53%) | inactive (68%) |
LCK | inactive (101.94%) | inactive (102%) |
SRM | inactive (106.97%) | - |
YES | inactive (97.06%) | inactive (117%) |
LYN | inactive (101.55%) | inactive (105%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BMX | inactive (95.79%) | inactive (86%) |
BTK | inactive (103.68%) | inactive (99%) |
ITK | inactive (94.78%) | inactive (101%) |
TEC | inactive (122.8%) | - |
TXK | inactive (104.19%) | inactive (109%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
KIT | inactive (93.23%) | inactive (110%) |
FLT3 | inactive (91.51%) | inactive (107%) |
FMS | inactive (100.64%) | inactive (110%) |
PDGFRb | inactive (104.57%) | inactive (113%) |
PDGFRa | inactive (94.96%) | inactive (120%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CSK | inactive (106.57%) | inactive (114%) |
CTK | inactive (93.92%) | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DDR2 | inactive (92.57%) | inactive (129%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EGFR | inactive (97.34%) | inactive (125%) |
ErbB2 | inactive (95.64%) | - |
ErbB4 | inactive (83.68%) | inactive (88%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EphA1 | inactive (104.65%) | inactive (87%) |
EphA2 | inactive (105.74%) | inactive (104%) |
EphA3 | inactive (106.8%) | inactive (106%) |
EphA4 | inactive (107.56%) | inactive (109%) |
EphA5 | inactive (99.4%) | inactive (102%) |
EphA6 | inactive (103.94%) | - |
EphA7 | inactive (98.21%) | inactive (99%) |
EphA8 | inactive (100.67%) | inactive (96%) |
EphB1 | inactive (107.69%) | inactive (108%) |
EphB2 | inactive (114.42%) | inactive (108%) |
EphB3 | inactive (99.98%) | inactive (106%) |
EphB4 | inactive (89.72%) | inactive (111%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FAK | inactive (97.66%) | inactive (116%) |
PYK2 | inactive (95.35%) | inactive (127%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FER | inactive (91.59%) | inactive (109%) |
FES | inactive (104.57%) | inactive (111%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FGFR1 | inactive (92.72%) | inactive (121%) |
FGFR2 | inactive (104.71%) | inactive (111%) |
FGFR3 | inactive (98.91%) | inactive (123%) |
FGFR4 | inactive (84.58%) | inactive (112%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FLT1 | inactive (97.89%) | inactive (85%) |
FLT4 | inactive (118.69%) | inactive (91%) |
KDR | inactive (94.17%) | inactive (100%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IGF1R | inactive (104.59%) | inactive (121%) |
IRR | inactive (100.86%) | inactive (125%) |
INSR | inactive (90.5%) | inactive (110%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
JAK1 | inactive (109.24%) | - |
JAK2 | inactive (93.84%) | inactive (97%) |
JAK3 | inactive (95.27%) | inactive (103%) |
TYK2 | inactive (101.03%) | - |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MUSK | inactive (78.91%) | inactive (88%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RET | inactive (97.28%) | inactive (103%) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RON | inactive (98.95%) | inactive (96%) |
MET | inactive (91.39%) | inactive (117%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ROS | inactive (81.55%) | inactive (88%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SYK | inactive (98.6%) | inactive (118%) |
ZAP70 | inactive (105.27%) | inactive (94%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TIE2 | inactive (100.83%) | inactive (77%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TRKA | inactive (96.95%) | inactive (91%) |
TRKB | inactive (107.23%) | inactive (134%) |
TRKC | inactive (100.04%) | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK1 | inactive (100.45%) | - |
ALK2 | inactive (94.67%) | - |
ALK4 | inactive (98.8%) | inactive (127%) |
TGFbR1 | inactive (102.54%) | inactive (87%) |
TGFbR2 | inactive (118.62%) | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ARAF | inactive (97.72%) | - |
BRAF | inactive (94.03%) | - |
RAF1 | inactive (93.18%) | inactive (73%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IRAK1 | inactive (127.47%) | inactive (76%) |
IRAK4 | inactive (108.74%) | inactive (94%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LIMK1 | inactive (92.04%) | inactive (98%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LRRK2 | inactive (92.77%) | - |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MLK1 | inactive (83.31%) | inactive (74%) |
MLK2 | inactive (101.47%) | - |
MLK3 | inactive (95.2%) | - |
TAK1 | inactive (95.45%) | inactive (85%) |
ZAK | inactive (102.26%) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RIPK2 | inactive (89.91%) | inactive (87%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NuaK1 | inactive (94.81%) | inactive (97%) |
BRSK1 | inactive (90.26%) | inactive (52%) |
BRSK2 | inactive (98.55%) | inactive (106%) |
CHK1 | inactive (103.94%) | inactive (89%) |
LKB1 | inactive (90.71%) | inactive (100%) |
MARK1 | inactive (94.52%) | inactive (81%) |
MARK3 | inactive (98.01%) | - |
MARK4 | inactive (94.72%) | - |
MELK | inactive (101.99%) | inactive (91%) |
PASK | inactive (101.02%) | inactive (99%) |
QIK | inactive (90.45%) | - |
NuaK2 | inactive (135.75%) | - |
MARK2 | inactive (101.83%) | inactive (112%) |
AMPKa1 | - | inactive (93%) |
AMPKa2 | - | inactive (122%) |
SIK | - | inactive (79%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK1a | inactive (108.47%) | inactive (106%) |
CaMK1b | inactive (98.45%) | - |
CaMK1d | inactive (106.54%) | inactive (101%) |
CaMK1g | inactive (98.96%) | - |
CaMK4 | inactive (101.41%) | inactive (118%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK2a | inactive (104.05%) | - |
CaMK2b | inactive (90.49%) | active (47%) |
CaMK2d | inactive (102.53%) | inactive (87%) |
CaMK2g | inactive (92.64%) | inactive (79%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CHK2 | inactive (99.27%) | inactive (86%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DAPK1 | inactive (97.69%) | inactive (85%) |
DAPK2 | inactive (107.99%) | inactive (100%) |
DRAK1 | inactive (93.01%) | inactive (102%) |
DAPK3 | inactive (100.54%) | inactive (110%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DCLK2 | inactive (98.08%) | inactive (75%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAPKAPK2 | inactive (101.09%) | inactive (90%) |
MAPKAPK3 | inactive (97.76%) | inactive (103%) |
MAPKAPK5 | inactive (96.14%) | inactive (87%) |
MNK1 | inactive (75.5%) | - |
MNK2 | active (39.18%) | active (35%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
smMLCK | inactive (96.75%) | inactive (72%) |
skMLCK | inactive (96.2%) | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PHKg1 | inactive (90.31%) | - |
PHKg2 | inactive (101.47%) | inactive (103%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PIM1 | inactive (93.51%) | inactive (97%) |
PIM2 | inactive (105.21%) | inactive (97%) |
PIM3 | inactive (103.16%) | inactive (91%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKD1 | inactive (95.5%) | inactive (87%) |
PKD3 | inactive (90.68%) | - |
PKD2 | inactive (95.75%) | inactive (104%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TSSK1 | inactive (103.46%) | inactive (94%) |
TSSK2 | inactive (96.9%) | inactive (100%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
STK33 | inactive (97.28%) | inactive (98%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP3K5 | inactive (108.72%) | inactive (93%) |
MAP3K2 | inactive (94.86%) | - |
MAP3K3 | inactive (103.27%) | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
COT | inactive (99%) | - |
NIK | inactive (112.07%) | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GCK | inactive (101.24%) | inactive (86%) |
HGK | inactive (54.35%) | - |
KHS1 | inactive (105.99%) | - |
LOK | inactive (93.71%) | inactive (86%) |
MINK | inactive (84.56%) | inactive (85%) |
MST1 | inactive (103.4%) | inactive (89%) |
MST2 | inactive (111.73%) | inactive (103%) |
MST3 | inactive (93.54%) | inactive (61%) |
MST4 | inactive (103.86%) | - |
OSR1 | inactive (97.2%) | - |
PAK1 | inactive (99.12%) | - |
PAK2 | inactive (83.99%) | inactive (98%) |
PAK3 | inactive (101.99%) | inactive (61%) |
PAK4 | inactive (96.71%) | inactive (93%) |
PAK5 | inactive (93.8%) | inactive (97%) |
PAK6 | inactive (104.2%) | inactive (106%) |
SLK | inactive (102.61%) | - |
YSK1 | inactive (117.25%) | - |
STLK3 | inactive (99.83%) | - |
TAO1 | inactive (88.42%) | inactive (100%) |
TAO2 | inactive (92.07%) | inactive (110%) |
TAO3 | inactive (102.73%) | inactive (98%) |
MYO3B | inactive (96.43%) | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP2K1 | inactive (96.46%) | inactive (87%) |
MAP2K2 | inactive (103.14%) | - |
MAP2K6 | inactive (106.28%) | inactive (77%) |
MAP2K7 | - | inactive (101%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AurA | inactive (78.03%) | inactive (99%) |
AurB | inactive (95.94%) | inactive (92%) |
AurC | inactive (93.08%) | inactive (66%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMKK1 | inactive (122.14%) | - |
CaMKK2 | inactive (112.65%) | - |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Haspin | inactive (62.34%) | active (48%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IKKa | inactive (107.26%) | inactive (97%) |
IKKb | inactive (101.79%) | inactive (105%) |
IKKe | inactive (96.45%) | - |
TBK1 | inactive (93.42%) | inactive (65%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NEK1 | inactive (101.39%) | - |
NEK11 | inactive (76.91%) | inactive (89%) |
NEK2 | inactive (105.61%) | inactive (78%) |
NEK4 | inactive (95.41%) | - |
NEK6 | inactive (93.41%) | inactive (95%) |
NEK7 | inactive (103.77%) | inactive (95%) |
NEK9 | inactive (101.07%) | - |
NEK3 | inactive (91.61%) | inactive (114%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PBK | inactive (97.13%) | - |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PLK1 | inactive (101.64%) | inactive (86%) |
PLK2 | inactive (99.9%) | inactive (107%) |
PLK3 | inactive (95.29%) | inactive (91%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SgK496 | inactive (95.95%) | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MPSK1 | inactive (110%) | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TTK | inactive (112.35%) | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ULK1 | inactive (83.76%) | - |
ULK2 | inactive (105.57%) | inactive (104%) |
ULK3 | inactive (82.98%) | inactive (104%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wee1 | inactive (89.31%) | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wnk2 | inactive (96.88%) | inactive (107%) |
Wnk3 | inactive (100.38%) | inactive (98%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TLK2 | inactive (95.84%) | inactive (103%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK1 | 7 | 6 | 4 |
VRK | 3 | 1 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK1d | inactive (105.34%) | inactive (85%) |
CK1g1 | inactive (79.19%) | inactive (96%) |
CK1g2 | inactive (95.04%) | inactive (107%) |
CK1g3 | inactive (107.96%) | inactive (110%) |
CK1a | inactive (100.32%) | - |
CK1e | inactive (100.02%) | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
VRK1 | inactive (101.45%) | - |
VRK2 | - | inactive (101%) |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK2 | 3 | 2 | 2 |
CLK | 4 | 4 | 2 |
DYRK | 10 | 9 | 4 |
MAPK | 14 | 10 | 10 |
GSK | 2 | 2 | 2 |
SRPK | 3 | 3 | 3 |
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK2a1 | inactive (95.01%) | inactive (78%) |
CK2a2 | inactive (94.95%) | inactive (126%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CLK1 | inactive (104.66%) | - |
CLK2 | inactive (100.85%) | inactive (112%) |
CLK3 | inactive (92.56%) | inactive (87%) |
CLK4 | inactive (101.2%) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DYRK1A | inactive (77.62%) | - |
DYRK1B | inactive (90.49%) | - |
DYRK2 | inactive (77.45%) | inactive (77%) |
DYRK3 | inactive (100.65%) | - |
DYRK4 | inactive (98.7%) | - |
HIPK1 | inactive (97.37%) | inactive (95%) |
HIPK2 | inactive (94.06%) | inactive (100%) |
HIPK3 | inactive (107.11%) | inactive (95%) |
HIPK4 | inactive (93.8%) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Erk1 | inactive (98.94%) | inactive (77%) |
Erk2 | inactive (100.2%) | inactive (101%) |
JNK3 | inactive (101.88%) | inactive (85%) |
NLK | inactive (95.08%) | inactive (96%) |
p38a | inactive (104.21%) | inactive (77%) |
p38b | inactive (111.71%) | inactive (96%) |
p38d | inactive (122.67%) | inactive (103%) |
p38g | inactive (103.92%) | inactive (100%) |
JNK1 | inactive (100.28%) | inactive (97%) |
JNK2 | inactive (103.25%) | inactive (107%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GSK3A | inactive (102.74%) | inactive (123%) |
GSK3B | inactive (103.59%) | inactive (94%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSSK1 | inactive (96.03%) | inactive (102%) |
SRPK1 | inactive (108.03%) | inactive (108%) |
SRPK2 | inactive (102.82%) | inactive (89%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
PDHK | 5 | 1 | - |
Alpha | 6 | - | 1 |
PIKK | 6 | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDHK1 | inactive (96.57%) | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
eEF2K | - | inactive (86%) |
Atypical - PIKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FRAP | - | inactive (109%) |