Compound Information
Test on : RBC, Metz, Millipore
Compound Name
RBC, Metz, Millipore : JNK Inhibitor VIII
Inchikey
Same : KQMPRSZTUSSXND-N
RBC, Metz, Millipore : KQMPRSZTUSSXND-UHFFFAOYSA-N
ChemSpider
RBC, Metz, Millipore : 9799348
Pubchem CID
RBC, Metz, Millipore : 11624601
ChEMBL
RBC, Metz, Millipore : CHEMBL210618
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PDK1 | inactive (94.6%) | inactive (>3981.07nM) | inactive (107%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
AKT1 | inactive (102.12%) | inactive (>7943.28nM) | inactive (113%) |
AKT2 | inactive (102.86%) | inactive (>7943.28nM) | inactive (111%) |
AKT3 | inactive (104.86%) | inactive (>10000nM) | inactive (95%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DMPK1 | inactive (99.54%) | - | inactive (97%) |
MRCKa | inactive (98.87%) | inactive (>10000nM) | inactive (113%) |
MRCKb | inactive (102.86%) | - | inactive (101%) |
ROCK1 | inactive (96.42%) | inactive (>10000nM) | inactive (116%) |
ROCK2 | inactive (93.12%) | inactive (>7943.28nM) | inactive (93%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
BARK1 | inactive (108.4%) | - | - |
BARK2 | inactive (105.6%) | - | - |
GPRK4 | inactive (99.75%) | - | - |
GPRK5 | inactive (95.41%) | - | inactive (99%) |
GPRK6 | inactive (98.85%) | - | inactive (93%) |
GPRK7 | inactive (113.88%) | - | inactive (96%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MSK1 | inactive (101.12%) | inactive (>1995.26nM) | inactive (102%) |
MSK2 | inactive (105.46%) | - | inactive (105%) |
p70S6K | inactive (103.7%) | inactive (3162.28nM) | inactive (140%) |
p70S6Kb | inactive (96%) | - | - |
RSK2 | inactive (95.65%) | inactive (>7943.28nM) | inactive (107%) |
RSK4 | inactive (94.32%) | - | inactive (96%) |
RSK1 | inactive (79.91%) | - | inactive (90%) |
RSK3 | inactive (98.83%) | - | inactive (103%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKACg | inactive (104.31%) | - | - |
PRKX | inactive (100.04%) | inactive (>1584.89nM) | inactive (86%) |
PKACa | inactive (104.16%) | inactive (>7943.28nM) | inactive (88%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKCa | inactive (99.92%) | - | inactive (107%) |
PKCd | inactive (96.91%) | inactive (>7943.28nM) | inactive (118%) |
PKCe | inactive (98.83%) | - | inactive (116%) |
PKCh | inactive (94.32%) | - | inactive (79%) |
PKCg | inactive (95.4%) | - | inactive (97%) |
PKCi | inactive (100.37%) | - | inactive (120%) |
PKCt | inactive (111.42%) | - | inactive (98%) |
PKCz | inactive (104.07%) | inactive (>7943.28nM) | inactive (115%) |
PKCb | inactive (104.8%) | - | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKG2 | inactive (114.28%) | inactive (>1584.89nM) | - |
PKG1 | inactive (101%) | inactive (>1995.26nM) | - |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKN1 | inactive (103.77%) | - | - |
PKN2 | inactive (99.71%) | inactive (>7943.28nM) | inactive (92%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
SGK1 | inactive (105.44%) | inactive (>10000nM) | inactive (79%) |
SGK2 | inactive (102%) | - | inactive (95%) |
SGK3 | inactive (108.61%) | - | inactive (110%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
NDR1 | inactive (101.8%) | - | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ABL1 | inactive (100.12%) | inactive (>630.96nM) | inactive (103%) |
ABL2 | inactive (101.69%) | - | inactive (106%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ACK | inactive (92.19%) | - | inactive (73%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ALK | inactive (92.9%) | - | inactive (81%) |
LTK | inactive (97.25%) | - | - |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
AXL | inactive (105.28%) | inactive (>1995.26nM) | inactive (96%) |
MER | inactive (83.86%) | - | inactive (98%) |
TYRO3 | inactive (101.51%) | - | inactive (105%) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
BLK | inactive (103.4%) | inactive (>1584.89nM) | inactive (108%) |
BRK | inactive (93.61%) | - | inactive (60%) |
SRC | inactive (94.69%) | inactive (>5011.87nM) | inactive (112%) |
FGR | inactive (93.59%) | - | inactive (83%) |
FRK | inactive (103.01%) | - | inactive (90%) |
FYN | inactive (101.17%) | inactive (>794.33nM) | inactive (84%) |
HCK | inactive (98.47%) | - | inactive (78%) |
LCK | inactive (101.96%) | inactive (>2511.89nM) | inactive (94%) |
SRM | inactive (107.75%) | - | - |
YES | inactive (99.25%) | - | inactive (76%) |
LYN | inactive (98.53%) | inactive (>1584.89nM) | inactive (69%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
BMX | inactive (98.37%) | - | inactive (83%) |
BTK | inactive (92.48%) | - | inactive (81%) |
ITK | inactive (104.51%) | inactive (>1584.89nM) | inactive (98%) |
TEC | inactive (99.15%) | - | - |
TXK | inactive (92.97%) | - | inactive (79%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
KIT | inactive (84.63%) | inactive (>1258.93nM) | inactive (106%) |
FLT3 | inactive (102.42%) | inactive (>2511.89nM) | inactive (94%) |
FMS | inactive (99.21%) | inactive (>2511.89nM) | inactive (94%) |
PDGFRb | inactive (103.91%) | - | inactive (94%) |
PDGFRa | inactive (97.11%) | - | inactive (106%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CSK | inactive (95.07%) | - | inactive (106%) |
CTK | inactive (88.59%) | - | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DDR2 | inactive (95.43%) | - | inactive (89%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
EGFR | inactive (100.5%) | inactive (>1995.26nM) | inactive (107%) |
ErbB2 | inactive (100.82%) | inactive (>1584.89nM) | - |
ErbB4 | inactive (98.61%) | inactive (>3981.07nM) | inactive (103%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
EphA1 | inactive (97.38%) | - | inactive (107%) |
EphA2 | inactive (103.21%) | inactive (>3162.28nM) | inactive (93%) |
EphA3 | inactive (94.75%) | - | inactive (96%) |
EphA4 | inactive (99.08%) | - | inactive (96%) |
EphA5 | inactive (112.31%) | - | inactive (88%) |
EphA6 | inactive (89.49%) | - | - |
EphA7 | inactive (108.1%) | - | inactive (105%) |
EphA8 | inactive (84.22%) | - | inactive (86%) |
EphB1 | inactive (94.44%) | - | inactive (105%) |
EphB2 | inactive (97.59%) | - | inactive (101%) |
EphB3 | inactive (95.9%) | - | inactive (103%) |
EphB4 | inactive (98.25%) | - | inactive (95%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FAK | inactive (97.55%) | inactive (>1584.89nM) | inactive (73%) |
PYK2 | inactive (107.57%) | inactive (>1584.89nM) | inactive (98%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FER | inactive (94.06%) | - | inactive (99%) |
FES | inactive (91.05%) | - | inactive (89%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FGFR1 | inactive (106.05%) | inactive (>5011.87nM) | inactive (113%) |
FGFR2 | inactive (109.97%) | - | inactive (100%) |
FGFR3 | inactive (99.03%) | inactive (>1995.26nM) | inactive (114%) |
FGFR4 | inactive (109.4%) | - | inactive (122%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FLT1 | inactive (85.5%) | inactive (>398.11nM) | inactive (100%) |
FLT4 | inactive (92.31%) | inactive (>6309.57nM) | inactive (95%) |
KDR | inactive (101.65%) | inactive (>7943.28nM) | inactive (92%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
IGF1R | inactive (104.75%) | inactive (>1000nM) | inactive (90%) |
IRR | - | - | inactive (99%) |
INSR | inactive (102.08%) | inactive (>5011.87nM) | inactive (98%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
JAK1 | inactive (109.91%) | - | - |
JAK2 | inactive (101.09%) | inactive (>1584.89nM) | inactive (98%) |
JAK3 | inactive (99.14%) | inactive (>1584.89nM) | inactive (103%) |
TYK2 | inactive (100.6%) | inactive (>1995.26nM) | - |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MUSK | inactive (103.61%) | - | inactive (82%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
RET | inactive (103.95%) | - | inactive (96%) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
RON | inactive (95.03%) | - | inactive (87%) |
MET | inactive (106.81%) | inactive (>3162.28nM) | inactive (133%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ROS | inactive (97.44%) | - | inactive (98%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
SYK | inactive (99.18%) | - | inactive (90%) |
ZAP70 | inactive (90.6%) | - | inactive (110%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TIE2 | inactive (100.96%) | - | inactive (109%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TRKA | inactive (101.74%) | inactive (>2511.89nM) | inactive (94%) |
TRKB | inactive (101.67%) | inactive (>5011.87nM) | inactive (118%) |
TRKC | inactive (101.74%) | - | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ALK1 | inactive (106.58%) | - | - |
ALK2 | inactive (95.25%) | - | - |
ALK4 | inactive (98.46%) | - | inactive (105%) |
TGFbR1 | inactive (97.78%) | - | inactive (109%) |
TGFbR2 | inactive (104.31%) | - | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ARAF | inactive (104.48%) | - | - |
BRAF | inactive (99.07%) | - | - |
RAF1 | inactive (91.77%) | - | inactive (74%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
IRAK1 | inactive (100.38%) | inactive (>7943.28nM) | inactive (94%) |
IRAK4 | inactive (94.93%) | inactive (>10000nM) | inactive (81%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
LIMK1 | inactive (102.82%) | inactive (>10000nM) | inactive (89%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
LRRK2 | inactive (90.54%) | - | - |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MLK1 | inactive (103.48%) | - | inactive (102%) |
MLK2 | inactive (91.34%) | - | - |
MLK3 | inactive (98.76%) | - | - |
TAK1 | inactive (96.62%) | - | inactive (95%) |
ZAK | inactive (90.45%) | inactive (>7943.28nM) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
RIPK2 | inactive (80.98%) | - | inactive (91%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
NuaK1 | inactive (96.12%) | - | inactive (111%) |
BRSK1 | inactive (95.66%) | inactive (>10000nM) | inactive (101%) |
BRSK2 | inactive (103.32%) | - | inactive (106%) |
CHK1 | inactive (151.2%) | inactive (>7943.28nM) | inactive (95%) |
LKB1 | inactive (96.36%) | - | inactive (96%) |
MARK1 | inactive (98.98%) | - | inactive (92%) |
MARK3 | inactive (94.82%) | inactive (>6309.57nM) | - |
MARK4 | inactive (96.9%) | - | - |
MELK | inactive (97.07%) | inactive (>1584.89nM) | inactive (96%) |
PASK | inactive (91.14%) | inactive (>1584.89nM) | inactive (115%) |
QIK | inactive (97.89%) | - | - |
NuaK2 | inactive (71.95%) | - | - |
MARK2 | inactive (99.76%) | inactive (>7943.28nM) | inactive (104%) |
AMPKa1 | - | inactive (>6309.57nM) | inactive (89%) |
AMPKa2 | - | - | inactive (91%) |
SIK | - | - | inactive (116%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CaMK1a | inactive (103.4%) | inactive (>7943.28nM) | inactive (97%) |
CaMK1b | inactive (96.54%) | - | - |
CaMK1d | inactive (107.78%) | - | inactive (105%) |
CaMK1g | inactive (100.14%) | - | - |
CaMK4 | inactive (99.14%) | - | inactive (91%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CaMK2a | inactive (103.8%) | - | - |
CaMK2b | inactive (98.09%) | inactive (>7943.28nM) | inactive (94%) |
CaMK2d | inactive (97.4%) | inactive (>6309.57nM) | inactive (107%) |
CaMK2g | inactive (100.78%) | inactive (>6309.57nM) | inactive (101%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CHK2 | inactive (102.41%) | inactive (>5011.87nM) | inactive (99%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DAPK1 | inactive (99.04%) | - | inactive (95%) |
DAPK2 | inactive (104.3%) | - | inactive (100%) |
DRAK1 | inactive (101.71%) | - | inactive (82%) |
DAPK3 | inactive (110.51%) | inactive (>1258.93nM) | inactive (98%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DCLK2 | inactive (98.12%) | - | inactive (138%) |
DCLK1 | - | inactive (>10000nM) | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MAPKAPK2 | inactive (102.69%) | inactive (>7943.28nM) | inactive (84%) |
MAPKAPK3 | inactive (101.06%) | inactive (>10000nM) | inactive (105%) |
MAPKAPK5 | inactive (86.53%) | inactive (>1584.89nM) | inactive (96%) |
MNK1 | inactive (104.89%) | - | - |
MNK2 | inactive (106.02%) | inactive (>10000nM) | inactive (100%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
smMLCK | inactive (96.47%) | - | inactive (113%) |
skMLCK | inactive (99.55%) | - | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PHKg1 | inactive (94.19%) | - | - |
PHKg2 | inactive (100.17%) | inactive (>5011.87nM) | inactive (118%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PIM1 | inactive (103.59%) | inactive (>10000nM) | inactive (95%) |
PIM2 | inactive (103.82%) | inactive (>1584.89nM) | inactive (142%) |
PIM3 | inactive (95.23%) | - | inactive (88%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PKD1 | inactive (88.41%) | - | inactive (90%) |
PKD3 | inactive (83.73%) | inactive (>10000nM) | - |
PKD2 | inactive (91.44%) | inactive (5011.87nM) | inactive (111%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TSSK1 | inactive (95.98%) | inactive (>1584.89nM) | inactive (97%) |
TSSK2 | inactive (91.16%) | inactive (>1584.89nM) | inactive (106%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
STK33 | inactive (97.72%) | - | inactive (107%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MAP3K5 | inactive (92.77%) | - | inactive (99%) |
MAP3K2 | inactive (92.45%) | - | - |
MAP3K3 | inactive (97.1%) | - | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
COT | inactive (96.92%) | - | - |
NIK | inactive (107.5%) | - | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
GCK | inactive (83.6%) | inactive (>6309.57nM) | inactive (89%) |
HGK | inactive (94.55%) | inactive (>10000nM) | - |
KHS1 | inactive (95.36%) | inactive (>7943.28nM) | - |
LOK | inactive (97.73%) | - | inactive (112%) |
MINK | inactive (97.42%) | inactive (>7943.28nM) | inactive (106%) |
MST1 | inactive (95.41%) | - | inactive (80%) |
MST2 | inactive (100%) | inactive (>7943.28nM) | inactive (108%) |
MST3 | inactive (99.52%) | - | inactive (92%) |
MST4 | inactive (103.74%) | - | - |
OSR1 | inactive (104.02%) | - | - |
PAK1 | inactive (101.61%) | inactive (>10000nM) | - |
PAK2 | inactive (100.81%) | - | inactive (106%) |
PAK3 | inactive (104.05%) | - | inactive (108%) |
PAK4 | inactive (91.85%) | inactive (>5011.87nM) | inactive (91%) |
PAK5 | inactive (107.02%) | - | inactive (118%) |
PAK6 | inactive (101.84%) | - | inactive (100%) |
SLK | inactive (103.01%) | inactive (>10000nM) | - |
YSK1 | inactive (94.5%) | - | - |
STLK3 | inactive (92.72%) | - | - |
TAO1 | inactive (109.03%) | inactive (>10000nM) | inactive (94%) |
TAO2 | inactive (99.42%) | - | inactive (105%) |
TAO3 | inactive (88.6%) | - | inactive (89%) |
MYO3B | inactive (101.86%) | - | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MAP2K1 | inactive (87.01%) | - | inactive (125%) |
MAP2K2 | inactive (90.26%) | - | - |
MAP2K6 | inactive (96.8%) | - | inactive (121%) |
MAP2K7 | - | - | active (11%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
AurA | inactive (103.91%) | inactive (>3981.07nM) | inactive (106%) |
AurB | inactive (104.97%) | inactive (>6309.57nM) | inactive (104%) |
AurC | inactive (97.39%) | - | inactive (78%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CaMKK1 | inactive (103.79%) | - | - |
CaMKK2 | inactive (85.03%) | - | - |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Haspin | inactive (98.94%) | - | inactive (110%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
IKKa | inactive (96.12%) | inactive (>3981.07nM) | inactive (115%) |
IKKb | inactive (101.74%) | inactive (>3162.28nM) | inactive (113%) |
IKKe | inactive (83.69%) | - | - |
TBK1 | inactive (96.64%) | - | inactive (79%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
NEK1 | inactive (95.24%) | - | - |
NEK11 | inactive (109.19%) | - | inactive (109%) |
NEK2 | inactive (87.71%) | inactive (>10000nM) | inactive (99%) |
NEK4 | inactive (93.17%) | inactive (>6309.57nM) | - |
NEK6 | inactive (98.1%) | - | inactive (111%) |
NEK7 | inactive (93.48%) | - | inactive (97%) |
NEK9 | inactive (95.92%) | - | - |
NEK3 | inactive (89.99%) | - | inactive (84%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PBK | inactive (115.59%) | inactive (>10000nM) | - |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PLK1 | inactive (95.34%) | inactive (>7943.28nM) | inactive (85%) |
PLK2 | inactive (104.9%) | - | inactive (100%) |
PLK3 | inactive (101.19%) | inactive (>7943.28nM) | inactive (102%) |
PLK4 | - | inactive (>3981.07nM) | - |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
SgK496 | inactive (97.36%) | - | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MPSK1 | inactive (94.05%) | - | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TTK | inactive (75.6%) | - | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
ULK1 | inactive (102.93%) | - | - |
ULK2 | inactive (109.91%) | - | inactive (113%) |
ULK3 | inactive (103.86%) | - | inactive (92%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Wee1 | inactive (88.15%) | - | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Wnk2 | inactive (103.8%) | - | inactive (94%) |
Wnk3 | inactive (93.28%) | - | inactive (92%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
TLK2 | inactive (100.2%) | - | inactive (92%) |
Other - CDC7
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CDC7 | - | inactive (>1258.93nM) | - |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz | Millipore |
---|
CK1 | 7 | 6 | 5 | 4 |
VRK | 3 | 1 | - | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CK1d | inactive (102.64%) | inactive (>7943.28nM) | inactive (104%) |
CK1g1 | inactive (97.66%) | inactive (>6309.57nM) | inactive (108%) |
CK1g2 | inactive (100.3%) | inactive (>7943.28nM) | inactive (111%) |
CK1g3 | inactive (104.81%) | - | inactive (115%) |
CK1a | inactive (88.42%) | inactive (>6309.57nM) | - |
CK1e | inactive (100.63%) | - | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
VRK1 | inactive (92.55%) | - | - |
VRK2 | - | - | inactive (89%) |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz | Millipore |
---|
CK2 | 3 | 2 | 1 | 2 |
CLK | 4 | 4 | 2 | 2 |
DYRK | 10 | 9 | 6 | 4 |
MAPK | 14 | 10 | 8 | 10 |
GSK | 2 | 2 | 2 | 2 |
SRPK | 3 | 3 | 1 | 3 |
CDK | 20 | - | 7 | - |
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CK2a1 | inactive (96.88%) | inactive (>6309.57nM) | inactive (98%) |
CK2a2 | inactive (105.81%) | - | inactive (100%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CLK1 | inactive (98.08%) | - | - |
CLK2 | inactive (96.13%) | inactive (>7943.28nM) | inactive (118%) |
CLK3 | inactive (100.55%) | - | inactive (98%) |
CLK4 | inactive (96.12%) | inactive (>10000nM) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
DYRK1A | inactive (98.52%) | inactive (>6309.57nM) | - |
DYRK1B | inactive (99.16%) | - | - |
DYRK2 | inactive (111.22%) | - | inactive (102%) |
DYRK3 | inactive (113.98%) | inactive (>6309.57nM) | - |
DYRK4 | inactive (92.63%) | - | - |
HIPK1 | inactive (105.27%) | - | inactive (110%) |
HIPK2 | inactive (106.4%) | inactive (>3162.28nM) | inactive (108%) |
HIPK3 | inactive (113.48%) | - | inactive (99%) |
HIPK4 | inactive (106.38%) | inactive (>7943.28nM) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
Erk1 | inactive (96.03%) | - | inactive (83%) |
Erk2 | inactive (92.62%) | inactive (5011.87nM) | inactive (96%) |
JNK3 | inactive (51.46%) | - | active (-2%) |
NLK | inactive (103.82%) | - | inactive (86%) |
p38a | inactive (93.85%) | - | inactive (98%) |
p38b | inactive (105.6%) | - | inactive (98%) |
p38d | inactive (106.05%) | inactive (>7943.28nM) | inactive (104%) |
p38g | inactive (94.69%) | inactive (>6309.57nM) | inactive (100%) |
JNK1 | active (28.12%) | active (2nM) | active (-16%) |
JNK2 | active (6.45%) | active (3.98nM) | active (-1%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
GSK3A | inactive (98.89%) | inactive (>7943.28nM) | inactive (99%) |
GSK3B | inactive (100.6%) | inactive (>6309.57nM) | inactive (105%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
MSSK1 | inactive (92.27%) | - | inactive (99%) |
SRPK1 | inactive (101.11%) | inactive (>7943.28nM) | inactive (97%) |
SRPK2 | inactive (97.85%) | - | inactive (93%) |
CMGC - CDK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
CDC2 | - | inactive (>7943.28nM) | - |
CDK2 | - | active (794.33nM) | - |
CDK5 | - | inactive (>10000nM) | - |
CDK8 | - | - | - |
CDK7 | - | - | - |
CDK9 | - | - | - |
CDK11 | - | inactive (>100000nM) | - |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Metz | Millipore |
---|
PDHK | 5 | 1 | - | - |
Alpha | 6 | - | 1 | 1 |
PIKK | 6 | - | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
PDHK1 | inactive (94.6%) | - | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
eEF2K | - | inactive (>3981.07nM) | inactive (88%) |
Atypical - PIKK
Bioactivity |
---|
Kinase | RBC | Metz | Millipore |
---|
FRAP | - | - | inactive (99%) |