Compound Information
Test on : RBC, Millipore
Compound Name
RBC : ZINC16052820
Millipore : CGK733
Inchikey
Same : HLCDNLNLQNYZTK-N
RBC : HLCDNLNLQNYZTK-NRFANRHFSA-N
Millipore : HLCDNLNLQNYZTK-UHFFFAOYSA-N
ChemSpider
RBC : 68894522
Millipore : 5037512
Pubchem CID
RBC : 92509771
Millipore : 6605258
ChEMBL
RBC : -
Millipore : CHEMBL1221601
RBC | Millipore |
| |
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDK1 | inactive (112.34%) | inactive (103%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AKT1 | inactive (117.84%) | inactive (108%) |
AKT2 | inactive (91.57%) | inactive (108%) |
AKT3 | inactive (106.46%) | inactive (98%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DMPK1 | inactive (85.51%) | inactive (71%) |
MRCKa | inactive (111.27%) | inactive (106%) |
MRCKb | inactive (97.19%) | inactive (97%) |
ROCK1 | inactive (99.79%) | inactive (110%) |
ROCK2 | inactive (109.24%) | inactive (99%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BARK1 | inactive (79.54%) | - |
BARK2 | inactive (98.34%) | - |
GPRK4 | inactive (101.14%) | - |
GPRK5 | inactive (105.02%) | inactive (90%) |
GPRK6 | inactive (97.5%) | inactive (100%) |
GPRK7 | inactive (101.35%) | inactive (86%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSK1 | inactive (112.54%) | inactive (112%) |
MSK2 | inactive (92.73%) | inactive (95%) |
p70S6K | inactive (91.93%) | inactive (141%) |
p70S6Kb | inactive (99.35%) | - |
RSK2 | inactive (96.16%) | inactive (108%) |
RSK4 | inactive (94.7%) | inactive (80%) |
RSK1 | inactive (105.02%) | inactive (108%) |
RSK3 | inactive (100.91%) | inactive (113%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKACg | - | - |
PRKX | inactive (105.54%) | inactive (82%) |
PKACa | inactive (101.77%) | inactive (105%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKCa | inactive (73.11%) | inactive (108%) |
PKCd | inactive (91.2%) | inactive (100%) |
PKCe | inactive (109.48%) | inactive (84%) |
PKCh | inactive (102.92%) | inactive (106%) |
PKCg | inactive (99.79%) | inactive (101%) |
PKCi | inactive (93.98%) | inactive (111%) |
PKCt | inactive (106.85%) | inactive (97%) |
PKCz | inactive (98.04%) | inactive (102%) |
PKCb | inactive (106.9%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKG2 | inactive (96.65%) | - |
PKG1 | inactive (100.3%) | - |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKN1 | inactive (92.84%) | - |
PKN2 | inactive (88.06%) | inactive (94%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SGK1 | inactive (93.14%) | inactive (110%) |
SGK2 | inactive (118.75%) | inactive (113%) |
SGK3 | inactive (85.77%) | inactive (110%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NDR1 | active (0%) | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ABL1 | inactive (101.16%) | inactive (109%) |
ABL2 | inactive (104.83%) | inactive (115%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ACK | inactive (97.96%) | inactive (100%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK | inactive (110.12%) | inactive (81%) |
LTK | inactive (91.54%) | - |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AXL | inactive (111.81%) | inactive (109%) |
MER | inactive (96.23%) | inactive (100%) |
TYRO3 | inactive (108.24%) | inactive (106%) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BLK | inactive (110.12%) | inactive (111%) |
BRK | inactive (87.82%) | inactive (107%) |
SRC | inactive (96.13%) | inactive (98%) |
FGR | inactive (84.52%) | inactive (105%) |
FRK | inactive (102.96%) | inactive (71%) |
FYN | inactive (91.22%) | inactive (104%) |
HCK | inactive (107.04%) | inactive (80%) |
LCK | inactive (91.85%) | inactive (95%) |
SRM | inactive (96.93%) | - |
YES | inactive (94.59%) | inactive (115%) |
LYN | inactive (102.7%) | inactive (89%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BMX | inactive (102.32%) | inactive (101%) |
BTK | inactive (103.86%) | inactive (87%) |
ITK | inactive (94.88%) | inactive (110%) |
TEC | inactive (200.7%) | - |
TXK | inactive (107.95%) | inactive (82%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
KIT | inactive (97.16%) | inactive (105%) |
FLT3 | inactive (99.31%) | inactive (99%) |
FMS | inactive (96.25%) | inactive (89%) |
PDGFRb | inactive (105.37%) | inactive (97%) |
PDGFRa | inactive (99.96%) | inactive (113%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CSK | inactive (99.26%) | inactive (95%) |
CTK | inactive (96.48%) | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DDR2 | inactive (96.36%) | inactive (102%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EGFR | inactive (108.01%) | inactive (105%) |
ErbB2 | inactive (94.8%) | - |
ErbB4 | inactive (103.36%) | inactive (105%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EphA1 | inactive (88.12%) | inactive (104%) |
EphA2 | inactive (103.34%) | inactive (107%) |
EphA3 | inactive (105.21%) | inactive (117%) |
EphA4 | inactive (101.07%) | inactive (96%) |
EphA5 | inactive (107.01%) | inactive (104%) |
EphA6 | - | - |
EphA7 | inactive (108.71%) | inactive (102%) |
EphA8 | inactive (103.76%) | inactive (103%) |
EphB1 | inactive (109.22%) | inactive (97%) |
EphB2 | inactive (100.73%) | inactive (111%) |
EphB3 | inactive (103.88%) | inactive (104%) |
EphB4 | inactive (101.48%) | inactive (109%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FAK | inactive (113.3%) | inactive (111%) |
PYK2 | inactive (101.9%) | inactive (108%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FER | inactive (104.38%) | inactive (117%) |
FES | inactive (103.88%) | inactive (108%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FGFR1 | inactive (97.73%) | inactive (106%) |
FGFR2 | inactive (97.7%) | inactive (109%) |
FGFR3 | inactive (96.77%) | inactive (121%) |
FGFR4 | inactive (100.02%) | inactive (118%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FLT1 | inactive (97.19%) | inactive (102%) |
FLT4 | inactive (102.34%) | inactive (93%) |
KDR | inactive (92.54%) | inactive (104%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IGF1R | inactive (93.7%) | inactive (76%) |
IRR | inactive (93.75%) | inactive (126%) |
INSR | inactive (100.43%) | inactive (115%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
JAK1 | inactive (105.82%) | - |
JAK2 | inactive (99.88%) | inactive (107%) |
JAK3 | inactive (110.11%) | inactive (107%) |
TYK2 | inactive (93.97%) | - |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MUSK | inactive (105.83%) | inactive (85%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RET | inactive (103.37%) | inactive (111%) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RON | inactive (101.79%) | inactive (88%) |
MET | inactive (100.75%) | inactive (105%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ROS | inactive (99.5%) | inactive (103%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SYK | inactive (104.17%) | inactive (94%) |
ZAP70 | inactive (94.24%) | inactive (126%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TIE2 | inactive (97.81%) | inactive (117%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TRKA | inactive (106.72%) | inactive (87%) |
TRKB | inactive (97.68%) | inactive (91%) |
TRKC | inactive (107.91%) | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK1 | inactive (106.69%) | - |
ALK2 | inactive (98.76%) | - |
ALK4 | inactive (105.78%) | inactive (94%) |
TGFbR1 | inactive (92.56%) | inactive (98%) |
TGFbR2 | inactive (91.65%) | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ARAF | inactive (108.75%) | - |
BRAF | inactive (102.23%) | - |
RAF1 | inactive (95.33%) | inactive (92%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IRAK1 | inactive (107.17%) | inactive (104%) |
IRAK4 | inactive (191.01%) | inactive (112%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LIMK1 | inactive (94.46%) | inactive (90%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LRRK2 | inactive (99.29%) | - |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MLK1 | inactive (93.98%) | inactive (102%) |
MLK2 | inactive (98.86%) | - |
MLK3 | inactive (102.03%) | - |
TAK1 | inactive (89.69%) | inactive (102%) |
ZAK | inactive (98.59%) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RIPK2 | inactive (97.43%) | inactive (92%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NuaK1 | inactive (95.31%) | inactive (105%) |
BRSK1 | inactive (98.31%) | inactive (91%) |
BRSK2 | inactive (101.91%) | inactive (93%) |
CHK1 | inactive (100.29%) | inactive (105%) |
LKB1 | inactive (94.2%) | inactive (98%) |
MARK1 | inactive (101.24%) | inactive (96%) |
MARK3 | inactive (103.59%) | - |
MARK4 | inactive (103.55%) | - |
MELK | inactive (101.84%) | inactive (76%) |
PASK | inactive (103.73%) | inactive (103%) |
QIK | inactive (112.05%) | - |
NuaK2 | inactive (108.3%) | - |
MARK2 | inactive (92.28%) | inactive (104%) |
AMPKa1 | - | inactive (90%) |
AMPKa2 | - | inactive (89%) |
SIK | - | inactive (136%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK1a | inactive (93.07%) | inactive (99%) |
CaMK1b | inactive (114.61%) | - |
CaMK1d | inactive (99.02%) | inactive (122%) |
CaMK1g | inactive (102.43%) | - |
CaMK4 | inactive (98.51%) | inactive (122%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK2a | inactive (95.99%) | - |
CaMK2b | inactive (103.83%) | inactive (91%) |
CaMK2d | inactive (102.37%) | inactive (99%) |
CaMK2g | inactive (107.12%) | inactive (99%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CHK2 | inactive (97.64%) | inactive (103%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DAPK1 | inactive (75.14%) | inactive (90%) |
DAPK2 | inactive (102.85%) | inactive (95%) |
DRAK1 | inactive (99.78%) | inactive (113%) |
DAPK3 | inactive (103.1%) | inactive (96%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DCLK2 | inactive (107.52%) | inactive (136%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAPKAPK2 | inactive (96.29%) | inactive (90%) |
MAPKAPK3 | inactive (105.75%) | inactive (113%) |
MAPKAPK5 | inactive (101.93%) | inactive (87%) |
MNK1 | inactive (100.23%) | - |
MNK2 | inactive (134.85%) | inactive (106%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
smMLCK | inactive (99.61%) | inactive (103%) |
skMLCK | inactive (104.46%) | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PHKg1 | inactive (104.08%) | - |
PHKg2 | inactive (108.95%) | inactive (110%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PIM1 | inactive (101.31%) | inactive (102%) |
PIM2 | inactive (117.25%) | inactive (90%) |
PIM3 | inactive (119.98%) | inactive (108%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKD1 | inactive (96.88%) | inactive (110%) |
PKD3 | inactive (98.52%) | - |
PKD2 | inactive (107.28%) | inactive (100%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TSSK1 | inactive (93.36%) | inactive (87%) |
TSSK2 | inactive (92.66%) | inactive (102%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
STK33 | inactive (99.58%) | inactive (98%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP3K5 | inactive (97.08%) | inactive (103%) |
MAP3K2 | inactive (96.77%) | - |
MAP3K3 | inactive (118.25%) | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
COT | inactive (105.06%) | - |
NIK | inactive (92.14%) | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GCK | inactive (110.73%) | inactive (88%) |
HGK | inactive (92.71%) | - |
KHS1 | inactive (91.02%) | - |
LOK | inactive (107.88%) | inactive (112%) |
MINK | inactive (109.92%) | inactive (113%) |
MST1 | inactive (96.16%) | inactive (92%) |
MST2 | inactive (106.85%) | inactive (98%) |
MST3 | inactive (92.83%) | inactive (86%) |
MST4 | inactive (89.3%) | - |
OSR1 | inactive (98.32%) | - |
PAK1 | inactive (86.03%) | - |
PAK2 | inactive (100.03%) | inactive (101%) |
PAK3 | inactive (91.87%) | inactive (90%) |
PAK4 | inactive (117.82%) | inactive (100%) |
PAK5 | inactive (103.8%) | inactive (106%) |
PAK6 | inactive (101.35%) | inactive (105%) |
SLK | inactive (95.19%) | - |
YSK1 | inactive (96.18%) | - |
STLK3 | inactive (77.03%) | - |
TAO1 | inactive (103.78%) | inactive (93%) |
TAO2 | inactive (103.18%) | inactive (91%) |
TAO3 | inactive (120.95%) | inactive (96%) |
MYO3B | active (0%) | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP2K1 | inactive (95.07%) | inactive (116%) |
MAP2K2 | inactive (82.25%) | - |
MAP2K6 | inactive (107.22%) | inactive (135%) |
MAP2K7 | - | inactive (108%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AurA | inactive (80.84%) | inactive (83%) |
AurB | inactive (95.3%) | inactive (110%) |
AurC | inactive (93.81%) | inactive (94%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMKK1 | inactive (127.6%) | - |
CaMKK2 | inactive (125.54%) | - |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Haspin | inactive (109.42%) | inactive (83%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IKKa | inactive (91.51%) | inactive (90%) |
IKKb | inactive (101.98%) | inactive (114%) |
IKKe | inactive (105.86%) | - |
TBK1 | inactive (98.66%) | inactive (96%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NEK1 | inactive (101.14%) | - |
NEK11 | inactive (92.16%) | inactive (86%) |
NEK2 | inactive (111.77%) | inactive (90%) |
NEK4 | inactive (87.84%) | - |
NEK6 | inactive (108.76%) | inactive (120%) |
NEK7 | inactive (101.54%) | inactive (108%) |
NEK9 | inactive (109.95%) | - |
NEK3 | inactive (96.21%) | inactive (94%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PBK | inactive (115.87%) | - |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PLK1 | inactive (111.48%) | inactive (102%) |
PLK2 | inactive (92.85%) | inactive (90%) |
PLK3 | inactive (94.42%) | inactive (100%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SgK496 | inactive (100.01%) | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MPSK1 | inactive (99.37%) | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TTK | inactive (96.94%) | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ULK1 | inactive (99.07%) | - |
ULK2 | inactive (106.38%) | inactive (96%) |
ULK3 | active (0%) | inactive (97%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wee1 | inactive (91.81%) | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wnk2 | inactive (117.03%) | inactive (107%) |
Wnk3 | inactive (108.2%) | inactive (104%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TLK2 | active (0%) | inactive (99%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK1 | 7 | 6 | 4 |
VRK | 3 | 1 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK1d | inactive (105.01%) | active (45%) |
CK1g1 | inactive (83.34%) | inactive (94%) |
CK1g2 | inactive (98.3%) | inactive (103%) |
CK1g3 | inactive (87.71%) | inactive (110%) |
CK1a | inactive (94.13%) | - |
CK1e | inactive (110.91%) | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
VRK1 | inactive (96.66%) | - |
VRK2 | - | inactive (108%) |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK2 | 3 | 2 | 2 |
CLK | 4 | 4 | 2 |
DYRK | 10 | 9 | 4 |
MAPK | 14 | 10 | 10 |
GSK | 2 | 2 | 2 |
SRPK | 3 | 3 | 3 |
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK2a1 | inactive (95.35%) | inactive (117%) |
CK2a2 | inactive (96.95%) | inactive (110%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CLK1 | inactive (106.06%) | - |
CLK2 | inactive (93.46%) | inactive (112%) |
CLK3 | inactive (123.63%) | inactive (94%) |
CLK4 | inactive (105.29%) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DYRK1A | inactive (99.76%) | - |
DYRK1B | inactive (102.83%) | - |
DYRK2 | inactive (102.33%) | inactive (98%) |
DYRK3 | inactive (100.06%) | - |
DYRK4 | inactive (103.79%) | - |
HIPK1 | inactive (108.33%) | inactive (99%) |
HIPK2 | inactive (118.21%) | inactive (104%) |
HIPK3 | inactive (105.36%) | inactive (96%) |
HIPK4 | inactive (103.61%) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Erk1 | inactive (119.72%) | inactive (82%) |
Erk2 | inactive (97.56%) | inactive (102%) |
JNK3 | inactive (96.24%) | inactive (92%) |
NLK | inactive (106.37%) | inactive (103%) |
p38a | inactive (100.65%) | inactive (105%) |
p38b | inactive (104.41%) | inactive (98%) |
p38d | inactive (107.27%) | inactive (95%) |
p38g | inactive (109.47%) | inactive (106%) |
JNK1 | inactive (82.12%) | inactive (120%) |
JNK2 | inactive (88.65%) | inactive (104%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GSK3A | inactive (104.77%) | inactive (108%) |
GSK3B | inactive (109.35%) | inactive (112%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSSK1 | inactive (97.98%) | inactive (98%) |
SRPK1 | inactive (99.27%) | inactive (107%) |
SRPK2 | inactive (102.67%) | inactive (116%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
PDHK | 5 | 1 | - |
Alpha | 6 | - | 1 |
PIKK | 6 | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDHK1 | inactive (112.34%) | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
eEF2K | - | inactive (116%) |
Atypical - PIKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FRAP | - | inactive (102%) |