Compound Information
Test on : DRx, RBC, Metz
Compound Name
DRx, RBC, Metz : Tozasertib
Inchikey
Same : GCIKSSRWRFVXBI-N
DRx, RBC, Metz : GCIKSSRWRFVXBI-UHFFFAOYSA-N
ChemSpider
DRx, RBC, Metz : 4591897
Pubchem CID
DRx, RBC, Metz : 5494449
ChEMBL
DRx, RBC, Metz : CHEMBL572878
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
Other
Other - NAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AAK1 | active (290nM) | - | - |
BIKE | active (65nM) | - | - |
GAK | inactive (3200nM) | - | - |
MPSK1 | active (610nM) | inactive (52.81%) | - |
Other - Aur
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AurA | active (3.9nM) | active (5.19%) | active (3.16nM) |
AurB | active (7.4nM) | active (4.89%) | active (5.01nM) |
AurC | active (6.3nM) | active (40.42%) | - |
Other - CAMKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CaMKK1 | inactive (4600nM) | inactive (85.96%) | - |
CaMKK2 | inactive (10001nM) | inactive (106.44%) | inactive (>2511.89nM) |
Other - PEK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
HRI | inactive (10001nM) | - | - |
PKR | inactive (10001nM) | - | - |
Other - IRE
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IRE1 | inactive (5600nM) | - | - |
Other - IKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IKKa | inactive (10001nM) | inactive (99.4%) | inactive (>3981.07nM) |
IKKb | inactive (10001nM) | inactive (84.93%) | inactive (>3162.28nM) |
IKKe | active (2600nM) | inactive (84.8%) | inactive (>3162.28nM) |
TBK1 | active (490nM) | inactive (90.53%) | inactive (>1995.26nM) |
Other - NEK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
NEK1 | inactive (10001nM) | inactive (67.64%) | - |
NEK11 | inactive (10001nM) | inactive (82.76%) | - |
NEK2 | inactive (10001nM) | inactive (104.59%) | inactive (>3981.07nM) |
NEK3 | inactive (10001nM) | inactive (95.05%) | - |
NEK4 | inactive (10001nM) | inactive (102.79%) | inactive (>6309.57nM) |
NEK5 | inactive (4200nM) | - | - |
NEK6 | inactive (10001nM) | inactive (94.17%) | - |
NEK7 | inactive (8700nM) | inactive (92.83%) | - |
NEK9 | inactive (10001nM) | inactive (101.75%) | - |
Other - WEE
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MYT1 | inactive (10001nM) | - | - |
Wee1 | inactive (3200nM) | inactive (100.44%) | - |
Wee1B | inactive (4200nM) | - | - |
Other - PLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PLK1 | inactive (10001nM) | inactive (95.25%) | inactive (>7943.28nM) |
PLK2 | inactive (10001nM) | inactive (103.79%) | - |
PLK3 | inactive (10001nM) | inactive (98.77%) | inactive (>7943.28nM) |
PLK4 | active (9.2nM) | - | active (25.12nM) |
Other - SgK496
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SgK496 | inactive (10001nM) | inactive (97.17%) | - |
Other - NKF1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SBK | inactive (10001nM) | - | - |
SgK110 | active (530nM) | - | - |
Other - NKF4
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CLIK1 | inactive (10001nM) | - | - |
Other - ULK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Fused | inactive (10001nM) | - | - |
ULK1 | inactive (10001nM) | inactive (99.23%) | - |
ULK2 | inactive (10001nM) | inactive (100.73%) | - |
ULK3 | active (310nM) | inactive (87.33%) | - |
Other - TLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TLK1 | inactive (4000nM) | - | - |
TLK2 | inactive (10001nM) | inactive (86.62%) | - |
Other - TTK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TTK | inactive (8100nM) | inactive (103.95%) | - |
Other - Haspin
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Haspin | - | inactive (67.95%) | - |
Other - TOPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PBK | - | inactive (106.56%) | inactive (>10000nM) |
Other - WNK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Wnk2 | - | inactive (96.01%) | - |
Wnk3 | - | inactive (93.33%) | - |
Other - CDC7
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CDC7 | - | - | inactive (>1258.93nM) |
TK
TK - Abl
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ABL1 | active (13nM) | active (13.76%) | active (15.85nM) |
ABL2 | active (4nM) | active (5.75%) | - |
TK - ALK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ALK | inactive (3100nM) | inactive (91.46%) | inactive (2511.89nM) |
LTK | inactive (7500nM) | inactive (84.19%) | active (501.19nM) |
TK - Axl
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AXL | active (210nM) | active (44.28%) | active (199.53nM) |
MER | active (1700nM) | inactive (106.16%) | - |
TYRO3 | inactive (10001nM) | inactive (84.99%) | inactive (1258.93nM) |
TK - Src
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
BLK | active (2200nM) | inactive (81.35%) | active (31.62nM) |
BRK | inactive (10001nM) | inactive (94.64%) | - |
FGR | active (790nM) | inactive (58.16%) | - |
FRK | inactive (3800nM) | inactive (101.33%) | - |
FYN | active (530nM) | inactive (72.15%) | inactive (3162.28nM) |
HCK | inactive (6200nM) | inactive (82.66%) | inactive (>3162.28nM) |
LCK | active (61nM) | active (12.26%) | active (125.89nM) |
LYN | active (650nM) | inactive (52.59%) | active (251.19nM) |
SRC | active (170nM) | active (26.73%) | active (158.49nM) |
SRM | inactive (10001nM) | inactive (95.94%) | - |
YES | active (470nM) | active (33.94%) | - |
TK - Tec
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
BMX | active (2600nM) | active (40.02%) | - |
BTK | inactive (4400nM) | inactive (63.59%) | inactive (1584.89nM) |
ITK | active (350nM) | inactive (98.73%) | active (63.1nM) |
TEC | inactive (8700nM) | inactive (112.07%) | - |
TXK | active (2700nM) | inactive (78.84%) | - |
TK - PDGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FMS | active (1800nM) | inactive (106.39%) | inactive (>2511.89nM) |
FLT3 | active (6.5nM) | active (6.67%) | active (398.11nM) |
KIT | active (240nM) | inactive (89.2%) | inactive (>5011.87nM) |
PDGFRa | active (1600nM) | inactive (71.36%) | inactive (>501.19nM) |
PDGFRb | active (310nM) | inactive (71.52%) | active (398.11nM) |
TK - Csk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CSK | inactive (4800nM) | inactive (78.13%) | - |
CTK | inactive (10001nM) | inactive (78.65%) | - |
TK - DDR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DDR1 | active (28nM) | - | - |
DDR2 | active (230nM) | inactive (61.87%) | - |
TK - EGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
EGFR | inactive (10001nM) | inactive (93.75%) | inactive (1584.89nM) |
ErbB2 | inactive (10001nM) | inactive (101.89%) | inactive (>1584.89nM) |
ErbB3 | inactive (7100nM) | - | - |
ErbB4 | inactive (10001nM) | inactive (93.12%) | inactive (>3981.07nM) |
TK - Eph
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
EphA1 | active (1000nM) | inactive (78.08%) | - |
EphA2 | active (840nM) | active (34.43%) | active (630.96nM) |
EphA3 | active (1500nM) | active (44.21%) | - |
EphA4 | inactive (4300nM) | inactive (72.07%) | - |
EphA5 | inactive (10001nM) | inactive (88.01%) | - |
EphA6 | inactive (4700nM) | active (48.38%) | - |
EphA7 | inactive (10001nM) | inactive (74.74%) | - |
EphA8 | active (500nM) | inactive (77.08%) | - |
EphB1 | active (1900nM) | inactive (69.66%) | - |
EphB2 | inactive (5600nM) | inactive (78.3%) | - |
EphB3 | inactive (10001nM) | inactive (62.17%) | - |
EphB4 | active (1700nM) | active (46.11%) | - |
EphB6 | active (28nM) | - | - |
TK - FAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FAK | inactive (10001nM) | inactive (100.26%) | inactive (>6309.57nM) |
PYK2 | active (2600nM) | inactive (95.49%) | inactive (>1584.89nM) |
TK - Fer
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FER | inactive (4200nM) | inactive (92.16%) | - |
FES | inactive (7400nM) | inactive (97.21%) | - |
TK - FGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FGFR1 | active (550nM) | inactive (73.95%) | active (794.33nM) |
FGFR2 | active (570nM) | inactive (66.37%) | - |
FGFR3 | active (860nM) | inactive (70.62%) | active (630.96nM) |
FGFR4 | inactive (7200nM) | inactive (87.76%) | - |
TK - VEGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FLT1 | active (100nM) | inactive (76.96%) | inactive (1258.93nM) |
FLT4 | active (1900nM) | inactive (55.43%) | inactive (1584.89nM) |
KDR | active (2000nM) | inactive (85.27%) | active (316.23nM) |
TK - InsR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IGF1R | active (740nM) | inactive (96.28%) | inactive (>1584.89nM) |
INSR | active (630nM) | active (43.5%) | active (1000nM) |
IRR | active (290nM) | inactive (52.37%) | - |
TK - JakA
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
JAK1 | inactive (5900nM) | inactive (91.86%) | - |
JAK2 | active (190nM) | inactive (75.53%) | active (251.19nM) |
JAK3 | active (630nM) | inactive (91.8%) | inactive (>5011.87nM) |
TYK2 | active (510nM) | inactive (67.67%) | active (199.53nM) |
TK - Met
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MET | active (670nM) | inactive (70.91%) | inactive (>794.33nM) |
RON | active (1300nM) | inactive (83.59%) | active (794.33nM) |
TK - Musk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MUSK | active (300nM) | inactive (102.8%) | - |
TK - Ret
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
RET | active (28nM) | active (3.91%) | active (12.59nM) |
TK - Sev
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ROS | active (610nM) | active (30.22%) | active (158.49nM) |
TK - Syk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SYK | active (1800nM) | inactive (99.19%) | - |
ZAP70 | inactive (10001nM) | inactive (105.66%) | - |
TK - Tie
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TIE1 | active (270nM) | - | - |
TIE2 | active (450nM) | active (27.77%) | - |
TK - Ack
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TNK1 | active (83nM) | - | - |
ACK | inactive (4400nM) | inactive (66.43%) | inactive (>3981.07nM) |
TK - Trk
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TRKA | active (38nM) | active (6.52%) | active (316.23nM) |
TRKB | active (240nM) | active (26.93%) | active (316.23nM) |
TRKC | active (200nM) | active (6.04%) | active (630.96nM) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ALK2 | active (1900nM) | inactive (162.3%) | inactive (1258.93nM) |
ALK4 | inactive (10001nM) | inactive (114.12%) | - |
ACTR2 | inactive (10001nM) | - | - |
ACTR2B | inactive (10001nM) | - | - |
ALK1 | inactive (9500nM) | inactive (99.46%) | - |
BMPR1A | inactive (10001nM) | - | - |
BMPR1B | active (1100nM) | - | - |
BMPR2 | inactive (7100nM) | - | - |
TGFbR1 | inactive (8400nM) | inactive (94.74%) | - |
TGFbR2 | inactive (10001nM) | inactive (101.73%) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SgK288 | inactive (5600nM) | - | - |
RIPK1 | active (20nM) | - | - |
RIPK2 | inactive (10001nM) | inactive (103.97%) | - |
ANKRD3 | active (300nM) | - | - |
TKL - RAF
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
BRAF | inactive (10001nM) | inactive (103.8%) | - |
RAF1 | inactive (10001nM) | inactive (117.18%) | - |
ARAF | - | inactive (122.73%) | - |
TKL - MLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DLK | active (190nM) | - | - |
LZK | active (180nM) | - | - |
MLK1 | active (390nM) | active (38.71%) | - |
MLK2 | active (1800nM) | inactive (61.05%) | active (398.11nM) |
MLK3 | active (680nM) | inactive (52.72%) | - |
TAK1 | active (2300nM) | inactive (90.73%) | - |
HH498 | inactive (10001nM) | - | - |
ZAK | active (2800nM) | inactive (91.04%) | inactive (7943.28nM) |
TKL - IRAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
IRAK1 | inactive (10001nM) | inactive (91.53%) | inactive (>7943.28nM) |
IRAK3 | inactive (10001nM) | - | - |
IRAK4 | inactive (3700nM) | inactive (78%) | inactive (2511.89nM) |
TKL - LISK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
LIMK1 | active (2600nM) | active (33.11%) | active (794.33nM) |
LIMK2 | active (2600nM) | - | - |
TESK1 | inactive (5600nM) | - | - |
TKL - LRRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
LRRK2 | inactive (10001nM) | inactive (56.37%) | active (630.96nM) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz |
---|
ABC1 | 5 | 2 | - | - |
PIKK | 6 | 1 | - | - |
RIO | 3 | 3 | - | - |
Alpha | 6 | 1 | - | 1 |
PDHK | 5 | - | 1 | - |
Atypical - ABC1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ADCK3 | inactive (10001nM) | - | - |
ADCK4 | inactive (10001nM) | - | - |
Atypical - PIKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
FRAP | inactive (10001nM) | - | - |
Atypical - RIO
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
RIOK1 | active (360nM) | - | - |
RIOK2 | active (250nM) | - | - |
RIOK3 | active (600nM) | - | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ChaK2 | inactive (10001nM) | - | - |
eEF2K | - | - | inactive (>3981.07nM) |
Atypical - PDHK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PDHK1 | - | inactive (82.71%) | - |
AGC
AGC - Akt
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AKT1 | inactive (10001nM) | inactive (99.19%) | inactive (>7943.28nM) |
AKT2 | inactive (10001nM) | inactive (103.23%) | inactive (>7943.28nM) |
AKT3 | inactive (10001nM) | inactive (85%) | inactive (>10000nM) |
AGC - DMPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CRIK | inactive (10001nM) | - | - |
DMPK1 | inactive (10001nM) | inactive (98.51%) | - |
DMPK2 | inactive (10001nM) | - | - |
MRCKa | inactive (10001nM) | inactive (75.25%) | inactive (>10000nM) |
MRCKb | inactive (10001nM) | inactive (101.05%) | - |
ROCK1 | inactive (10001nM) | inactive (109.68%) | inactive (>3981.07nM) |
ROCK2 | inactive (10001nM) | inactive (91.99%) | inactive (>3981.07nM) |
AGC - GRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
RHOK | inactive (10001nM) | - | - |
GPRK4 | active (400nM) | inactive (90.32%) | - |
GPRK7 | inactive (10001nM) | inactive (95.45%) | - |
BARK1 | - | inactive (107.32%) | - |
BARK2 | - | inactive (96.06%) | - |
GPRK5 | - | inactive (103.88%) | inactive (>3981.07nM) |
GPRK6 | - | inactive (103.97%) | - |
AGC - NDR
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
LATS1 | inactive (5500nM) | - | - |
LATS2 | inactive (6500nM) | - | - |
NDR1 | inactive (10001nM) | inactive (97.76%) | - |
NDR2 | inactive (6900nM) | - | - |
AGC - MAST
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAST1 | inactive (10001nM) | - | - |
AGC - PDK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PDK1 | inactive (10001nM) | inactive (82.71%) | inactive (2511.89nM) |
AGC - PKA
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKACa | inactive (10001nM) | inactive (98.11%) | inactive (>3981.07nM) |
PKACb | inactive (10001nM) | - | - |
PRKX | inactive (10001nM) | inactive (136.86%) | inactive (>3162.28nM) |
PKACg | - | inactive (112%) | - |
AGC - PKN
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKN1 | active (1500nM) | inactive (82.56%) | - |
PKN2 | inactive (5000nM) | inactive (99.8%) | inactive (5011.87nM) |
AGC - PKC
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKCd | inactive (10001nM) | inactive (97.51%) | inactive (>7943.28nM) |
PKCe | inactive (10001nM) | inactive (97.8%) | - |
PKCh | inactive (10001nM) | inactive (111.23%) | - |
PKCi | inactive (10001nM) | inactive (98.92%) | - |
PKCt | inactive (5300nM) | inactive (86.03%) | inactive (>1995.26nM) |
PKCa | - | inactive (81.97%) | - |
PKCg | - | inactive (94.16%) | inactive (>7943.28nM) |
PKCz | - | inactive (76.35%) | inactive (7943.28nM) |
PKCb | - | inactive (89.72%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKG1 | inactive (10001nM) | inactive (90.8%) | inactive (>1995.26nM) |
PKG2 | inactive (10001nM) | inactive (105.45%) | inactive (>1584.89nM) |
AGC - RSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
p70S6K | inactive (10001nM) | inactive (95.96%) | inactive (3162.28nM) |
MSK1 | - | inactive (85.7%) | inactive (>1995.26nM) |
MSK2 | - | inactive (100.03%) | - |
p70S6Kb | - | inactive (94.43%) | - |
RSK2 | - | inactive (82.13%) | inactive (>3981.07nM) |
RSK4 | - | inactive (90.73%) | - |
RSK1 | - | inactive (103.02%) | - |
RSK3 | - | inactive (76.05%) | - |
AGC - SGK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SGK3 | inactive (10001nM) | inactive (101.32%) | - |
SGK1 | - | inactive (115.85%) | inactive (>6309.57nM) |
SGK2 | - | inactive (95.47%) | - |
AGC - YANK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
YANK1 | inactive (10001nM) | - | - |
YANK2 | inactive (10001nM) | - | - |
YANK3 | inactive (10001nM) | - | - |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
AMPKa1 | active (1100nM) | - | inactive (2511.89nM) |
AMPKa2 | active (350nM) | - | - |
NuaK1 | active (200nM) | active (18.54%) | - |
BRSK1 | inactive (8400nM) | inactive (112.11%) | inactive (6309.57nM) |
BRSK2 | inactive (10001nM) | inactive (89.6%) | - |
CHK1 | inactive (8700nM) | inactive (77.09%) | inactive (>3162.28nM) |
HUNK | inactive (9800nM) | - | - |
LKB1 | active (1300nM) | inactive (101.84%) | - |
MARK1 | inactive (4900nM) | inactive (114.08%) | - |
MARK2 | active (1400nM) | inactive (117.58%) | active (1000nM) |
MARK3 | active (2500nM) | inactive (96.91%) | inactive (3981.07nM) |
MARK4 | inactive (4900nM) | inactive (87.42%) | active (1000nM) |
MELK | active (240nM) | inactive (53.45%) | active (39.81nM) |
NIM1 | inactive (10001nM) | - | - |
QSK | inactive (10001nM) | - | - |
SIK | active (2500nM) | - | - |
QIK | active (1700nM) | inactive (79.95%) | active (1000nM) |
NuaK2 | active (530nM) | inactive (77.54%) | - |
SNRK | inactive (10001nM) | - | - |
PASK | - | inactive (99.17%) | inactive (>1584.89nM) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CaMK1a | inactive (7000nM) | inactive (102.98%) | inactive (>7943.28nM) |
CaMK1d | inactive (4900nM) | inactive (110.07%) | inactive (>2511.89nM) |
CaMK1g | inactive (6500nM) | inactive (110.87%) | - |
CaMK4 | inactive (10001nM) | inactive (93.9%) | - |
CaMK1b | - | inactive (99.01%) | - |
CAMK - CAMK2
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CaMK2a | inactive (10001nM) | inactive (84.06%) | inactive (>3981.07nM) |
CaMK2b | inactive (10001nM) | inactive (118.49%) | inactive (>7943.28nM) |
CaMK2d | inactive (10001nM) | inactive (87.11%) | inactive (>6309.57nM) |
CaMK2g | inactive (10001nM) | inactive (108.93%) | inactive (>6309.57nM) |
CAMK - CASK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CASK | inactive (10001nM) | - | - |
CAMK - RAD53
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CHK2 | inactive (10001nM) | inactive (100.31%) | inactive (>2511.89nM) |
CAMK - DAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DAPK1 | inactive (10001nM) | inactive (102.24%) | - |
DAPK2 | inactive (10001nM) | inactive (98.15%) | - |
DAPK3 | inactive (9900nM) | inactive (109.32%) | inactive (>5011.87nM) |
DRAK1 | inactive (9000nM) | inactive (104.23%) | - |
DRAK2 | inactive (10001nM) | - | - |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DCLK1 | inactive (10001nM) | - | inactive (>10000nM) |
DCLK2 | inactive (10001nM) | inactive (99.15%) | - |
DCLK3 | inactive (3600nM) | - | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAPKAPK2 | inactive (3800nM) | inactive (100.53%) | inactive (>7943.28nM) |
MAPKAPK5 | inactive (10001nM) | inactive (95.8%) | inactive (>1584.89nM) |
MNK1 | inactive (10001nM) | inactive (92.83%) | - |
MNK2 | inactive (5200nM) | inactive (97.61%) | inactive (>10000nM) |
MAPKAPK3 | - | inactive (97.71%) | inactive (>10000nM) |
CAMK - MLCK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
caMLCK | active (15nM) | - | - |
smMLCK | inactive (10001nM) | inactive (96.96%) | - |
skMLCK | active (43nM) | active (18.9%) | - |
SgK085 | active (2200nM) | - | - |
CAMK - PHK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PHKg1 | active (2200nM) | inactive (69.92%) | - |
PHKg2 | inactive (4400nM) | inactive (90.55%) | inactive (>5011.87nM) |
CAMK - PIM
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PIM1 | inactive (10001nM) | inactive (98.61%) | inactive (>6309.57nM) |
PIM2 | inactive (10001nM) | inactive (97.31%) | inactive (>1584.89nM) |
PIM3 | inactive (10001nM) | inactive (101.1%) | - |
CAMK - PKD
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PKD1 | inactive (10001nM) | inactive (101.68%) | - |
PKD2 | inactive (10001nM) | inactive (77.31%) | inactive (5011.87nM) |
PKD3 | inactive (10001nM) | inactive (86.63%) | inactive (>3981.07nM) |
CAMK - STK33
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
STK33 | inactive (10001nM) | inactive (90.11%) | - |
CAMK - TSSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
TSSK1 | inactive (10001nM) | inactive (90.51%) | inactive (>1584.89nM) |
TSSK2 | - | inactive (83.85%) | inactive (>1584.89nM) |
STE
STE - STE11
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAP3K5 | inactive (10001nM) | inactive (102.08%) | - |
MAP3K6 | inactive (10001nM) | - | - |
MAP3K1 | inactive (10001nM) | - | - |
MAP3K7 | inactive (10001nM) | - | - |
MAP3K2 | active (1100nM) | inactive (116.44%) | - |
MAP3K3 | active (1900nM) | inactive (113.49%) | - |
MAP3K4 | active (2500nM) | - | - |
MAP3K8 | active (51nM) | - | - |
STE - STE20
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
HPK1 | active (72nM) | - | - |
LOK | active (120nM) | active (40.6%) | - |
GCK | active (2600nM) | inactive (102.33%) | inactive (>3162.28nM) |
KHS2 | active (290nM) | - | - |
HGK | active (2400nM) | inactive (92.78%) | inactive (>5011.87nM) |
KHS1 | active (83nM) | active (18.29%) | active (158.49nM) |
MINK | active (1100nM) | inactive (83.04%) | inactive (6309.57nM) |
MST1 | active (200nM) | active (48.86%) | - |
MST2 | active (510nM) | inactive (80.23%) | inactive (>2511.89nM) |
MST3 | inactive (3600nM) | inactive (96.73%) | - |
MST4 | inactive (3500nM) | inactive (130.05%) | - |
MYO3A | inactive (10001nM) | - | - |
MYO3B | inactive (10001nM) | inactive (92.78%) | - |
OSR1 | inactive (10001nM) | inactive (99.47%) | - |
PAK1 | inactive (4400nM) | inactive (100.47%) | inactive (7943.28nM) |
PAK2 | inactive (5700nM) | inactive (93.08%) | - |
PAK3 | inactive (3300nM) | inactive (87.68%) | - |
PAK4 | inactive (4300nM) | inactive (85.44%) | inactive (3981.07nM) |
PAK6 | inactive (9700nM) | inactive (103.93%) | - |
PAK5 | inactive (3300nM) | inactive (91.71%) | - |
SLK | active (82nM) | inactive (59.59%) | active (501.19nM) |
STLK3 | inactive (10001nM) | inactive (94.85%) | - |
TAO1 | active (290nM) | active (44.65%) | active (79.43nM) |
TAO2 | active (430nM) | active (18.65%) | - |
TAO3 | active (81nM) | inactive (76.3%) | - |
TNIK | active (1800nM) | - | - |
YSK1 | inactive (4800nM) | inactive (94.76%) | - |
STE - STE7
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
MAP2K1 | active (1800nM) | inactive (89.67%) | inactive (1258.93nM) |
MAP2K2 | active (2000nM) | inactive (91.34%) | inactive (1995.26nM) |
MAP2K3 | inactive (10001nM) | - | - |
MAP2K4 | inactive (10001nM) | - | - |
MAP2K5 | active (260nM) | - | - |
MAP2K6 | active (2600nM) | inactive (98.64%) | - |
MAP2K7 | inactive (10001nM) | - | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
COT | - | inactive (114.59%) | - |
NIK | - | inactive (110.51%) | - |
CMGC
CMGC - CDK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
PITSLRE | active (290nM) | - | - |
CHED | inactive (10001nM) | - | - |
CDK11 | inactive (10001nM) | - | active (199.53nM) |
PCTAIRE1 | active (230nM) | - | - |
PCTAIRE2 | inactive (5600nM) | - | - |
PCTAIRE3 | inactive (10001nM) | - | - |
PFTAIRE2 | inactive (10001nM) | - | - |
PFTAIRE1 | inactive (10001nM) | - | - |
CDC2 | - | - | inactive (>7943.28nM) |
CDK2 | - | - | inactive (>7943.28nM) |
CDK5 | - | - | inactive (>3162.28nM) |
CDK8 | - | - | inactive (>3981.07nM) |
CDK7 | - | - | inactive (>3981.07nM) |
CDK9 | - | - | inactive (>1584.89nM) |
CMGC - CDKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CDKL1 | inactive (10001nM) | - | - |
CDKL2 | active (49nM) | - | - |
CDKL3 | active (350nM) | - | - |
CDKL5 | active (2800nM) | - | - |
CMGC - CLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CLK1 | inactive (10001nM) | inactive (106.46%) | - |
CLK2 | inactive (10001nM) | inactive (88%) | inactive (>3981.07nM) |
CLK3 | inactive (10001nM) | inactive (109.96%) | - |
CLK4 | inactive (10001nM) | inactive (90.04%) | inactive (>3162.28nM) |
CMGC - CK2
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CK2a1 | inactive (10001nM) | inactive (114.11%) | inactive (>6309.57nM) |
CK2a2 | inactive (10001nM) | inactive (120.5%) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
DYRK1A | inactive (10001nM) | inactive (98.44%) | inactive (>1995.26nM) |
DYRK1B | inactive (10001nM) | inactive (98.82%) | inactive (>2511.89nM) |
DYRK2 | inactive (10001nM) | inactive (101.31%) | - |
HIPK1 | inactive (10001nM) | inactive (98.59%) | - |
HIPK2 | inactive (10001nM) | inactive (101.95%) | inactive (>3162.28nM) |
HIPK3 | inactive (10001nM) | inactive (99.11%) | - |
HIPK4 | inactive (10001nM) | inactive (95.26%) | inactive (>7943.28nM) |
PRP4 | active (2500nM) | - | - |
DYRK3 | - | inactive (105.47%) | inactive (>6309.57nM) |
DYRK4 | - | inactive (97.44%) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
Erk1 | inactive (10001nM) | inactive (96.05%) | - |
Erk2 | inactive (10001nM) | inactive (91.22%) | inactive (>7943.28nM) |
Erk3 | inactive (10001nM) | - | - |
Erk4 | inactive (10001nM) | - | - |
Erk5 | inactive (6800nM) | - | - |
Erk7 | inactive (10001nM) | - | - |
JNK1 | inactive (10001nM) | inactive (95.39%) | inactive (>5011.87nM) |
JNK2 | inactive (10001nM) | inactive (108.41%) | inactive (>3981.07nM) |
JNK3 | active (2800nM) | inactive (106.54%) | inactive (1995.26nM) |
NLK | inactive (10001nM) | inactive (102.52%) | - |
p38a | inactive (10001nM) | inactive (97.15%) | inactive (>3981.07nM) |
p38b | inactive (10001nM) | inactive (93.48%) | - |
p38d | inactive (10001nM) | inactive (89.5%) | inactive (>7943.28nM) |
p38g | inactive (10001nM) | inactive (96.22%) | inactive (>6309.57nM) |
CMGC - GSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
GSK3A | inactive (10001nM) | inactive (101.05%) | inactive (>3981.07nM) |
GSK3B | inactive (10001nM) | inactive (104.07%) | inactive (>3981.07nM) |
CMGC - RCK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
ICK | inactive (10001nM) | - | - |
MAK | inactive (10001nM) | - | - |
CMGC - SRPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
SRPK1 | active (82nM) | inactive (96.44%) | inactive (>7943.28nM) |
SRPK2 | active (680nM) | inactive (94.65%) | - |
MSSK1 | active (240nM) | inactive (105.34%) | - |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz |
---|
CK1 | 7 | 7 | 6 | 5 |
VRK | 3 | 1 | 1 | - |
CK1 - CK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
CK1a | inactive (10001nM) | inactive (96.67%) | inactive (>3981.07nM) |
CK1a2 | inactive (10001nM) | - | - |
CK1d | inactive (10001nM) | inactive (92.6%) | inactive (>7943.28nM) |
CK1e | inactive (10001nM) | inactive (98.78%) | - |
CK1g1 | inactive (10001nM) | inactive (99.08%) | inactive (>6309.57nM) |
CK1g2 | inactive (10001nM) | inactive (96.15%) | inactive (>7943.28nM) |
CK1g3 | inactive (10001nM) | inactive (100.26%) | - |
CK1 - VRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz |
---|
VRK2 | inactive (10001nM) | - | - |
VRK1 | - | inactive (107.36%) | - |