Compound Information
Test on : RBC, Millipore
Compound Name
RBC : N-(3-chlorophenyl)-3-[[3,5-dimethyl-4-[(4-methyl-1-piperazinyl)-oxomethyl]-1H-pyrrol-2-yl]methylidene]-N-methyl-2-oxo-1H-indole-5-sulfonamide
Millipore : SU11274
Inchikey
Same : FPYJSJDOHRDAMT-N
RBC : FPYJSJDOHRDAMT-UHFFFAOYSA-N
Millipore : FPYJSJDOHRDAMT-KQWNVCNZSA-N
ChemSpider
RBC : 26470841
Millipore : 7828213
Pubchem CID
RBC : 53396327
Millipore : 9549297
ChEMBL
RBC : -
Millipore : CHEMBL261641
RBC | Millipore |
| |
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDK1 | inactive (114.1%) | inactive (109%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AKT1 | inactive (98.8%) | inactive (103%) |
AKT2 | inactive (102.27%) | inactive (106%) |
AKT3 | inactive (106.6%) | inactive (103%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DMPK1 | inactive (113.44%) | inactive (51%) |
MRCKa | inactive (104.84%) | inactive (110%) |
MRCKb | inactive (113.19%) | inactive (99%) |
ROCK1 | inactive (83.99%) | inactive (123%) |
ROCK2 | inactive (58.23%) | inactive (71%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BARK1 | inactive (104.62%) | - |
BARK2 | inactive (102.85%) | - |
GPRK4 | inactive (103.37%) | - |
GPRK5 | inactive (98.93%) | inactive (102%) |
GPRK6 | inactive (89.65%) | inactive (100%) |
GPRK7 | inactive (86.75%) | inactive (65%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSK1 | inactive (94.14%) | inactive (123%) |
MSK2 | inactive (108.6%) | inactive (102%) |
p70S6K | inactive (83.7%) | inactive (66%) |
p70S6Kb | inactive (98.38%) | - |
RSK2 | inactive (76.79%) | active (44%) |
RSK4 | inactive (67.79%) | inactive (81%) |
RSK1 | inactive (54.36%) | inactive (95%) |
RSK3 | inactive (75.37%) | inactive (93%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKACg | inactive (111.08%) | - |
PRKX | inactive (103.92%) | inactive (99%) |
PKACa | inactive (100.17%) | inactive (86%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKCa | inactive (91.91%) | inactive (103%) |
PKCd | inactive (95.29%) | inactive (97%) |
PKCe | inactive (99.07%) | inactive (97%) |
PKCh | inactive (88.66%) | inactive (111%) |
PKCg | inactive (94.77%) | inactive (105%) |
PKCi | inactive (98.71%) | inactive (88%) |
PKCt | inactive (106.8%) | inactive (106%) |
PKCz | inactive (94.54%) | inactive (100%) |
PKCb | inactive (99.11%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKG2 | inactive (104.19%) | - |
PKG1 | inactive (97.08%) | - |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKN1 | inactive (86.39%) | - |
PKN2 | inactive (85.39%) | active (41%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SGK1 | inactive (102.98%) | inactive (94%) |
SGK2 | inactive (103.4%) | inactive (106%) |
SGK3 | inactive (101.3%) | inactive (114%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NDR1 | inactive (101.72%) | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ABL1 | inactive (89.15%) | inactive (110%) |
ABL2 | inactive (73.2%) | inactive (76%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ACK | inactive (65.43%) | inactive (79%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK | inactive (77.66%) | inactive (66%) |
LTK | active (45.52%) | - |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AXL | inactive (66.5%) | active (13%) |
MER | active (21.36%) | active (1%) |
TYRO3 | active (34.71%) | active (48%) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BLK | inactive (51.66%) | active (16%) |
BRK | inactive (91.25%) | inactive (102%) |
SRC | inactive (53.34%) | inactive (77%) |
FGR | active (39.24%) | active (35%) |
FRK | inactive (95.39%) | inactive (107%) |
FYN | inactive (67.08%) | inactive (86%) |
HCK | inactive (63.52%) | inactive (53%) |
LCK | active (29.32%) | inactive (53%) |
SRM | inactive (104.33%) | - |
YES | active (26.98%) | active (14%) |
LYN | active (39.12%) | active (23%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BMX | inactive (97.29%) | inactive (86%) |
BTK | inactive (93.08%) | inactive (101%) |
ITK | inactive (87.35%) | inactive (81%) |
TEC | inactive (86.72%) | - |
TXK | inactive (101.83%) | inactive (111%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
KIT | inactive (51.27%) | active (31%) |
FLT3 | active (26.46%) | inactive (67%) |
FMS | inactive (64.88%) | active (17%) |
PDGFRb | inactive (76.41%) | inactive (83%) |
PDGFRa | inactive (72.78%) | active (48%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CSK | inactive (78.21%) | inactive (119%) |
CTK | inactive (100.24%) | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DDR2 | inactive (105.16%) | inactive (99%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EGFR | inactive (97.09%) | inactive (114%) |
ErbB2 | inactive (91.5%) | - |
ErbB4 | inactive (105.39%) | inactive (110%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EphA1 | inactive (107.68%) | inactive (85%) |
EphA2 | inactive (97.81%) | inactive (99%) |
EphA3 | inactive (103.1%) | inactive (110%) |
EphA4 | inactive (80.67%) | inactive (97%) |
EphA5 | inactive (96.41%) | inactive (98%) |
EphA6 | active (24%) | - |
EphA7 | inactive (85.81%) | inactive (96%) |
EphA8 | inactive (91.65%) | inactive (102%) |
EphB1 | inactive (84.55%) | inactive (103%) |
EphB2 | inactive (91.81%) | inactive (91%) |
EphB3 | inactive (98.6%) | inactive (112%) |
EphB4 | inactive (95.38%) | inactive (108%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FAK | inactive (96.8%) | inactive (129%) |
PYK2 | inactive (57.71%) | active (43%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FER | inactive (81.03%) | inactive (107%) |
FES | inactive (95.99%) | inactive (127%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FGFR1 | inactive (79.96%) | inactive (55%) |
FGFR2 | inactive (74.12%) | inactive (62%) |
FGFR3 | inactive (74.15%) | inactive (74%) |
FGFR4 | inactive (104.01%) | inactive (102%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FLT1 | inactive (74.65%) | active (37%) |
FLT4 | inactive (55.06%) | active (45%) |
KDR | inactive (79.42%) | inactive (51%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IGF1R | inactive (103.31%) | inactive (129%) |
IRR | inactive (93.05%) | inactive (110%) |
INSR | inactive (98.84%) | inactive (104%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
JAK1 | inactive (68.04%) | - |
JAK2 | active (40.6%) | active (35%) |
JAK3 | active (47.02%) | inactive (54%) |
TYK2 | inactive (75.14%) | - |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MUSK | inactive (84.19%) | active (46%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RET | active (23.04%) | active (20%) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RON | inactive (102.57%) | inactive (61%) |
MET | active (1.18%) | active (2%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ROS | inactive (69.56%) | inactive (96%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SYK | inactive (96.73%) | inactive (124%) |
ZAP70 | inactive (94.35%) | inactive (98%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TIE2 | inactive (90.84%) | active (43%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TRKA | active (7.81%) | active (0%) |
TRKB | active (35.73%) | active (15%) |
TRKC | active (5.93%) | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK1 | inactive (102.66%) | - |
ALK2 | inactive (96.82%) | - |
ALK4 | inactive (102.15%) | inactive (131%) |
TGFbR1 | inactive (103.45%) | inactive (86%) |
TGFbR2 | inactive (127.42%) | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ARAF | inactive (119.58%) | - |
BRAF | inactive (91.88%) | - |
RAF1 | inactive (114.06%) | inactive (97%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IRAK1 | inactive (57.69%) | active (37%) |
IRAK4 | inactive (65.54%) | inactive (64%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LIMK1 | inactive (87.91%) | inactive (93%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LRRK2 | active (6.63%) | - |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MLK1 | inactive (95.18%) | inactive (79%) |
MLK2 | inactive (74.04%) | - |
MLK3 | inactive (79.15%) | - |
TAK1 | inactive (79.77%) | inactive (88%) |
ZAK | inactive (97.35%) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RIPK2 | inactive (92.72%) | inactive (99%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NuaK1 | active (15.9%) | active (30%) |
BRSK1 | inactive (100.51%) | inactive (71%) |
BRSK2 | inactive (89.04%) | inactive (79%) |
CHK1 | inactive (89.71%) | inactive (91%) |
LKB1 | inactive (89.9%) | inactive (105%) |
MARK1 | inactive (62.52%) | active (44%) |
MARK3 | active (41.9%) | - |
MARK4 | active (36.22%) | - |
MELK | inactive (78.94%) | inactive (71%) |
PASK | inactive (105.92%) | inactive (121%) |
QIK | inactive (86.01%) | - |
NuaK2 | inactive (61.94%) | - |
MARK2 | active (44.14%) | active (48%) |
AMPKa1 | - | active (25%) |
AMPKa2 | - | active (33%) |
SIK | - | inactive (79%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK1a | inactive (95.78%) | inactive (95%) |
CaMK1b | inactive (100.94%) | - |
CaMK1d | inactive (137.51%) | inactive (97%) |
CaMK1g | inactive (92.48%) | - |
CaMK4 | inactive (96.18%) | inactive (97%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK2a | inactive (73.81%) | - |
CaMK2b | inactive (89.78%) | inactive (97%) |
CaMK2d | inactive (68.35%) | active (44%) |
CaMK2g | inactive (118.81%) | active (46%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CHK2 | inactive (85.08%) | inactive (84%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DAPK1 | inactive (105.72%) | inactive (98%) |
DAPK2 | inactive (111.07%) | inactive (100%) |
DRAK1 | inactive (97.04%) | inactive (128%) |
DAPK3 | inactive (105.56%) | inactive (105%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DCLK2 | inactive (90.37%) | inactive (85%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAPKAPK2 | inactive (103.87%) | inactive (96%) |
MAPKAPK3 | inactive (96.94%) | inactive (107%) |
MAPKAPK5 | inactive (77.6%) | inactive (129%) |
MNK1 | inactive (104.92%) | - |
MNK2 | inactive (106.48%) | inactive (105%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
smMLCK | inactive (84.3%) | inactive (76%) |
skMLCK | inactive (73.79%) | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PHKg1 | active (45.19%) | - |
PHKg2 | inactive (96%) | inactive (92%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PIM1 | inactive (102.86%) | inactive (92%) |
PIM2 | inactive (103.21%) | inactive (101%) |
PIM3 | inactive (106.06%) | inactive (93%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKD1 | inactive (61.8%) | inactive (87%) |
PKD3 | active (42.7%) | - |
PKD2 | inactive (58.26%) | inactive (107%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TSSK1 | active (21.73%) | active (40%) |
TSSK2 | inactive (96.28%) | inactive (93%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
STK33 | inactive (67.88%) | inactive (84%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP3K5 | inactive (104.67%) | inactive (81%) |
MAP3K2 | inactive (68.53%) | - |
MAP3K3 | inactive (63.63%) | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
COT | inactive (82.94%) | - |
NIK | inactive (109.36%) | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GCK | inactive (53.53%) | active (33%) |
HGK | active (40.9%) | - |
KHS1 | active (5.06%) | - |
LOK | active (9.05%) | active (13%) |
MINK | inactive (68.68%) | inactive (65%) |
MST1 | active (49.13%) | inactive (82%) |
MST2 | inactive (78.61%) | inactive (89%) |
MST3 | active (49.57%) | active (21%) |
MST4 | inactive (63.52%) | - |
OSR1 | inactive (115.8%) | - |
PAK1 | inactive (87.74%) | - |
PAK2 | inactive (96.2%) | inactive (99%) |
PAK3 | inactive (93.53%) | active (45%) |
PAK4 | inactive (101.29%) | inactive (95%) |
PAK5 | inactive (97.09%) | inactive (98%) |
PAK6 | inactive (108.38%) | inactive (93%) |
SLK | active (13.61%) | - |
YSK1 | inactive (91%) | - |
STLK3 | inactive (84.75%) | - |
TAO1 | active (41.89%) | active (34%) |
TAO2 | active (21.85%) | active (19%) |
TAO3 | inactive (61.55%) | active (26%) |
MYO3B | inactive (72.51%) | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP2K1 | inactive (89.26%) | active (43%) |
MAP2K2 | inactive (99.55%) | - |
MAP2K6 | inactive (91.9%) | inactive (73%) |
MAP2K7 | - | inactive (101%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AurA | active (27.55%) | active (5%) |
AurB | active (19.22%) | active (3%) |
AurC | active (37.94%) | active (18%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMKK1 | inactive (93.26%) | - |
CaMKK2 | inactive (75.16%) | - |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Haspin | inactive (101.93%) | inactive (90%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IKKa | inactive (100.02%) | inactive (101%) |
IKKb | inactive (107.18%) | inactive (104%) |
IKKe | inactive (74.18%) | - |
TBK1 | inactive (60.43%) | inactive (60%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NEK1 | active (23.52%) | - |
NEK11 | inactive (102.94%) | inactive (76%) |
NEK2 | inactive (50.8%) | active (39%) |
NEK4 | inactive (79.74%) | - |
NEK6 | inactive (103.56%) | inactive (95%) |
NEK7 | inactive (90.33%) | inactive (101%) |
NEK9 | inactive (92.52%) | - |
NEK3 | inactive (98.66%) | inactive (107%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PBK | inactive (103.76%) | - |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PLK1 | inactive (96.86%) | inactive (93%) |
PLK2 | inactive (96.4%) | inactive (101%) |
PLK3 | inactive (94.97%) | inactive (100%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SgK496 | inactive (97.19%) | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MPSK1 | inactive (95.41%) | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TTK | inactive (90.7%) | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ULK1 | active (5.17%) | - |
ULK2 | active (16.84%) | active (14%) |
ULK3 | inactive (55.29%) | active (30%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wee1 | inactive (81.85%) | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wnk2 | inactive (111.59%) | inactive (116%) |
Wnk3 | - | inactive (111%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TLK2 | inactive (95.83%) | inactive (106%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK1 | 7 | 6 | 4 |
VRK | 3 | 1 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK1d | inactive (83.5%) | inactive (69%) |
CK1g1 | inactive (104.34%) | inactive (99%) |
CK1g2 | inactive (99.69%) | inactive (77%) |
CK1g3 | inactive (93.31%) | inactive (84%) |
CK1a | inactive (79.16%) | - |
CK1e | inactive (76.14%) | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
VRK1 | inactive (87.28%) | - |
VRK2 | - | inactive (112%) |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK2 | 3 | 2 | 2 |
CLK | 4 | 4 | 2 |
DYRK | 10 | 9 | 4 |
MAPK | 14 | 10 | 10 |
GSK | 2 | 2 | 2 |
SRPK | 3 | 3 | 3 |
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK2a1 | inactive (78.8%) | inactive (84%) |
CK2a2 | inactive (84.58%) | inactive (121%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CLK1 | - | - |
CLK2 | active (5.1%) | active (7%) |
CLK3 | inactive (71.07%) | inactive (51%) |
CLK4 | active (34.31%) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DYRK1A | inactive (94.06%) | - |
DYRK1B | inactive (98.87%) | - |
DYRK2 | inactive (101.22%) | inactive (86%) |
DYRK3 | - | - |
DYRK4 | inactive (96.06%) | - |
HIPK1 | inactive (103.81%) | inactive (100%) |
HIPK2 | inactive (104.6%) | inactive (78%) |
HIPK3 | inactive (102.55%) | inactive (78%) |
HIPK4 | inactive (102.88%) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Erk1 | inactive (106.49%) | inactive (90%) |
Erk2 | inactive (85.1%) | inactive (93%) |
JNK3 | inactive (99.03%) | inactive (97%) |
NLK | inactive (105.73%) | inactive (111%) |
p38a | inactive (86.24%) | inactive (94%) |
p38b | inactive (103.39%) | inactive (104%) |
p38d | inactive (100.26%) | inactive (106%) |
p38g | inactive (99.82%) | inactive (107%) |
JNK1 | inactive (86.94%) | inactive (108%) |
JNK2 | inactive (77.97%) | inactive (106%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GSK3A | inactive (98.44%) | inactive (109%) |
GSK3B | inactive (96.1%) | inactive (100%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSSK1 | inactive (84.77%) | inactive (105%) |
SRPK1 | inactive (77.32%) | inactive (72%) |
SRPK2 | inactive (60.55%) | inactive (65%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
PDHK | 5 | 1 | - |
Alpha | 6 | - | 1 |
PIKK | 6 | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDHK1 | inactive (114.1%) | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
eEF2K | - | inactive (79%) |
Atypical - PIKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FRAP | - | inactive (88%) |