Compound Information
Test on : RBC, Millipore
Compound Name
RBC : 2-amino-4-(4-hydroxyphenyl)buta-1,3-diene-1,1,3-tricarbonitrile
Millipore : Tyrphostin AG 112
Inchikey
Same : DXVJRTIPBNBLLB-N
RBC : DXVJRTIPBNBLLB-UHFFFAOYSA-N
Millipore : DXVJRTIPBNBLLB-BJMVGYQFSA-N
ChemSpider
RBC : 1964
Millipore : 4485966
Pubchem CID
RBC : 2045
Millipore : 5328804
ChEMBL
RBC : -
Millipore : CHEMBL76589
RBC | Millipore |
| |
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDK1 | inactive (99.38%) | inactive (106%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AKT1 | inactive (99.24%) | inactive (112%) |
AKT2 | inactive (92.82%) | inactive (118%) |
AKT3 | inactive (95.76%) | inactive (103%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DMPK1 | inactive (100.63%) | inactive (103%) |
MRCKa | inactive (96.21%) | inactive (90%) |
MRCKb | inactive (108.57%) | inactive (96%) |
ROCK1 | inactive (100.47%) | inactive (112%) |
ROCK2 | inactive (98.26%) | inactive (105%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BARK1 | inactive (103.62%) | - |
BARK2 | inactive (96.67%) | - |
GPRK4 | inactive (99.58%) | - |
GPRK5 | inactive (113.24%) | inactive (101%) |
GPRK6 | inactive (107.38%) | inactive (94%) |
GPRK7 | inactive (104.49%) | inactive (98%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSK1 | inactive (96.72%) | inactive (122%) |
MSK2 | inactive (99.71%) | inactive (91%) |
p70S6K | inactive (89.49%) | inactive (66%) |
p70S6Kb | inactive (96.83%) | - |
RSK2 | inactive (94.56%) | active (49%) |
RSK4 | inactive (103.62%) | inactive (94%) |
RSK1 | inactive (93.78%) | inactive (108%) |
RSK3 | inactive (96.16%) | inactive (94%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKACg | inactive (96.8%) | - |
PRKX | inactive (93.75%) | inactive (99%) |
PKACa | inactive (100.23%) | inactive (82%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKCa | inactive (97.35%) | inactive (109%) |
PKCd | inactive (93.7%) | inactive (102%) |
PKCe | inactive (89.32%) | inactive (95%) |
PKCh | inactive (90.32%) | inactive (118%) |
PKCg | inactive (105.06%) | inactive (113%) |
PKCi | inactive (97.41%) | inactive (81%) |
PKCt | inactive (99.78%) | inactive (101%) |
PKCz | inactive (105.36%) | inactive (94%) |
PKCb | inactive (111.01%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKG2 | inactive (86.94%) | - |
PKG1 | inactive (91.27%) | - |
AGC - PKN
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKN1 | inactive (88.98%) | - |
PKN2 | inactive (96.89%) | inactive (101%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SGK1 | inactive (96.11%) | inactive (95%) |
SGK2 | inactive (109.74%) | inactive (93%) |
SGK3 | inactive (103.38%) | inactive (115%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NDR1 | inactive (96.92%) | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ABL1 | inactive (102.76%) | inactive (87%) |
ABL2 | inactive (94.9%) | inactive (93%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ACK | inactive (98.05%) | inactive (84%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK | inactive (108.52%) | inactive (88%) |
LTK | inactive (92.47%) | - |
TK - Axl
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AXL | inactive (93.67%) | inactive (92%) |
MER | inactive (93.49%) | inactive (110%) |
TYRO3 | inactive (99.26%) | inactive (104%) |
TK - Src
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BLK | inactive (101.03%) | inactive (103%) |
BRK | inactive (84.85%) | inactive (102%) |
SRC | inactive (92.35%) | inactive (83%) |
FGR | inactive (98.74%) | inactive (109%) |
FRK | inactive (98.95%) | inactive (102%) |
FYN | inactive (98.4%) | inactive (104%) |
HCK | inactive (98.65%) | inactive (84%) |
LCK | inactive (95.06%) | inactive (116%) |
SRM | inactive (107.15%) | - |
YES | inactive (100.21%) | inactive (114%) |
LYN | inactive (92.18%) | inactive (93%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
BMX | inactive (79.96%) | inactive (104%) |
BTK | inactive (99.7%) | inactive (94%) |
ITK | inactive (98.67%) | inactive (95%) |
TEC | inactive (94.66%) | - |
TXK | inactive (100.08%) | inactive (78%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
KIT | inactive (92.44%) | inactive (104%) |
FLT3 | inactive (92.2%) | inactive (100%) |
FMS | inactive (98.05%) | inactive (79%) |
PDGFRb | inactive (98.84%) | inactive (99%) |
PDGFRa | inactive (97.78%) | inactive (119%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CSK | inactive (97.58%) | inactive (100%) |
CTK | inactive (92.52%) | - |
TK - DDR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DDR2 | inactive (97.6%) | inactive (116%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EGFR | inactive (78.67%) | inactive (109%) |
ErbB2 | inactive (90.08%) | - |
ErbB4 | inactive (92.74%) | inactive (95%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
EphA1 | inactive (103.18%) | inactive (91%) |
EphA2 | inactive (99.95%) | inactive (102%) |
EphA3 | inactive (98.31%) | inactive (110%) |
EphA4 | inactive (96%) | inactive (111%) |
EphA5 | inactive (94.26%) | inactive (125%) |
EphA6 | inactive (98.65%) | - |
EphA7 | inactive (90.53%) | inactive (91%) |
EphA8 | inactive (102.3%) | inactive (98%) |
EphB1 | inactive (88.34%) | inactive (100%) |
EphB2 | inactive (97.08%) | inactive (115%) |
EphB3 | inactive (99.53%) | inactive (118%) |
EphB4 | inactive (88.13%) | inactive (116%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FAK | inactive (98.5%) | inactive (132%) |
PYK2 | inactive (97.39%) | inactive (129%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FER | inactive (91.11%) | inactive (112%) |
FES | inactive (101.47%) | inactive (96%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FGFR1 | inactive (95.29%) | inactive (100%) |
FGFR2 | inactive (102.27%) | inactive (113%) |
FGFR3 | inactive (98.87%) | inactive (99%) |
FGFR4 | inactive (91.09%) | inactive (135%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FLT1 | inactive (90.65%) | inactive (96%) |
FLT4 | inactive (95.91%) | inactive (94%) |
KDR | inactive (97.2%) | inactive (105%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IGF1R | inactive (90.56%) | inactive (106%) |
IRR | inactive (99.88%) | inactive (142%) |
INSR | inactive (94.16%) | inactive (113%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
JAK1 | inactive (99.4%) | - |
JAK2 | inactive (101.85%) | inactive (101%) |
JAK3 | inactive (102.08%) | inactive (101%) |
TYK2 | inactive (97.35%) | - |
TK - Musk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MUSK | inactive (103.36%) | inactive (102%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RET | inactive (109.83%) | inactive (93%) |
TK - Met
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RON | inactive (101.52%) | inactive (113%) |
MET | inactive (116.93%) | inactive (101%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ROS | inactive (97.13%) | inactive (95%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SYK | inactive (100.81%) | inactive (116%) |
ZAP70 | inactive (96.04%) | inactive (128%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TIE2 | inactive (104.15%) | inactive (84%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TRKA | inactive (101.99%) | inactive (121%) |
TRKB | inactive (95.37%) | inactive (99%) |
TRKC | inactive (95.5%) | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ALK1 | inactive (88.83%) | - |
ALK2 | inactive (93.8%) | - |
ALK4 | inactive (100.84%) | inactive (122%) |
TGFbR1 | inactive (92.98%) | inactive (91%) |
TGFbR2 | inactive (113.24%) | - |
TKL - RAF
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ARAF | inactive (90.77%) | - |
BRAF | inactive (90.14%) | - |
RAF1 | inactive (86.32%) | inactive (92%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IRAK1 | inactive (122.98%) | inactive (103%) |
IRAK4 | inactive (92.61%) | inactive (109%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LIMK1 | inactive (89.86%) | inactive (106%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
LRRK2 | inactive (97.09%) | - |
TKL - MLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MLK1 | inactive (94.41%) | inactive (99%) |
MLK2 | inactive (97.96%) | - |
MLK3 | inactive (94.75%) | - |
TAK1 | inactive (94.77%) | inactive (102%) |
ZAK | inactive (95.68%) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
RIPK2 | inactive (95.48%) | inactive (103%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NuaK1 | inactive (92.31%) | inactive (105%) |
BRSK1 | inactive (99.25%) | inactive (72%) |
BRSK2 | inactive (101.45%) | inactive (106%) |
CHK1 | inactive (98.32%) | inactive (90%) |
LKB1 | inactive (96.5%) | inactive (105%) |
MARK1 | inactive (110.82%) | inactive (89%) |
MARK3 | inactive (96.47%) | - |
MARK4 | inactive (94.33%) | - |
MELK | inactive (101.03%) | inactive (70%) |
PASK | inactive (82.87%) | inactive (99%) |
QIK | inactive (87.65%) | - |
NuaK2 | inactive (121.73%) | - |
MARK2 | inactive (91.29%) | inactive (103%) |
AMPKa1 | - | inactive (92%) |
AMPKa2 | - | inactive (100%) |
SIK | - | inactive (90%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK1a | inactive (97.21%) | inactive (109%) |
CaMK1b | inactive (97.35%) | - |
CaMK1d | inactive (98.87%) | inactive (109%) |
CaMK1g | inactive (104.41%) | - |
CaMK4 | inactive (97.24%) | inactive (110%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMK2a | inactive (103%) | - |
CaMK2b | inactive (93.29%) | inactive (96%) |
CaMK2d | inactive (91.1%) | inactive (108%) |
CaMK2g | inactive (89.42%) | inactive (116%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CHK2 | inactive (95.53%) | inactive (88%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DAPK1 | inactive (92.65%) | inactive (85%) |
DAPK2 | inactive (95.7%) | inactive (99%) |
DRAK1 | inactive (72.83%) | inactive (91%) |
DAPK3 | inactive (91.05%) | inactive (103%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DCLK2 | inactive (100.61%) | inactive (94%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAPKAPK2 | inactive (91.3%) | inactive (94%) |
MAPKAPK3 | inactive (99.9%) | inactive (139%) |
MAPKAPK5 | inactive (94.23%) | inactive (101%) |
MNK1 | inactive (77.2%) | - |
MNK2 | inactive (79.12%) | inactive (99%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
smMLCK | inactive (100.99%) | inactive (68%) |
skMLCK | inactive (99.44%) | - |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PHKg1 | inactive (92.48%) | - |
PHKg2 | inactive (96.67%) | inactive (96%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PIM1 | inactive (102.73%) | inactive (80%) |
PIM2 | inactive (88.17%) | inactive (104%) |
PIM3 | inactive (91.3%) | inactive (102%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PKD1 | inactive (101.34%) | inactive (93%) |
PKD3 | inactive (91.94%) | - |
PKD2 | inactive (100.4%) | inactive (101%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TSSK1 | inactive (111.45%) | inactive (98%) |
TSSK2 | inactive (94.63%) | inactive (85%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
STK33 | inactive (93.23%) | inactive (97%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP3K5 | inactive (103.02%) | inactive (81%) |
MAP3K2 | inactive (102.3%) | - |
MAP3K3 | inactive (78.57%) | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
COT | inactive (96.04%) | - |
NIK | inactive (107.9%) | - |
STE - STE20
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GCK | inactive (100.43%) | inactive (84%) |
HGK | inactive (91.18%) | - |
KHS1 | inactive (99.58%) | - |
LOK | inactive (92.43%) | inactive (98%) |
MINK | inactive (97.74%) | inactive (89%) |
MST1 | inactive (99.14%) | inactive (106%) |
MST2 | inactive (95.25%) | inactive (108%) |
MST3 | inactive (103.45%) | inactive (71%) |
MST4 | inactive (101%) | - |
OSR1 | inactive (72.18%) | - |
PAK1 | inactive (90.87%) | - |
PAK2 | inactive (85.99%) | inactive (88%) |
PAK3 | inactive (98.39%) | inactive (82%) |
PAK4 | inactive (85.58%) | inactive (98%) |
PAK5 | inactive (94.55%) | inactive (95%) |
PAK6 | inactive (97.01%) | inactive (100%) |
SLK | inactive (102.11%) | - |
YSK1 | inactive (90.38%) | - |
STLK3 | inactive (90.31%) | - |
TAO1 | inactive (93.16%) | inactive (101%) |
TAO2 | inactive (97.26%) | inactive (104%) |
TAO3 | inactive (101.91%) | inactive (99%) |
MYO3B | inactive (88.11%) | - |
STE - STE7
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MAP2K1 | inactive (93.68%) | inactive (104%) |
MAP2K2 | inactive (102.52%) | - |
MAP2K6 | inactive (93.97%) | inactive (91%) |
MAP2K7 | - | inactive (94%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
AurA | inactive (89.64%) | inactive (83%) |
AurB | inactive (90.96%) | inactive (81%) |
AurC | inactive (101.2%) | inactive (105%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CaMKK1 | inactive (104.21%) | - |
CaMKK2 | inactive (91.56%) | - |
Other - Haspin
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Haspin | inactive (90.13%) | inactive (88%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
IKKa | inactive (94%) | inactive (96%) |
IKKb | inactive (101.81%) | inactive (99%) |
IKKe | inactive (91.04%) | - |
TBK1 | inactive (91.1%) | inactive (82%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
NEK1 | inactive (95.71%) | - |
NEK11 | inactive (97.24%) | inactive (75%) |
NEK2 | inactive (102.08%) | inactive (91%) |
NEK4 | inactive (93.27%) | - |
NEK6 | inactive (97.33%) | inactive (102%) |
NEK7 | inactive (98.86%) | inactive (116%) |
NEK9 | inactive (97.92%) | - |
NEK3 | inactive (97.96%) | inactive (115%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PBK | inactive (96.42%) | - |
Other - PLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PLK1 | inactive (60.78%) | inactive (79%) |
PLK2 | inactive (99.88%) | inactive (104%) |
PLK3 | inactive (63.63%) | inactive (79%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
SgK496 | inactive (92.92%) | - |
Other - NAK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MPSK1 | inactive (109.02%) | - |
Other - TTK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TTK | inactive (94.43%) | - |
Other - ULK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
ULK1 | inactive (89.28%) | - |
ULK2 | inactive (104.53%) | inactive (108%) |
ULK3 | inactive (67.82%) | inactive (100%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wee1 | inactive (93.67%) | - |
Other - WNK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Wnk2 | inactive (103.32%) | inactive (103%) |
Wnk3 | inactive (99.81%) | inactive (96%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
TLK2 | inactive (89.4%) | inactive (100%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK1 | 7 | 6 | 4 |
VRK | 3 | 1 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK1d | inactive (98.68%) | inactive (82%) |
CK1g1 | inactive (93.41%) | inactive (83%) |
CK1g2 | inactive (103.53%) | inactive (85%) |
CK1g3 | inactive (100.38%) | inactive (90%) |
CK1a | inactive (85.02%) | - |
CK1e | inactive (92.37%) | - |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
VRK1 | inactive (103.11%) | - |
VRK2 | - | inactive (100%) |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
CK2 | 3 | 2 | 2 |
CLK | 4 | 4 | 2 |
DYRK | 10 | 9 | 4 |
MAPK | 14 | 10 | 10 |
GSK | 2 | 2 | 2 |
SRPK | 3 | 3 | 3 |
CMGC - CK2
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CK2a1 | inactive (103.88%) | inactive (91%) |
CK2a2 | inactive (101.63%) | inactive (120%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
CLK1 | inactive (96.53%) | - |
CLK2 | inactive (100.16%) | inactive (109%) |
CLK3 | inactive (100.29%) | inactive (87%) |
CLK4 | inactive (100.71%) | - |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
DYRK1A | inactive (95.86%) | - |
DYRK1B | inactive (101.14%) | - |
DYRK2 | inactive (116.76%) | inactive (85%) |
DYRK3 | inactive (97.66%) | - |
DYRK4 | inactive (106.57%) | - |
HIPK1 | inactive (103.27%) | inactive (97%) |
HIPK2 | inactive (101.75%) | inactive (91%) |
HIPK3 | inactive (102.35%) | inactive (98%) |
HIPK4 | inactive (99.75%) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
Erk1 | inactive (101.32%) | inactive (80%) |
Erk2 | inactive (100.51%) | inactive (118%) |
JNK3 | inactive (98.79%) | inactive (96%) |
NLK | inactive (96.73%) | inactive (101%) |
p38a | inactive (104.48%) | inactive (78%) |
p38b | inactive (100.14%) | inactive (104%) |
p38d | inactive (103.44%) | inactive (118%) |
p38g | inactive (92.62%) | inactive (101%) |
JNK1 | inactive (100.2%) | inactive (114%) |
JNK2 | inactive (104.78%) | inactive (108%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
GSK3A | inactive (91.14%) | inactive (103%) |
GSK3B | inactive (89.48%) | inactive (83%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
MSSK1 | inactive (96.37%) | inactive (119%) |
SRPK1 | inactive (99.97%) | inactive (100%) |
SRPK2 | inactive (88.8%) | inactive (101%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC | Millipore |
---|
PDHK | 5 | 1 | - |
Alpha | 6 | - | 1 |
PIKK | 6 | - | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
PDHK1 | inactive (99.38%) | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
eEF2K | - | inactive (101%) |
Atypical - PIKK
Bioactivity |
---|
Kinase | RBC | Millipore |
---|
FRAP | - | inactive (104%) |