Compound Information
Test on : RBC
Compound Name : -
Inchikey : DGCXNBUJPWPMJJ-UHFFFAOYSA-N
CANNOT FIND
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC |
---|
PDK1 | inactive (79.01%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC |
---|
AKT1 | inactive (79.72%) |
AKT2 | inactive (55.76%) |
AKT3 | inactive (81.23%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC |
---|
DMPK1 | inactive (84.81%) |
MRCKa | inactive (91.6%) |
MRCKb | inactive (82.64%) |
ROCK1 | inactive (94.52%) |
ROCK2 | inactive (81.7%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC |
---|
BARK1 | inactive (106.01%) |
BARK2 | inactive (106.45%) |
GPRK4 | inactive (68.41%) |
GPRK5 | inactive (74.28%) |
GPRK6 | inactive (57.97%) |
GPRK7 | inactive (78.09%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC |
---|
MSK1 | inactive (68.68%) |
MSK2 | inactive (72.22%) |
p70S6K | inactive (85.77%) |
p70S6Kb | inactive (86.31%) |
RSK2 | inactive (75.05%) |
RSK4 | inactive (62.34%) |
RSK1 | inactive (53.07%) |
RSK3 | inactive (89.1%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC |
---|
PKACg | inactive (88.55%) |
PRKX | inactive (94.3%) |
PKACa | inactive (76.62%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC |
---|
PKCa | inactive (91.4%) |
PKCd | inactive (102.3%) |
PKCe | inactive (99.04%) |
PKCh | active (49.23%) |
PKCg | inactive (59.32%) |
PKCi | inactive (85.7%) |
PKCt | inactive (83.03%) |
PKCz | inactive (99.13%) |
PKCb | active (29.29%) |
AGC - PKG
Bioactivity |
---|
Kinase | RBC |
---|
PKG2 | inactive (140.02%) |
PKG1 | inactive (108.7%) |
AGC - PKN
Bioactivity |
---|
Kinase | RBC |
---|
PKN1 | inactive (97.53%) |
PKN2 | inactive (77.06%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC |
---|
SGK1 | inactive (67.19%) |
SGK2 | inactive (75.08%) |
SGK3 | inactive (90.42%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC |
---|
NDR1 | active (46.64%) |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC |
---|
ABL1 | inactive (89.75%) |
ABL2 | inactive (89.72%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC |
---|
ACK | active (44.94%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC |
---|
ALK | inactive (83.46%) |
LTK | inactive (176.61%) |
TK - Axl
Bioactivity |
---|
Kinase | RBC |
---|
AXL | active (10.31%) |
MER | inactive (93.13%) |
TYRO3 | active (33.29%) |
TK - Src
Bioactivity |
---|
Kinase | RBC |
---|
BLK | inactive (108.61%) |
BRK | inactive (110.8%) |
SRC | inactive (80.4%) |
FGR | inactive (79.76%) |
FRK | active (33.88%) |
FYN | inactive (76.23%) |
HCK | inactive (83.96%) |
LCK | inactive (70.48%) |
SRM | active (6.34%) |
YES | inactive (89.15%) |
LYN | inactive (85.17%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC |
---|
BMX | inactive (79.03%) |
BTK | inactive (90.55%) |
ITK | inactive (71.48%) |
TEC | active (2.44%) |
TXK | inactive (90.82%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC |
---|
KIT | active (22.16%) |
FLT3 | inactive (100.02%) |
FMS | active (11.63%) |
PDGFRb | active (11.35%) |
PDGFRa | active (44.11%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC |
---|
CSK | inactive (84.76%) |
CTK | inactive (99.68%) |
TK - DDR
Bioactivity |
---|
Kinase | RBC |
---|
DDR2 | inactive (58.71%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC |
---|
EGFR | active (36.99%) |
ErbB2 | active (22.24%) |
ErbB4 | inactive (50.2%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC |
---|
EphA1 | inactive (73.05%) |
EphA2 | inactive (100.02%) |
EphA3 | inactive (81.64%) |
EphA4 | inactive (61.06%) |
EphA5 | inactive (81.54%) |
EphA6 | inactive (105.72%) |
EphA7 | inactive (81.95%) |
EphA8 | inactive (92.57%) |
EphB1 | inactive (89.47%) |
EphB2 | inactive (86.1%) |
EphB3 | inactive (90.17%) |
EphB4 | inactive (97.09%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC |
---|
FAK | inactive (87.03%) |
PYK2 | inactive (52.06%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC |
---|
FER | inactive (89.09%) |
FES | inactive (87.55%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC |
---|
FGFR1 | active (24.22%) |
FGFR2 | inactive (59.36%) |
FGFR3 | active (26.7%) |
FGFR4 | inactive (57.97%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC |
---|
FLT1 | active (3.06%) |
FLT4 | active (5.79%) |
KDR | active (1.95%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC |
---|
IGF1R | inactive (91.14%) |
IRR | inactive (86.7%) |
INSR | active (32.26%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC |
---|
JAK1 | inactive (101.04%) |
JAK2 | inactive (82.55%) |
JAK3 | inactive (90.38%) |
TYK2 | inactive (77.21%) |
TK - Musk
Bioactivity |
---|
Kinase | RBC |
---|
MUSK | inactive (107.07%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC |
---|
RET | inactive (100.61%) |
TK - Met
Bioactivity |
---|
Kinase | RBC |
---|
RON | inactive (93.63%) |
MET | inactive (83.28%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC |
---|
ROS | inactive (91.12%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC |
---|
SYK | inactive (94.76%) |
ZAP70 | inactive (68.23%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC |
---|
TIE2 | active (4.27%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC |
---|
TRKA | inactive (76.65%) |
TRKB | active (29.41%) |
TRKC | inactive (87.2%) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC |
---|
ALK1 | inactive (104.78%) |
ALK2 | inactive (93.07%) |
ALK4 | inactive (112.88%) |
TGFbR1 | inactive (106.54%) |
TGFbR2 | inactive (93.37%) |
TKL - RAF
Bioactivity |
---|
Kinase | RBC |
---|
ARAF | inactive (104.07%) |
BRAF | inactive (84.9%) |
RAF1 | inactive (76.07%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC |
---|
IRAK1 | inactive (77.56%) |
IRAK4 | inactive (96.9%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC |
---|
LIMK1 | inactive (64.99%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC |
---|
LRRK2 | inactive (85.55%) |
TKL - MLK
Bioactivity |
---|
Kinase | RBC |
---|
MLK1 | inactive (63.33%) |
MLK2 | inactive (94.65%) |
MLK3 | inactive (68.99%) |
TAK1 | inactive (89.85%) |
ZAK | inactive (69.78%) |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC |
---|
RIPK2 | inactive (100.59%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC |
---|
NuaK1 | inactive (89.81%) |
BRSK1 | inactive (84.77%) |
BRSK2 | inactive (66.74%) |
CHK1 | inactive (111.86%) |
LKB1 | inactive (99.09%) |
MARK1 | inactive (98.16%) |
MARK3 | inactive (78.06%) |
MARK4 | inactive (88.09%) |
MELK | inactive (55.73%) |
PASK | inactive (73.39%) |
QIK | inactive (106.16%) |
NuaK2 | inactive (92.54%) |
MARK2 | inactive (94.22%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC |
---|
CaMK1a | inactive (68.72%) |
CaMK1b | inactive (83.38%) |
CaMK1d | inactive (93.94%) |
CaMK1g | active (28.49%) |
CaMK4 | inactive (85.38%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC |
---|
CaMK2a | inactive (84.71%) |
CaMK2b | inactive (85.15%) |
CaMK2d | inactive (93%) |
CaMK2g | inactive (91.13%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC |
---|
CHK2 | inactive (54.72%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC |
---|
DAPK1 | inactive (92.17%) |
DAPK2 | inactive (83.39%) |
DRAK1 | inactive (83.76%) |
DAPK3 | inactive (96.2%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC |
---|
DCLK2 | inactive (86.48%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC |
---|
MAPKAPK2 | inactive (103.99%) |
MAPKAPK3 | inactive (76.03%) |
MAPKAPK5 | inactive (66.86%) |
MNK1 | inactive (79.34%) |
MNK2 | inactive (78.25%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC |
---|
smMLCK | inactive (94.12%) |
skMLCK | inactive (88.14%) |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC |
---|
PHKg1 | inactive (92.46%) |
PHKg2 | inactive (96.12%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC |
---|
PIM1 | inactive (94.08%) |
PIM2 | inactive (92.78%) |
PIM3 | inactive (93.34%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC |
---|
PKD1 | inactive (86.5%) |
PKD3 | inactive (83.44%) |
PKD2 | inactive (91.69%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC |
---|
TSSK1 | inactive (88.74%) |
TSSK2 | inactive (74.99%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC |
---|
STK33 | inactive (107.01%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC |
---|
MAP3K5 | inactive (105.96%) |
MAP3K2 | inactive (82.96%) |
MAP3K3 | inactive (133.52%) |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC |
---|
COT | inactive (75.89%) |
NIK | inactive (123.52%) |
STE - STE20
Bioactivity |
---|
Kinase | RBC |
---|
GCK | inactive (79.4%) |
HGK | inactive (89.01%) |
KHS1 | inactive (78.69%) |
LOK | inactive (84.33%) |
MINK | inactive (91.22%) |
MST1 | inactive (87.83%) |
MST2 | inactive (97.45%) |
MST3 | inactive (101.44%) |
MST4 | inactive (91.75%) |
OSR1 | inactive (83.01%) |
PAK1 | inactive (96.13%) |
PAK2 | inactive (96.25%) |
PAK3 | inactive (97.12%) |
PAK4 | inactive (91.38%) |
PAK5 | inactive (93.4%) |
PAK6 | inactive (108.04%) |
SLK | inactive (92.42%) |
YSK1 | inactive (100.73%) |
STLK3 | inactive (89.2%) |
TAO1 | inactive (90.22%) |
TAO2 | inactive (91.93%) |
TAO3 | inactive (90.85%) |
MYO3B | inactive (88.38%) |
STE - STE7
Bioactivity |
---|
Kinase | RBC |
---|
MAP2K1 | inactive (88.68%) |
MAP2K2 | inactive (94.69%) |
MAP2K6 | inactive (85.66%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC |
---|
AurA | inactive (71.37%) |
AurB | inactive (84.73%) |
AurC | inactive (95.42%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC |
---|
CaMKK1 | inactive (74.94%) |
CaMKK2 | inactive (76.86%) |
Other - Haspin
Bioactivity |
---|
Kinase | RBC |
---|
Haspin | inactive (79.2%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC |
---|
IKKa | inactive (71.99%) |
IKKb | inactive (73.35%) |
IKKe | inactive (89.18%) |
TBK1 | inactive (87%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC |
---|
NEK1 | active (46.3%) |
NEK11 | inactive (87.97%) |
NEK2 | inactive (77.71%) |
NEK4 | inactive (96.08%) |
NEK6 | inactive (96.28%) |
NEK7 | inactive (83.56%) |
NEK9 | inactive (118.9%) |
NEK3 | inactive (110.66%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC |
---|
PBK | inactive (64.47%) |
Other - PLK
Bioactivity |
---|
Kinase | RBC |
---|
PLK1 | active (28.6%) |
PLK2 | active (37.27%) |
PLK3 | active (28.53%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC |
---|
SgK496 | inactive (81.53%) |
Other - NAK
Bioactivity |
---|
Kinase | RBC |
---|
MPSK1 | inactive (80.54%) |
Other - TTK
Bioactivity |
---|
Kinase | RBC |
---|
TTK | inactive (124.72%) |
Other - ULK
Bioactivity |
---|
Kinase | RBC |
---|
ULK1 | inactive (107.47%) |
ULK2 | inactive (104.74%) |
ULK3 | inactive (103.29%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC |
---|
Wee1 | inactive (70.86%) |
Other - WNK
Bioactivity |
---|
Kinase | RBC |
---|
Wnk2 | inactive (142.58%) |
Wnk3 | inactive (116.13%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC |
---|
TLK2 | inactive (100.15%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
CK1 | 7 | 6 |
VRK | 3 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC |
---|
CK1d | inactive (86.84%) |
CK1g1 | inactive (85.15%) |
CK1g2 | inactive (82.19%) |
CK1g3 | inactive (80.34%) |
CK1a | inactive (85.8%) |
CK1e | inactive (80.56%) |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC |
---|
VRK1 | inactive (90.53%) |
CMGC
CMGC - CK2
Bioactivity |
---|
Kinase | RBC |
---|
CK2a1 | inactive (101.45%) |
CK2a2 | inactive (76.2%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC |
---|
CLK1 | inactive (79.43%) |
CLK2 | inactive (92.11%) |
CLK3 | inactive (81.21%) |
CLK4 | inactive (78.26%) |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC |
---|
DYRK1A | inactive (95.05%) |
DYRK1B | inactive (81.04%) |
DYRK2 | inactive (113.32%) |
DYRK3 | inactive (88.62%) |
DYRK4 | inactive (88.52%) |
HIPK1 | inactive (99.29%) |
HIPK2 | inactive (106.78%) |
HIPK3 | inactive (100.97%) |
HIPK4 | inactive (97.9%) |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC |
---|
Erk1 | inactive (86.96%) |
Erk2 | inactive (87.51%) |
JNK3 | inactive (55%) |
NLK | inactive (98.16%) |
p38a | inactive (88.61%) |
p38b | inactive (101.11%) |
p38d | inactive (95.57%) |
p38g | inactive (92.53%) |
JNK1 | inactive (78.33%) |
JNK2 | inactive (51.94%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC |
---|
GSK3A | inactive (88.72%) |
GSK3B | inactive (83.49%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC |
---|
MSSK1 | inactive (89.39%) |
SRPK1 | inactive (109.24%) |
SRPK2 | inactive (95.77%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
PDHK | 5 | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC |
---|
PDHK1 | inactive (79.01%) |