Compound Information
Test on : DRx, RBC, Metz, Millipore
Compound Name
DRx : UNII-WS78QR6DSV
RBC : UNII-2Z5A7553WW
Metz, Millipore : 152121-47-6
Inchikey
Same : CDMGBJANTYXAIV-N
DRx : CDMGBJANTYXAIV-HHHXNRCGSA-N
RBC : CDMGBJANTYXAIV-MHZLTWQESA-N
Metz, Millipore : CDMGBJANTYXAIV-UHFFFAOYSA-N
ChemSpider
DRx : -
RBC : 7822386
Metz, Millipore : 153453
Pubchem CID
DRx : 40467016
RBC : 9543416
Metz, Millipore : 176155
ChEMBL
DRx : -
RBC : -
Metz, Millipore : CHEMBL10
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
Other
Other - NAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
AAK1 | inactive (10001nM) | - | - | - |
BIKE | inactive (10001nM) | - | - | - |
GAK | active (19nM) | - | - | - |
MPSK1 | inactive (10001nM) | inactive (111.28%) | - | - |
Other - Aur
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
AurA | inactive (10001nM) | inactive (99.54%) | inactive (>3981.07nM) | inactive (117%) |
AurB | inactive (10001nM) | inactive (87.68%) | inactive (>5011.87nM) | inactive (102%) |
AurC | inactive (10001nM) | inactive (98.48%) | - | inactive (115%) |
Other - CAMKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CaMKK1 | inactive (10001nM) | inactive (125.29%) | - | - |
CaMKK2 | inactive (10001nM) | inactive (110.44%) | inactive (>2511.89nM) | - |
Other - PEK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
HRI | inactive (10001nM) | - | - | - |
PKR | inactive (10001nM) | - | - | - |
Other - IRE
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
IRE1 | inactive (10001nM) | - | - | - |
Other - IKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
IKKa | inactive (10001nM) | inactive (100.2%) | inactive (>3981.07nM) | inactive (113%) |
IKKb | inactive (10001nM) | inactive (106.32%) | inactive (>3162.28nM) | inactive (104%) |
IKKe | inactive (10001nM) | inactive (98.04%) | inactive (>3162.28nM) | - |
TBK1 | inactive (10001nM) | inactive (99.67%) | inactive (>3162.28nM) | inactive (124%) |
Other - NEK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
NEK1 | inactive (10001nM) | inactive (94.69%) | - | - |
NEK11 | inactive (10001nM) | inactive (81.28%) | - | inactive (90%) |
NEK2 | inactive (10001nM) | inactive (104.97%) | inactive (>6309.57nM) | inactive (114%) |
NEK3 | inactive (10001nM) | inactive (92.23%) | - | inactive (104%) |
NEK4 | inactive (10001nM) | inactive (98.23%) | inactive (>6309.57nM) | - |
NEK5 | inactive (10001nM) | - | - | - |
NEK6 | inactive (10001nM) | inactive (103.44%) | - | inactive (112%) |
NEK7 | inactive (10001nM) | inactive (98.85%) | - | inactive (101%) |
NEK9 | inactive (10001nM) | inactive (99.07%) | - | - |
Other - WEE
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
MYT1 | inactive (10001nM) | - | - | - |
Wee1 | inactive (10001nM) | inactive (92.08%) | - | - |
Wee1B | inactive (10001nM) | - | - | - |
Other - PLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PLK1 | inactive (10001nM) | inactive (100.46%) | inactive (>7943.28nM) | inactive (117%) |
PLK2 | inactive (10001nM) | inactive (95.63%) | - | inactive (116%) |
PLK3 | inactive (10001nM) | inactive (97.26%) | inactive (>7943.28nM) | inactive (90%) |
PLK4 | inactive (10001nM) | - | inactive (>3981.07nM) | - |
Other - SgK496
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
SgK496 | inactive (10001nM) | inactive (100.47%) | - | - |
Other - NKF1
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
SBK | inactive (10001nM) | - | - | - |
SgK110 | inactive (10001nM) | - | - | - |
Other - NKF4
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CLIK1 | inactive (10001nM) | - | - | - |
Other - ULK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
Fused | active (1300nM) | - | - | - |
ULK1 | inactive (10001nM) | inactive (89.28%) | - | - |
ULK2 | inactive (10001nM) | inactive (83.55%) | - | inactive (120%) |
ULK3 | inactive (10001nM) | inactive (83.19%) | - | inactive (104%) |
Other - TLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
TLK1 | inactive (10001nM) | - | - | - |
TLK2 | inactive (10001nM) | inactive (96.45%) | - | inactive (113%) |
Other - TTK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
TTK | active (2500nM) | inactive (99.86%) | - | - |
Other - Haspin
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
Haspin | - | inactive (88.25%) | - | inactive (88%) |
Other - TOPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PBK | - | inactive (101.95%) | inactive (>10000nM) | - |
Other - WNK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
Wnk2 | - | inactive (102.51%) | - | inactive (117%) |
Wnk3 | - | inactive (98.96%) | - | inactive (110%) |
Other - CDC7
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CDC7 | - | - | inactive (>1258.93nM) | - |
TK
TK - Abl
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
ABL1 | inactive (10001nM) | inactive (96.97%) | inactive (>3162.28nM) | inactive (89%) |
ABL2 | inactive (10001nM) | inactive (91.52%) | - | inactive (86%) |
TK - ALK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
ALK | inactive (10001nM) | inactive (104.76%) | inactive (>6309.57nM) | inactive (122%) |
LTK | inactive (10001nM) | inactive (100.82%) | inactive (>2511.89nM) | - |
TK - Axl
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
AXL | inactive (10001nM) | inactive (100.5%) | inactive (>1995.26nM) | inactive (122%) |
MER | inactive (10001nM) | inactive (93.87%) | - | inactive (117%) |
TYRO3 | inactive (10001nM) | inactive (96.99%) | inactive (>3162.28nM) | inactive (107%) |
TK - Src
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
BLK | inactive (10001nM) | inactive (101.66%) | inactive (>1584.89nM) | inactive (101%) |
BRK | inactive (3900nM) | inactive (54.21%) | inactive (>2511.89nM) | inactive (59%) |
FGR | inactive (10001nM) | inactive (92.68%) | - | inactive (87%) |
FRK | active (1800nM) | inactive (87.25%) | active (251.19nM) | inactive (71%) |
FYN | inactive (10001nM) | inactive (89.81%) | inactive (>3981.07nM) | inactive (76%) |
HCK | inactive (10001nM) | inactive (96.07%) | inactive (>3162.28nM) | inactive (105%) |
LCK | active (2800nM) | inactive (94.98%) | inactive (5011.87nM) | inactive (79%) |
LYN | inactive (10001nM) | inactive (91.81%) | inactive (>1584.89nM) | active (47%) |
SRC | inactive (5300nM) | inactive (92.59%) | inactive (>1995.26nM) | inactive (112%) |
SRM | inactive (10001nM) | inactive (101.85%) | inactive (>1584.89nM) | - |
YES | inactive (10001nM) | inactive (92.65%) | - | inactive (110%) |
TK - Tec
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
BMX | inactive (10001nM) | inactive (94.38%) | - | inactive (81%) |
BTK | inactive (10001nM) | inactive (97.23%) | inactive (>6309.57nM) | inactive (94%) |
ITK | inactive (10001nM) | inactive (97.02%) | inactive (>1584.89nM) | inactive (100%) |
TEC | inactive (10001nM) | inactive (113.37%) | - | - |
TXK | inactive (4500nM) | inactive (63.94%) | - | inactive (77%) |
TK - PDGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
FMS | inactive (10001nM) | inactive (95.52%) | inactive (>2511.89nM) | inactive (109%) |
FLT3 | inactive (10001nM) | inactive (91.51%) | inactive (>2511.89nM) | inactive (91%) |
KIT | inactive (10001nM) | inactive (91.32%) | inactive (>3981.07nM) | inactive (119%) |
PDGFRa | inactive (10001nM) | inactive (98.82%) | inactive (>3162.28nM) | inactive (110%) |
PDGFRb | inactive (10001nM) | inactive (102.78%) | inactive (>1995.26nM) | inactive (120%) |
TK - Csk
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CSK | inactive (10001nM) | inactive (87.66%) | - | inactive (103%) |
CTK | inactive (10001nM) | inactive (95.59%) | inactive (>1995.26nM) | - |
TK - DDR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
DDR1 | active (1000nM) | - | - | - |
DDR2 | inactive (5000nM) | inactive (103.2%) | - | inactive (94%) |
TK - EGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
EGFR | active (1700nM) | inactive (86.51%) | inactive (>1258.93nM) | active (1%) |
ErbB2 | inactive (10001nM) | inactive (94.56%) | inactive (>1258.93nM) | - |
ErbB3 | inactive (10001nM) | - | - | - |
ErbB4 | inactive (4800nM) | inactive (66.83%) | inactive (>3981.07nM) | inactive (115%) |
TK - Eph
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
EphA1 | inactive (10001nM) | inactive (97.01%) | - | inactive (90%) |
EphA2 | inactive (10001nM) | inactive (94.76%) | inactive (>6309.57nM) | inactive (95%) |
EphA3 | inactive (10001nM) | inactive (96.08%) | - | inactive (105%) |
EphA4 | inactive (10001nM) | inactive (95.55%) | - | inactive (110%) |
EphA5 | inactive (10001nM) | inactive (89.53%) | - | inactive (96%) |
EphA6 | active (1200nM) | inactive (57.15%) | - | - |
EphA7 | inactive (10001nM) | inactive (83.06%) | - | inactive (102%) |
EphA8 | inactive (10001nM) | inactive (101.16%) | - | inactive (91%) |
EphB1 | inactive (10001nM) | inactive (93.02%) | - | inactive (106%) |
EphB2 | inactive (10001nM) | inactive (108.29%) | - | inactive (101%) |
EphB3 | inactive (10001nM) | inactive (96.65%) | - | inactive (114%) |
EphB4 | inactive (10001nM) | inactive (91.1%) | - | inactive (107%) |
EphB6 | inactive (3100nM) | - | - | - |
TK - FAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
FAK | inactive (10001nM) | inactive (95.52%) | inactive (>6309.57nM) | inactive (125%) |
PYK2 | inactive (10001nM) | inactive (92.53%) | inactive (>1584.89nM) | inactive (115%) |
TK - Fer
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
FER | inactive (10001nM) | inactive (95.05%) | inactive (>1584.89nM) | inactive (107%) |
FES | inactive (10001nM) | inactive (97.29%) | inactive (>1995.26nM) | inactive (112%) |
TK - FGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
FGFR1 | inactive (10001nM) | inactive (90.72%) | inactive (>3981.07nM) | inactive (142%) |
FGFR2 | inactive (10001nM) | inactive (103.46%) | - | inactive (99%) |
FGFR3 | inactive (10001nM) | inactive (96.97%) | inactive (>1995.26nM) | inactive (115%) |
FGFR4 | inactive (10001nM) | inactive (73.79%) | - | inactive (110%) |
TK - VEGFR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
FLT1 | inactive (10001nM) | inactive (95.16%) | inactive (>3981.07nM) | inactive (101%) |
FLT4 | inactive (10001nM) | inactive (119.2%) | inactive (6309.57nM) | inactive (93%) |
KDR | inactive (10001nM) | inactive (99.23%) | inactive (>2511.89nM) | inactive (107%) |
TK - InsR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
IGF1R | inactive (10001nM) | inactive (94.32%) | inactive (>1995.26nM) | inactive (102%) |
INSR | inactive (10001nM) | inactive (88.9%) | inactive (>5011.87nM) | inactive (94%) |
IRR | inactive (10001nM) | inactive (100.3%) | - | inactive (109%) |
TK - JakA
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
JAK1 | inactive (10001nM) | inactive (105.36%) | - | - |
JAK2 | inactive (10001nM) | inactive (99.5%) | inactive (>2511.89nM) | inactive (112%) |
JAK3 | inactive (10001nM) | inactive (93.85%) | inactive (>5011.87nM) | inactive (107%) |
TYK2 | inactive (10001nM) | inactive (101.56%) | inactive (>1995.26nM) | - |
TK - Met
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
MET | inactive (10001nM) | inactive (102.77%) | inactive (>2511.89nM) | inactive (123%) |
RON | inactive (10001nM) | inactive (100.98%) | inactive (>3981.07nM) | inactive (105%) |
TK - Musk
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
MUSK | inactive (10001nM) | inactive (90.33%) | - | inactive (143%) |
TK - Ret
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
RET | inactive (10001nM) | inactive (85.05%) | inactive (>3162.28nM) | inactive (90%) |
TK - Sev
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
ROS | inactive (10001nM) | inactive (94.41%) | inactive (>2511.89nM) | inactive (117%) |
TK - Syk
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
SYK | inactive (10001nM) | inactive (98%) | inactive (>1584.89nM) | inactive (112%) |
ZAP70 | inactive (10001nM) | inactive (94.42%) | - | inactive (124%) |
TK - Tie
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
TIE1 | inactive (10001nM) | - | - | - |
TIE2 | inactive (10001nM) | inactive (94.53%) | - | inactive (102%) |
TK - Ack
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
TNK1 | inactive (10001nM) | - | - | - |
ACK | inactive (10001nM) | inactive (82.11%) | inactive (>3981.07nM) | inactive (93%) |
TK - Trk
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
TRKA | inactive (10001nM) | inactive (100.47%) | inactive (>2511.89nM) | inactive (121%) |
TRKB | inactive (10001nM) | inactive (103.95%) | inactive (>3981.07nM) | inactive (94%) |
TRKC | inactive (10001nM) | inactive (97.97%) | inactive (>2511.89nM) | - |
TKL
TKL
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz | Millipore |
---|
STKR | 12 | 10 | 5 | 1 | 2 |
RIPK | 5 | 4 | 1 | - | 1 |
RAF | 5 | 2 | 3 | 1 | 1 |
MLK | 10 | 8 | 5 | 2 | 2 |
IRAK | 4 | 3 | 2 | 2 | 2 |
LISK | 4 | 3 | 1 | 1 | 1 |
LRRK | 2 | 1 | 1 | 1 | - |
TKL - STKR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
ALK2 | inactive (10001nM) | inactive (97.44%) | inactive (>3981.07nM) | - |
ALK4 | active (3000nM) | inactive (127.24%) | - | inactive (87%) |
ACTR2 | inactive (10001nM) | - | - | - |
ACTR2B | inactive (10001nM) | - | - | - |
ALK1 | inactive (10001nM) | inactive (97.67%) | - | - |
BMPR1A | inactive (10001nM) | - | - | - |
BMPR1B | inactive (3300nM) | - | - | - |
BMPR2 | inactive (10001nM) | - | - | - |
TGFbR1 | inactive (7100nM) | inactive (100.51%) | - | inactive (130%) |
TGFbR2 | active (1800nM) | inactive (144.37%) | - | - |
TKL - RIPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
SgK288 | inactive (10001nM) | - | - | - |
RIPK1 | inactive (10001nM) | - | - | - |
RIPK2 | active (24nM) | active (49.08%) | - | active (24%) |
ANKRD3 | inactive (10001nM) | - | - | - |
TKL - RAF
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
BRAF | active (710nM) | inactive (78.79%) | - | - |
RAF1 | active (980nM) | active (41.08%) | - | active (17%) |
ARAF | - | active (42.66%) | - | - |
TKL - MLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
DLK | inactive (10001nM) | - | - | - |
LZK | inactive (10001nM) | - | - | - |
MLK1 | inactive (10001nM) | inactive (95.04%) | - | inactive (101%) |
MLK2 | inactive (10001nM) | inactive (103.83%) | inactive (>3162.28nM) | - |
MLK3 | inactive (10001nM) | inactive (96.4%) | - | - |
TAK1 | inactive (10001nM) | inactive (94.04%) | - | inactive (106%) |
HH498 | inactive (3500nM) | - | - | - |
ZAK | inactive (4400nM) | inactive (100.35%) | inactive (>7943.28nM) | - |
TKL - IRAK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
IRAK1 | inactive (10001nM) | inactive (129.36%) | inactive (>7943.28nM) | inactive (108%) |
IRAK3 | inactive (10001nM) | - | - | - |
IRAK4 | inactive (10001nM) | inactive (129.61%) | inactive (>10000nM) | inactive (113%) |
TKL - LISK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
LIMK1 | inactive (10001nM) | inactive (91.32%) | inactive (>6309.57nM) | inactive (110%) |
LIMK2 | inactive (10001nM) | - | - | - |
TESK1 | inactive (10001nM) | - | - | - |
TKL - LRRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
LRRK2 | inactive (10001nM) | inactive (100.3%) | inactive (>2511.89nM) | - |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz | Millipore |
---|
ABC1 | 5 | 2 | - | - | - |
PIKK | 6 | 1 | - | - | 1 |
RIO | 3 | 3 | - | - | - |
Alpha | 6 | 1 | - | 1 | 1 |
PDHK | 5 | - | 1 | - | - |
Atypical - ABC1
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
ADCK3 | inactive (10001nM) | - | - | - |
ADCK4 | inactive (3100nM) | - | - | - |
Atypical - PIKK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
FRAP | inactive (10001nM) | - | - | inactive (106%) |
Atypical - RIO
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
RIOK1 | inactive (10001nM) | - | - | - |
RIOK2 | inactive (10001nM) | - | - | - |
RIOK3 | inactive (10001nM) | - | - | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
ChaK2 | inactive (10001nM) | - | - | - |
eEF2K | - | - | inactive (>3981.07nM) | inactive (111%) |
Atypical - PDHK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PDHK1 | - | inactive (96.32%) | - | - |
AGC
AGC - Akt
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
AKT1 | inactive (10001nM) | inactive (102.38%) | inactive (>7943.28nM) | inactive (102%) |
AKT2 | inactive (10001nM) | inactive (96.78%) | inactive (>7943.28nM) | inactive (107%) |
AKT3 | inactive (10001nM) | inactive (101.55%) | inactive (>10000nM) | inactive (117%) |
AGC - DMPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CRIK | active (420nM) | - | - | - |
DMPK1 | inactive (10001nM) | inactive (103.44%) | - | inactive (122%) |
DMPK2 | active (400nM) | - | - | - |
MRCKa | inactive (6200nM) | inactive (94.26%) | inactive (>10000nM) | inactive (106%) |
MRCKb | active (2700nM) | inactive (104.55%) | - | inactive (113%) |
ROCK1 | inactive (10001nM) | inactive (101.65%) | inactive (>3981.07nM) | inactive (70%) |
ROCK2 | inactive (10001nM) | inactive (98.4%) | inactive (>5011.87nM) | inactive (119%) |
AGC - GRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
RHOK | inactive (10001nM) | - | - | - |
GPRK4 | inactive (10001nM) | inactive (95.46%) | - | - |
GPRK7 | inactive (10001nM) | inactive (107.14%) | - | inactive (109%) |
BARK1 | - | inactive (101.31%) | - | - |
BARK2 | - | inactive (98.22%) | - | - |
GPRK5 | - | inactive (104.29%) | inactive (>3981.07nM) | inactive (109%) |
GPRK6 | - | inactive (102.24%) | - | inactive (107%) |
AGC - NDR
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
LATS1 | inactive (10001nM) | - | - | - |
LATS2 | inactive (10001nM) | - | - | - |
NDR1 | inactive (10001nM) | inactive (104.52%) | - | - |
NDR2 | inactive (10001nM) | - | - | - |
AGC - MAST
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
MAST1 | inactive (10001nM) | - | - | - |
AGC - PDK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PDK1 | inactive (10001nM) | inactive (96.32%) | inactive (>3981.07nM) | inactive (117%) |
AGC - PKA
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PKACa | inactive (10001nM) | inactive (98.88%) | inactive (>2511.89nM) | inactive (105%) |
PKACb | inactive (10001nM) | - | - | - |
PRKX | inactive (10001nM) | inactive (99.32%) | inactive (>3162.28nM) | inactive (98%) |
PKACg | - | inactive (106.67%) | - | - |
AGC - PKN
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PKN1 | inactive (10001nM) | inactive (96.5%) | - | - |
PKN2 | inactive (10001nM) | inactive (95.81%) | inactive (>7943.28nM) | inactive (103%) |
AGC - PKC
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PKCd | inactive (10001nM) | inactive (106.86%) | inactive (>7943.28nM) | inactive (105%) |
PKCe | inactive (10001nM) | inactive (114.99%) | - | inactive (125%) |
PKCh | inactive (10001nM) | inactive (95.75%) | - | inactive (79%) |
PKCi | inactive (10001nM) | inactive (95.16%) | inactive (>5011.87nM) | inactive (105%) |
PKCt | inactive (10001nM) | inactive (111.33%) | inactive (>2511.89nM) | inactive (105%) |
PKCa | - | inactive (92.33%) | - | inactive (107%) |
PKCg | - | inactive (89.98%) | inactive (>7943.28nM) | inactive (104%) |
PKCz | - | inactive (103.25%) | inactive (>7943.28nM) | inactive (108%) |
PKCb | - | inactive (97.89%) | - | - |
AGC - PKG
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PKG1 | inactive (10001nM) | inactive (94.32%) | inactive (>1995.26nM) | - |
PKG2 | inactive (10001nM) | inactive (92.67%) | inactive (>1584.89nM) | - |
AGC - RSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
p70S6K | inactive (10001nM) | inactive (97.39%) | inactive (>6309.57nM) | inactive (103%) |
MSK1 | - | inactive (103.5%) | inactive (>1995.26nM) | inactive (97%) |
MSK2 | - | inactive (99.59%) | inactive (>1584.89nM) | inactive (102%) |
p70S6Kb | - | inactive (97.16%) | - | - |
RSK2 | - | inactive (95.69%) | inactive (>3981.07nM) | inactive (108%) |
RSK4 | - | inactive (110.23%) | - | inactive (114%) |
RSK1 | - | inactive (99.88%) | - | inactive (107%) |
RSK3 | - | inactive (101.78%) | - | inactive (86%) |
AGC - SGK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
SGK3 | inactive (10001nM) | inactive (101.06%) | - | inactive (120%) |
SGK1 | - | inactive (97.33%) | inactive (>7943.28nM) | inactive (96%) |
SGK2 | - | inactive (106.05%) | - | inactive (114%) |
AGC - YANK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
YANK1 | active (1300nM) | - | - | - |
YANK2 | active (2100nM) | - | - | - |
YANK3 | inactive (10001nM) | - | - | - |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
AMPKa1 | inactive (10001nM) | - | inactive (>3162.28nM) | inactive (109%) |
AMPKa2 | inactive (10001nM) | - | - | inactive (104%) |
NuaK1 | inactive (10001nM) | inactive (94.42%) | - | inactive (97%) |
BRSK1 | inactive (10001nM) | inactive (97.86%) | inactive (>10000nM) | inactive (104%) |
BRSK2 | inactive (10001nM) | inactive (101.42%) | - | inactive (102%) |
CHK1 | inactive (10001nM) | inactive (97.33%) | inactive (>5011.87nM) | inactive (104%) |
HUNK | inactive (10001nM) | - | - | - |
LKB1 | inactive (10001nM) | inactive (81.56%) | - | inactive (109%) |
MARK1 | inactive (10001nM) | inactive (104.61%) | - | inactive (105%) |
MARK2 | inactive (10001nM) | inactive (99.08%) | inactive (>7943.28nM) | inactive (108%) |
MARK3 | inactive (10001nM) | inactive (100.64%) | inactive (>6309.57nM) | - |
MARK4 | inactive (10001nM) | inactive (98.46%) | inactive (>5011.87nM) | - |
MELK | inactive (10001nM) | inactive (101.56%) | inactive (>1995.26nM) | inactive (107%) |
NIM1 | inactive (10001nM) | - | - | - |
QSK | inactive (3900nM) | - | - | - |
SIK | inactive (10001nM) | - | - | inactive (132%) |
QIK | inactive (10001nM) | inactive (82.14%) | active (1000nM) | - |
NuaK2 | inactive (10001nM) | inactive (130.93%) | - | - |
SNRK | inactive (10001nM) | - | - | - |
PASK | - | inactive (99.07%) | - | inactive (113%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CaMK1a | inactive (10001nM) | inactive (105.96%) | inactive (>6309.57nM) | inactive (115%) |
CaMK1d | inactive (10001nM) | inactive (104.66%) | inactive (>2511.89nM) | inactive (138%) |
CaMK1g | inactive (10001nM) | inactive (99.25%) | - | - |
CaMK4 | inactive (10001nM) | inactive (101.38%) | - | inactive (113%) |
CaMK1b | - | inactive (102.1%) | - | - |
CAMK - CAMK2
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CaMK2a | inactive (10001nM) | inactive (100.77%) | inactive (>3981.07nM) | - |
CaMK2b | inactive (10001nM) | inactive (97.58%) | inactive (>7943.28nM) | inactive (114%) |
CaMK2d | inactive (10001nM) | inactive (102.59%) | inactive (>6309.57nM) | inactive (108%) |
CaMK2g | inactive (10001nM) | inactive (82.16%) | inactive (>6309.57nM) | inactive (103%) |
CAMK - CASK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CASK | inactive (10001nM) | - | - | - |
CAMK - RAD53
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CHK2 | inactive (10001nM) | inactive (99.55%) | inactive (>6309.57nM) | inactive (90%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
DAPK1 | inactive (10001nM) | inactive (90.35%) | - | inactive (85%) |
DAPK2 | inactive (10001nM) | inactive (101.83%) | - | inactive (90%) |
DAPK3 | inactive (10001nM) | inactive (95.46%) | inactive (>5011.87nM) | inactive (98%) |
DRAK1 | inactive (10001nM) | inactive (98.95%) | inactive (>3981.07nM) | inactive (123%) |
DRAK2 | inactive (10001nM) | - | - | - |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
DCLK1 | inactive (10001nM) | - | inactive (>10000nM) | - |
DCLK2 | inactive (10001nM) | inactive (99.84%) | - | inactive (132%) |
DCLK3 | inactive (10001nM) | - | - | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
MAPKAPK2 | inactive (10001nM) | inactive (98.28%) | inactive (>7943.28nM) | inactive (104%) |
MAPKAPK5 | inactive (10001nM) | inactive (92.54%) | inactive (>1584.89nM) | inactive (145%) |
MNK1 | inactive (10001nM) | inactive (98.53%) | - | - |
MNK2 | inactive (10001nM) | inactive (94.42%) | inactive (>10000nM) | inactive (103%) |
MAPKAPK3 | - | inactive (101.04%) | inactive (>10000nM) | inactive (104%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
caMLCK | inactive (10001nM) | - | - | - |
smMLCK | inactive (10001nM) | inactive (101.39%) | - | inactive (118%) |
skMLCK | inactive (10001nM) | inactive (99.89%) | - | - |
SgK085 | inactive (10001nM) | - | - | - |
CAMK - PHK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PHKg1 | inactive (10001nM) | inactive (94.09%) | - | - |
PHKg2 | inactive (10001nM) | inactive (102.45%) | inactive (>5011.87nM) | inactive (109%) |
CAMK - PIM
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PIM1 | inactive (10001nM) | inactive (102.72%) | inactive (>6309.57nM) | inactive (84%) |
PIM2 | inactive (10001nM) | inactive (104.07%) | inactive (>1584.89nM) | inactive (125%) |
PIM3 | inactive (10001nM) | inactive (98.09%) | inactive (>7943.28nM) | inactive (107%) |
CAMK - PKD
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PKD1 | inactive (10001nM) | inactive (95.77%) | - | inactive (123%) |
PKD2 | inactive (10001nM) | inactive (95.8%) | inactive (6309.57nM) | inactive (105%) |
PKD3 | inactive (10001nM) | inactive (84.13%) | inactive (>3981.07nM) | - |
CAMK - STK33
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
STK33 | inactive (10001nM) | inactive (98.12%) | - | inactive (106%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
TSSK1 | inactive (10001nM) | inactive (108.37%) | inactive (>1584.89nM) | inactive (106%) |
TSSK2 | - | inactive (95.71%) | inactive (>1584.89nM) | inactive (94%) |
STE
STE
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz | Millipore |
---|
STE11 | 8 | 8 | 3 | - | 1 |
STE20 | 31 | 27 | 23 | 9 | 14 |
STE7 | 7 | 7 | 3 | 2 | 3 |
STE-Unique | 2 | - | 2 | - | - |
STE - STE11
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
MAP3K5 | inactive (10001nM) | inactive (106.75%) | - | inactive (138%) |
MAP3K6 | inactive (10001nM) | - | - | - |
MAP3K1 | inactive (10001nM) | - | - | - |
MAP3K7 | inactive (10001nM) | - | - | - |
MAP3K2 | inactive (10001nM) | inactive (95.26%) | - | - |
MAP3K3 | inactive (10001nM) | inactive (101.55%) | - | - |
MAP3K4 | inactive (10001nM) | - | - | - |
MAP3K8 | inactive (10001nM) | - | - | - |
STE - STE20
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
HPK1 | inactive (10001nM) | - | - | - |
LOK | inactive (10001nM) | inactive (89.15%) | - | inactive (109%) |
GCK | inactive (10001nM) | inactive (105.78%) | inactive (>2511.89nM) | inactive (104%) |
KHS2 | inactive (10001nM) | - | - | - |
HGK | inactive (3700nM) | inactive (95.76%) | active (398.11nM) | - |
KHS1 | inactive (10001nM) | inactive (99.49%) | inactive (>7943.28nM) | - |
MINK | inactive (10001nM) | inactive (107%) | inactive (2511.89nM) | inactive (112%) |
MST1 | inactive (10001nM) | inactive (101.46%) | - | inactive (111%) |
MST2 | inactive (10001nM) | inactive (102.19%) | inactive (>5011.87nM) | inactive (104%) |
MST3 | inactive (10001nM) | inactive (98.95%) | - | inactive (115%) |
MST4 | inactive (10001nM) | inactive (96.75%) | - | - |
MYO3A | inactive (10001nM) | - | - | - |
MYO3B | inactive (10001nM) | inactive (104.3%) | - | - |
OSR1 | inactive (10001nM) | inactive (101.87%) | - | - |
PAK1 | inactive (10001nM) | inactive (99.17%) | inactive (>10000nM) | - |
PAK2 | inactive (10001nM) | inactive (77.95%) | - | inactive (110%) |
PAK3 | inactive (10001nM) | inactive (101.97%) | - | inactive (114%) |
PAK4 | inactive (10001nM) | inactive (91.99%) | inactive (>5011.87nM) | inactive (106%) |
PAK6 | inactive (10001nM) | inactive (76.68%) | - | inactive (110%) |
PAK5 | inactive (10001nM) | inactive (103.94%) | - | inactive (105%) |
SLK | inactive (3700nM) | inactive (94.07%) | inactive (1995.26nM) | - |
STLK3 | inactive (10001nM) | inactive (93.94%) | - | - |
TAO1 | inactive (10001nM) | inactive (97.91%) | inactive (>5011.87nM) | inactive (100%) |
TAO2 | inactive (10001nM) | inactive (93.98%) | - | inactive (111%) |
TAO3 | inactive (10001nM) | inactive (102.73%) | - | inactive (108%) |
TNIK | active (820nM) | - | - | - |
YSK1 | inactive (10001nM) | inactive (111.12%) | - | - |
STE - STE7
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
MAP2K1 | inactive (10001nM) | inactive (94.76%) | inactive (>3162.28nM) | inactive (113%) |
MAP2K2 | inactive (9600nM) | inactive (99.87%) | inactive (>3981.07nM) | - |
MAP2K3 | inactive (10001nM) | - | - | - |
MAP2K4 | inactive (10001nM) | - | - | - |
MAP2K5 | active (1400nM) | - | - | - |
MAP2K6 | inactive (10001nM) | inactive (101.98%) | - | active (43%) |
MAP2K7 | inactive (10001nM) | - | - | inactive (86%) |
STE - STE-Unique
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
COT | - | inactive (92.12%) | - | - |
NIK | - | inactive (117.93%) | - | - |
CMGC
CMGC
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz | Millipore |
---|
CDK | 20 | 8 | - | 7 | - |
CDKL | 5 | 4 | - | - | - |
CLK | 4 | 4 | 4 | 2 | 2 |
CK2 | 3 | 2 | 2 | 1 | 2 |
DYRK | 10 | 8 | 9 | 6 | 4 |
MAPK | 14 | 14 | 10 | 8 | 10 |
GSK | 2 | 2 | 2 | 2 | 2 |
RCK | 3 | 2 | - | - | - |
SRPK | 3 | 3 | 3 | 1 | 3 |
CMGC - CDK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
PITSLRE | inactive (10001nM) | - | - | - |
CHED | inactive (10001nM) | - | - | - |
CDK11 | inactive (10001nM) | - | - | - |
PCTAIRE1 | inactive (10001nM) | - | - | - |
PCTAIRE2 | inactive (10001nM) | - | - | - |
PCTAIRE3 | inactive (10001nM) | - | - | - |
PFTAIRE2 | inactive (10001nM) | - | - | - |
PFTAIRE1 | inactive (10001nM) | - | - | - |
CDC2 | - | - | inactive (>7943.28nM) | - |
CDK2 | - | - | inactive (>7943.28nM) | - |
CDK5 | - | - | inactive (>3162.28nM) | - |
CDK8 | - | - | inactive (>3981.07nM) | - |
CDK7 | - | - | inactive (>3981.07nM) | - |
CDK9 | - | - | inactive (>1584.89nM) | - |
CMGC - CDKL
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CDKL1 | inactive (10001nM) | - | - | - |
CDKL2 | inactive (10001nM) | - | - | - |
CDKL3 | inactive (10001nM) | - | - | - |
CDKL5 | inactive (10001nM) | - | - | - |
CMGC - CLK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CLK1 | inactive (10001nM) | inactive (101.4%) | - | - |
CLK2 | inactive (10001nM) | inactive (107.64%) | inactive (>3981.07nM) | inactive (114%) |
CLK3 | inactive (10001nM) | inactive (99.14%) | - | inactive (98%) |
CLK4 | inactive (10001nM) | inactive (98.72%) | inactive (>2511.89nM) | - |
CMGC - CK2
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CK2a1 | inactive (10001nM) | inactive (86.24%) | inactive (>6309.57nM) | inactive (100%) |
CK2a2 | inactive (10001nM) | inactive (104.29%) | - | inactive (122%) |
CMGC - DYRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
DYRK1A | inactive (10001nM) | inactive (95.56%) | inactive (>1995.26nM) | - |
DYRK1B | inactive (10001nM) | inactive (104.04%) | inactive (>2511.89nM) | - |
DYRK2 | inactive (10001nM) | inactive (98.74%) | - | inactive (115%) |
HIPK1 | inactive (10001nM) | inactive (103.63%) | - | inactive (102%) |
HIPK2 | inactive (10001nM) | inactive (101.86%) | inactive (>3162.28nM) | inactive (110%) |
HIPK3 | inactive (10001nM) | inactive (103.04%) | - | inactive (110%) |
HIPK4 | inactive (10001nM) | inactive (93.49%) | inactive (>7943.28nM) | - |
PRP4 | inactive (10001nM) | - | - | - |
DYRK3 | - | inactive (98.98%) | inactive (>6309.57nM) | - |
DYRK4 | - | inactive (99.2%) | inactive (>7943.28nM) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
Erk1 | inactive (10001nM) | inactive (100.57%) | - | inactive (124%) |
Erk2 | inactive (10001nM) | inactive (94.7%) | inactive (>7943.28nM) | inactive (118%) |
Erk3 | inactive (10001nM) | - | - | - |
Erk4 | inactive (10001nM) | - | - | - |
Erk5 | inactive (10001nM) | - | - | - |
Erk7 | inactive (10001nM) | - | - | - |
JNK1 | active (1100nM) | inactive (96.09%) | inactive (1258.93nM) | inactive (111%) |
JNK2 | active (130nM) | inactive (100.4%) | active (199.53nM) | inactive (74%) |
JNK3 | active (35nM) | inactive (113.93%) | active (25.12nM) | active (20%) |
NLK | active (25nM) | inactive (53.79%) | - | inactive (62%) |
p38a | active (12nM) | active (22.82%) | active (19.95nM) | active (5%) |
p38b | active (70nM) | inactive (68.92%) | - | active (24%) |
p38d | inactive (10001nM) | inactive (105.91%) | inactive (>7943.28nM) | inactive (111%) |
p38g | active (1500nM) | inactive (104.61%) | inactive (>6309.57nM) | inactive (114%) |
CMGC - GSK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
GSK3A | inactive (10001nM) | inactive (94.13%) | inactive (>3981.07nM) | inactive (86%) |
GSK3B | active (1700nM) | inactive (80.24%) | inactive (1584.89nM) | inactive (93%) |
CMGC - RCK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
ICK | inactive (10001nM) | - | - | - |
MAK | inactive (10001nM) | - | - | - |
CMGC - SRPK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
SRPK1 | inactive (10001nM) | inactive (99.53%) | inactive (>7943.28nM) | inactive (112%) |
SRPK2 | inactive (10001nM) | inactive (101.92%) | - | inactive (112%) |
MSSK1 | inactive (10001nM) | inactive (99.4%) | - | inactive (102%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Metz | Millipore |
---|
CK1 | 7 | 7 | 6 | 5 | 4 |
VRK | 3 | 1 | 1 | - | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
CK1a | active (75nM) | inactive (63.9%) | active (316.23nM) | - |
CK1a2 | active (1700nM) | - | - | - |
CK1d | active (37nM) | active (13.93%) | active (39.81nM) | active (11%) |
CK1e | active (100nM) | active (30.97%) | - | - |
CK1g1 | inactive (10001nM) | inactive (95.71%) | inactive (>6309.57nM) | inactive (119%) |
CK1g2 | inactive (10001nM) | inactive (95.65%) | inactive (>7943.28nM) | inactive (120%) |
CK1g3 | inactive (10001nM) | inactive (103.23%) | inactive (>6309.57nM) | inactive (125%) |
CK1 - VRK
Bioactivity |
---|
Kinase | DRx | RBC | Metz | Millipore |
---|
VRK2 | inactive (10001nM) | - | - | inactive (114%) |
VRK1 | - | inactive (95.83%) | - | - |