Compound Information
Test on : DRx, RBC, Millipore
Compound Name
DRx, RBC : C35H30N4O4
Millipore : N-Benzoylstaurosporine
Inchikey
Same : BMGQWWVMWDBQGC-N
DRx, RBC : BMGQWWVMWDBQGC-PZFYLCKJSA-N
Millipore : BMGQWWVMWDBQGC-UHFFFAOYSA-N
ChemSpider
DRx, RBC : 21435595
Millipore : 19416722
Pubchem CID
DRx, RBC : 24202429
Millipore : 16760627
ChEMBL
DRx, RBC : CHEMBL338448
Millipore : -
DRx, RBC | Millipore |
| |
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
Other
Other - NAK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
AAK1 | active (48nM) | - | - |
BIKE | active (220nM) | - | - |
GAK | active (380nM) | - | - |
MPSK1 | active (280nM) | active (47.89%) | - |
Other - Aur
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
AurA | active (120nM) | active (4.48%) | active (-3%) |
AurB | active (62nM) | active (2.96%) | active (1%) |
AurC | active (170nM) | active (12.02%) | inactive (62%) |
Other - CAMKK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
CaMKK1 | active (130nM) | active (20.39%) | - |
CaMKK2 | active (73nM) | active (3.9%) | - |
Other - PEK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
HRI | inactive (10001nM) | - | - |
PKR | inactive (6900nM) | - | - |
Other - IRE
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
IRE1 | active (2300nM) | - | - |
Other - IKK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
IKKa | inactive (3800nM) | inactive (89.61%) | inactive (101%) |
IKKb | inactive (6300nM) | inactive (97.85%) | inactive (89%) |
IKKe | active (160nM) | active (9.85%) | - |
TBK1 | active (9.3nM) | active (3.22%) | active (2%) |
Other - NEK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
NEK1 | inactive (10001nM) | inactive (66.2%) | - |
NEK11 | inactive (10001nM) | inactive (97.99%) | active (47%) |
NEK2 | inactive (10001nM) | inactive (100.82%) | inactive (82%) |
NEK3 | inactive (10001nM) | inactive (106.59%) | inactive (102%) |
NEK4 | inactive (10001nM) | inactive (97.59%) | - |
NEK5 | inactive (10001nM) | - | - |
NEK6 | inactive (10001nM) | inactive (109.97%) | inactive (93%) |
NEK7 | inactive (10001nM) | inactive (101.49%) | inactive (91%) |
NEK9 | inactive (10001nM) | inactive (64.36%) | - |
Other - WEE
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
MYT1 | inactive (10001nM) | - | - |
Wee1 | inactive (4600nM) | inactive (89.34%) | - |
Wee1B | inactive (10001nM) | - | - |
Other - PLK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
PLK1 | inactive (10001nM) | inactive (95.41%) | inactive (87%) |
PLK2 | inactive (10001nM) | inactive (97.47%) | inactive (100%) |
PLK3 | inactive (10001nM) | inactive (95.26%) | inactive (95%) |
PLK4 | active (66nM) | - | - |
Other - SgK496
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
SgK496 | inactive (4700nM) | inactive (96.44%) | - |
Other - NKF1
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
SBK | inactive (10001nM) | - | - |
SgK110 | inactive (10001nM) | - | - |
Other - NKF4
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
CLIK1 | inactive (10001nM) | - | - |
Other - ULK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
Fused | inactive (10001nM) | - | - |
ULK1 | inactive (10001nM) | inactive (99.21%) | - |
ULK2 | inactive (10001nM) | inactive (95.75%) | inactive (96%) |
ULK3 | active (1300nM) | active (37%) | active (17%) |
Other - TLK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
TLK1 | inactive (10001nM) | - | - |
TLK2 | inactive (10001nM) | inactive (75.02%) | inactive (95%) |
Other - TTK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
TTK | active (350nM) | inactive (55.02%) | - |
Other - Haspin
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
Haspin | - | inactive (70.17%) | inactive (78%) |
Other - TOPK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
PBK | - | - | - |
Other - WNK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
Wnk2 | - | inactive (111.01%) | inactive (90%) |
Wnk3 | - | inactive (91.37%) | inactive (91%) |
TK
TK - Abl
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
ABL1 | inactive (10001nM) | inactive (82.69%) | inactive (89%) |
ABL2 | inactive (10001nM) | inactive (76.26%) | inactive (77%) |
TK - ALK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
ALK | active (270nM) | active (49.16%) | active (32%) |
LTK | active (3000nM) | inactive (50.06%) | - |
TK - Axl
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
AXL | active (620nM) | inactive (106.06%) | active (14%) |
MER | active (2900nM) | inactive (78.66%) | active (8%) |
TYRO3 | inactive (10001nM) | inactive (98.76%) | inactive (83%) |
TK - Src
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
BLK | active (500nM) | active (48.75%) | active (7%) |
BRK | inactive (10001nM) | inactive (96.23%) | inactive (98%) |
FGR | active (730nM) | active (17.37%) | active (7%) |
FRK | active (2400nM) | inactive (65.84%) | active (33%) |
FYN | active (2100nM) | active (33.96%) | active (6%) |
HCK | active (720nM) | active (14.9%) | active (7%) |
LCK | active (280nM) | active (19.75%) | active (13%) |
LYN | inactive (4200nM) | active (28.88%) | active (6%) |
SRC | active (1200nM) | active (39.58%) | active (40%) |
SRM | inactive (10001nM) | inactive (97.64%) | - |
YES | active (950nM) | active (20.6%) | active (5%) |
TK - Tec
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
BMX | inactive (10001nM) | active (31.99%) | active (12%) |
BTK | inactive (10001nM) | inactive (60.53%) | inactive (60%) |
ITK | inactive (10001nM) | inactive (70.61%) | inactive (56%) |
TEC | inactive (10001nM) | inactive (106.49%) | - |
TXK | inactive (10001nM) | inactive (71.72%) | inactive (82%) |
TK - PDGFR
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
FMS | active (330nM) | active (6.65%) | active (0%) |
FLT3 | active (11nM) | active (2.41%) | active (1%) |
KIT | active (220nM) | active (37.42%) | inactive (65%) |
PDGFRa | active (380nM) | active (29.97%) | inactive (54%) |
PDGFRb | active (110nM) | active (14.8%) | active (46%) |
TK - Csk
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
CSK | inactive (8700nM) | inactive (55.05%) | inactive (82%) |
CTK | inactive (10001nM) | inactive (112.76%) | - |
TK - DDR
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
DDR1 | inactive (7200nM) | - | - |
DDR2 | inactive (10001nM) | inactive (379.86%) | inactive (106%) |
TK - EGFR
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
EGFR | active (1300nM) | inactive (78.54%) | inactive (101%) |
ErbB2 | inactive (10001nM) | inactive (86.66%) | - |
ErbB3 | inactive (10001nM) | - | - |
ErbB4 | inactive (3100nM) | inactive (98.17%) | inactive (67%) |
TK - Eph
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
EphA1 | inactive (10001nM) | inactive (93.51%) | inactive (87%) |
EphA2 | inactive (10001nM) | inactive (92.29%) | inactive (97%) |
EphA3 | inactive (10001nM) | inactive (94.06%) | inactive (97%) |
EphA4 | inactive (10001nM) | inactive (96.93%) | inactive (103%) |
EphA5 | inactive (10001nM) | inactive (95.82%) | inactive (97%) |
EphA6 | inactive (10001nM) | inactive (79.52%) | - |
EphA7 | inactive (10001nM) | inactive (87.23%) | inactive (94%) |
EphA8 | inactive (10001nM) | inactive (94.08%) | inactive (94%) |
EphB1 | inactive (10001nM) | inactive (96.36%) | inactive (97%) |
EphB2 | inactive (10001nM) | inactive (94.02%) | inactive (111%) |
EphB3 | inactive (10001nM) | inactive (90.52%) | inactive (119%) |
EphB4 | inactive (10001nM) | inactive (109.52%) | inactive (107%) |
EphB6 | inactive (3100nM) | - | - |
TK - FAK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
FAK | inactive (10001nM) | inactive (87.45%) | inactive (90%) |
PYK2 | active (660nM) | inactive (58.16%) | active (16%) |
TK - Fer
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
FER | active (1200nM) | active (22.36%) | active (26%) |
FES | inactive (10001nM) | active (48.3%) | active (15%) |
TK - FGFR
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
FGFR1 | active (1600nM) | active (36.08%) | active (5%) |
FGFR2 | active (2400nM) | active (49.5%) | active (21%) |
FGFR3 | active (1700nM) | inactive (57.53%) | active (34%) |
FGFR4 | inactive (10001nM) | inactive (84.15%) | inactive (71%) |
TK - VEGFR
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
FLT1 | active (450nM) | active (37.01%) | active (4%) |
FLT4 | active (670nM) | active (10.86%) | active (1%) |
KDR | inactive (3200nM) | active (30.59%) | active (3%) |
TK - InsR
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
IGF1R | inactive (10001nM) | inactive (97.11%) | inactive (115%) |
INSR | inactive (10001nM) | inactive (106.22%) | inactive (87%) |
IRR | inactive (10001nM) | inactive (96.17%) | inactive (98%) |
TK - JakA
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
JAK1 | active (670nM) | active (16.26%) | - |
JAK2 | active (94nM) | active (8.94%) | active (7%) |
JAK3 | active (12nM) | active (0.78%) | active (1%) |
TYK2 | active (250nM) | active (8.26%) | - |
TK - Met
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
MET | active (690nM) | inactive (89.4%) | active (35%) |
RON | inactive (10001nM) | inactive (101.13%) | active (47%) |
TK - Musk
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
MUSK | inactive (10001nM) | active (44.61%) | active (32%) |
TK - Ret
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
RET | active (350nM) | active (15.6%) | active (8%) |
TK - Sev
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
ROS | active (430nM) | active (6.53%) | inactive (63%) |
TK - Syk
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
SYK | active (88nM) | active (16.82%) | active (2%) |
ZAP70 | active (2600nM) | inactive (65.4%) | inactive (70%) |
TK - Tie
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
TIE1 | active (1400nM) | - | - |
TIE2 | active (1900nM) | inactive (95.83%) | inactive (133%) |
TK - Ack
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
TNK1 | active (83nM) | - | - |
ACK | active (120nM) | active (0.49%) | active (11%) |
TK - Trk
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
TRKA | active (380nM) | active (5.85%) | active (0%) |
TRKB | active (310nM) | active (12.82%) | active (23%) |
TRKC | active (1700nM) | active (3.76%) | - |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
ALK2 | inactive (10001nM) | inactive (95.46%) | - |
ALK4 | inactive (10001nM) | inactive (101.69%) | inactive (128%) |
ACTR2 | inactive (10001nM) | - | - |
ACTR2B | inactive (10001nM) | - | - |
ALK1 | inactive (10001nM) | inactive (94.34%) | - |
BMPR1A | inactive (10001nM) | - | - |
BMPR1B | inactive (10001nM) | - | - |
BMPR2 | inactive (10001nM) | - | - |
TGFbR1 | inactive (10001nM) | inactive (98.73%) | inactive (85%) |
TGFbR2 | inactive (10001nM) | inactive (99.06%) | - |
TKL - RIPK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
SgK288 | inactive (10001nM) | - | - |
RIPK1 | inactive (10001nM) | - | - |
RIPK2 | inactive (10001nM) | inactive (82.76%) | inactive (88%) |
ANKRD3 | inactive (10001nM) | - | - |
TKL - RAF
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
BRAF | inactive (10001nM) | inactive (106.05%) | - |
RAF1 | inactive (10001nM) | inactive (114.23%) | inactive (80%) |
ARAF | - | inactive (121.61%) | - |
TKL - MLK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
DLK | inactive (10001nM) | - | - |
LZK | active (2800nM) | - | - |
MLK1 | active (15nM) | active (0.45%) | active (1%) |
MLK2 | active (790nM) | active (3.15%) | - |
MLK3 | active (17nM) | active (1.38%) | - |
TAK1 | active (130nM) | active (19%) | active (39%) |
HH498 | inactive (10001nM) | - | - |
ZAK | inactive (10001nM) | inactive (94.19%) | - |
TKL - IRAK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
IRAK1 | inactive (10001nM) | inactive (86.31%) | inactive (85%) |
IRAK3 | active (180nM) | - | - |
IRAK4 | inactive (10001nM) | inactive (71.45%) | inactive (53%) |
TKL - LISK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
LIMK1 | inactive (10001nM) | active (19.6%) | active (22%) |
LIMK2 | inactive (10001nM) | - | - |
TESK1 | inactive (10001nM) | - | - |
TKL - LRRK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
LRRK2 | active (570nM) | active (8.46%) | - |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Millipore |
---|
ABC1 | 5 | 2 | - | - |
PIKK | 6 | 1 | - | 1 |
RIO | 3 | 3 | - | - |
Alpha | 6 | 1 | - | 1 |
PDHK | 5 | - | 1 | - |
Atypical - ABC1
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
ADCK3 | inactive (10001nM) | - | - |
ADCK4 | inactive (10001nM) | - | - |
Atypical - PIKK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
FRAP | inactive (10001nM) | - | inactive (95%) |
Atypical - RIO
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
RIOK1 | active (1200nM) | - | - |
RIOK2 | active (97nM) | - | - |
RIOK3 | active (420nM) | - | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
ChaK2 | inactive (10001nM) | - | - |
eEF2K | - | - | inactive (83%) |
Atypical - PDHK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
PDHK1 | - | active (21.75%) | - |
AGC
AGC - Akt
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
AKT1 | active (950nM) | inactive (81.28%) | inactive (97%) |
AKT2 | active (780nM) | inactive (77.21%) | inactive (80%) |
AKT3 | inactive (4400nM) | inactive (55.13%) | active (22%) |
AGC - DMPK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
CRIK | inactive (10001nM) | - | - |
DMPK1 | inactive (3800nM) | inactive (112.42%) | inactive (98%) |
DMPK2 | inactive (10001nM) | - | - |
MRCKa | inactive (10001nM) | inactive (95.98%) | inactive (93%) |
MRCKb | inactive (10001nM) | inactive (95.89%) | inactive (85%) |
ROCK1 | inactive (7800nM) | inactive (85.32%) | inactive (110%) |
ROCK2 | active (2300nM) | inactive (80.88%) | inactive (79%) |
AGC - GRK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
RHOK | active (85nM) | - | - |
GPRK4 | active (110nM) | inactive (94.4%) | - |
GPRK7 | active (48nM) | active (15.55%) | active (8%) |
BARK1 | - | inactive (101.85%) | - |
BARK2 | - | inactive (97.46%) | - |
GPRK5 | - | inactive (93.32%) | inactive (82%) |
GPRK6 | - | inactive (60.82%) | inactive (79%) |
AGC - NDR
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
LATS1 | active (1100nM) | - | - |
LATS2 | active (2200nM) | - | - |
NDR1 | inactive (10001nM) | inactive (83.79%) | - |
NDR2 | inactive (10001nM) | - | - |
AGC - MAST
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
MAST1 | active (190nM) | - | - |
AGC - PDK1
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
PDK1 | active (190nM) | active (21.75%) | active (2%) |
AGC - PKA
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
PKACa | active (720nM) | active (34%) | active (13%) |
PKACb | active (240nM) | - | - |
PRKX | active (960nM) | inactive (55.36%) | active (24%) |
PKACg | - | inactive (58.08%) | - |
AGC - PKN
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
PKN1 | active (9.3nM) | active (1.37%) | - |
PKN2 | active (15nM) | active (11.43%) | active (2%) |
AGC - PKC
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
PKCd | active (320nM) | active (10.93%) | active (21%) |
PKCe | active (540nM) | active (10.68%) | active (42%) |
PKCh | active (290nM) | active (20.43%) | inactive (84%) |
PKCi | inactive (10001nM) | inactive (96.43%) | inactive (79%) |
PKCt | active (920nM) | inactive (76.87%) | active (15%) |
PKCa | - | active (27.72%) | active (36%) |
PKCg | - | active (35.59%) | active (15%) |
PKCz | - | inactive (98.6%) | inactive (101%) |
PKCb | - | active (9.54%) | - |
AGC - PKG
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
PKG1 | active (250nM) | active (8.37%) | - |
PKG2 | active (74nM) | active (-9.42%) | - |
AGC - RSK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
p70S6K | active (1300nM) | active (19.36%) | active (4%) |
MSK1 | - | active (13.22%) | active (13%) |
MSK2 | - | active (16.77%) | active (12%) |
p70S6Kb | - | inactive (55.91%) | - |
RSK2 | - | active (3.19%) | active (1%) |
RSK4 | - | active (1.15%) | active (0%) |
RSK1 | - | active (0.43%) | active (1%) |
RSK3 | - | active (3.06%) | active (0%) |
AGC - SGK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
SGK3 | active (1400nM) | inactive (93.47%) | inactive (87%) |
SGK1 | - | inactive (81.87%) | inactive (57%) |
SGK2 | - | inactive (99.01%) | inactive (80%) |
AGC - YANK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
YANK1 | active (2400nM) | - | - |
YANK2 | inactive (10001nM) | - | - |
YANK3 | inactive (10001nM) | - | - |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
AMPKa1 | active (180nM) | - | active (10%) |
AMPKa2 | active (460nM) | - | active (1%) |
NuaK1 | active (41nM) | active (2.71%) | active (7%) |
BRSK1 | active (1200nM) | active (21.12%) | active (3%) |
BRSK2 | active (650nM) | active (16.4%) | active (4%) |
CHK1 | active (1300nM) | inactive (53%) | inactive (59%) |
HUNK | active (240nM) | - | - |
LKB1 | active (350nM) | inactive (94.82%) | inactive (95%) |
MARK1 | active (170nM) | active (4.09%) | active (1%) |
MARK2 | active (100nM) | active (3.53%) | active (0%) |
MARK3 | active (21nM) | active (4.76%) | - |
MARK4 | active (370nM) | active (3.16%) | - |
MELK | active (280nM) | active (4.87%) | active (5%) |
NIM1 | inactive (10001nM) | - | - |
QSK | active (98nM) | - | - |
SIK | active (160nM) | - | active (4%) |
QIK | active (560nM) | active (11.7%) | - |
NuaK2 | active (63nM) | active (26.19%) | - |
SNRK | inactive (10001nM) | - | - |
PASK | - | inactive (90.86%) | inactive (85%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
CaMK1a | active (2000nM) | inactive (93%) | inactive (84%) |
CaMK1d | active (670nM) | inactive (80.82%) | active (42%) |
CaMK1g | active (1800nM) | inactive (96.65%) | - |
CaMK4 | inactive (10001nM) | inactive (102.97%) | inactive (98%) |
CaMK1b | - | inactive (92.86%) | - |
CAMK - CAMK2
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
CaMK2a | active (20nM) | active (36.75%) | - |
CaMK2b | active (210nM) | inactive (57.36%) | active (18%) |
CaMK2d | active (36nM) | active (17.3%) | active (5%) |
CaMK2g | active (140nM) | active (43.92%) | active (10%) |
CAMK - CASK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
CASK | inactive (10001nM) | - | - |
CAMK - RAD53
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
CHK2 | inactive (10001nM) | inactive (85.05%) | inactive (79%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
DAPK1 | inactive (4700nM) | inactive (84.03%) | inactive (63%) |
DAPK2 | active (890nM) | inactive (104.92%) | inactive (71%) |
DAPK3 | active (1800nM) | inactive (82.6%) | inactive (56%) |
DRAK1 | active (1900nM) | inactive (62.87%) | active (16%) |
DRAK2 | inactive (4700nM) | - | - |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
DCLK1 | inactive (10001nM) | - | - |
DCLK2 | inactive (10001nM) | inactive (101.11%) | inactive (75%) |
DCLK3 | inactive (10001nM) | - | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
MAPKAPK2 | inactive (10001nM) | inactive (97.78%) | inactive (75%) |
MAPKAPK5 | inactive (10001nM) | inactive (91.96%) | inactive (102%) |
MNK1 | inactive (10001nM) | inactive (92.74%) | - |
MNK2 | active (950nM) | inactive (58.06%) | active (44%) |
MAPKAPK3 | - | inactive (91.52%) | inactive (68%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
caMLCK | active (2300nM) | - | - |
smMLCK | active (2000nM) | active (27.34%) | active (13%) |
skMLCK | inactive (10001nM) | inactive (83.53%) | - |
SgK085 | active (640nM) | - | - |
CAMK - PHK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
PHKg1 | active (900nM) | active (2.34%) | - |
PHKg2 | active (1400nM) | inactive (79.71%) | active (44%) |
CAMK - PIM
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
PIM1 | active (560nM) | active (41.18%) | active (33%) |
PIM2 | inactive (3100nM) | inactive (98.8%) | inactive (80%) |
PIM3 | active (560nM) | inactive (60.75%) | inactive (93%) |
CAMK - PKD
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
PKD1 | inactive (10001nM) | inactive (71.55%) | inactive (85%) |
PKD2 | inactive (6300nM) | inactive (62.87%) | inactive (101%) |
PKD3 | inactive (3200nM) | active (44.88%) | - |
CAMK - STK33
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
STK33 | active (190nM) | active (46.43%) | active (25%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
TSSK1 | inactive (4800nM) | active (8.24%) | active (15%) |
TSSK2 | - | inactive (89.09%) | inactive (51%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
MAP3K5 | inactive (10001nM) | inactive (100.89%) | inactive (96%) |
MAP3K6 | inactive (10001nM) | - | - |
MAP3K1 | inactive (10001nM) | - | - |
MAP3K7 | inactive (10001nM) | - | - |
MAP3K2 | active (140nM) | active (30.16%) | - |
MAP3K3 | active (210nM) | active (31.04%) | - |
MAP3K4 | inactive (10001nM) | - | - |
MAP3K8 | active (15nM) | - | - |
STE - STE20
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
HPK1 | active (2100nM) | - | - |
LOK | active (590nM) | active (19.25%) | active (21%) |
GCK | active (2500nM) | active (5.17%) | active (4%) |
KHS2 | active (120nM) | - | - |
HGK | active (650nM) | active (7.25%) | - |
KHS1 | active (1100nM) | active (7.01%) | - |
MINK | active (170nM) | active (29.21%) | inactive (52%) |
MST1 | active (40nM) | active (5.58%) | active (1%) |
MST2 | active (220nM) | active (1.93%) | active (3%) |
MST3 | inactive (10001nM) | active (39.1%) | active (17%) |
MST4 | inactive (10001nM) | active (23.82%) | - |
MYO3A | inactive (10001nM) | - | - |
MYO3B | inactive (10001nM) | inactive (53.74%) | - |
OSR1 | inactive (10001nM) | inactive (98.17%) | - |
PAK1 | active (2100nM) | active (35.1%) | - |
PAK2 | inactive (3300nM) | inactive (66.62%) | inactive (72%) |
PAK3 | active (180nM) | inactive (54.74%) | active (33%) |
PAK4 | inactive (10001nM) | inactive (92.89%) | inactive (64%) |
PAK6 | inactive (10001nM) | inactive (96.4%) | active (49%) |
PAK5 | inactive (10001nM) | inactive (90.4%) | inactive (52%) |
SLK | active (220nM) | active (30.49%) | - |
STLK3 | inactive (10001nM) | inactive (96.05%) | - |
TAO1 | inactive (10001nM) | inactive (60.77%) | active (50%) |
TAO2 | inactive (10001nM) | inactive (86.22%) | inactive (83%) |
TAO3 | inactive (10001nM) | active (38.08%) | active (42%) |
TNIK | active (1600nM) | - | - |
YSK1 | active (1800nM) | inactive (54.97%) | - |
STE - STE7
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
MAP2K1 | inactive (10001nM) | inactive (108.98%) | inactive (74%) |
MAP2K2 | inactive (10001nM) | inactive (81.5%) | - |
MAP2K3 | inactive (5300nM) | - | - |
MAP2K4 | inactive (4800nM) | - | - |
MAP2K5 | inactive (10001nM) | - | - |
MAP2K6 | inactive (6500nM) | inactive (91.43%) | inactive (52%) |
MAP2K7 | inactive (10001nM) | - | inactive (111%) |
STE - STE-Unique
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
COT | - | inactive (99.62%) | - |
NIK | - | inactive (113.31%) | - |
CMGC
CMGC - CDK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
PITSLRE | inactive (10001nM) | - | - |
CHED | inactive (10001nM) | - | - |
CDK11 | inactive (7200nM) | - | - |
PCTAIRE1 | inactive (10001nM) | - | - |
PCTAIRE2 | inactive (10001nM) | - | - |
PCTAIRE3 | inactive (10001nM) | - | - |
PFTAIRE2 | inactive (10001nM) | - | - |
PFTAIRE1 | inactive (10001nM) | - | - |
CMGC - CDKL
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
CDKL1 | inactive (10001nM) | - | - |
CDKL2 | inactive (10001nM) | - | - |
CDKL3 | inactive (10001nM) | - | - |
CDKL5 | inactive (10001nM) | - | - |
CMGC - CLK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
CLK1 | active (350nM) | inactive (55.8%) | - |
CLK2 | active (860nM) | active (36.04%) | active (17%) |
CLK3 | inactive (3600nM) | inactive (89.58%) | inactive (51%) |
CLK4 | active (410nM) | active (22.59%) | - |
CMGC - CK2
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
CK2a1 | inactive (10001nM) | inactive (100.64%) | inactive (73%) |
CK2a2 | inactive (10001nM) | inactive (87.85%) | inactive (117%) |
CMGC - DYRK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
DYRK1A | active (100nM) | active (32.24%) | - |
DYRK1B | active (330nM) | active (35.6%) | - |
DYRK2 | inactive (10001nM) | inactive (108.17%) | inactive (90%) |
HIPK1 | inactive (10001nM) | inactive (101.41%) | inactive (95%) |
HIPK2 | inactive (3100nM) | inactive (106.09%) | inactive (75%) |
HIPK3 | active (2300nM) | inactive (93.33%) | inactive (80%) |
HIPK4 | active (950nM) | inactive (90.54%) | - |
PRP4 | active (55nM) | - | - |
DYRK3 | - | inactive (98.5%) | - |
DYRK4 | - | inactive (96.41%) | - |
CMGC - MAPK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
Erk1 | inactive (10001nM) | inactive (88.35%) | inactive (75%) |
Erk2 | inactive (10001nM) | inactive (88.85%) | inactive (101%) |
Erk3 | inactive (10001nM) | - | - |
Erk4 | inactive (10001nM) | - | - |
Erk5 | inactive (10001nM) | - | - |
Erk7 | inactive (10001nM) | - | - |
JNK1 | inactive (4400nM) | inactive (88.29%) | inactive (92%) |
JNK2 | inactive (5000nM) | inactive (82.67%) | inactive (99%) |
JNK3 | inactive (3600nM) | inactive (98.94%) | active (50%) |
NLK | inactive (10001nM) | inactive (96.93%) | inactive (90%) |
p38a | inactive (10001nM) | inactive (93.71%) | inactive (71%) |
p38b | inactive (10001nM) | inactive (97.63%) | inactive (86%) |
p38d | inactive (10001nM) | inactive (103.88%) | inactive (92%) |
p38g | inactive (10001nM) | inactive (95.84%) | inactive (104%) |
CMGC - GSK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
GSK3A | active (2500nM) | active (27.39%) | active (17%) |
GSK3B | active (1800nM) | active (49.79%) | active (39%) |
CMGC - RCK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
ICK | inactive (5900nM) | - | - |
MAK | inactive (10001nM) | - | - |
CMGC - SRPK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
SRPK1 | active (42nM) | inactive (97.13%) | inactive (78%) |
SRPK2 | active (330nM) | inactive (83.15%) | inactive (64%) |
MSSK1 | active (80nM) | inactive (93.27%) | inactive (96%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC | Millipore |
---|
CK1 | 7 | 7 | 6 | 4 |
VRK | 3 | 1 | 1 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
CK1a | inactive (10001nM) | inactive (96.25%) | - |
CK1a2 | inactive (10001nM) | - | - |
CK1d | inactive (10001nM) | inactive (100.59%) | inactive (80%) |
CK1e | inactive (10001nM) | inactive (96.57%) | - |
CK1g1 | inactive (10001nM) | inactive (102.98%) | inactive (66%) |
CK1g2 | inactive (10001nM) | inactive (98.3%) | inactive (82%) |
CK1g3 | inactive (10001nM) | inactive (95.34%) | inactive (66%) |
CK1 - VRK
Bioactivity |
---|
Kinase | DRx | RBC | Millipore |
---|
VRK2 | inactive (10001nM) | - | inactive (99%) |
VRK1 | - | inactive (90.82%) | - |