Compound Information
Test on : DRx, RBC
Compound Name
DRx, RBC : Lapatinib
Inchikey
Same : BCFGMOOMADDAQU-N
DRx, RBC : BCFGMOOMADDAQU-UHFFFAOYSA-N
ChemSpider
DRx, RBC : 181006
Pubchem CID
DRx, RBC : 208908
ChEMBL
DRx, RBC : CHEMBL554
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
Other
Other - NAK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
AAK1 | inactive (10001nM) | - |
BIKE | inactive (10001nM) | - |
GAK | inactive (10001nM) | - |
MPSK1 | inactive (10001nM) | inactive (97.06%) |
Other - Aur
Bioactivity |
---|
Kinase | DRx | RBC |
---|
AurA | inactive (10001nM) | inactive (81.49%) |
AurB | inactive (10001nM) | inactive (98.44%) |
AurC | inactive (10001nM) | inactive (90.92%) |
Other - CAMKK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CaMKK1 | inactive (10001nM) | inactive (98.79%) |
CaMKK2 | inactive (10001nM) | inactive (100.79%) |
Other - PEK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
HRI | inactive (10001nM) | - |
PKR | inactive (10001nM) | - |
Other - IRE
Bioactivity |
---|
Kinase | DRx | RBC |
---|
IRE1 | inactive (10001nM) | - |
Other - IKK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
IKKa | inactive (10001nM) | inactive (99.5%) |
IKKb | inactive (10001nM) | inactive (81.01%) |
IKKe | inactive (10001nM) | inactive (94.87%) |
TBK1 | inactive (10001nM) | inactive (103.46%) |
Other - NEK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
NEK1 | inactive (10001nM) | inactive (71.77%) |
NEK11 | inactive (10001nM) | inactive (106.63%) |
NEK2 | inactive (10001nM) | inactive (118.31%) |
NEK3 | inactive (10001nM) | inactive (99.56%) |
NEK4 | inactive (10001nM) | inactive (98.09%) |
NEK5 | inactive (10001nM) | - |
NEK6 | inactive (10001nM) | inactive (93.72%) |
NEK7 | inactive (10001nM) | inactive (98.65%) |
NEK9 | inactive (10001nM) | inactive (100.44%) |
Other - WEE
Bioactivity |
---|
Kinase | DRx | RBC |
---|
MYT1 | inactive (10001nM) | - |
Wee1 | inactive (10001nM) | inactive (97.55%) |
Wee1B | inactive (10001nM) | - |
Other - PLK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PLK1 | inactive (10001nM) | inactive (98.98%) |
PLK2 | inactive (10001nM) | inactive (102.7%) |
PLK3 | inactive (10001nM) | inactive (104.8%) |
PLK4 | inactive (10001nM) | - |
Other - SgK496
Bioactivity |
---|
Kinase | DRx | RBC |
---|
SgK496 | inactive (10001nM) | inactive (108.08%) |
Other - NKF1
Bioactivity |
---|
Kinase | DRx | RBC |
---|
SBK | inactive (10001nM) | - |
SgK110 | inactive (10001nM) | - |
Other - NKF4
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CLIK1 | inactive (10001nM) | - |
Other - ULK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
Fused | inactive (10001nM) | - |
ULK1 | inactive (10001nM) | inactive (95.44%) |
ULK2 | inactive (10001nM) | inactive (104.49%) |
ULK3 | inactive (10001nM) | inactive (105.75%) |
Other - TLK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
TLK1 | inactive (10001nM) | - |
TLK2 | inactive (10001nM) | inactive (83.9%) |
Other - TTK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
TTK | inactive (10001nM) | inactive (101.94%) |
Other - Haspin
Bioactivity |
---|
Kinase | DRx | RBC |
---|
Haspin | - | inactive (66.53%) |
Other - TOPK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PBK | - | inactive (105.09%) |
Other - WNK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
Wnk2 | - | inactive (101.7%) |
Wnk3 | - | inactive (103.92%) |
TK
TK - Abl
Bioactivity |
---|
Kinase | DRx | RBC |
---|
ABL1 | inactive (10001nM) | inactive (96.38%) |
ABL2 | inactive (10001nM) | inactive (97.29%) |
TK - ALK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
ALK | inactive (10001nM) | inactive (103.81%) |
LTK | inactive (10001nM) | inactive (99.99%) |
TK - Axl
Bioactivity |
---|
Kinase | DRx | RBC |
---|
AXL | inactive (10001nM) | inactive (96.24%) |
MER | inactive (10001nM) | inactive (95.36%) |
TYRO3 | inactive (10001nM) | inactive (98.94%) |
TK - Src
Bioactivity |
---|
Kinase | DRx | RBC |
---|
BLK | inactive (10001nM) | inactive (95.9%) |
BRK | inactive (10001nM) | inactive (102.82%) |
FGR | inactive (10001nM) | inactive (84.83%) |
FRK | inactive (10001nM) | inactive (104.48%) |
FYN | inactive (10001nM) | inactive (99.38%) |
HCK | inactive (10001nM) | inactive (86.48%) |
LCK | inactive (10001nM) | inactive (94.17%) |
LYN | inactive (10001nM) | inactive (104.19%) |
SRC | inactive (10001nM) | inactive (102.48%) |
SRM | inactive (10001nM) | inactive (97.95%) |
YES | inactive (10001nM) | inactive (84.66%) |
TK - Tec
Bioactivity |
---|
Kinase | DRx | RBC |
---|
BMX | inactive (10001nM) | inactive (105.29%) |
BTK | inactive (10001nM) | inactive (102.77%) |
ITK | inactive (10001nM) | inactive (98.35%) |
TEC | inactive (10001nM) | inactive (101.36%) |
TXK | inactive (10001nM) | inactive (109.7%) |
TK - PDGFR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
FMS | inactive (10001nM) | inactive (105.74%) |
FLT3 | inactive (10001nM) | inactive (92.55%) |
KIT | inactive (10001nM) | inactive (98.45%) |
PDGFRa | inactive (10001nM) | inactive (107.54%) |
PDGFRb | inactive (10001nM) | inactive (92.02%) |
TK - Csk
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CSK | inactive (10001nM) | inactive (105.72%) |
CTK | inactive (10001nM) | inactive (75.94%) |
TK - DDR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
DDR1 | inactive (10001nM) | - |
DDR2 | inactive (10001nM) | inactive (107%) |
TK - EGFR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
EGFR | active (2.4nM) | active (8.02%) |
ErbB2 | active (7nM) | active (9.57%) |
ErbB3 | inactive (5500nM) | - |
ErbB4 | active (54nM) | active (11.19%) |
TK - Eph
Bioactivity |
---|
Kinase | DRx | RBC |
---|
EphA1 | inactive (10001nM) | inactive (99.3%) |
EphA2 | inactive (10001nM) | inactive (99.03%) |
EphA3 | inactive (10001nM) | inactive (98.18%) |
EphA4 | inactive (10001nM) | inactive (101.24%) |
EphA5 | inactive (10001nM) | inactive (103.29%) |
EphA6 | inactive (10001nM) | inactive (115.41%) |
EphA7 | inactive (10001nM) | inactive (95.62%) |
EphA8 | inactive (10001nM) | inactive (99.49%) |
EphB1 | inactive (10001nM) | inactive (103.96%) |
EphB2 | inactive (10001nM) | inactive (101.23%) |
EphB3 | inactive (10001nM) | - |
EphB4 | inactive (10001nM) | inactive (94.09%) |
EphB6 | inactive (10001nM) | - |
TK - FAK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
FAK | inactive (10001nM) | inactive (104.49%) |
PYK2 | inactive (10001nM) | inactive (101.12%) |
TK - Fer
Bioactivity |
---|
Kinase | DRx | RBC |
---|
FER | inactive (10001nM) | inactive (94.63%) |
FES | inactive (10001nM) | inactive (103.76%) |
TK - FGFR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
FGFR1 | inactive (10001nM) | inactive (102.48%) |
FGFR2 | inactive (10001nM) | inactive (96.42%) |
FGFR3 | inactive (10001nM) | inactive (96.72%) |
FGFR4 | inactive (10001nM) | inactive (96.63%) |
TK - VEGFR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
FLT1 | inactive (10001nM) | inactive (100.37%) |
FLT4 | inactive (10001nM) | inactive (93.25%) |
KDR | inactive (10001nM) | inactive (96.6%) |
TK - InsR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
IGF1R | inactive (10001nM) | inactive (87.43%) |
INSR | inactive (10001nM) | inactive (104.76%) |
IRR | inactive (10001nM) | inactive (103.83%) |
TK - JakA
Bioactivity |
---|
Kinase | DRx | RBC |
---|
JAK1 | inactive (10001nM) | inactive (98.04%) |
JAK2 | inactive (10001nM) | inactive (100.99%) |
JAK3 | inactive (10001nM) | inactive (96.24%) |
TYK2 | inactive (10001nM) | inactive (95.53%) |
TK - Met
Bioactivity |
---|
Kinase | DRx | RBC |
---|
MET | inactive (10001nM) | inactive (84.12%) |
RON | inactive (10001nM) | inactive (92.2%) |
TK - Musk
Bioactivity |
---|
Kinase | DRx | RBC |
---|
MUSK | inactive (10001nM) | inactive (96.55%) |
TK - Ret
Bioactivity |
---|
Kinase | DRx | RBC |
---|
RET | inactive (10001nM) | inactive (99.77%) |
TK - Sev
Bioactivity |
---|
Kinase | DRx | RBC |
---|
ROS | inactive (10001nM) | inactive (106.93%) |
TK - Syk
Bioactivity |
---|
Kinase | DRx | RBC |
---|
SYK | inactive (10001nM) | inactive (113.43%) |
ZAP70 | inactive (10001nM) | inactive (92.5%) |
TK - Tie
Bioactivity |
---|
Kinase | DRx | RBC |
---|
TIE1 | inactive (10001nM) | - |
TIE2 | inactive (10001nM) | inactive (93.25%) |
TK - Ack
Bioactivity |
---|
Kinase | DRx | RBC |
---|
TNK1 | inactive (10001nM) | - |
ACK | inactive (10001nM) | inactive (97.52%) |
TK - Trk
Bioactivity |
---|
Kinase | DRx | RBC |
---|
TRKA | inactive (10001nM) | inactive (99.17%) |
TRKB | inactive (10001nM) | inactive (98.77%) |
TRKC | inactive (10001nM) | inactive (103.09%) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
ALK2 | inactive (10001nM) | inactive (105.52%) |
ALK4 | inactive (10001nM) | inactive (98.68%) |
ACTR2 | inactive (10001nM) | - |
ACTR2B | inactive (10001nM) | - |
ALK1 | inactive (10001nM) | inactive (104.52%) |
BMPR1A | inactive (10001nM) | - |
BMPR1B | inactive (10001nM) | - |
BMPR2 | inactive (10001nM) | - |
TGFbR1 | inactive (10001nM) | inactive (100.71%) |
TGFbR2 | inactive (10001nM) | inactive (96.1%) |
TKL - RIPK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
SgK288 | inactive (10001nM) | - |
RIPK1 | inactive (10001nM) | - |
RIPK2 | inactive (3600nM) | inactive (109.98%) |
ANKRD3 | inactive (10001nM) | - |
TKL - RAF
Bioactivity |
---|
Kinase | DRx | RBC |
---|
BRAF | inactive (10001nM) | inactive (92.41%) |
RAF1 | inactive (10001nM) | inactive (85.88%) |
ARAF | - | inactive (84.96%) |
TKL - MLK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
DLK | inactive (10001nM) | - |
LZK | inactive (10001nM) | - |
MLK1 | inactive (10001nM) | inactive (111.64%) |
MLK2 | inactive (10001nM) | inactive (107.65%) |
MLK3 | inactive (10001nM) | inactive (105.99%) |
TAK1 | inactive (10001nM) | inactive (89.01%) |
HH498 | inactive (10001nM) | - |
ZAK | inactive (10001nM) | inactive (96.71%) |
TKL - IRAK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
IRAK1 | inactive (10001nM) | inactive (98.82%) |
IRAK3 | inactive (10001nM) | - |
IRAK4 | inactive (10001nM) | inactive (91.45%) |
TKL - LISK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
LIMK1 | inactive (10001nM) | inactive (95.18%) |
LIMK2 | inactive (10001nM) | - |
TESK1 | inactive (10001nM) | - |
TKL - LRRK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
LRRK2 | inactive (10001nM) | inactive (76.86%) |
Atypical
Atypical - ABC1
Bioactivity |
---|
Kinase | DRx | RBC |
---|
ADCK3 | inactive (10001nM) | - |
ADCK4 | inactive (10001nM) | - |
Atypical - PIKK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
FRAP | inactive (10001nM) | - |
Atypical - RIO
Bioactivity |
---|
Kinase | DRx | RBC |
---|
RIOK1 | inactive (10001nM) | - |
RIOK2 | inactive (10001nM) | - |
RIOK3 | inactive (10001nM) | - |
Atypical - Alpha
Bioactivity |
---|
Kinase | DRx | RBC |
---|
ChaK2 | inactive (10001nM) | - |
Atypical - PDHK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PDHK1 | - | inactive (86.38%) |
AGC
AGC - Akt
Bioactivity |
---|
Kinase | DRx | RBC |
---|
AKT1 | inactive (10001nM) | inactive (95.6%) |
AKT2 | inactive (10001nM) | inactive (104.99%) |
AKT3 | inactive (10001nM) | inactive (83.52%) |
AGC - DMPK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CRIK | inactive (10001nM) | - |
DMPK1 | inactive (10001nM) | inactive (94.68%) |
DMPK2 | inactive (10001nM) | - |
MRCKa | inactive (10001nM) | inactive (88.21%) |
MRCKb | inactive (10001nM) | inactive (95.74%) |
ROCK1 | inactive (10001nM) | inactive (108.09%) |
ROCK2 | inactive (10001nM) | inactive (92.72%) |
AGC - GRK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
RHOK | inactive (10001nM) | - |
GPRK4 | inactive (10001nM) | inactive (90.28%) |
GPRK7 | inactive (10001nM) | inactive (95.82%) |
BARK1 | - | inactive (94.85%) |
BARK2 | - | inactive (96.7%) |
GPRK5 | - | inactive (97.19%) |
GPRK6 | - | inactive (101.48%) |
AGC - NDR
Bioactivity |
---|
Kinase | DRx | RBC |
---|
LATS1 | inactive (10001nM) | - |
LATS2 | inactive (10001nM) | - |
NDR1 | inactive (10001nM) | inactive (101.13%) |
NDR2 | inactive (10001nM) | - |
AGC - MAST
Bioactivity |
---|
Kinase | DRx | RBC |
---|
MAST1 | inactive (10001nM) | - |
AGC - PDK1
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PDK1 | inactive (10001nM) | inactive (86.38%) |
AGC - PKA
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PKACa | inactive (10001nM) | inactive (95.98%) |
PKACb | inactive (10001nM) | - |
PRKX | inactive (10001nM) | inactive (111.23%) |
PKACg | - | inactive (109.58%) |
AGC - PKN
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PKN1 | inactive (10001nM) | inactive (105.68%) |
PKN2 | inactive (10001nM) | inactive (92.02%) |
AGC - PKC
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PKCd | inactive (10001nM) | inactive (102.62%) |
PKCe | inactive (10001nM) | inactive (98.01%) |
PKCh | inactive (10001nM) | inactive (110.16%) |
PKCi | inactive (10001nM) | inactive (106.35%) |
PKCt | inactive (10001nM) | inactive (72.45%) |
PKCa | - | inactive (83.03%) |
PKCg | - | inactive (79.34%) |
PKCz | - | inactive (79.68%) |
PKCb | - | inactive (99.84%) |
AGC - PKG
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PKG1 | inactive (10001nM) | inactive (95.37%) |
PKG2 | inactive (10001nM) | inactive (107.5%) |
AGC - RSK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
p70S6K | inactive (10001nM) | inactive (95.72%) |
MSK1 | - | inactive (98.31%) |
MSK2 | - | inactive (93.44%) |
p70S6Kb | - | inactive (100.35%) |
RSK2 | - | inactive (104.62%) |
RSK4 | - | inactive (107.71%) |
RSK1 | - | inactive (105.13%) |
RSK3 | - | inactive (83.98%) |
AGC - SGK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
SGK3 | inactive (10001nM) | inactive (101.69%) |
SGK1 | - | inactive (127.66%) |
SGK2 | - | inactive (105.63%) |
AGC - YANK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
YANK1 | inactive (10001nM) | - |
YANK2 | inactive (10001nM) | - |
YANK3 | inactive (10001nM) | - |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | DRx | RBC |
---|
AMPKa1 | inactive (10001nM) | - |
AMPKa2 | inactive (10001nM) | - |
NuaK1 | inactive (10001nM) | inactive (108.13%) |
BRSK1 | inactive (10001nM) | inactive (98.57%) |
BRSK2 | inactive (10001nM) | inactive (106.01%) |
CHK1 | inactive (10001nM) | inactive (100.47%) |
HUNK | inactive (10001nM) | - |
LKB1 | inactive (10001nM) | inactive (105.81%) |
MARK1 | inactive (10001nM) | inactive (148.99%) |
MARK2 | inactive (10001nM) | inactive (137.16%) |
MARK3 | inactive (10001nM) | inactive (95.85%) |
MARK4 | inactive (10001nM) | inactive (103.54%) |
MELK | inactive (10001nM) | inactive (88.53%) |
NIM1 | inactive (10001nM) | - |
QSK | inactive (10001nM) | - |
SIK | inactive (10001nM) | - |
QIK | inactive (10001nM) | inactive (100.8%) |
NuaK2 | inactive (10001nM) | inactive (95.11%) |
SNRK | inactive (10001nM) | - |
PASK | - | inactive (100.75%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CaMK1a | inactive (10001nM) | inactive (101.92%) |
CaMK1d | inactive (10001nM) | inactive (103.79%) |
CaMK1g | inactive (10001nM) | inactive (102.36%) |
CaMK4 | inactive (10001nM) | inactive (107.16%) |
CaMK1b | - | inactive (98.08%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CaMK2a | inactive (10001nM) | inactive (98.58%) |
CaMK2b | inactive (10001nM) | inactive (93.76%) |
CaMK2d | inactive (10001nM) | inactive (92.46%) |
CaMK2g | inactive (10001nM) | inactive (110.85%) |
CAMK - CASK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CASK | inactive (10001nM) | - |
CAMK - RAD53
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CHK2 | inactive (10001nM) | inactive (96.83%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
DAPK1 | inactive (10001nM) | inactive (107.11%) |
DAPK2 | inactive (10001nM) | inactive (103.43%) |
DAPK3 | inactive (10001nM) | inactive (97.41%) |
DRAK1 | inactive (10001nM) | inactive (89.71%) |
DRAK2 | inactive (10001nM) | - |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | DRx | RBC |
---|
DCLK1 | inactive (10001nM) | - |
DCLK2 | inactive (10001nM) | inactive (101%) |
DCLK3 | inactive (10001nM) | - |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
MAPKAPK2 | inactive (10001nM) | inactive (94.71%) |
MAPKAPK5 | inactive (10001nM) | inactive (92.78%) |
MNK1 | inactive (10001nM) | inactive (94.53%) |
MNK2 | inactive (10001nM) | inactive (97.27%) |
MAPKAPK3 | - | inactive (102.69%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
caMLCK | inactive (10001nM) | - |
smMLCK | inactive (10001nM) | inactive (90.72%) |
skMLCK | inactive (10001nM) | inactive (108.21%) |
SgK085 | inactive (10001nM) | - |
CAMK - PHK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PHKg1 | inactive (10001nM) | inactive (95.71%) |
PHKg2 | inactive (10001nM) | inactive (99.47%) |
CAMK - PIM
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PIM1 | inactive (10001nM) | inactive (99%) |
PIM2 | inactive (10001nM) | inactive (101.64%) |
PIM3 | inactive (10001nM) | inactive (93.7%) |
CAMK - PKD
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PKD1 | inactive (10001nM) | inactive (99.43%) |
PKD2 | inactive (10001nM) | inactive (86.41%) |
PKD3 | inactive (10001nM) | inactive (88.55%) |
CAMK - STK33
Bioactivity |
---|
Kinase | DRx | RBC |
---|
STK33 | inactive (10001nM) | inactive (94.74%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
TSSK1 | inactive (10001nM) | inactive (79.03%) |
TSSK2 | - | inactive (89.86%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | DRx | RBC |
---|
MAP3K5 | inactive (10001nM) | inactive (104.9%) |
MAP3K6 | inactive (10001nM) | - |
MAP3K1 | inactive (10001nM) | - |
MAP3K7 | inactive (10001nM) | - |
MAP3K2 | inactive (10001nM) | inactive (123.21%) |
MAP3K3 | inactive (10001nM) | inactive (109.83%) |
MAP3K4 | inactive (10001nM) | - |
MAP3K8 | inactive (10001nM) | - |
STE - STE20
Bioactivity |
---|
Kinase | DRx | RBC |
---|
HPK1 | inactive (10001nM) | - |
LOK | inactive (4400nM) | inactive (94.79%) |
GCK | inactive (10001nM) | inactive (104.14%) |
KHS2 | inactive (10001nM) | - |
HGK | inactive (10001nM) | inactive (111.21%) |
KHS1 | inactive (10001nM) | inactive (109.07%) |
MINK | inactive (10001nM) | inactive (110.74%) |
MST1 | inactive (10001nM) | inactive (99.36%) |
MST2 | inactive (10001nM) | inactive (93.75%) |
MST3 | inactive (10001nM) | inactive (106.39%) |
MST4 | inactive (10001nM) | inactive (109.93%) |
MYO3A | inactive (10001nM) | - |
MYO3B | inactive (10001nM) | inactive (96.08%) |
OSR1 | inactive (10001nM) | inactive (104.51%) |
PAK1 | inactive (10001nM) | inactive (110.31%) |
PAK2 | inactive (10001nM) | inactive (101.75%) |
PAK3 | inactive (10001nM) | inactive (104.93%) |
PAK4 | inactive (10001nM) | inactive (89.93%) |
PAK6 | inactive (10001nM) | inactive (106.47%) |
PAK5 | inactive (10001nM) | inactive (98.52%) |
SLK | inactive (3300nM) | inactive (85.06%) |
STLK3 | inactive (10001nM) | inactive (100.2%) |
TAO1 | inactive (10001nM) | inactive (98.81%) |
TAO2 | inactive (10001nM) | inactive (105.04%) |
TAO3 | inactive (10001nM) | inactive (100.98%) |
TNIK | inactive (10001nM) | - |
YSK1 | inactive (10001nM) | inactive (102.05%) |
STE - STE7
Bioactivity |
---|
Kinase | DRx | RBC |
---|
MAP2K1 | inactive (10001nM) | inactive (104.87%) |
MAP2K2 | inactive (10001nM) | inactive (106.04%) |
MAP2K3 | inactive (10001nM) | - |
MAP2K4 | inactive (10001nM) | - |
MAP2K5 | active (1100nM) | - |
MAP2K6 | inactive (10001nM) | inactive (95.37%) |
MAP2K7 | inactive (4400nM) | - |
STE - STE-Unique
Bioactivity |
---|
Kinase | DRx | RBC |
---|
COT | - | inactive (99.73%) |
NIK | - | inactive (108.8%) |
CMGC
CMGC - CDK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
PITSLRE | inactive (10001nM) | - |
CHED | inactive (10001nM) | - |
CDK11 | inactive (10001nM) | - |
PCTAIRE1 | inactive (10001nM) | - |
PCTAIRE2 | inactive (10001nM) | - |
PCTAIRE3 | inactive (10001nM) | - |
PFTAIRE2 | inactive (10001nM) | - |
PFTAIRE1 | inactive (10001nM) | - |
CMGC - CDKL
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CDKL1 | inactive (10001nM) | - |
CDKL2 | inactive (10001nM) | - |
CDKL3 | inactive (10001nM) | - |
CDKL5 | inactive (10001nM) | - |
CMGC - CLK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CLK1 | inactive (10001nM) | inactive (107.26%) |
CLK2 | inactive (10001nM) | inactive (95.11%) |
CLK3 | inactive (10001nM) | inactive (107.13%) |
CLK4 | inactive (10001nM) | inactive (114.72%) |
CMGC - CK2
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CK2a1 | inactive (10001nM) | inactive (120.84%) |
CK2a2 | inactive (10001nM) | inactive (100.76%) |
CMGC - DYRK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
DYRK1A | inactive (10001nM) | inactive (101.44%) |
DYRK1B | inactive (10001nM) | inactive (93.07%) |
DYRK2 | inactive (10001nM) | inactive (102.31%) |
HIPK1 | inactive (10001nM) | inactive (97.06%) |
HIPK2 | inactive (10001nM) | inactive (104.05%) |
HIPK3 | inactive (10001nM) | inactive (99.06%) |
HIPK4 | inactive (10001nM) | inactive (108.49%) |
PRP4 | inactive (10001nM) | - |
DYRK3 | - | inactive (90.17%) |
DYRK4 | - | inactive (102.58%) |
CMGC - MAPK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
Erk1 | inactive (10001nM) | inactive (94.8%) |
Erk2 | inactive (10001nM) | inactive (101.88%) |
Erk3 | inactive (10001nM) | - |
Erk4 | inactive (10001nM) | - |
Erk5 | inactive (10001nM) | - |
Erk7 | inactive (10001nM) | - |
JNK1 | inactive (10001nM) | inactive (91.95%) |
JNK2 | inactive (10001nM) | inactive (98.14%) |
JNK3 | inactive (10001nM) | inactive (100.4%) |
NLK | inactive (10001nM) | inactive (108.16%) |
p38a | inactive (10001nM) | inactive (100.89%) |
p38b | inactive (10001nM) | inactive (100.65%) |
p38d | inactive (10001nM) | inactive (91.11%) |
p38g | inactive (10001nM) | inactive (95.02%) |
CMGC - GSK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
GSK3A | inactive (10001nM) | inactive (105.21%) |
GSK3B | inactive (10001nM) | inactive (102.88%) |
CMGC - RCK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
ICK | inactive (10001nM) | - |
MAK | inactive (10001nM) | - |
CMGC - SRPK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
SRPK1 | inactive (10001nM) | inactive (100.37%) |
SRPK2 | inactive (10001nM) | inactive (87.97%) |
MSSK1 | inactive (10001nM) | inactive (103.58%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | DRx | RBC |
---|
CK1 | 7 | 7 | 6 |
VRK | 3 | 1 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | DRx | RBC |
---|
CK1a | inactive (10001nM) | inactive (104.15%) |
CK1a2 | inactive (10001nM) | - |
CK1d | inactive (10001nM) | inactive (91.19%) |
CK1e | inactive (10001nM) | inactive (99.39%) |
CK1g1 | inactive (10001nM) | inactive (104.78%) |
CK1g2 | inactive (10001nM) | inactive (99.53%) |
CK1g3 | inactive (10001nM) | inactive (104.2%) |
CK1 - VRK
Bioactivity |
---|
Kinase | DRx | RBC |
---|
VRK2 | inactive (10001nM) | - |
VRK1 | - | inactive (100.72%) |