Compound Information
Test on : RBC
Compound Name : -
Inchikey : AXPBLFXFGVEGKU-UHFFFAOYSA-N
CANNOT FIND
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
Bioactivity |
---|
Kinase | RBC |
---|
PDK1 | inactive (89.8%) |
AGC - Akt
Bioactivity |
---|
Kinase | RBC |
---|
AKT1 | inactive (94.41%) |
AKT2 | inactive (104.2%) |
AKT3 | inactive (90.66%) |
AGC - DMPK
Bioactivity |
---|
Kinase | RBC |
---|
DMPK1 | inactive (98.73%) |
MRCKa | inactive (112.35%) |
MRCKb | inactive (88.17%) |
ROCK1 | inactive (104.99%) |
ROCK2 | inactive (85.02%) |
AGC - GRK
Bioactivity |
---|
Kinase | RBC |
---|
BARK1 | inactive (97.31%) |
BARK2 | inactive (99.17%) |
GPRK4 | inactive (92.4%) |
GPRK5 | inactive (108.56%) |
GPRK6 | inactive (99.5%) |
GPRK7 | inactive (100.85%) |
AGC - RSK
Bioactivity |
---|
Kinase | RBC |
---|
MSK1 | inactive (90.78%) |
MSK2 | inactive (101.44%) |
p70S6K | inactive (87.67%) |
p70S6Kb | inactive (107.29%) |
RSK2 | inactive (80.14%) |
RSK4 | inactive (62.05%) |
RSK1 | inactive (80.42%) |
RSK3 | active (44.2%) |
AGC - PKA
Bioactivity |
---|
Kinase | RBC |
---|
PKACg | inactive (99.22%) |
PRKX | inactive (110.05%) |
PKACa | inactive (73.81%) |
AGC - PKC
Bioactivity |
---|
Kinase | RBC |
---|
PKCa | active (49.46%) |
PKCd | active (40.27%) |
PKCe | inactive (78.02%) |
PKCh | inactive (102.43%) |
PKCg | inactive (93.64%) |
PKCi | inactive (99.38%) |
PKCt | inactive (71.53%) |
PKCz | inactive (89.75%) |
PKCb | inactive (88.37%) |
AGC - PKG
Bioactivity |
---|
Kinase | RBC |
---|
PKG2 | inactive (108.94%) |
PKG1 | inactive (85.45%) |
AGC - PKN
Bioactivity |
---|
Kinase | RBC |
---|
PKN1 | inactive (74.18%) |
PKN2 | inactive (105.37%) |
AGC - SGK
Bioactivity |
---|
Kinase | RBC |
---|
SGK1 | inactive (125.57%) |
SGK2 | inactive (103.19%) |
SGK3 | inactive (94.38%) |
AGC - NDR
Bioactivity |
---|
Kinase | RBC |
---|
NDR1 | inactive (85.07%) |
TK
TK - Abl
Bioactivity |
---|
Kinase | RBC |
---|
ABL1 | active (1.8%) |
ABL2 | active (2.19%) |
TK - Ack
Bioactivity |
---|
Kinase | RBC |
---|
ACK | active (3.54%) |
TK - ALK
Bioactivity |
---|
Kinase | RBC |
---|
ALK | inactive (65.99%) |
LTK | inactive (57.74%) |
TK - Axl
Bioactivity |
---|
Kinase | RBC |
---|
AXL | active (37.63%) |
MER | active (28.92%) |
TYRO3 | active (47.75%) |
TK - Src
Bioactivity |
---|
Kinase | RBC |
---|
BLK | active (20.73%) |
BRK | inactive (93.08%) |
SRC | active (6.05%) |
FGR | active (11.49%) |
FRK | active (29.2%) |
FYN | active (29.42%) |
HCK | active (11.88%) |
LCK | active (1.88%) |
SRM | inactive (90.65%) |
YES | active (7.29%) |
LYN | active (2.13%) |
TK - Tec
Bioactivity |
---|
Kinase | RBC |
---|
BMX | active (14.48%) |
BTK | active (5.69%) |
ITK | inactive (103.18%) |
TEC | inactive (96.11%) |
TXK | active (27.53%) |
TK - PDGFR
Bioactivity |
---|
Kinase | RBC |
---|
KIT | inactive (93.64%) |
FLT3 | active (30.26%) |
FMS | active (43.09%) |
PDGFRb | inactive (74.83%) |
PDGFRa | inactive (86.95%) |
TK - Csk
Bioactivity |
---|
Kinase | RBC |
---|
CSK | active (12.33%) |
CTK | inactive (139.74%) |
TK - DDR
Bioactivity |
---|
Kinase | RBC |
---|
DDR2 | inactive (104.75%) |
TK - EGFR
Bioactivity |
---|
Kinase | RBC |
---|
EGFR | active (3.84%) |
ErbB2 | active (32.95%) |
ErbB4 | active (1.53%) |
TK - Eph
Bioactivity |
---|
Kinase | RBC |
---|
EphA1 | inactive (97.72%) |
EphA2 | active (9.58%) |
EphA3 | active (31.66%) |
EphA4 | active (27.01%) |
EphA5 | active (37.14%) |
EphA6 | active (4.38%) |
EphA7 | inactive (77.15%) |
EphA8 | active (10.52%) |
EphB1 | active (11.8%) |
EphB2 | active (17.43%) |
EphB3 | active (49.42%) |
EphB4 | active (12.48%) |
TK - FAK
Bioactivity |
---|
Kinase | RBC |
---|
FAK | inactive (95.96%) |
PYK2 | active (32.56%) |
TK - Fer
Bioactivity |
---|
Kinase | RBC |
---|
FER | inactive (54.64%) |
FES | active (35.71%) |
TK - FGFR
Bioactivity |
---|
Kinase | RBC |
---|
FGFR1 | inactive (64.42%) |
FGFR2 | inactive (58.1%) |
FGFR3 | inactive (82.57%) |
FGFR4 | inactive (94.06%) |
TK - VEGFR
Bioactivity |
---|
Kinase | RBC |
---|
FLT1 | active (44.54%) |
FLT4 | active (44.1%) |
KDR | inactive (65.28%) |
TK - InsR
Bioactivity |
---|
Kinase | RBC |
---|
IGF1R | inactive (91.55%) |
IRR | active (36.9%) |
INSR | inactive (69.81%) |
TK - JakA
Bioactivity |
---|
Kinase | RBC |
---|
JAK1 | inactive (98.99%) |
JAK2 | inactive (97.42%) |
JAK3 | inactive (88.5%) |
TYK2 | inactive (98.13%) |
TK - Musk
Bioactivity |
---|
Kinase | RBC |
---|
MUSK | inactive (81.66%) |
TK - Ret
Bioactivity |
---|
Kinase | RBC |
---|
RET | active (18.94%) |
TK - Met
Bioactivity |
---|
Kinase | RBC |
---|
RON | inactive (85.41%) |
MET | inactive (84.5%) |
TK - Sev
Bioactivity |
---|
Kinase | RBC |
---|
ROS | inactive (95.39%) |
TK - Syk
Bioactivity |
---|
Kinase | RBC |
---|
SYK | active (21.1%) |
ZAP70 | inactive (100.93%) |
TK - Tie
Bioactivity |
---|
Kinase | RBC |
---|
TIE2 | inactive (82.65%) |
TK - Trk
Bioactivity |
---|
Kinase | RBC |
---|
TRKA | inactive (105.65%) |
TRKB | inactive (69.15%) |
TRKC | active (15.25%) |
TKL
TKL - STKR
Bioactivity |
---|
Kinase | RBC |
---|
ALK1 | inactive (67.65%) |
ALK2 | inactive (93.27%) |
ALK4 | inactive (104.76%) |
TGFbR1 | inactive (99.05%) |
TGFbR2 | inactive (95.73%) |
TKL - RAF
Bioactivity |
---|
Kinase | RBC |
---|
ARAF | inactive (109.13%) |
BRAF | inactive (91.75%) |
RAF1 | inactive (104.98%) |
TKL - IRAK
Bioactivity |
---|
Kinase | RBC |
---|
IRAK1 | inactive (91.27%) |
IRAK4 | inactive (63.15%) |
TKL - LISK
Bioactivity |
---|
Kinase | RBC |
---|
LIMK1 | inactive (96.41%) |
TKL - LRRK
Bioactivity |
---|
Kinase | RBC |
---|
LRRK2 | active (30.12%) |
TKL - MLK
Bioactivity |
---|
Kinase | RBC |
---|
MLK1 | active (16.48%) |
MLK2 | active (22.88%) |
MLK3 | active (13.47%) |
TAK1 | active (28.29%) |
ZAK | inactive (67.65%) |
TKL - RIPK
Bioactivity |
---|
Kinase | RBC |
---|
RIPK2 | inactive (111.13%) |
CAMK
CAMK - CAMKL
Bioactivity |
---|
Kinase | RBC |
---|
NuaK1 | active (11.43%) |
BRSK1 | inactive (97.53%) |
BRSK2 | inactive (94.2%) |
CHK1 | active (38.9%) |
LKB1 | inactive (98.07%) |
MARK1 | inactive (108.81%) |
MARK3 | inactive (65.36%) |
MARK4 | inactive (60.56%) |
MELK | active (25.8%) |
PASK | inactive (108.82%) |
QIK | active (1.93%) |
NuaK2 | inactive (59.47%) |
MARK2 | inactive (99.92%) |
CAMK - CAMK1
Bioactivity |
---|
Kinase | RBC |
---|
CaMK1a | inactive (68.94%) |
CaMK1b | inactive (109.23%) |
CaMK1d | active (16.57%) |
CaMK1g | inactive (82.66%) |
CaMK4 | inactive (90.66%) |
CAMK - CAMK2
Bioactivity |
---|
Kinase | RBC |
---|
CaMK2a | inactive (92.7%) |
CaMK2b | inactive (86.25%) |
CaMK2d | inactive (94.59%) |
CaMK2g | inactive (130.84%) |
CAMK - RAD53
Bioactivity |
---|
Kinase | RBC |
---|
CHK2 | active (21.7%) |
CAMK - DAPK
Bioactivity |
---|
Kinase | RBC |
---|
DAPK1 | inactive (105.76%) |
DAPK2 | inactive (82.86%) |
DRAK1 | inactive (107.35%) |
DAPK3 | inactive (106.92%) |
CAMK - DCAMKL
Bioactivity |
---|
Kinase | RBC |
---|
DCLK2 | inactive (98.39%) |
CAMK - MAPKAPK
Bioactivity |
---|
Kinase | RBC |
---|
MAPKAPK2 | inactive (94.74%) |
MAPKAPK3 | inactive (98.22%) |
MAPKAPK5 | inactive (94.74%) |
MNK1 | inactive (96.92%) |
MNK2 | inactive (98.7%) |
CAMK - MLCK
Bioactivity |
---|
Kinase | RBC |
---|
smMLCK | inactive (72.04%) |
skMLCK | active (32.05%) |
CAMK - PHK
Bioactivity |
---|
Kinase | RBC |
---|
PHKg1 | inactive (52.08%) |
PHKg2 | inactive (102.96%) |
CAMK - PIM
Bioactivity |
---|
Kinase | RBC |
---|
PIM1 | inactive (99.16%) |
PIM2 | inactive (111.49%) |
PIM3 | inactive (97.69%) |
CAMK - PKD
Bioactivity |
---|
Kinase | RBC |
---|
PKD1 | active (43.71%) |
PKD3 | active (42.25%) |
PKD2 | active (35.54%) |
CAMK - TSSK
Bioactivity |
---|
Kinase | RBC |
---|
TSSK1 | inactive (79.24%) |
TSSK2 | inactive (83.89%) |
CAMK - STK33
Bioactivity |
---|
Kinase | RBC |
---|
STK33 | inactive (63.55%) |
STE
STE - STE11
Bioactivity |
---|
Kinase | RBC |
---|
MAP3K5 | inactive (95.7%) |
MAP3K2 | active (23.47%) |
MAP3K3 | active (11.8%) |
STE - STE-Unique
Bioactivity |
---|
Kinase | RBC |
---|
COT | inactive (100.88%) |
NIK | inactive (129.16%) |
STE - STE20
Bioactivity |
---|
Kinase | RBC |
---|
GCK | active (3.16%) |
HGK | active (1.03%) |
KHS1 | active (1.72%) |
LOK | active (12.61%) |
MINK | active (1.21%) |
MST1 | active (7.4%) |
MST2 | active (13.86%) |
MST3 | active (11.02%) |
MST4 | active (5.9%) |
OSR1 | inactive (100.06%) |
PAK1 | active (11.68%) |
PAK2 | inactive (69.37%) |
PAK3 | active (9.9%) |
PAK4 | inactive (95.78%) |
PAK5 | inactive (83.64%) |
PAK6 | inactive (104.67%) |
SLK | active (21.59%) |
YSK1 | active (10.1%) |
STLK3 | inactive (93.6%) |
TAO1 | inactive (52.78%) |
TAO2 | inactive (65.41%) |
TAO3 | inactive (71.33%) |
MYO3B | active (40.28%) |
STE - STE7
Bioactivity |
---|
Kinase | RBC |
---|
MAP2K1 | inactive (65.35%) |
MAP2K2 | active (8.43%) |
MAP2K6 | inactive (93.44%) |
Other
Other - Aur
Bioactivity |
---|
Kinase | RBC |
---|
AurA | inactive (86.04%) |
AurB | inactive (83.15%) |
AurC | inactive (82.1%) |
Other - CAMKK
Bioactivity |
---|
Kinase | RBC |
---|
CaMKK1 | inactive (84.79%) |
CaMKK2 | inactive (85.13%) |
Other - Haspin
Bioactivity |
---|
Kinase | RBC |
---|
Haspin | inactive (65.6%) |
Other - IKK
Bioactivity |
---|
Kinase | RBC |
---|
IKKa | inactive (98.1%) |
IKKb | inactive (95.36%) |
IKKe | inactive (75.45%) |
TBK1 | inactive (65.68%) |
Other - NEK
Bioactivity |
---|
Kinase | RBC |
---|
NEK1 | active (15.17%) |
NEK11 | inactive (93.98%) |
NEK2 | active (8.56%) |
NEK4 | active (32.6%) |
NEK6 | inactive (85.32%) |
NEK7 | inactive (94.61%) |
NEK9 | inactive (94.04%) |
NEK3 | inactive (85.88%) |
Other - TOPK
Bioactivity |
---|
Kinase | RBC |
---|
PBK | inactive (104.39%) |
Other - PLK
Bioactivity |
---|
Kinase | RBC |
---|
PLK1 | inactive (93.81%) |
PLK2 | inactive (100.07%) |
PLK3 | inactive (98.49%) |
Other - SgK496
Bioactivity |
---|
Kinase | RBC |
---|
SgK496 | inactive (104.48%) |
Other - NAK
Bioactivity |
---|
Kinase | RBC |
---|
MPSK1 | inactive (85.12%) |
Other - TTK
Bioactivity |
---|
Kinase | RBC |
---|
TTK | inactive (109.96%) |
Other - ULK
Bioactivity |
---|
Kinase | RBC |
---|
ULK1 | inactive (79.11%) |
ULK2 | inactive (92.25%) |
ULK3 | inactive (100.34%) |
Other - WEE
Bioactivity |
---|
Kinase | RBC |
---|
Wee1 | active (40.47%) |
Other - WNK
Bioactivity |
---|
Kinase | RBC |
---|
Wnk2 | inactive (94.23%) |
Wnk3 | inactive (91.81%) |
Other - TLK
Bioactivity |
---|
Kinase | RBC |
---|
TLK2 | inactive (92.16%) |
CK1
CK1
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
CK1 | 7 | 6 |
VRK | 3 | 1 |
CK1 - CK1
Bioactivity |
---|
Kinase | RBC |
---|
CK1d | active (10.86%) |
CK1g1 | inactive (95.69%) |
CK1g2 | inactive (98.25%) |
CK1g3 | inactive (98.29%) |
CK1a | active (49.52%) |
CK1e | active (11.44%) |
CK1 - VRK
Bioactivity |
---|
Kinase | RBC |
---|
VRK1 | inactive (100.25%) |
CMGC
CMGC - CK2
Bioactivity |
---|
Kinase | RBC |
---|
CK2a1 | inactive (115.6%) |
CK2a2 | inactive (108.03%) |
CMGC - CLK
Bioactivity |
---|
Kinase | RBC |
---|
CLK1 | inactive (81.01%) |
CLK2 | inactive (69.3%) |
CLK3 | inactive (94.93%) |
CLK4 | inactive (76.63%) |
CMGC - DYRK
Bioactivity |
---|
Kinase | RBC |
---|
DYRK1A | inactive (99.39%) |
DYRK1B | inactive (97.05%) |
DYRK2 | inactive (104.26%) |
DYRK3 | inactive (91.76%) |
DYRK4 | inactive (97.93%) |
HIPK1 | inactive (96.28%) |
HIPK2 | inactive (89.05%) |
HIPK3 | inactive (93.5%) |
HIPK4 | inactive (74.57%) |
CMGC - MAPK
Bioactivity |
---|
Kinase | RBC |
---|
Erk1 | inactive (98.9%) |
Erk2 | inactive (93.66%) |
JNK3 | inactive (105.52%) |
NLK | inactive (101.16%) |
p38a | inactive (88.59%) |
p38b | inactive (101.09%) |
p38d | inactive (91.24%) |
p38g | inactive (99.94%) |
JNK1 | inactive (105.13%) |
JNK2 | inactive (108.01%) |
CMGC - GSK
Bioactivity |
---|
Kinase | RBC |
---|
GSK3A | inactive (102.67%) |
GSK3B | inactive (99.88%) |
CMGC - SRPK
Bioactivity |
---|
Kinase | RBC |
---|
MSSK1 | inactive (105.59%) |
SRPK1 | inactive (98.45%) |
SRPK2 | inactive (100.54%) |
Atypical
Atypical
Test Member No. in Family |
---|
Family | no. Member on 518kinase | RBC |
---|
PDHK | 5 | 1 |
Atypical - PDHK
Bioactivity |
---|
Kinase | RBC |
---|
PDHK1 | inactive (89.8%) |