Q9UF33 EphA6


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Group: TK
Family: Eph
PDB Structure Num: 0
FDA approved drugs from DrugBank: Fostamatinib






structureFDA kinase druginchikeykinase profiling data countkinase profiling labelChEMBL data countChEMBL labelvote label
BPNUQXPIQBZCMR-LJQANCHMSA-N1inactive--inactive
WJEOLQLKVOPQFV-UHFFFAOYSA-N2inactive--inactive
MPVGZUGXCQEXTM-UHFFFAOYSA-N1active--active
CVWXJKQAOSCOAB-UHFFFAOYSA-N1inactive--inactive
RITAVMQDGBJQJZ-UHFFFAOYSA-N1inactive--inactive
RAHBGWKEPAQNFF-UHFFFAOYSA-N1active--active
ODPGGGTTYSGTGO-UHFFFAOYSA-N1active--active
OVPNQJVDAFNBDN-UHFFFAOYSA-N1inactive--inactive
QYZOGCMHVIGURT-UHFFFAOYSA-N1inactive--inactive
XXJWYDDUDKYVKI-UHFFFAOYSA-N1active--active
CYOHGALHFOKKQC-UHFFFAOYSA-N1inactive--inactive
XQVVPGYIWAGRNI-QFIPXVFZSA-N1inactive--inactive
-FCLPVPNWFDOVKL-DQSJHHFOSA-N1active--active
ULXXDDBFHOBEHA-INIZCTEOSA-N1active--active
MVCOAUNKQVWQHZ-UHFFFAOYSA-N1active--active
PSPFQEBFYXJZEV-UHFFFAOYSA-N1inactive--inactive
OUSFTKFNBAZUKL-UHFFFAOYSA-N1inactive--inactive
WCWUXEGQKLTGDX-NSHDSACASA-N1active--active
UIARLYUEJFELEN-FMLDBKJISA-N1active--active
-KCOYQXZDFIIGCY-CZIZESTLSA-N1inactive--inactive
YABJJWZLRMPFSI-UHFFFAOYSA-N1active--active
OMZCMEYTWSXEPZ-UHFFFAOYSA-N1active--active
GFMMXOIFOQCCGU-UHFFFAOYSA-N1inactive--inactive
UJLAWZDWDVHWOW-DGCLKSJQSA-N1inactive--inactive
CrizotinibKTEIFNKAUNYNJU-GFCCVEGCSA-N1active--active
DasatinibZBNZXTGUTAYRHI-UHFFFAOYSA-N2exclude--exclude
ErlotinibAAKJLRGGTJKAMG-UHFFFAOYSA-N2active--active
CXQHYVUVSFXTMY-UHFFFAOYSA-N1active--active
BIIVYFLTOXDAOV-YVEFUNNKSA-N1inactive--inactive
DEZZLWQELQORIU-UHFFFAOYSA-N1inactive--inactive
LHNIIDJUOCFXAP-UHFFFAOYSA-N1inactive--inactive
GefitinibXGALLCVXEZPNRQ-UHFFFAOYSA-N2active--active
-XWFUWIOJOVXAMS-FXIRQEPWSA-N1inactive--inactive
ZHJGWYRLJUCMRT-QGZVFWFLSA-N1inactive--inactive
KGPGFQWBCSZGEL-ZDUSSCGKSA-N1inactive--inactive
MYQAUKPBNJWPIE-UHFFFAOYSA-N1inactive--inactive
JWNPDZNEKVCWMY-UHFFFAOYSA-N1inactive--inactive
ImatinibKTUFNOKKBVMGRW-UHFFFAOYSA-N2inactive--inactive
RuxolitinibHFNKQEVNSGCOJV-OAHLLOKOSA-N1inactive--inactive
-OLESUNNHPSUJLS-UHFFFAOYSA-N1inactive--inactive
SHPFDGWALWEPGS-UHFFFAOYSA-N1inactive--inactive
YYLKKYCXAOBSRM-UHFFFAOYSA-N1active--active
LapatinibBCFGMOOMADDAQU-UHFFFAOYSA-N2inactive--inactive
UUADYKVKJIMIPA-UHFFFAOYSA-N1inactive--inactive
ZCBUQCWBWNUWSU-SFHVURJKSA-N1inactive--inactive
ZNOLRTPMNMPLHY-UHFFFAOYSA-N1inactive--inactive
UXXQOJXBIDBUAC-UHFFFAOYSA-N2inactive--inactive
HHFBDROWDBDFBR-UHFFFAOYSA-N1active--active
NilotinibHHZIURLSWUIHRB-UHFFFAOYSA-N2active--active
PazopanibCUIHSIWYWATEQL-UHFFFAOYSA-N2inactive--inactive
VAARYSWULJUGST-UHFFFAOYSA-N1active--active
OYONTEXKYJZFHA-OAQYLSRUSA-N1inactive--inactive
TUVCWJQQGGETHL-UHFFFAOYSA-N2inactive--inactive
BMGQWWVMWDBQGC-PZFYLCKJSA-N2inactive--inactive
YZDJQTHVDDOVHR-UHFFFAOYSA-N1inactive--inactive
-MTICIDWIKCANDD-UHFFFAOYSA-N1active--active
YCOYDOIWSSHVCK-UHFFFAOYSA-N2inactive--inactive
TamatinibNHHQJBCNYHBUSI-UHFFFAOYSA-N1active--active
JRNJNYBQQYBCLE-UHFFFAOYSA-N1inactive--inactive
CDMGBJANTYXAIV-HHHXNRCGSA-N1active--active
BCZUAADEACICHN-UHFFFAOYSA-N1inactive--inactive
BosutinibUBPYILGKFZZVDX-UHFFFAOYSA-N1active--active
SorafenibMLDQJTXFUGDVEO-UHFFFAOYSA-N2active--active
HKSZLNNOFSGOKW-FYTWVXJKSA-N1active--active
CTNPALGJUAXMMC-PMFHANACSA-N1active--active
SunitinibWINHZLLDWRZWRT-ATVHPVEESA-N2active--active
QQWUGDVOUVUTOY-UHFFFAOYSA-N1active--active
UJIAQDJKSXQLIT-UHFFFAOYSA-N1inactive--inactive
JOOXLOJCABQBSG-UHFFFAOYSA-N1inactive--inactive
VandetanibUHTHHESEBZOYNR-UHFFFAOYSA-N2active--active
GCIKSSRWRFVXBI-UHFFFAOYSA-N2exclude--exclude
VEPKQEUBKLEPRA-UHFFFAOYSA-N1inactive--inactive
NJTUORMLOPXPBY-UHFFFAOYSA-N1inactive--inactive
ODZGYELAMAOARP-UHFFFAOYSA-N1inactive--inactive
ZUDPNBZMAJGYTE-UHFFFAOYSA-N1inactive--inactive
AVLYNJZZQYEFEA-UHFFFAOYSA-N1inactive--inactive
KQMPRSZTUSSXND-UHFFFAOYSA-N1inactive--inactive
ZXVUBPLDUMSDOE-UHFFFAOYSA-N1inactive--inactive
KOZFSFOOLUUIGY-IYYJOCMQSA-N1inactive--inactive
QQUXFYAWXPMDOE-UHFFFAOYSA-N1inactive--inactive
-BLLBARDQJSOSJD-PGUFJCEWSA-N1inactive--inactive
LLLQTDSSHZREGW-UHFFFAOYSA-N1inactive--inactive
FMETVQKSDIOGPX-UHFFFAOYSA-N1inactive--inactive
CZQHHVNHHHRRDU-UHFFFAOYSA-N1inactive--inactive
NGAGMBNBKCDCDJ-UHFFFAOYSA-N1inactive--inactive
-NHBMKTBZZSJUGA-HKRCYGBASA-N1inactive--inactive
GYQSWJNGTWVFOL-UHFFFAOYSA-N1inactive--inactive
JLOXTZFYJNCPIS-UHFFFAOYSA-N1inactive--inactive
FPYJSJDOHRDAMT-UHFFFAOYSA-N1active--active
UQPMANVRZYYQMD-UHFFFAOYSA-N1active--active
ODYAQBDIXCVKAE-UHFFFAOYSA-N1inactive--inactive
IBAKVEUZKHOWNG-UHFFFAOYSA-N1inactive--inactive
VXPWQNBKEIVYIS-OAHLLOKOSA-N1inactive--inactive
DZFBYHUKZSRPHU-UHFFFAOYSA-N1inactive--inactive
QFWCYNPOPKQOKV-UHFFFAOYSA-N1inactive--inactive
BGIYKDUASORTBB-UHFFFAOYSA-N1inactive--inactive
KFHMLBXBRCITHF-UHFFFAOYSA-N1inactive--inactive
WUPUZEMRHDROEO-UHFFFAOYSA-N1inactive--inactive
CZDUJGOCEPWCNA-UHFFFAOYSA-N1inactive--inactive
INTPTKHSGKBHHW-UHFFFAOYSA-N1inactive--inactive
ZDNURMVOKAERHZ-UHFFFAOYSA-N1inactive--inactive
PEPCXHNLEXQQSE-UHFFFAOYSA-N1active--active
-DGCXNBUJPWPMJJ-UHFFFAOYSA-N1inactive--inactive
VFBGXTUGODTSPK-UHFFFAOYSA-N1active--active
ZJFMARHFPUZEKI-UHFFFAOYSA-N1inactive--inactive
SQWZFLMPDUSYGV-UHFFFAOYSA-N1inactive--inactive
SRLVNYDXMUGOFI-UHFFFAOYSA-N1inactive--inactive
KKDPIZPUTYIBFX-UHFFFAOYSA-N1inactive--inactive
GDQXJQSQYMMKRA-UHFFFAOYSA-N1active--active
RONQPWQYDRPRGG-UHFFFAOYSA-N1inactive--inactive
KIWODJBCHRADND-UHFFFAOYSA-N1inactive--inactive
PMXCMJLOPOFPBT-OAHLLOKOSA-N1inactive--inactive
-QFJCIRLUMZQUOT-JRLVRMFHSA-N1inactive--inactive
LLJRXVHJOJRCSM-UHFFFAOYSA-N1inactive--inactive
CMKMGFAUKPAOMG-AWEZNQCLSA-N1inactive--inactive
FXGHOAZJQNLNFD-KRWDZBQOSA-N1inactive--inactive
-XFXDYDZBKXMGBX-HOTGVXAUSA-N1inactive--inactive
-NJNKPVPFGLGHPA-UHFFFAOYSA-N1inactive--inactive
CDMGBJANTYXAIV-MHZLTWQESA-N1inactive--inactive
VSPFURGQAYMVAN-UHFFFAOYSA-N1inactive--inactive
OTPNDVKVEAIXTI-IYBDPMFKSA-N1inactive--inactive
BHWCZLOXTLWZAQ-UHFFFAOYSA-N1inactive--inactive
YOELZIQOLWZLQC-UHFFFAOYSA-N1inactive--inactive
ZFGXZJKLOFCECI-UHFFFAOYSA-N1inactive--inactive
DMWVGXGXHPOEPT-UHFFFAOYSA-N1inactive--inactive
HKSZLNNOFSGOKW-HMWZOHBLSA-N1active--active
WNRSTFUVBWNELX-UHFFFAOYSA-N1inactive--inactive
LOGJQOUIVKBFGH-UHFFFAOYSA-N1inactive--inactive
QNUKRWAIZMBVCU-UHFFFAOYSA-N1inactive--inactive
XPLJEFSRINKZLC-UHFFFAOYSA-N1active--active
MLKHXLFEYOOYEY-UHFFFAOYSA-N1active--active
LCACSMNPIITJGG-UHFFFAOYSA-N1inactive--inactive
KFLWBZPSJQPRDD-UHFFFAOYSA-N1inactive--inactive
NMEUKWOOQOHUNA-UHFFFAOYSA-N1inactive--inactive
IBCXZJCWDGCXQT-UHFFFAOYSA-N1inactive--inactive
BTUOOXPZOVNPMF-UHFFFAOYSA-N1inactive--inactive
UOHFCPXBKJPCAD-UHFFFAOYSA-N1inactive--inactive
TUCIOBMMDDOEMM-UHFFFAOYSA-N1inactive--inactive
DXVJRTIPBNBLLB-UHFFFAOYSA-N1inactive--inactive
FQNCLVJEQCJWSU-UHFFFAOYSA-N1inactive--inactive
QNOXYUNHIGOWNY-UHFFFAOYSA-N1inactive--inactive
GFNNBHLJANVSQV-UHFFFAOYSA-N1active--active
PMUJUSJUVIXDQC-UHFFFAOYSA-N1inactive--inactive
GGPZCOONYBPZEW-UHFFFAOYSA-N1inactive--inactive
-YUWFTONEHHSMEI-CZUORRHYSA-N1inactive--inactive
RFHPWPWVGFSLOP-UHFFFAOYSA-N1inactive--inactive
WUWDLXZGHZSWQZ-UHFFFAOYSA-N1inactive--inactive
HBWLNACPIFKNIP-UHFFFAOYSA-N1inactive--inactive
-QDLHCMPXEPAAMD-BLNDMVMCSA-N1inactive--inactive
-BLQHLDXMMWHXIT-YSZXOBSOSA-N1inactive--inactive
-AXPBLFXFGVEGKU-UHFFFAOYSA-N1active--active
PIQCTGMSNWUMAF-UHFFFAOYSA-N1active--active
ZTFBIUXIQYRUNT-MDWZMJQESA-N1inactive--inactive
BTIHMVBBUGXLCJ-OAHLLOKOSA-N1inactive--inactive
UJLAWZDWDVHWOW-AAEUAGOBSA-N1inactive--inactive
FYSRKRZDBHOFAY-UHFFFAOYSA-N1inactive--inactive
ITOFPJRDSCGOSA-KZLRUDJFSA-N--1inactiveinactive
KHFTUYLQBLIIEQ-ZSSZZUKFSA-N--1inactiveinactive
ZEHBZHZMQSHZFI-UHFFFAOYSA-N--1inactiveinactive