| | BPNUQXPIQBZCMR-LJQANCHMSA-N | 1 | inactive | - | - | inactive |
| | WJEOLQLKVOPQFV-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | MPVGZUGXCQEXTM-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | CVWXJKQAOSCOAB-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | RITAVMQDGBJQJZ-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | RAHBGWKEPAQNFF-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | ODPGGGTTYSGTGO-UHFFFAOYSA-N | 1 | active | - | - | active |
| | OVPNQJVDAFNBDN-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | QYZOGCMHVIGURT-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | XXJWYDDUDKYVKI-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | CYOHGALHFOKKQC-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | XQVVPGYIWAGRNI-QFIPXVFZSA-N | 1 | inactive | - | - | inactive |
- | | FCLPVPNWFDOVKL-DQSJHHFOSA-N | 1 | inactive | - | - | inactive |
| | ULXXDDBFHOBEHA-INIZCTEOSA-N | 1 | inactive | - | - | inactive |
| | MVCOAUNKQVWQHZ-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | PSPFQEBFYXJZEV-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | OUSFTKFNBAZUKL-UHFFFAOYSA-N | 1 | active | - | - | active |
| | WCWUXEGQKLTGDX-NSHDSACASA-N | 1 | inactive | - | - | inactive |
| | UIARLYUEJFELEN-FMLDBKJISA-N | 1 | inactive | - | - | inactive |
- | | KCOYQXZDFIIGCY-CZIZESTLSA-N | 1 | inactive | - | - | inactive |
| | YABJJWZLRMPFSI-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | OMZCMEYTWSXEPZ-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | GFMMXOIFOQCCGU-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | UJLAWZDWDVHWOW-DGCLKSJQSA-N | 1 | inactive | - | - | inactive |
| Crizotinib | KTEIFNKAUNYNJU-GFCCVEGCSA-N | 1 | inactive | - | - | inactive |
| Dasatinib | ZBNZXTGUTAYRHI-UHFFFAOYSA-N | 1 | active | - | - | active |
| Erlotinib | AAKJLRGGTJKAMG-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | CXQHYVUVSFXTMY-UHFFFAOYSA-N | 1 | active | - | - | active |
| | BIIVYFLTOXDAOV-YVEFUNNKSA-N | 1 | inactive | - | - | inactive |
| | DEZZLWQELQORIU-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | LHNIIDJUOCFXAP-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| Gefitinib | XGALLCVXEZPNRQ-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
- | | XWFUWIOJOVXAMS-FXIRQEPWSA-N | 1 | inactive | - | - | inactive |
| | ZHJGWYRLJUCMRT-QGZVFWFLSA-N | 1 | inactive | - | - | inactive |
| | KGPGFQWBCSZGEL-ZDUSSCGKSA-N | 1 | active | - | - | active |
| | MYQAUKPBNJWPIE-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | JWNPDZNEKVCWMY-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| Imatinib | KTUFNOKKBVMGRW-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| Ruxolitinib | HFNKQEVNSGCOJV-OAHLLOKOSA-N | 1 | inactive | - | - | inactive |
- | | OLESUNNHPSUJLS-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | SHPFDGWALWEPGS-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | YYLKKYCXAOBSRM-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| Lapatinib | BCFGMOOMADDAQU-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | UUADYKVKJIMIPA-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | ZCBUQCWBWNUWSU-SFHVURJKSA-N | 1 | inactive | - | - | inactive |
| | ZNOLRTPMNMPLHY-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | UXXQOJXBIDBUAC-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | HHFBDROWDBDFBR-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| Nilotinib | HHZIURLSWUIHRB-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| Pazopanib | CUIHSIWYWATEQL-UHFFFAOYSA-N | 1 | active | - | - | active |
| | VAARYSWULJUGST-UHFFFAOYSA-N | 1 | active | - | - | active |
| | OYONTEXKYJZFHA-OAQYLSRUSA-N | 1 | inactive | - | - | inactive |
| | TUVCWJQQGGETHL-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | BMGQWWVMWDBQGC-PZFYLCKJSA-N | 1 | inactive | - | - | inactive |
| | YZDJQTHVDDOVHR-UHFFFAOYSA-N | 1 | active | - | - | active |
- | | MTICIDWIKCANDD-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | YCOYDOIWSSHVCK-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| Tamatinib | NHHQJBCNYHBUSI-UHFFFAOYSA-N | 1 | active | - | - | active |
| | JRNJNYBQQYBCLE-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | CDMGBJANTYXAIV-HHHXNRCGSA-N | 1 | active | - | - | active |
| | BCZUAADEACICHN-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| Bosutinib | UBPYILGKFZZVDX-UHFFFAOYSA-N | 1 | active | - | - | active |
| Sorafenib | MLDQJTXFUGDVEO-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | HKSZLNNOFSGOKW-FYTWVXJKSA-N | 1 | inactive | - | - | inactive |
| | CTNPALGJUAXMMC-PMFHANACSA-N | 1 | inactive | - | - | inactive |
| Sunitinib | WINHZLLDWRZWRT-ATVHPVEESA-N | 1 | inactive | - | - | inactive |
| | QQWUGDVOUVUTOY-UHFFFAOYSA-N | 1 | active | - | - | active |
| | UJIAQDJKSXQLIT-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | JOOXLOJCABQBSG-UHFFFAOYSA-N | 1 | active | - | - | active |
| Vandetanib | UHTHHESEBZOYNR-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | GCIKSSRWRFVXBI-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |
| | VEPKQEUBKLEPRA-UHFFFAOYSA-N | 1 | inactive | - | - | inactive |