Q15835 RHOK


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Group: AGC
Family: GRK
PDB Structure Num: 0






structureFDA kinase druginchikeykinase profiling data countkinase profiling labelChEMBL data countChEMBL labelvote label
BPNUQXPIQBZCMR-LJQANCHMSA-N1inactive--inactive
WJEOLQLKVOPQFV-UHFFFAOYSA-N1inactive--inactive
MPVGZUGXCQEXTM-UHFFFAOYSA-N1inactive--inactive
CVWXJKQAOSCOAB-UHFFFAOYSA-N1inactive--inactive
RITAVMQDGBJQJZ-UHFFFAOYSA-N1inactive--inactive
RAHBGWKEPAQNFF-UHFFFAOYSA-N1inactive--inactive
ODPGGGTTYSGTGO-UHFFFAOYSA-N1inactive--inactive
OVPNQJVDAFNBDN-UHFFFAOYSA-N1inactive--inactive
QYZOGCMHVIGURT-UHFFFAOYSA-N1inactive--inactive
XXJWYDDUDKYVKI-UHFFFAOYSA-N1inactive--inactive
CYOHGALHFOKKQC-UHFFFAOYSA-N1inactive--inactive
XQVVPGYIWAGRNI-QFIPXVFZSA-N1inactive--inactive
-FCLPVPNWFDOVKL-DQSJHHFOSA-N1active--active
ULXXDDBFHOBEHA-INIZCTEOSA-N1inactive--inactive
MVCOAUNKQVWQHZ-UHFFFAOYSA-N1inactive--inactive
PSPFQEBFYXJZEV-UHFFFAOYSA-N1inactive--inactive
OUSFTKFNBAZUKL-UHFFFAOYSA-N1inactive--inactive
WCWUXEGQKLTGDX-NSHDSACASA-N1inactive--inactive
UIARLYUEJFELEN-FMLDBKJISA-N1active--active
-KCOYQXZDFIIGCY-CZIZESTLSA-N1active--active
YABJJWZLRMPFSI-UHFFFAOYSA-N1inactive--inactive
OMZCMEYTWSXEPZ-UHFFFAOYSA-N1inactive--inactive
GFMMXOIFOQCCGU-UHFFFAOYSA-N1inactive--inactive
UJLAWZDWDVHWOW-DGCLKSJQSA-N1inactive--inactive
CrizotinibKTEIFNKAUNYNJU-GFCCVEGCSA-N1inactive--inactive
DasatinibZBNZXTGUTAYRHI-UHFFFAOYSA-N1inactive--inactive
ErlotinibAAKJLRGGTJKAMG-UHFFFAOYSA-N1inactive--inactive
CXQHYVUVSFXTMY-UHFFFAOYSA-N1inactive--inactive
BIIVYFLTOXDAOV-YVEFUNNKSA-N1active--active
DEZZLWQELQORIU-UHFFFAOYSA-N1inactive--inactive
LHNIIDJUOCFXAP-UHFFFAOYSA-N1inactive--inactive
GefitinibXGALLCVXEZPNRQ-UHFFFAOYSA-N1inactive--inactive
-XWFUWIOJOVXAMS-FXIRQEPWSA-N1active--active
ZHJGWYRLJUCMRT-QGZVFWFLSA-N1inactive--inactive
KGPGFQWBCSZGEL-ZDUSSCGKSA-N1active--active
MYQAUKPBNJWPIE-UHFFFAOYSA-N1inactive--inactive
JWNPDZNEKVCWMY-UHFFFAOYSA-N1inactive--inactive
ImatinibKTUFNOKKBVMGRW-UHFFFAOYSA-N1inactive--inactive
RuxolitinibHFNKQEVNSGCOJV-OAHLLOKOSA-N1active--active
-OLESUNNHPSUJLS-UHFFFAOYSA-N1active--active
SHPFDGWALWEPGS-UHFFFAOYSA-N1inactive--inactive
YYLKKYCXAOBSRM-UHFFFAOYSA-N1inactive--inactive
LapatinibBCFGMOOMADDAQU-UHFFFAOYSA-N1inactive--inactive
UUADYKVKJIMIPA-UHFFFAOYSA-N1active--active
ZCBUQCWBWNUWSU-SFHVURJKSA-N1active--active
ZNOLRTPMNMPLHY-UHFFFAOYSA-N1inactive--inactive
UXXQOJXBIDBUAC-UHFFFAOYSA-N1inactive--inactive
HHFBDROWDBDFBR-UHFFFAOYSA-N1inactive--inactive
NilotinibHHZIURLSWUIHRB-UHFFFAOYSA-N1inactive--inactive
PazopanibCUIHSIWYWATEQL-UHFFFAOYSA-N1inactive--inactive
VAARYSWULJUGST-UHFFFAOYSA-N1inactive--inactive
OYONTEXKYJZFHA-OAQYLSRUSA-N1active--active
TUVCWJQQGGETHL-UHFFFAOYSA-N1inactive--inactive
BMGQWWVMWDBQGC-PZFYLCKJSA-N1active--active
YZDJQTHVDDOVHR-UHFFFAOYSA-N1inactive--inactive
-MTICIDWIKCANDD-UHFFFAOYSA-N1active--active
YCOYDOIWSSHVCK-UHFFFAOYSA-N1inactive--inactive
TamatinibNHHQJBCNYHBUSI-UHFFFAOYSA-N1active--active
JRNJNYBQQYBCLE-UHFFFAOYSA-N1inactive--inactive
CDMGBJANTYXAIV-HHHXNRCGSA-N1inactive--inactive
BCZUAADEACICHN-UHFFFAOYSA-N1inactive--inactive
BosutinibUBPYILGKFZZVDX-UHFFFAOYSA-N1inactive--inactive
SorafenibMLDQJTXFUGDVEO-UHFFFAOYSA-N1inactive--inactive
HKSZLNNOFSGOKW-FYTWVXJKSA-N1active--active
CTNPALGJUAXMMC-PMFHANACSA-N1active--active
SunitinibWINHZLLDWRZWRT-ATVHPVEESA-N1active--active
QQWUGDVOUVUTOY-UHFFFAOYSA-N1active--active
UJIAQDJKSXQLIT-UHFFFAOYSA-N1inactive--inactive
JOOXLOJCABQBSG-UHFFFAOYSA-N1inactive--inactive
VandetanibUHTHHESEBZOYNR-UHFFFAOYSA-N1inactive--inactive
GCIKSSRWRFVXBI-UHFFFAOYSA-N1inactive--inactive
VEPKQEUBKLEPRA-UHFFFAOYSA-N1inactive--inactive
VWBSMGFTNCQOMB-UHFFFAOYSA-N--1inactiveinactive
BLMBNKDQXGINRE-UHFFFAOYSA-N--1inactiveinactive
JNVSJVSIHCPPTE-UHFFFAOYSA-N--1inactiveinactive
BXTYCBBDHNQJNG-UHFFFAOYSA-N--1inactiveinactive
UGYAZGXSMRGKRD-UHFFFAOYSA-N--1activeactive
ASPDMKGCEMLVBM-UHFFFAOYSA-N--1inactiveinactive
WFOVEDJTASPCIR-UHFFFAOYSA-N--1inactiveinactive
DMNINFHJFPFPIZ-UHFFFAOYSA-N--1activeactive
ZEHBZHZMQSHZFI-UHFFFAOYSA-N--1inactiveinactive
IDOAXNXBZZZOFX-UHFFFAOYSA-N--1inactiveinactive
GJTSGDBPSODHKH-UHFFFAOYSA-N--1inactiveinactive
YJQKIQOVJOGHMP-UHFFFAOYSA-N--1inactiveinactive
VUCAOBMPSJTWFL-UHFFFAOYSA-N--1inactiveinactive
QTCMCOOGSCOKGD-UHFFFAOYSA-N--1inactiveinactive
KQJWWWZXJNOLQF-UHFFFAOYSA-N--1inactiveinactive
JPDACOLMZSWYPX-UHFFFAOYSA-N--1inactiveinactive
FQDUDXKZLXZCSH-UHFFFAOYSA-N--1inactiveinactive
XXNLGEQPVDKVAF-UHFFFAOYSA-N--1inactiveinactive
XMXZNJPJVZOVGR-UHFFFAOYSA-N--1inactiveinactive
WYUIOBMKPJWABA-UHFFFAOYSA-N--1inactiveinactive
ISUFLCGFYQDRGM-UHFFFAOYSA-N--1inactiveinactive
VGSYMGCEDYSPMI-UHFFFAOYSA-N--1inactiveinactive
IGPLDYDCTCCRIM-UHFFFAOYSA-N--1inactiveinactive
SJWYJDDFSFWNTR-UHFFFAOYSA-N--1inactiveinactive
WTXKZWYFQBECHP-UHFFFAOYSA-N--1inactiveinactive
BSBBIWMXRBLRGQ-UHFFFAOYSA-N--1inactiveinactive
GDCBQWYGIXMEOS-UHFFFAOYSA-N--1inactiveinactive
CBBCUNUDUOFOKM-UHFFFAOYSA-N--1inactiveinactive
HEAIGWIZTYAQTC-UHFFFAOYSA-N--1inactiveinactive
AHOUBRCZNHFOSL-YOEHRIQHSA-N--1inactiveinactive
WGESQHUBLPGDDK-UHFFFAOYSA-N--1inactiveinactive
XWJOKKXDMHSILW-UHFFFAOYSA-N--1inactiveinactive
ARSZMAAOVNYKQN-UHFFFAOYSA-N--1inactiveinactive
MSYSXAOSMCNJKL-UHFFFAOYSA-N--1inactiveinactive