Q12852 DLK


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Group: TKL
Family: MLK
PDB Structure Num: 5
FDA approved drugs from DrugBank: Fostamatinib






structureFDA kinase druginchikeykinase profiling data countkinase profiling labelChEMBL data countChEMBL labelvote label
BPNUQXPIQBZCMR-LJQANCHMSA-N1inactive--inactive
WJEOLQLKVOPQFV-UHFFFAOYSA-N1inactive--inactive
MPVGZUGXCQEXTM-UHFFFAOYSA-N1inactive--inactive
CVWXJKQAOSCOAB-UHFFFAOYSA-N1inactive--inactive
RITAVMQDGBJQJZ-UHFFFAOYSA-N1active--active
RAHBGWKEPAQNFF-UHFFFAOYSA-N1inactive--inactive
ODPGGGTTYSGTGO-UHFFFAOYSA-N1active--active
OVPNQJVDAFNBDN-UHFFFAOYSA-N1inactive--inactive
QYZOGCMHVIGURT-UHFFFAOYSA-N1inactive--inactive
XXJWYDDUDKYVKI-UHFFFAOYSA-N1inactive--inactive
CYOHGALHFOKKQC-UHFFFAOYSA-N1inactive--inactive
XQVVPGYIWAGRNI-QFIPXVFZSA-N1inactive--inactive
-FCLPVPNWFDOVKL-DQSJHHFOSA-N1active--active
ULXXDDBFHOBEHA-INIZCTEOSA-N1inactive--inactive
MVCOAUNKQVWQHZ-UHFFFAOYSA-N1inactive--inactive
PSPFQEBFYXJZEV-UHFFFAOYSA-N1inactive--inactive
OUSFTKFNBAZUKL-UHFFFAOYSA-N1inactive--inactive
WCWUXEGQKLTGDX-NSHDSACASA-N1inactive--inactive
UIARLYUEJFELEN-FMLDBKJISA-N1active--active
-KCOYQXZDFIIGCY-CZIZESTLSA-N1active--active
YABJJWZLRMPFSI-UHFFFAOYSA-N1inactive--inactive
OMZCMEYTWSXEPZ-UHFFFAOYSA-N1inactive--inactive
GFMMXOIFOQCCGU-UHFFFAOYSA-N1inactive--inactive
UJLAWZDWDVHWOW-DGCLKSJQSA-N1inactive--inactive
CrizotinibKTEIFNKAUNYNJU-GFCCVEGCSA-N1active--active
DasatinibZBNZXTGUTAYRHI-UHFFFAOYSA-N1inactive--inactive
ErlotinibAAKJLRGGTJKAMG-UHFFFAOYSA-N1inactive--inactive
CXQHYVUVSFXTMY-UHFFFAOYSA-N1active--active
BIIVYFLTOXDAOV-YVEFUNNKSA-N1inactive--inactive
DEZZLWQELQORIU-UHFFFAOYSA-N1inactive--inactive
LHNIIDJUOCFXAP-UHFFFAOYSA-N1inactive--inactive
GefitinibXGALLCVXEZPNRQ-UHFFFAOYSA-N1inactive--inactive
-XWFUWIOJOVXAMS-FXIRQEPWSA-N1inactive--inactive
ZHJGWYRLJUCMRT-QGZVFWFLSA-N1inactive--inactive
KGPGFQWBCSZGEL-ZDUSSCGKSA-N1inactive--inactive
MYQAUKPBNJWPIE-UHFFFAOYSA-N1inactive--inactive
JWNPDZNEKVCWMY-UHFFFAOYSA-N1active--active
ImatinibKTUFNOKKBVMGRW-UHFFFAOYSA-N1inactive--inactive
RuxolitinibHFNKQEVNSGCOJV-OAHLLOKOSA-N1inactive--inactive
-OLESUNNHPSUJLS-UHFFFAOYSA-N1active--active
SHPFDGWALWEPGS-UHFFFAOYSA-N1inactive--inactive
YYLKKYCXAOBSRM-UHFFFAOYSA-N1active--active
LapatinibBCFGMOOMADDAQU-UHFFFAOYSA-N1inactive--inactive
UUADYKVKJIMIPA-UHFFFAOYSA-N1inactive--inactive
ZCBUQCWBWNUWSU-SFHVURJKSA-N1inactive--inactive
ZNOLRTPMNMPLHY-UHFFFAOYSA-N1inactive--inactive
UXXQOJXBIDBUAC-UHFFFAOYSA-N1inactive--inactive
HHFBDROWDBDFBR-UHFFFAOYSA-N1inactive--inactive
NilotinibHHZIURLSWUIHRB-UHFFFAOYSA-N1inactive--inactive
PazopanibCUIHSIWYWATEQL-UHFFFAOYSA-N1inactive--inactive
VAARYSWULJUGST-UHFFFAOYSA-N1inactive--inactive
OYONTEXKYJZFHA-OAQYLSRUSA-N1active--active
TUVCWJQQGGETHL-UHFFFAOYSA-N1inactive--inactive
BMGQWWVMWDBQGC-PZFYLCKJSA-N1inactive--inactive
YZDJQTHVDDOVHR-UHFFFAOYSA-N1inactive--inactive
-MTICIDWIKCANDD-UHFFFAOYSA-N1inactive--inactive
YCOYDOIWSSHVCK-UHFFFAOYSA-N1inactive--inactive
TamatinibNHHQJBCNYHBUSI-UHFFFAOYSA-N1inactive--inactive
JRNJNYBQQYBCLE-UHFFFAOYSA-N1inactive--inactive
CDMGBJANTYXAIV-HHHXNRCGSA-N1inactive--inactive
BCZUAADEACICHN-UHFFFAOYSA-N1inactive--inactive
BosutinibUBPYILGKFZZVDX-UHFFFAOYSA-N1active--active
SorafenibMLDQJTXFUGDVEO-UHFFFAOYSA-N1inactive--inactive
HKSZLNNOFSGOKW-FYTWVXJKSA-N1active--active
CTNPALGJUAXMMC-PMFHANACSA-N1active--active
SunitinibWINHZLLDWRZWRT-ATVHPVEESA-N1active--active
QQWUGDVOUVUTOY-UHFFFAOYSA-N1active--active
UJIAQDJKSXQLIT-UHFFFAOYSA-N1inactive--inactive
JOOXLOJCABQBSG-UHFFFAOYSA-N1inactive--inactive
VandetanibUHTHHESEBZOYNR-UHFFFAOYSA-N1inactive--inactive
GCIKSSRWRFVXBI-UHFFFAOYSA-N1active--active
VEPKQEUBKLEPRA-UHFFFAOYSA-N1inactive--inactive
BOWCRFQTJJGHST-UHFFFAOYSA-N--1inactiveinactive
MVRFKJDYYPKRFL-UHFFFAOYSA-N--1inactiveinactive
FLOSXXAKVKYADW-UHFFFAOYSA-N--1activeactive
ROSFWOBLBMDAEV-UHFFFAOYSA-N--1inactiveinactive
GQHCEFMDGMWZFB-UHFFFAOYSA-N--1activeactive
BLBAMJMJBNCHSZ-UHFFFAOYSA-N--1inactiveinactive
SUZLQCNSEYYNFG-UHFFFAOYSA-N--1inactiveinactive
ZJTFBJWIKGEKQC-UHFFFAOYSA-N--1activeactive
SKVWGAYKWDVXNG-UHFFFAOYSA-N--1activeactive
LXJPOSRRJBJZRJ-UHFFFAOYSA-N--1activeactive
FBTGAWKEJSISFL-UHFFFAOYSA-N--1activeactive
JAXBPMVTQNGQOE-UHFFFAOYSA-N--1activeactive
OTWFDDLIAWFRHM-UHFFFAOYSA-N--1activeactive
HINMBDRVCLOXLD-UHFFFAOYSA-N--1activeactive
XWCUFVJABJEBOS-UHFFFAOYSA-N--1activeactive
OZCJURDLKWBQAU-UHFFFAOYSA-N--1activeactive
KSRDBIJRCOLMNC-UHFFFAOYSA-N--1activeactive
RHFIAUKMKYHHFA-UHFFFAOYSA-N--1activeactive
WNGHVWGFYUFTLS-UHFFFAOYSA-N--1activeactive
DLCJUPPKXMYZCU-UHFFFAOYSA-N--1activeactive
LRIIFYKTGXAZMR-UHFFFAOYSA-N--1activeactive
SYJRRKLEZAGNOV-UHFFFAOYSA-N--1activeactive
LNGNXKRWIDCEAU-UHFFFAOYSA-N--1inactiveinactive
JUWMQAMEXATQIU-UHFFFAOYSA-N--1activeactive
ZWBJERDJEJXJAD-UHFFFAOYSA-N--1activeactive
GMTAOJMPNXLKJI-UHFFFAOYSA-N--1inactiveinactive
YRPUWZXFERSRBH-UHFFFAOYSA-N--1inactiveinactive
KOFKETXAQRCNNS-UHFFFAOYSA-N--1inactiveinactive
BPCISKGSUMOXTI-UHFFFAOYSA-N--1activeactive
HPCAFTNDPHAAGH-UHFFFAOYSA-N--1inactiveinactive
ZBHXJFIKXIBKBY-UHFFFAOYSA-N--1inactiveinactive
ZDBCVOUBHOHGIX-UHFFFAOYSA-N--1inactiveinactive
ZEHBZHZMQSHZFI-UHFFFAOYSA-N--1inactiveinactive