P53671 LIMK2


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Group: TKL
Family: LISK
PDB Structure Num: 2
FDA approved drugs from DrugBank: Fostamatinib






structureFDA kinase druginchikeykinase profiling data countkinase profiling labelChEMBL data countChEMBL labelvote label
BPNUQXPIQBZCMR-LJQANCHMSA-N1inactive--inactive
WJEOLQLKVOPQFV-UHFFFAOYSA-N1inactive--inactive
MPVGZUGXCQEXTM-UHFFFAOYSA-N1inactive--inactive
CVWXJKQAOSCOAB-UHFFFAOYSA-N1inactive--inactive
RITAVMQDGBJQJZ-UHFFFAOYSA-N1inactive--inactive
RAHBGWKEPAQNFF-UHFFFAOYSA-N1inactive--inactive
ODPGGGTTYSGTGO-UHFFFAOYSA-N1active--active
OVPNQJVDAFNBDN-UHFFFAOYSA-N1inactive--inactive
QYZOGCMHVIGURT-UHFFFAOYSA-N1inactive--inactive
XXJWYDDUDKYVKI-UHFFFAOYSA-N1inactive--inactive
CYOHGALHFOKKQC-UHFFFAOYSA-N1inactive--inactive
XQVVPGYIWAGRNI-QFIPXVFZSA-N1inactive--inactive
-FCLPVPNWFDOVKL-DQSJHHFOSA-N1inactive--inactive
ULXXDDBFHOBEHA-INIZCTEOSA-N1inactive--inactive
MVCOAUNKQVWQHZ-UHFFFAOYSA-N1inactive--inactive
PSPFQEBFYXJZEV-UHFFFAOYSA-N1inactive--inactive
OUSFTKFNBAZUKL-UHFFFAOYSA-N1inactive--inactive
WCWUXEGQKLTGDX-NSHDSACASA-N1inactive--inactive
UIARLYUEJFELEN-FMLDBKJISA-N1inactive--inactive
-KCOYQXZDFIIGCY-CZIZESTLSA-N1inactive--inactive
YABJJWZLRMPFSI-UHFFFAOYSA-N1inactive--inactive
OMZCMEYTWSXEPZ-UHFFFAOYSA-N1inactive--inactive
GFMMXOIFOQCCGU-UHFFFAOYSA-N1inactive--inactive
UJLAWZDWDVHWOW-DGCLKSJQSA-N1inactive--inactive
CrizotinibKTEIFNKAUNYNJU-GFCCVEGCSA-N1active--active
DasatinibZBNZXTGUTAYRHI-UHFFFAOYSA-N1active--active
ErlotinibAAKJLRGGTJKAMG-UHFFFAOYSA-N1inactive--inactive
CXQHYVUVSFXTMY-UHFFFAOYSA-N1active--active
BIIVYFLTOXDAOV-YVEFUNNKSA-N1inactive--inactive
DEZZLWQELQORIU-UHFFFAOYSA-N1inactive--inactive
LHNIIDJUOCFXAP-UHFFFAOYSA-N1inactive--inactive
GefitinibXGALLCVXEZPNRQ-UHFFFAOYSA-N1inactive--inactive
-XWFUWIOJOVXAMS-FXIRQEPWSA-N1inactive--inactive
ZHJGWYRLJUCMRT-QGZVFWFLSA-N1inactive--inactive
KGPGFQWBCSZGEL-ZDUSSCGKSA-N1inactive--inactive
MYQAUKPBNJWPIE-UHFFFAOYSA-N1inactive--inactive
JWNPDZNEKVCWMY-UHFFFAOYSA-N1inactive--inactive
ImatinibKTUFNOKKBVMGRW-UHFFFAOYSA-N1inactive--inactive
RuxolitinibHFNKQEVNSGCOJV-OAHLLOKOSA-N1inactive--inactive
-OLESUNNHPSUJLS-UHFFFAOYSA-N1inactive--inactive
SHPFDGWALWEPGS-UHFFFAOYSA-N1active--active
YYLKKYCXAOBSRM-UHFFFAOYSA-N1inactive--inactive
LapatinibBCFGMOOMADDAQU-UHFFFAOYSA-N1inactive--inactive
UUADYKVKJIMIPA-UHFFFAOYSA-N1inactive--inactive
ZCBUQCWBWNUWSU-SFHVURJKSA-N1inactive--inactive
ZNOLRTPMNMPLHY-UHFFFAOYSA-N1inactive--inactive
UXXQOJXBIDBUAC-UHFFFAOYSA-N1inactive--inactive
HHFBDROWDBDFBR-UHFFFAOYSA-N1inactive--inactive
NilotinibHHZIURLSWUIHRB-UHFFFAOYSA-N1inactive--inactive
PazopanibCUIHSIWYWATEQL-UHFFFAOYSA-N1active--active
VAARYSWULJUGST-UHFFFAOYSA-N1active--active
OYONTEXKYJZFHA-OAQYLSRUSA-N1inactive--inactive
TUVCWJQQGGETHL-UHFFFAOYSA-N1inactive--inactive
BMGQWWVMWDBQGC-PZFYLCKJSA-N1inactive--inactive
YZDJQTHVDDOVHR-UHFFFAOYSA-N1active--active
-MTICIDWIKCANDD-UHFFFAOYSA-N1inactive--inactive
YCOYDOIWSSHVCK-UHFFFAOYSA-N1inactive--inactive
TamatinibNHHQJBCNYHBUSI-UHFFFAOYSA-N1active--active
JRNJNYBQQYBCLE-UHFFFAOYSA-N1inactive--inactive
CDMGBJANTYXAIV-HHHXNRCGSA-N1inactive--inactive
BCZUAADEACICHN-UHFFFAOYSA-N1inactive--inactive
BosutinibUBPYILGKFZZVDX-UHFFFAOYSA-N1inactive--inactive
SorafenibMLDQJTXFUGDVEO-UHFFFAOYSA-N1inactive--inactive
HKSZLNNOFSGOKW-FYTWVXJKSA-N1inactive--inactive
CTNPALGJUAXMMC-PMFHANACSA-N1inactive--inactive
SunitinibWINHZLLDWRZWRT-ATVHPVEESA-N1inactive--inactive
QQWUGDVOUVUTOY-UHFFFAOYSA-N1active--active
UJIAQDJKSXQLIT-UHFFFAOYSA-N1inactive--inactive
JOOXLOJCABQBSG-UHFFFAOYSA-N1inactive--inactive
VandetanibUHTHHESEBZOYNR-UHFFFAOYSA-N1inactive--inactive
GCIKSSRWRFVXBI-UHFFFAOYSA-N1active--active
VEPKQEUBKLEPRA-UHFFFAOYSA-N1inactive--inactive
RZCBPADGHYZXSD-ZDUSSCGKSA-N--1activeactive
DHODDWMFDDAHDC-INIZCTEOSA-N--1activeactive
XDNKWMQFUPMOCW-KRWDZBQOSA-N--1activeactive
KXDMWKDZFFHEHC-UHFFFAOYSA-N--1activeactive
FXQYSASDTKPUOS-UHFFFAOYSA-N--1activeactive
YXANFBAJHKQOBF-UHFFFAOYSA-N--1inactiveinactive
SDZJESDWVOOOKS-HNNXBMFYSA-N--1activeactive
SLUWFPJROQKLET-UHFFFAOYSA-N--1activeactive
KKSNLMSTPZRCCK-KRWDZBQOSA-N--1activeactive
MVPARBNSRQJBEM-HNNXBMFYSA-N--2activeactive
KSECQYDNQYAZMQ-AWEZNQCLSA-N--1activeactive
SYMCODQMUIIHQO-UHFFFAOYSA-N--1inactiveinactive
LITGTHZJNKGRSE-CABCVRRESA-N--1activeactive
VHPPTKHCXNGNDC-UHFFFAOYSA-N--1inactiveinactive
GRLGLNJPPWPUSU-OKILXGFUSA-N--1activeactive
JQXGSDPBFXEDBN-LBPRGKRZSA-N--1activeactive
GSNIGRNYQGRXBW-HNNXBMFYSA-N--1activeactive
XTTGFHVGRVSEQJ-AWEZNQCLSA-N--1activeactive
QXOXJENITDQYCG-GOSISDBHSA-N--1activeactive
XMIUKXIQHLXPBO-AWEZNQCLSA-N--1activeactive
BCNLLDVODACBHT-INIZCTEOSA-N--1activeactive
BLMCSSLGKGQBHN-UHFFFAOYSA-N--1activeactive
DCEWGZDEKYCLOP-UHFFFAOYSA-N--1activeactive
CPJGIRFFPLPFGW-CYBMUJFWSA-N--1activeactive
ZZABGZFZUJBLLS-AWEZNQCLSA-N--1activeactive
QRCVBFDDXGCPTD-UHFFFAOYSA-N--1activeactive
LSXPHTSMOQWNKP-SFHVURJKSA-N--1activeactive
CPJGIRFFPLPFGW-ZDUSSCGKSA-N--1activeactive
LLTNWTYFGBIZTB-AWEZNQCLSA-N--1activeactive
SPKWLNDBVFRGKM-INIZCTEOSA-N--2activeactive
ZQWSKCMUBPPXNS-UHFFFAOYSA-N--1activeactive
IQWWRYFXGXTCRB-UHFFFAOYSA-N--1activeactive
YUZYPXOGQFDMIJ-UHFFFAOYSA-N--1inactiveinactive
JMAQIAGPIUIAPQ-UHFFFAOYSA-N--1inactiveinactive
CZFWUZDEOVCKHA-LBPRGKRZSA-N--1activeactive
RFPNUIOUJIEGLY-UHFFFAOYSA-N--1inactiveinactive
KJFJUZUMQQERFW-HNNXBMFYSA-N--1activeactive
XYAAKAODCJCORG-ZDUSSCGKSA-N--1activeactive
RHTZFHQZNIEKPG-AWEZNQCLSA-N--1activeactive
ZYOHQBDYDFWQRU-UHFFFAOYSA-N--1activeactive
SHQFPLWVQBAKMP-KRWDZBQOSA-N--1activeactive
APWWGLHVZKSZOE-UHFFFAOYSA-N--1inactiveinactive
XLVDNAJPINHYSI-UHFFFAOYSA-N--1inactiveinactive
QWETWPHULIMRMN-UHFFFAOYSA-N--1inactiveinactive
SOHUUAAKBLRJIV-UHFFFAOYSA-N--1inactiveinactive
VVKQZMUJMLYYGY-UHFFFAOYSA-N--1activeactive
XCZSICUSGXTGKT-UHFFFAOYSA-N--1activeactive
BOOBTTZFNINJRN-UHFFFAOYSA-N--1inactiveinactive
QPSPUIQBHBHIQQ-UHFFFAOYSA-N--1inactiveinactive
BQIFRQYAMVYLOP-UHFFFAOYSA-N--1inactiveinactive
MVJBIZDRJOFXBG-UHFFFAOYSA-N--1inactiveinactive
RJDOGMOZKFERKX-UHFFFAOYSA-N--1activeactive
BVUPEIDHNYSDAC-UHFFFAOYSA-N--1activeactive
UNMJHZVVYMTJHP-UHFFFAOYSA-N--1activeactive
FFDIPAAUHNHALW-UHFFFAOYSA-N--1activeactive
WTRAMLNUHRBZEC-UHFFFAOYSA-N--1activeactive
RYXLLTGGHCFCFK-UHFFFAOYSA-N--1activeactive
ZEMLGPJIQJHESM-UHFFFAOYSA-N--1activeactive
WUCYRTXFXRZKSV-UHFFFAOYSA-N--2excludeexclude
NSNKKSURBOMEKE-UHFFFAOYSA-N--1activeactive
MTHYJGOTWRWQBV-UHFFFAOYSA-N--1activeactive
VCVUTSJXFBAJEE-UHFFFAOYSA-N--1activeactive
XACSASLXEAYEEO-UHFFFAOYSA-N--1activeactive
IMBPDUMBJKDSPJ-UHFFFAOYSA-N--1activeactive
LAVCNMCLMYEWTG-UHFFFAOYSA-N--1inactiveinactive
UNWYGJWQCPQFQS-UHFFFAOYSA-N--1activeactive
GKMZBTXNOFZJEL-UHFFFAOYSA-N--1activeactive
KSBGCPVPRWKTMY-UHFFFAOYSA-N--1activeactive
TUFSMSWPRKEYRO-UHFFFAOYSA-N--1inactiveinactive
BPIQRPNLTNOFEM-UHFFFAOYSA-N--1activeactive
OUEWYQINKGAXHX-UHFFFAOYSA-N--1inactiveinactive
QTQJYAAVROMTLX-UHFFFAOYSA-N--1inactiveinactive
GSKLEHKWVKSVHN-UHFFFAOYSA-N--1activeactive
QXOLGUWNZPMDNR-UHFFFAOYSA-N--1activeactive
FYTAJCOXVSKAQF-UHFFFAOYSA-N--1activeactive
CFNAVCPPRDKPBH-UHFFFAOYSA-N--1inactiveinactive
CQXHFGYFIHOEFD-UHFFFAOYSA-N--1activeactive
KDSVANHTYAGFHO-UHFFFAOYSA-N--1activeactive
JBNJAADAOPJAQV-UHFFFAOYSA-N--1activeactive
LJBXWGVECYNLLM-UHFFFAOYSA-N--1activeactive
BRWPJGJHJUEZTD-UHFFFAOYSA-N--1inactiveinactive
RBJHDGSFXKINKF-UHFFFAOYSA-N--1inactiveinactive
SRGYPZUCDIFDTE-UHFFFAOYSA-N--1activeactive
WGWSXJXDEVNYRU-KRWDZBQOSA-N--1activeactive
WGWSXJXDEVNYRU-QGZVFWFLSA-N--1activeactive
HSFGCMJKYHQRQQ-UHFFFAOYSA-N--1activeactive
YHLIDLWSAGDBKL-UHFFFAOYSA-N--1activeactive
CJLCYOXEAFXEGB-UHFFFAOYSA-N--1activeactive
KRFJFFSNMVTINU-UHFFFAOYSA-N--1activeactive
GBLCVNINRYFFJV-UHFFFAOYSA-N--1inactiveinactive
CUFGKGXAWMMGOM-UHFFFAOYSA-N--1inactiveinactive
WGKJGIIWRDYVJF-UHFFFAOYSA-N--1inactiveinactive
WJXSOMFZMISVNK-UHFFFAOYSA-N--1activeactive
DMUATXJZGOPROG-UHFFFAOYSA-N--1activeactive
OQHGYDFCYFPABG-UHFFFAOYSA-N--1activeactive
OGBRRCBVEXWMQF-HOTGVXAUSA-N--1activeactive
VQYKTJZUIGNLQB-AWEZNQCLSA-N--1activeactive
AFUATWMQZAOHQC-AWEZNQCLSA-N--1activeactive
MCTDUQPDBRONSD-HNNXBMFYSA-N--1inactiveinactive
OGBRRCBVEXWMQF-JKSUJKDBSA-N--1activeactive
PIHWOKGTWVJGMD-UHFFFAOYSA-N--1activeactive
JBNLRXGSIJBDMC-UHFFFAOYSA-N--1activeactive
SPFGMXTXKGFEMU-UHFFFAOYSA-N--1activeactive
VCYAIYACPTUHNX-YJBOKZPZSA-N--1activeactive
VCYAIYACPTUHNX-QAPCUYQASA-N--1activeactive
XIMVZDIPXNUARA-UHFFFAOYSA-N--1activeactive
UFFGIZGDBJFJBO-UHFFFAOYSA-N--1activeactive
BYJACWIXRRGPAO-UHFFFAOYSA-N--1activeactive
NDUMDYQFHRPXEL-UHFFFAOYSA-N--1activeactive
JFKVNPYSINXUEZ-UHFFFAOYSA-N--1activeactive
HMZQIUFZSWXUEG-UHFFFAOYSA-N--1activeactive
PNEHHQFPYPNPDP-UHFFFAOYSA-N--1activeactive
PAOJADRMYANSIV-UHFFFAOYSA-N--1activeactive
TVCSBVZJGSWVFO-UHFFFAOYSA-N--1activeactive
PWPNYABQEOGNNC-UHFFFAOYSA-N--4activeactive
IVUGBSGLHRJSSP-UHFFFAOYSA-N--1activeactive
UEWMYTIDOPPABK-UHFFFAOYSA-N--1activeactive
CWTWMAPTTBKMQQ-UHFFFAOYSA-N--1activeactive
XKNKSXHITXPWPU-UHFFFAOYSA-N--1activeactive
NXEVMWHFSSQBGY-UHFFFAOYSA-N--1activeactive
OYYKGCKVVURSQO-UHFFFAOYSA-N--1activeactive
IWAGHIAOERSNDT-UHFFFAOYSA-N--1activeactive
UXIGAYGUDGBPOS-UHFFFAOYSA-N--1activeactive
LBMPEUDJKWLTOC-UHFFFAOYSA-N--1activeactive
DEEIBAOTOOOOIG-UHFFFAOYSA-N--1activeactive
SNUDLLACDRMNDB-UHFFFAOYSA-N--1activeactive
PQVIVJUHYDLYRA-UHFFFAOYSA-N--1activeactive
UMDIEKHQTFPTBH-UHFFFAOYSA-N--1activeactive
ZCVGUOHAEJQFRY-UHFFFAOYSA-N--1activeactive
SOGKOUURZPAQPP-UHFFFAOYSA-N--1activeactive
VUTDBZFATUOXQL-UHFFFAOYSA-N--1activeactive
UMQNZSBIZJEBSD-UHFFFAOYSA-N--1activeactive
SGTQAYSNMALFSG-UHFFFAOYSA-N--1inactiveinactive
NEAFSODAYAUEGX-UHFFFAOYSA-N--1activeactive
WLWQRWYWHSJFFX-UHFFFAOYSA-N--1inactiveinactive
WRWOUEHJMWGBKY-UHFFFAOYSA-N--1activeactive
UVPTTYAFVRRFMP-UHFFFAOYSA-N--1activeactive
HXOGWFKVKCOUQG-UHFFFAOYSA-N--1activeactive
SXLCBECQMMDJSN-UHFFFAOYSA-N--1activeactive
RKAKGPYRNHXPDK-UHFFFAOYSA-N--1activeactive
PRNCXCNGOBQGGJ-UHFFFAOYSA-N--1activeactive
SEZBMVMOFIKXMB-UHFFFAOYSA-N--1activeactive
YTTBQAOPTOOIMN-UHFFFAOYSA-N--1activeactive
UIQNMIISGRIHIY-UHFFFAOYSA-N--1activeactive
XJGIAMVUFKIMTL-UHFFFAOYSA-N--1activeactive
UYPFVVTZNUIZNF-UHFFFAOYSA-N--1activeactive
HNIKKHODIZOTRI-UHFFFAOYSA-N--1activeactive
LKTNBFFMIICAFJ-UHFFFAOYSA-N--1activeactive
FQQRNYQTYDWOME-UHFFFAOYSA-N--1activeactive
PUQNSBRQHFAIKU-UHFFFAOYSA-N--1activeactive
AXYJYZXEBHIVPM-UHFFFAOYSA-N--1activeactive
XSRLKVPNDGGLCH-UHFFFAOYSA-N--1activeactive
HZRAQVDLSJCYGZ-UHFFFAOYSA-N--1activeactive
IQXFPGQRIPGJOH-UHFFFAOYSA-N--1activeactive
DGTREGXOFARCHY-UHFFFAOYSA-N--1activeactive
IIALFTYNTCYIML-UHFFFAOYSA-N--1activeactive
VUFXATHBRBCDNJ-UHFFFAOYSA-N--1activeactive
SYBULHVKMWRDDE-UHFFFAOYSA-N--1activeactive
GMFFUPZRKJLVKX-UHFFFAOYSA-N--1activeactive
NSLDDYUWZNXJFD-UHFFFAOYSA-N--1activeactive
UBHGJJDCAJQFBE-UHFFFAOYSA-N--1activeactive
PPPVIZUATMDNBM-UHFFFAOYSA-N--1activeactive
OIUPPGARAHMBQU-UHFFFAOYSA-N--1inactiveinactive
ZMFPALFDOPHLTO-UHFFFAOYSA-N--1activeactive
MDGXORCOVUOYBS-UHFFFAOYSA-N--1activeactive
DTVFQHOXYKFHFO-UHFFFAOYSA-N--1activeactive
YDQAHDMMKNYRCW-UHFFFAOYSA-N--1activeactive
GNHKGIMYNFCSPS-UHFFFAOYSA-N--1activeactive
BOOROEDYUBEHOH-UHFFFAOYSA-N--1activeactive
UJCLBWBWMXJXCM-UHFFFAOYSA-N--1activeactive
FKBLDGUTNDFWSK-UHFFFAOYSA-N--1activeactive
NSIGCPZYQUUXPW-UHFFFAOYSA-N--1activeactive
PERUSYKRJXRDST-UHFFFAOYSA-N--1activeactive
XGIDKOVZVAXJDJ-UHFFFAOYSA-N--1activeactive
AYRNUIDFFNFELA-UHFFFAOYSA-N--1activeactive
AJUWMHFAMFBWMN-UHFFFAOYSA-N--1activeactive
GXYLCVUZDYCVMB-UHFFFAOYSA-N--1activeactive
LPHIVAHXWKFNCZ-UHFFFAOYSA-N--1activeactive
YZEBEKHXMANRDT-UHFFFAOYSA-N--1activeactive
AGNADDDFSLVLRJ-UHFFFAOYSA-N--1activeactive
YCGVEGHRSHKVFO-UHFFFAOYSA-N--1activeactive
IAJWNLCFVHFJCR-UHFFFAOYSA-N--1activeactive
XEVVSMANPWGFNP-UHFFFAOYSA-N--1activeactive
KFGVCKLINBSYTQ-UHFFFAOYSA-N--1activeactive
PUQFAZBAPCKZKN-UHFFFAOYSA-N--1activeactive
DRRUMZPUGPNKLX-UHFFFAOYSA-N--1activeactive
QSSKKSGGXPWDPC-UHFFFAOYSA-N--1activeactive
HFBCKXXEXNDPEJ-UHFFFAOYSA-N--1activeactive
PAOKFNVXQHEMAT-UHFFFAOYSA-N--1activeactive
IWTYIWZMOWXLSU-UHFFFAOYSA-N--1activeactive
ZQYHTGNJVMVCGP-UHFFFAOYSA-N--1activeactive
GBGCCWYYTLPKCJ-UHFFFAOYSA-N--1activeactive
QQXFHZXFOXVCFA-UHFFFAOYSA-N--1activeactive
GIOJSCUMPYUYQD-UHFFFAOYSA-N--1activeactive
DSWZDIKQFDCBGM-UHFFFAOYSA-N--1activeactive
HBVOISKDRNXOAW-LBPRGKRZSA-N--1inactiveinactive
HGEMEBXHIFACIK-UHFFFAOYSA-N--1inactiveinactive
OBCMZHZSMUJYNB-UHFFFAOYSA-N--1inactiveinactive
NWNKAJGVSLONKZ-UHFFFAOYSA-N--1inactiveinactive
UBFBUNVMPQVTNN-UHFFFAOYSA-N--1inactiveinactive
IADPZBONWBWIJL-UHFFFAOYSA-N--1inactiveinactive
AVMSOILXAYKHOD-UHFFFAOYSA-N--1inactiveinactive
FJPRCIGXYORUGN-UHFFFAOYSA-N--1inactiveinactive
XMQJTVUUGGWRNA-UHFFFAOYSA-N--1inactiveinactive
AUHOGGLIKKHJMN-UHFFFAOYSA-N--1inactiveinactive
IDQFWWKUZNCJCP-UHFFFAOYSA-N--1inactiveinactive
DFNYHODYPRNKAK-UHFFFAOYSA-N--1inactiveinactive
ZEHBZHZMQSHZFI-UHFFFAOYSA-N--1inactiveinactive