P22612 PKACg


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Group: AGC
Family: PKA
PDB Structure Num: 0






structureFDA kinase druginchikeykinase profiling data countkinase profiling labelChEMBL data countChEMBL labelvote label
NJTUORMLOPXPBY-UHFFFAOYSA-N1inactive--inactive
ODZGYELAMAOARP-UHFFFAOYSA-N1inactive--inactive
ZUDPNBZMAJGYTE-UHFFFAOYSA-N1inactive--inactive
AVLYNJZZQYEFEA-UHFFFAOYSA-N1inactive--inactive
KQMPRSZTUSSXND-UHFFFAOYSA-N1inactive--inactive
ZXVUBPLDUMSDOE-UHFFFAOYSA-N1inactive--inactive
KOZFSFOOLUUIGY-IYYJOCMQSA-N1active--active
QQUXFYAWXPMDOE-UHFFFAOYSA-N1inactive--inactive
-BLLBARDQJSOSJD-PGUFJCEWSA-N1inactive--inactive
LLLQTDSSHZREGW-UHFFFAOYSA-N1inactive--inactive
FMETVQKSDIOGPX-UHFFFAOYSA-N1inactive--inactive
NGAGMBNBKCDCDJ-UHFFFAOYSA-N1inactive--inactive
-NHBMKTBZZSJUGA-HKRCYGBASA-N1inactive--inactive
GYQSWJNGTWVFOL-UHFFFAOYSA-N1inactive--inactive
JLOXTZFYJNCPIS-UHFFFAOYSA-N1inactive--inactive
FPYJSJDOHRDAMT-UHFFFAOYSA-N1inactive--inactive
UQPMANVRZYYQMD-UHFFFAOYSA-N1inactive--inactive
ODYAQBDIXCVKAE-UHFFFAOYSA-N1inactive--inactive
IBAKVEUZKHOWNG-UHFFFAOYSA-N1inactive--inactive
VXPWQNBKEIVYIS-OAHLLOKOSA-N1inactive--inactive
DZFBYHUKZSRPHU-UHFFFAOYSA-N1inactive--inactive
QFWCYNPOPKQOKV-UHFFFAOYSA-N1inactive--inactive
BGIYKDUASORTBB-UHFFFAOYSA-N1inactive--inactive
KFHMLBXBRCITHF-UHFFFAOYSA-N1inactive--inactive
WUPUZEMRHDROEO-UHFFFAOYSA-N1inactive--inactive
CZDUJGOCEPWCNA-UHFFFAOYSA-N1inactive--inactive
INTPTKHSGKBHHW-UHFFFAOYSA-N1inactive--inactive
ZDNURMVOKAERHZ-UHFFFAOYSA-N1inactive--inactive
PEPCXHNLEXQQSE-UHFFFAOYSA-N1inactive--inactive
-DGCXNBUJPWPMJJ-UHFFFAOYSA-N1inactive--inactive
VFBGXTUGODTSPK-UHFFFAOYSA-N1inactive--inactive
ZJFMARHFPUZEKI-UHFFFAOYSA-N1inactive--inactive
TUVCWJQQGGETHL-UHFFFAOYSA-N1inactive--inactive
SQWZFLMPDUSYGV-UHFFFAOYSA-N1inactive--inactive
SRLVNYDXMUGOFI-UHFFFAOYSA-N1inactive--inactive
GDQXJQSQYMMKRA-UHFFFAOYSA-N1inactive--inactive
BMGQWWVMWDBQGC-PZFYLCKJSA-N1inactive--inactive
RONQPWQYDRPRGG-UHFFFAOYSA-N1inactive--inactive
KIWODJBCHRADND-UHFFFAOYSA-N1inactive--inactive
PMXCMJLOPOFPBT-OAHLLOKOSA-N1inactive--inactive
-QFJCIRLUMZQUOT-JRLVRMFHSA-N1inactive--inactive
LLJRXVHJOJRCSM-UHFFFAOYSA-N1inactive--inactive
CMKMGFAUKPAOMG-AWEZNQCLSA-N1inactive--inactive
FXGHOAZJQNLNFD-KRWDZBQOSA-N1inactive--inactive
-XFXDYDZBKXMGBX-HOTGVXAUSA-N1inactive--inactive
-NJNKPVPFGLGHPA-UHFFFAOYSA-N1inactive--inactive
CDMGBJANTYXAIV-MHZLTWQESA-N1inactive--inactive
VSPFURGQAYMVAN-UHFFFAOYSA-N1inactive--inactive
OTPNDVKVEAIXTI-IYBDPMFKSA-N1active--active
BHWCZLOXTLWZAQ-UHFFFAOYSA-N1inactive--inactive
YOELZIQOLWZLQC-UHFFFAOYSA-N1inactive--inactive
ZFGXZJKLOFCECI-UHFFFAOYSA-N1inactive--inactive
DMWVGXGXHPOEPT-UHFFFAOYSA-N1inactive--inactive
HKSZLNNOFSGOKW-HMWZOHBLSA-N1active--active
WNRSTFUVBWNELX-UHFFFAOYSA-N1inactive--inactive
LOGJQOUIVKBFGH-UHFFFAOYSA-N1inactive--inactive
QNUKRWAIZMBVCU-UHFFFAOYSA-N1inactive--inactive
XPLJEFSRINKZLC-UHFFFAOYSA-N1inactive--inactive
MLKHXLFEYOOYEY-UHFFFAOYSA-N1inactive--inactive
LCACSMNPIITJGG-UHFFFAOYSA-N1inactive--inactive
KFLWBZPSJQPRDD-UHFFFAOYSA-N1inactive--inactive
NMEUKWOOQOHUNA-UHFFFAOYSA-N1inactive--inactive
IBCXZJCWDGCXQT-UHFFFAOYSA-N1inactive--inactive
BTUOOXPZOVNPMF-UHFFFAOYSA-N1inactive--inactive
UOHFCPXBKJPCAD-UHFFFAOYSA-N1inactive--inactive
TUCIOBMMDDOEMM-UHFFFAOYSA-N1inactive--inactive
DXVJRTIPBNBLLB-UHFFFAOYSA-N1inactive--inactive
FQNCLVJEQCJWSU-UHFFFAOYSA-N1inactive--inactive
QNOXYUNHIGOWNY-UHFFFAOYSA-N1inactive--inactive
GFNNBHLJANVSQV-UHFFFAOYSA-N1inactive--inactive
PMUJUSJUVIXDQC-UHFFFAOYSA-N1inactive--inactive
GGPZCOONYBPZEW-UHFFFAOYSA-N1inactive--inactive
-YUWFTONEHHSMEI-CZUORRHYSA-N1inactive--inactive
RFHPWPWVGFSLOP-UHFFFAOYSA-N1inactive--inactive
WUWDLXZGHZSWQZ-UHFFFAOYSA-N1inactive--inactive
HBWLNACPIFKNIP-UHFFFAOYSA-N1inactive--inactive
-QDLHCMPXEPAAMD-BLNDMVMCSA-N1inactive--inactive
-BLQHLDXMMWHXIT-YSZXOBSOSA-N1inactive--inactive
-AXPBLFXFGVEGKU-UHFFFAOYSA-N1inactive--inactive
DasatinibZBNZXTGUTAYRHI-UHFFFAOYSA-N1inactive--inactive
PIQCTGMSNWUMAF-UHFFFAOYSA-N1inactive--inactive
ErlotinibAAKJLRGGTJKAMG-UHFFFAOYSA-N1inactive--inactive
GefitinibXGALLCVXEZPNRQ-UHFFFAOYSA-N1inactive--inactive
ImatinibKTUFNOKKBVMGRW-UHFFFAOYSA-N1inactive--inactive
LapatinibBCFGMOOMADDAQU-UHFFFAOYSA-N1inactive--inactive
WJEOLQLKVOPQFV-UHFFFAOYSA-N1inactive--inactive
ZTFBIUXIQYRUNT-MDWZMJQESA-N1inactive--inactive
NilotinibHHZIURLSWUIHRB-UHFFFAOYSA-N1inactive--inactive
PazopanibCUIHSIWYWATEQL-UHFFFAOYSA-N1inactive--inactive
BTIHMVBBUGXLCJ-OAHLLOKOSA-N1inactive--inactive
SorafenibMLDQJTXFUGDVEO-UHFFFAOYSA-N1inactive--inactive
SunitinibWINHZLLDWRZWRT-ATVHPVEESA-N1inactive--inactive
UXXQOJXBIDBUAC-UHFFFAOYSA-N1inactive--inactive
UJLAWZDWDVHWOW-AAEUAGOBSA-N1inactive--inactive
GCIKSSRWRFVXBI-UHFFFAOYSA-N1inactive--inactive
VandetanibUHTHHESEBZOYNR-UHFFFAOYSA-N1inactive--inactive
YCOYDOIWSSHVCK-UHFFFAOYSA-N1inactive--inactive
FYSRKRZDBHOFAY-UHFFFAOYSA-N1inactive--inactive
ZEHBZHZMQSHZFI-UHFFFAOYSA-N--1inactiveinactive