P19525 PKR


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Group: Other
Family: PEK
PDB Structure Num: 2
FDA approved drugs from DrugBank: Fostamatinib






structureFDA kinase druginchikeykinase profiling data countkinase profiling labelChEMBL data countChEMBL labelvote label
BPNUQXPIQBZCMR-LJQANCHMSA-N1active--active
WJEOLQLKVOPQFV-UHFFFAOYSA-N1inactive--inactive
MPVGZUGXCQEXTM-UHFFFAOYSA-N1inactive--inactive
CVWXJKQAOSCOAB-UHFFFAOYSA-N1inactive--inactive
RITAVMQDGBJQJZ-UHFFFAOYSA-N1inactive--inactive
RAHBGWKEPAQNFF-UHFFFAOYSA-N1inactive--inactive
ODPGGGTTYSGTGO-UHFFFAOYSA-N1active--active
OVPNQJVDAFNBDN-UHFFFAOYSA-N1inactive--inactive
QYZOGCMHVIGURT-UHFFFAOYSA-N1inactive--inactive
XXJWYDDUDKYVKI-UHFFFAOYSA-N1inactive--inactive
CYOHGALHFOKKQC-UHFFFAOYSA-N1inactive--inactive
XQVVPGYIWAGRNI-QFIPXVFZSA-N1active--active
-FCLPVPNWFDOVKL-DQSJHHFOSA-N1inactive--inactive
ULXXDDBFHOBEHA-INIZCTEOSA-N1inactive--inactive
MVCOAUNKQVWQHZ-UHFFFAOYSA-N1inactive--inactive
PSPFQEBFYXJZEV-UHFFFAOYSA-N1inactive--inactive
OUSFTKFNBAZUKL-UHFFFAOYSA-N1inactive--inactive
WCWUXEGQKLTGDX-NSHDSACASA-N1inactive--inactive
UIARLYUEJFELEN-FMLDBKJISA-N1active--active
-KCOYQXZDFIIGCY-CZIZESTLSA-N1active--active
YABJJWZLRMPFSI-UHFFFAOYSA-N1active--active
OMZCMEYTWSXEPZ-UHFFFAOYSA-N1inactive--inactive
GFMMXOIFOQCCGU-UHFFFAOYSA-N1inactive--inactive
UJLAWZDWDVHWOW-DGCLKSJQSA-N1inactive--inactive
CrizotinibKTEIFNKAUNYNJU-GFCCVEGCSA-N1active--active
DasatinibZBNZXTGUTAYRHI-UHFFFAOYSA-N1inactive--inactive
ErlotinibAAKJLRGGTJKAMG-UHFFFAOYSA-N1active--active
CXQHYVUVSFXTMY-UHFFFAOYSA-N1inactive--inactive
BIIVYFLTOXDAOV-YVEFUNNKSA-N1inactive--inactive
DEZZLWQELQORIU-UHFFFAOYSA-N1inactive--inactive
LHNIIDJUOCFXAP-UHFFFAOYSA-N1inactive--inactive
GefitinibXGALLCVXEZPNRQ-UHFFFAOYSA-N1inactive--inactive
-XWFUWIOJOVXAMS-FXIRQEPWSA-N1inactive--inactive
ZHJGWYRLJUCMRT-QGZVFWFLSA-N1inactive--inactive
KGPGFQWBCSZGEL-ZDUSSCGKSA-N1active--active
MYQAUKPBNJWPIE-UHFFFAOYSA-N1inactive--inactive
JWNPDZNEKVCWMY-UHFFFAOYSA-N1inactive--inactive
ImatinibKTUFNOKKBVMGRW-UHFFFAOYSA-N1inactive--inactive
RuxolitinibHFNKQEVNSGCOJV-OAHLLOKOSA-N1inactive--inactive
-OLESUNNHPSUJLS-UHFFFAOYSA-N1inactive--inactive
SHPFDGWALWEPGS-UHFFFAOYSA-N1inactive--inactive
YYLKKYCXAOBSRM-UHFFFAOYSA-N1inactive--inactive
LapatinibBCFGMOOMADDAQU-UHFFFAOYSA-N1inactive--inactive
UUADYKVKJIMIPA-UHFFFAOYSA-N1inactive--inactive
ZCBUQCWBWNUWSU-SFHVURJKSA-N1inactive--inactive
ZNOLRTPMNMPLHY-UHFFFAOYSA-N1inactive--inactive
UXXQOJXBIDBUAC-UHFFFAOYSA-N1inactive--inactive
HHFBDROWDBDFBR-UHFFFAOYSA-N1inactive--inactive
NilotinibHHZIURLSWUIHRB-UHFFFAOYSA-N1inactive--inactive
PazopanibCUIHSIWYWATEQL-UHFFFAOYSA-N1active--active
VAARYSWULJUGST-UHFFFAOYSA-N1inactive--inactive
OYONTEXKYJZFHA-OAQYLSRUSA-N1inactive--inactive
TUVCWJQQGGETHL-UHFFFAOYSA-N1inactive--inactive
BMGQWWVMWDBQGC-PZFYLCKJSA-N1inactive--inactive
YZDJQTHVDDOVHR-UHFFFAOYSA-N1inactive--inactive
-MTICIDWIKCANDD-UHFFFAOYSA-N1active--active
YCOYDOIWSSHVCK-UHFFFAOYSA-N1inactive--inactive
TamatinibNHHQJBCNYHBUSI-UHFFFAOYSA-N1active--active
JRNJNYBQQYBCLE-UHFFFAOYSA-N1inactive--inactive
CDMGBJANTYXAIV-HHHXNRCGSA-N1inactive--inactive
BCZUAADEACICHN-UHFFFAOYSA-N1inactive--inactive
BosutinibUBPYILGKFZZVDX-UHFFFAOYSA-N1inactive--inactive
SorafenibMLDQJTXFUGDVEO-UHFFFAOYSA-N1inactive--inactive
HKSZLNNOFSGOKW-FYTWVXJKSA-N1active--active
CTNPALGJUAXMMC-PMFHANACSA-N1active--active
SunitinibWINHZLLDWRZWRT-ATVHPVEESA-N1active--active
QQWUGDVOUVUTOY-UHFFFAOYSA-N1inactive--inactive
UJIAQDJKSXQLIT-UHFFFAOYSA-N1inactive--inactive
JOOXLOJCABQBSG-UHFFFAOYSA-N1active--active
VandetanibUHTHHESEBZOYNR-UHFFFAOYSA-N1inactive--inactive
GCIKSSRWRFVXBI-UHFFFAOYSA-N1inactive--inactive
VEPKQEUBKLEPRA-UHFFFAOYSA-N1inactive--inactive
UQPMANVRZYYQMD-UHFFFAOYSA-N--1inactiveinactive
PDVPLITVGXYXQU-KMKOMSMNSA-N--1inactiveinactive
KRIUNPBAQZGFQA-UHFFFAOYSA-N--1inactiveinactive
GNMXUYVFIVLAKI-UHFFFAOYSA-N--1inactiveinactive
ODZGYELAMAOARP-UHFFFAOYSA-N--1inactiveinactive
UUGQYFCRDPAFOP-UHFFFAOYSA-N--1inactiveinactive
LGJQFSLZOOSXTP-UHFFFAOYSA-N--1inactiveinactive
PUXMBOXMRGPILZ-ONNFQVAWSA-N--1inactiveinactive
UAWHUQSICLSVSY-UHFFFAOYSA-N--1inactiveinactive
KSHCLQFURMFDBK-ZROIWOOFSA-N--1inactiveinactive
HUTBIXFQVWPMKE-UHFFFAOYSA-N--1inactiveinactive
QXBNZWFQOKPAKZ-UHFFFAOYSA-N--1inactiveinactive
KDXIEQMFERTUAI-UHFFFAOYSA-N--1inactiveinactive
MRNZRCFFJZCLOS-UHFFFAOYSA-N--1inactiveinactive
IQMMQBXFNFNXIC-UHFFFAOYSA-N--1inactiveinactive
JOVQZEWRPNCLSA-UHFFFAOYSA-N--1inactiveinactive
FVHUOYBIHLPABI-UHFFFAOYSA-N--1inactiveinactive
BWTONTRMGUMYCX-UHFFFAOYSA-N--1inactiveinactive
FZKFDCYCUKXFBX-UHFFFAOYSA-N--1inactiveinactive
KQUMSCLXYMDAOX-UVTDQMKNSA-N--1inactiveinactive
NMYWWVYRHFAXHI-UHFFFAOYSA-N--1inactiveinactive
GZJNSLMEYSKTPA-UHFFFAOYSA-N--1inactiveinactive
MZDDMOLLGAAVBD-UHFFFAOYSA-N--1inactiveinactive
WGKPNAVGGMGMTL-UHFFFAOYSA-N--1inactiveinactive
IDAWNFCAFDXMER-UHFFFAOYSA-N--1inactiveinactive
ZZFSPQUVXYVZBC-UHFFFAOYSA-N--1inactiveinactive
ONQZNKLIEZTNIM-UHFFFAOYSA-N--1inactiveinactive
GDABVIQLKTYCHW-UHFFFAOYSA-N--1inactiveinactive
NSDAFAJEQZDUKI-UHFFFAOYSA-N--1inactiveinactive
BCTMUESPJWRRDU-UHFFFAOYSA-N--1inactiveinactive
GUBLLHZACKGVEX-UHFFFAOYSA-N--1activeactive
WSJZCTDJZGZIAP-UHFFFAOYSA-N--1inactiveinactive
XHEQSRJCJTWWAH-UHFFFAOYSA-N--1inactiveinactive
IYCHUTRJMZNBCE-UHFFFAOYSA-N--1inactiveinactive
BQLQSBPWPRNBFU-UHFFFAOYSA-N--1activeactive
BOFVTRSIQAXJSC-UHFFFAOYSA-N--1inactiveinactive
LTJDXJWAQOFQTN-UHFFFAOYSA-N--1inactiveinactive
HHIOEAVLBGCWLW-UHFFFAOYSA-N--1inactiveinactive
WDDGPIPVHUVNNS-UHFFFAOYSA-N--1inactiveinactive
AIHCHKBEOSNNLJ-UHFFFAOYSA-N--1inactiveinactive
NONAINIKZPCPPP-UHFFFAOYSA-N--1inactiveinactive
MHFAEQWEFZACHX-UHFFFAOYSA-N--1activeactive
XTWJVEUGFKGHSO-UHFFFAOYSA-N--1inactiveinactive
NIARUGPUHUTYPQ-UHFFFAOYSA-N--1inactiveinactive
UICHPPPBILRQKP-UHFFFAOYSA-N--1inactiveinactive
NJHWAIFJPXUVQO-UHFFFAOYSA-N--1activeactive
NTXPFFQYJAPSSK-UHFFFAOYSA-N--1inactiveinactive
WJZHVBZSCOLDKV-BJMVGYQFSA-N--1inactiveinactive
NMEUKWOOQOHUNA-UHFFFAOYSA-N--1activeactive
SAYGKHKXGCPTLX-UHFFFAOYSA-N--1activeactive
QNUKRWAIZMBVCU-WCIBSUBMSA-N--1inactiveinactive
DWHVZCLBMTZRQM-UHFFFAOYSA-N--1inactiveinactive
ARIOBGGRZJITQX-UHFFFAOYSA-N--1inactiveinactive
SVJQCVOKYJWUBC-OWOJBTEDSA-N--1inactiveinactive
XZEFMZCNXDQXOZ-UHFFFAOYSA-N--1inactiveinactive
JYCUVOXSZBECAY-UHFFFAOYSA-N--1inactiveinactive
UTBSBSOBZHXMHI-LSDHHAIUSA-N--1inactiveinactive
JBOXDNIWQACYPW-UHFFFAOYSA-N--1inactiveinactive
RDTDWGQDFJPTPD-UHFFFAOYSA-N--1inactiveinactive
WJZHVBZSCOLDKV-YHYXMXQVSA-N--1inactiveinactive
VPVLEBIVXZSOMQ-UHFFFAOYSA-N--1inactiveinactive
DDLZLOKCJHBUHD-WAVHTBQISA-N--1inactiveinactive
XHBVYDAKJHETMP-UHFFFAOYSA-N--1inactiveinactive
NMFKDDRQSNVETB-UHFFFAOYSA-N--1inactiveinactive
PRWSIEBRGXYXAJ-UHFFFAOYSA-N--1inactiveinactive
QAEKSWBVYBVLNO-UHFFFAOYSA-N--1activeactive
HFOKVVVCWLIUBP-UHFFFAOYSA-N--1activeactive
PVNWAPAWLNSQHB-UHFFFAOYSA-N--1inactiveinactive
MYKOWOGZBMOVBJ-UHFFFAOYSA-N--1activeactive
FQCPPVRJPILDIK-UHFFFAOYSA-N--1activeactive
RKUMZEVCWKZXFV-LCLDVOFVSA-N--1activeactive
AVLYNJZZQYEFEA-XDJHFCHBSA-N--1activeactive
WXUJAQBSBZLVEV-UHFFFAOYSA-N--1activeactive
KOZFSFOOLUUIGY-IYYJOCMQSA-N--1activeactive
AJSVUPMRZUQVSP-UHFFFAOYSA-N--1inactiveinactive
UCLNOBIGZZFHPP-UHFFFAOYSA-N--1inactiveinactive
ONUYJQFXGBVWOF-UHFFFAOYSA-N--1inactiveinactive
ZEDPEYMNHKLBHO-UHFFFAOYSA-N--1inactiveinactive
RESGOFFFUMERHK-UHFFFAOYSA-N--1inactiveinactive
DREKZLFTJPAMIG-UHFFFAOYSA-N--1inactiveinactive
ZPHRLKSOOXFGCC-UHFFFAOYSA-N--1inactiveinactive
SFTXEEPNVPAHDL-UHFFFAOYSA-N--1inactiveinactive
BZRCPNHODFSVAV-UHFFFAOYSA-N--1inactiveinactive
VILDFORHSQQFIZ-UHFFFAOYSA-N--1inactiveinactive
NYVUSSXLPQHLMH-UHFFFAOYSA-N--1inactiveinactive
KMNCFOUKJYOZIF-KRWDZBQOSA-N--1inactiveinactive