O94768 DRAK2


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Group: CAMK
Family: DAPK
PDB Structure Num: 3
FDA approved drugs from DrugBank: Fostamatinib






structureFDA kinase druginchikeykinase profiling data countkinase profiling labelChEMBL data countChEMBL labelvote label
BPNUQXPIQBZCMR-LJQANCHMSA-N1inactive--inactive
WJEOLQLKVOPQFV-UHFFFAOYSA-N1inactive--inactive
MPVGZUGXCQEXTM-UHFFFAOYSA-N1inactive--inactive
CVWXJKQAOSCOAB-UHFFFAOYSA-N1inactive--inactive
RITAVMQDGBJQJZ-UHFFFAOYSA-N1inactive--inactive
RAHBGWKEPAQNFF-UHFFFAOYSA-N1inactive--inactive
ODPGGGTTYSGTGO-UHFFFAOYSA-N1inactive--inactive
OVPNQJVDAFNBDN-UHFFFAOYSA-N1inactive--inactive
QYZOGCMHVIGURT-UHFFFAOYSA-N1inactive--inactive
XXJWYDDUDKYVKI-UHFFFAOYSA-N1inactive--inactive
CYOHGALHFOKKQC-UHFFFAOYSA-N1inactive--inactive
XQVVPGYIWAGRNI-QFIPXVFZSA-N1inactive--inactive
-FCLPVPNWFDOVKL-DQSJHHFOSA-N1active--active
ULXXDDBFHOBEHA-INIZCTEOSA-N1inactive--inactive
MVCOAUNKQVWQHZ-UHFFFAOYSA-N1inactive--inactive
PSPFQEBFYXJZEV-UHFFFAOYSA-N1inactive--inactive
OUSFTKFNBAZUKL-UHFFFAOYSA-N1inactive--inactive
WCWUXEGQKLTGDX-NSHDSACASA-N1inactive--inactive
UIARLYUEJFELEN-FMLDBKJISA-N1active--active
-KCOYQXZDFIIGCY-CZIZESTLSA-N1active--active
YABJJWZLRMPFSI-UHFFFAOYSA-N1inactive--inactive
OMZCMEYTWSXEPZ-UHFFFAOYSA-N1inactive--inactive
GFMMXOIFOQCCGU-UHFFFAOYSA-N1inactive--inactive
UJLAWZDWDVHWOW-DGCLKSJQSA-N1inactive--inactive
CrizotinibKTEIFNKAUNYNJU-GFCCVEGCSA-N1inactive--inactive
DasatinibZBNZXTGUTAYRHI-UHFFFAOYSA-N1inactive--inactive
ErlotinibAAKJLRGGTJKAMG-UHFFFAOYSA-N1inactive--inactive
CXQHYVUVSFXTMY-UHFFFAOYSA-N1inactive--inactive
BIIVYFLTOXDAOV-YVEFUNNKSA-N1active--active
DEZZLWQELQORIU-UHFFFAOYSA-N1inactive--inactive
LHNIIDJUOCFXAP-UHFFFAOYSA-N1inactive--inactive
GefitinibXGALLCVXEZPNRQ-UHFFFAOYSA-N1inactive--inactive
-XWFUWIOJOVXAMS-FXIRQEPWSA-N1inactive--inactive
ZHJGWYRLJUCMRT-QGZVFWFLSA-N1inactive--inactive
KGPGFQWBCSZGEL-ZDUSSCGKSA-N1inactive--inactive
MYQAUKPBNJWPIE-UHFFFAOYSA-N1inactive--inactive
JWNPDZNEKVCWMY-UHFFFAOYSA-N1active--active
ImatinibKTUFNOKKBVMGRW-UHFFFAOYSA-N1inactive--inactive
RuxolitinibHFNKQEVNSGCOJV-OAHLLOKOSA-N1inactive--inactive
-OLESUNNHPSUJLS-UHFFFAOYSA-N1inactive--inactive
SHPFDGWALWEPGS-UHFFFAOYSA-N1inactive--inactive
YYLKKYCXAOBSRM-UHFFFAOYSA-N1active--active
LapatinibBCFGMOOMADDAQU-UHFFFAOYSA-N1inactive--inactive
UUADYKVKJIMIPA-UHFFFAOYSA-N1inactive--inactive
ZCBUQCWBWNUWSU-SFHVURJKSA-N1inactive--inactive
ZNOLRTPMNMPLHY-UHFFFAOYSA-N1inactive--inactive
UXXQOJXBIDBUAC-UHFFFAOYSA-N1inactive--inactive
HHFBDROWDBDFBR-UHFFFAOYSA-N1active--active
NilotinibHHZIURLSWUIHRB-UHFFFAOYSA-N1inactive--inactive
PazopanibCUIHSIWYWATEQL-UHFFFAOYSA-N1inactive--inactive
VAARYSWULJUGST-UHFFFAOYSA-N1inactive--inactive
OYONTEXKYJZFHA-OAQYLSRUSA-N1inactive--inactive
TUVCWJQQGGETHL-UHFFFAOYSA-N1inactive--inactive
BMGQWWVMWDBQGC-PZFYLCKJSA-N1inactive--inactive
YZDJQTHVDDOVHR-UHFFFAOYSA-N1inactive--inactive
-MTICIDWIKCANDD-UHFFFAOYSA-N1inactive--inactive
YCOYDOIWSSHVCK-UHFFFAOYSA-N1inactive--inactive
TamatinibNHHQJBCNYHBUSI-UHFFFAOYSA-N1active--active
JRNJNYBQQYBCLE-UHFFFAOYSA-N1inactive--inactive
CDMGBJANTYXAIV-HHHXNRCGSA-N1inactive--inactive
BCZUAADEACICHN-UHFFFAOYSA-N1inactive--inactive
BosutinibUBPYILGKFZZVDX-UHFFFAOYSA-N1inactive--inactive
SorafenibMLDQJTXFUGDVEO-UHFFFAOYSA-N1inactive--inactive
HKSZLNNOFSGOKW-FYTWVXJKSA-N1active--active
CTNPALGJUAXMMC-PMFHANACSA-N1active--active
SunitinibWINHZLLDWRZWRT-ATVHPVEESA-N1active--active
QQWUGDVOUVUTOY-UHFFFAOYSA-N1inactive--inactive
UJIAQDJKSXQLIT-UHFFFAOYSA-N1inactive--inactive
JOOXLOJCABQBSG-UHFFFAOYSA-N1active--active
VandetanibUHTHHESEBZOYNR-UHFFFAOYSA-N1inactive--inactive
GCIKSSRWRFVXBI-UHFFFAOYSA-N1inactive--inactive
VEPKQEUBKLEPRA-UHFFFAOYSA-N1inactive--inactive
HGVYGHNZFIZVJT-UHFFFAOYSA-N--10inactiveinactive
HHLFERIUOTYKKU-UHFFFAOYSA-N--1inactiveinactive
RJIBTAMXAXHIAN-WAVHTBQISA-N--1inactiveinactive
GTQDKQRZKDDFGV-YPKPFQOOSA-N--1inactiveinactive
HBDSHCUSXQATPO-BGBJRWHRSA-N--1inactiveinactive
VVFCWFGNLTVHBL-CULIEIDSSA-N--1activeactive
QSDUMEKQISKWQM-CULIEIDSSA-N--1activeactive
PKYSCANLQNSBRH-NXGRKYSHSA-N--1activeactive
NSLIISQPJWPBAP-NZYJOVLSSA-N--1inactiveinactive
JGIGRRQUXCRVAK-IVGNLCKYSA-N--1activeactive
ZDXPORXWNAYWMZ-NZYJOVLSSA-N--1activeactive
HRSFSLVREYGRTM-IVGNLCKYSA-N--1activeactive
CZBQLMXEBSGXMK-IVGNLCKYSA-N--1activeactive
FKTPDWVDAWOMKC-UWXFNJGLSA-N--1activeactive
QAKSDJAWBXZYIT-JGPRMFOVSA-N--1inactiveinactive
HNDDKCMMUKHMOJ-NZYJOVLSSA-N--1inactiveinactive
AJRHRTCKQYIHHC-NXGRKYSHSA-N--1inactiveinactive
WXRNDKRLCQNQGX-FYDYZTLLSA-N--1inactiveinactive
ZOGGXBYOGQYIGW-IVGNLCKYSA-N--1inactiveinactive
HNIJOTMYVHYZJU-KMQMGNEHSA-N--1inactiveinactive
YQMFNWQNASFQAE-PLWLMNJCSA-N--1activeactive
FNCKZBZRSNSOLA-DWRRPZAGSA-N--1activeactive
XKQNBVAZAFAZFL-FTCCNZMVSA-N--1activeactive
QVJYGMLAIWRCFT-IHDYSDQQSA-N--1activeactive
UKVQMBJHWHGXOI-YPKPFQOOSA-N--1inactiveinactive
SQVBZWHGFBQRIR-WAVHTBQISA-N--1activeactive
PPOMQCAGVJQMEO-KPKJPENVSA-N--1inactiveinactive
OMUOMODZGKSORV-UVTDQMKNSA-N--1inactiveinactive
HCBULGQMULJTCM-ZSOIEALJSA-N--1inactiveinactive
BAYNHPXTNUSVIZ-ZROIWOOFSA-N--1inactiveinactive
AEPSDRVBEQFMLF-ZROIWOOFSA-N--1inactiveinactive
KNIKQAVPAFENMU-DHDCSXOGSA-N--1inactiveinactive
ATBRARWQWMQOEN-YBEGLDIGSA-N--1inactiveinactive
PABHGTXTQNQAPY-DHDCSXOGSA-N--1inactiveinactive
YHQBGGPEHALTKN-WQLSENKSSA-N--1inactiveinactive
PSVKQCKKLNUATG-UHFFFAOYSA-N--1inactiveinactive
YXPXYQXOOXUZLZ-PXNMLYILSA-N--1inactiveinactive
AOFDQEDHVOKUFO-DHDCSXOGSA-N--1inactiveinactive
NQHUQXMJCCDBSX-PXNMLYILSA-N--1inactiveinactive
QOGATBHPUPKBAD-JYRVWZFOSA-N--1inactiveinactive
CSVRKWMMYHBDKY-NSIKDUERSA-N--1inactiveinactive
XTUZRMCFFDJVLS-NDENLUEZSA-N--1inactiveinactive
XHFUEVVGKXHXPF-YVLHZVERSA-N--1inactiveinactive
FZBSZGXBRMAIPS-YBEGLDIGSA-N--1inactiveinactive
DYVAQTMXYZUFFL-PXNMLYILSA-N--1inactiveinactive
NORFRKRCIQFVJD-ZDLGFXPLSA-N--1activeactive
OBAKMFMBKXLTLJ-PXNMLYILSA-N--1inactiveinactive
NWAHAIOCXQFRPG-PXNMLYILSA-N--1inactiveinactive
IOJLBZJSULGZLY-CHHVJCJISA-N--1activeactive
CUAZFPPQWBQEFF-DHDCSXOGSA-N--1inactiveinactive
XJCSNCIQDUDMHE-YBEGLDIGSA-N--1inactiveinactive
GVKSTKQNQPMUJE-NVMNQCDNSA-N--1inactiveinactive
VYUMGAYDBBSNOO-PXNMLYILSA-N--1inactiveinactive
AUECCDDNJJIIJF-PDGQHHTCSA-N--1inactiveinactive
NOGLEZQEVPFGIZ-MFOYZWKCSA-N--1inactiveinactive
DULXFJCYVHXCMJ-BOPFTXTBSA-N--1inactiveinactive
QVPVIPBBHLHJJU-UHFFFAOYSA-N--1inactiveinactive
IGMWARPFGPVLJG-YVLHZVERSA-N--1inactiveinactive
BYUZPFPHQROZAU-MFOYZWKCSA-N--1activeactive
FDPUZRVMPWKWJI-PXNMLYILSA-N--1inactiveinactive
RGNXWPVNPFAADO-NSIKDUERSA-N--1inactiveinactive
FJYHPGCVLUAPLZ-YBEGLDIGSA-N--1inactiveinactive
MJWLCXWVFUXXNZ-UHFFFAOYSA-N--1activeactive
UWSYIZWDFUFMFV-YPKPFQOOSA-N--1inactiveinactive
WXFDRTZMBRMEOV-PFONDFGASA-N--1inactiveinactive
ANUNRTRKLZJBSN-YPKPFQOOSA-N--1inactiveinactive
OVLIPPSTFCMHMB-DTYMOMKHSA-N--1inactiveinactive
CRDNMYFJWFXOCH-YPKPFQOOSA-N--1inactiveinactive
SJYIDCVIUAFSFM-OWBHPGMISA-N--1inactiveinactive
ZPHLLQOZLTUSKY-SQFISAMPSA-N--1inactiveinactive
DJHRGLWVHIZNHI-PEZBUJJGSA-N--1inactiveinactive
QPWNOSITQGGYFW-OWBHPGMISA-N--1inactiveinactive