O14976 GAK


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Group: Other
Family: NAK
PDB Structure Num: 6
FDA approved drugs from DrugBank: Fostamatinib






structureFDA kinase druginchikeykinase profiling data countkinase profiling labelChEMBL data countChEMBL labelvote label
BPNUQXPIQBZCMR-LJQANCHMSA-N1active--active
WJEOLQLKVOPQFV-UHFFFAOYSA-N1inactive--inactive
MPVGZUGXCQEXTM-UHFFFAOYSA-N1active--active
CVWXJKQAOSCOAB-UHFFFAOYSA-N1inactive--inactive
RITAVMQDGBJQJZ-UHFFFAOYSA-N1active--active
RAHBGWKEPAQNFF-UHFFFAOYSA-N1inactive--inactive
ODPGGGTTYSGTGO-UHFFFAOYSA-N1active--active
OVPNQJVDAFNBDN-UHFFFAOYSA-N1inactive--inactive
QYZOGCMHVIGURT-UHFFFAOYSA-N1inactive--inactive
XXJWYDDUDKYVKI-UHFFFAOYSA-N1active--active
CYOHGALHFOKKQC-UHFFFAOYSA-N1inactive--inactive
XQVVPGYIWAGRNI-QFIPXVFZSA-N1active--active
-FCLPVPNWFDOVKL-DQSJHHFOSA-N1inactive--inactive
ULXXDDBFHOBEHA-INIZCTEOSA-N1active--active
MVCOAUNKQVWQHZ-UHFFFAOYSA-N1inactive--inactive
PSPFQEBFYXJZEV-UHFFFAOYSA-N1inactive--inactive
OUSFTKFNBAZUKL-UHFFFAOYSA-N1active--active
WCWUXEGQKLTGDX-NSHDSACASA-N1inactive--inactive
UIARLYUEJFELEN-FMLDBKJISA-N1active--active
-KCOYQXZDFIIGCY-CZIZESTLSA-N1active--active
YABJJWZLRMPFSI-UHFFFAOYSA-N1inactive--inactive
OMZCMEYTWSXEPZ-UHFFFAOYSA-N1active--active
GFMMXOIFOQCCGU-UHFFFAOYSA-N1inactive--inactive
UJLAWZDWDVHWOW-DGCLKSJQSA-N1inactive--inactive
CrizotinibKTEIFNKAUNYNJU-GFCCVEGCSA-N1inactive--inactive
DasatinibZBNZXTGUTAYRHI-UHFFFAOYSA-N1active--active
ErlotinibAAKJLRGGTJKAMG-UHFFFAOYSA-N1active--active
CXQHYVUVSFXTMY-UHFFFAOYSA-N1inactive--inactive
BIIVYFLTOXDAOV-YVEFUNNKSA-N1active--active
DEZZLWQELQORIU-UHFFFAOYSA-N1inactive--inactive
LHNIIDJUOCFXAP-UHFFFAOYSA-N1active--active
GefitinibXGALLCVXEZPNRQ-UHFFFAOYSA-N1active--active
-XWFUWIOJOVXAMS-FXIRQEPWSA-N1active--active
ZHJGWYRLJUCMRT-QGZVFWFLSA-N1inactive--inactive
KGPGFQWBCSZGEL-ZDUSSCGKSA-N1inactive--inactive
MYQAUKPBNJWPIE-UHFFFAOYSA-N1inactive--inactive
JWNPDZNEKVCWMY-UHFFFAOYSA-N1active--active
ImatinibKTUFNOKKBVMGRW-UHFFFAOYSA-N1active--active
RuxolitinibHFNKQEVNSGCOJV-OAHLLOKOSA-N1active--active
-OLESUNNHPSUJLS-UHFFFAOYSA-N1active--active
SHPFDGWALWEPGS-UHFFFAOYSA-N1active--active
YYLKKYCXAOBSRM-UHFFFAOYSA-N1active--active
LapatinibBCFGMOOMADDAQU-UHFFFAOYSA-N1inactive--inactive
UUADYKVKJIMIPA-UHFFFAOYSA-N1inactive--inactive
ZCBUQCWBWNUWSU-SFHVURJKSA-N1active--active
ZNOLRTPMNMPLHY-UHFFFAOYSA-N1inactive--inactive
UXXQOJXBIDBUAC-UHFFFAOYSA-N1inactive--inactive
HHFBDROWDBDFBR-UHFFFAOYSA-N1inactive--inactive
NilotinibHHZIURLSWUIHRB-UHFFFAOYSA-N1inactive--inactive
PazopanibCUIHSIWYWATEQL-UHFFFAOYSA-N1active--active
VAARYSWULJUGST-UHFFFAOYSA-N1active--active
OYONTEXKYJZFHA-OAQYLSRUSA-N1active--active
TUVCWJQQGGETHL-UHFFFAOYSA-N1inactive--inactive
BMGQWWVMWDBQGC-PZFYLCKJSA-N1active--active
YZDJQTHVDDOVHR-UHFFFAOYSA-N1inactive--inactive
-MTICIDWIKCANDD-UHFFFAOYSA-N1active--active
YCOYDOIWSSHVCK-UHFFFAOYSA-N1inactive--inactive
TamatinibNHHQJBCNYHBUSI-UHFFFAOYSA-N1active--active
JRNJNYBQQYBCLE-UHFFFAOYSA-N1inactive--inactive
CDMGBJANTYXAIV-HHHXNRCGSA-N1active--active
BCZUAADEACICHN-UHFFFAOYSA-N1inactive--inactive
BosutinibUBPYILGKFZZVDX-UHFFFAOYSA-N1active--active
SorafenibMLDQJTXFUGDVEO-UHFFFAOYSA-N1inactive--inactive
HKSZLNNOFSGOKW-FYTWVXJKSA-N1active--active
CTNPALGJUAXMMC-PMFHANACSA-N1active--active
SunitinibWINHZLLDWRZWRT-ATVHPVEESA-N1active--active
QQWUGDVOUVUTOY-UHFFFAOYSA-N1active--active
UJIAQDJKSXQLIT-UHFFFAOYSA-N1active--active
JOOXLOJCABQBSG-UHFFFAOYSA-N1active--active
VandetanibUHTHHESEBZOYNR-UHFFFAOYSA-N1active--active
GCIKSSRWRFVXBI-UHFFFAOYSA-N1inactive--inactive
VEPKQEUBKLEPRA-UHFFFAOYSA-N1inactive--inactive
CDMGBJANTYXAIV-UHFFFAOYSA-N--2activeactive