Q9H2K8 TAO3


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Group: STE
Family: STE20
PDB Structure Num: 1
FDA approved drugs from DrugBank: Fostamatinib






structure FDA kinase druginchikeydata countactive numinactive numsame percentagevote label
BPNUQXPIQBZCMR-LJQANCHMSA-N110100%active
WJEOLQLKVOPQFV-UHFFFAOYSA-N202100%inactive
MPVGZUGXCQEXTM-UHFFFAOYSA-N110100%active
CVWXJKQAOSCOAB-UHFFFAOYSA-N101100%inactive
RITAVMQDGBJQJZ-UHFFFAOYSA-N101100%inactive
RAHBGWKEPAQNFF-UHFFFAOYSA-N101100%inactive
ODPGGGTTYSGTGO-UHFFFAOYSA-N110100%active
OVPNQJVDAFNBDN-UHFFFAOYSA-N110100%active
QYZOGCMHVIGURT-UHFFFAOYSA-N101100%inactive
XXJWYDDUDKYVKI-UHFFFAOYSA-N101100%inactive
CYOHGALHFOKKQC-UHFFFAOYSA-N101100%inactive
XQVVPGYIWAGRNI-QFIPXVFZSA-N110100%active
-FCLPVPNWFDOVKL-DQSJHHFOSA-N101100%inactive
ULXXDDBFHOBEHA-INIZCTEOSA-N101100%inactive
MVCOAUNKQVWQHZ-UHFFFAOYSA-N101100%inactive
PSPFQEBFYXJZEV-UHFFFAOYSA-N101100%inactive
OUSFTKFNBAZUKL-UHFFFAOYSA-N110100%active
WCWUXEGQKLTGDX-NSHDSACASA-N101100%inactive
UIARLYUEJFELEN-FMLDBKJISA-N110100%active
-KCOYQXZDFIIGCY-CZIZESTLSA-N101100%inactive
YABJJWZLRMPFSI-UHFFFAOYSA-N110100%active
OMZCMEYTWSXEPZ-UHFFFAOYSA-N101100%inactive
GFMMXOIFOQCCGU-UHFFFAOYSA-N101100%inactive
UJLAWZDWDVHWOW-DGCLKSJQSA-N101100%inactive
CrizotinibKTEIFNKAUNYNJU-GFCCVEGCSA-N110100%active
DasatinibZBNZXTGUTAYRHI-UHFFFAOYSA-N21150%exclude
ErlotinibAAKJLRGGTJKAMG-UHFFFAOYSA-N202100%inactive
CXQHYVUVSFXTMY-UHFFFAOYSA-N101100%inactive
BIIVYFLTOXDAOV-YVEFUNNKSA-N110100%active
DEZZLWQELQORIU-UHFFFAOYSA-N101100%inactive
LHNIIDJUOCFXAP-UHFFFAOYSA-N101100%inactive
GefitinibXGALLCVXEZPNRQ-UHFFFAOYSA-N202100%inactive
-XWFUWIOJOVXAMS-FXIRQEPWSA-N110100%active
ZHJGWYRLJUCMRT-QGZVFWFLSA-N110100%active
KGPGFQWBCSZGEL-ZDUSSCGKSA-N101100%inactive
MYQAUKPBNJWPIE-UHFFFAOYSA-N303100%inactive
JWNPDZNEKVCWMY-UHFFFAOYSA-N101100%inactive
ImatinibKTUFNOKKBVMGRW-UHFFFAOYSA-N202100%inactive
RuxolitinibHFNKQEVNSGCOJV-OAHLLOKOSA-N110100%active
-OLESUNNHPSUJLS-UHFFFAOYSA-N110100%active
SHPFDGWALWEPGS-UHFFFAOYSA-N101100%inactive
YYLKKYCXAOBSRM-UHFFFAOYSA-N110100%active
LapatinibBCFGMOOMADDAQU-UHFFFAOYSA-N202100%inactive
UUADYKVKJIMIPA-UHFFFAOYSA-N101100%inactive
ZCBUQCWBWNUWSU-SFHVURJKSA-N110100%active
ZNOLRTPMNMPLHY-UHFFFAOYSA-N101100%inactive
UXXQOJXBIDBUAC-UHFFFAOYSA-N202100%inactive
HHFBDROWDBDFBR-UHFFFAOYSA-N101100%inactive
NilotinibHHZIURLSWUIHRB-UHFFFAOYSA-N21150%exclude
PazopanibCUIHSIWYWATEQL-UHFFFAOYSA-N21150%exclude
VAARYSWULJUGST-UHFFFAOYSA-N110100%active
OYONTEXKYJZFHA-OAQYLSRUSA-N110100%active
TUVCWJQQGGETHL-UHFFFAOYSA-N303100%inactive
BMGQWWVMWDBQGC-PZFYLCKJSA-N21150%exclude
YZDJQTHVDDOVHR-UHFFFAOYSA-N101100%inactive
-MTICIDWIKCANDD-UHFFFAOYSA-N110100%active
YCOYDOIWSSHVCK-UHFFFAOYSA-N202100%inactive
TamatinibNHHQJBCNYHBUSI-UHFFFAOYSA-N101100%inactive
JRNJNYBQQYBCLE-UHFFFAOYSA-N110100%active
CDMGBJANTYXAIV-HHHXNRCGSA-N101100%inactive
BCZUAADEACICHN-UHFFFAOYSA-N101100%inactive
BosutinibUBPYILGKFZZVDX-UHFFFAOYSA-N110100%active
SorafenibMLDQJTXFUGDVEO-UHFFFAOYSA-N21150%exclude
HKSZLNNOFSGOKW-FYTWVXJKSA-N110100%active
CTNPALGJUAXMMC-PMFHANACSA-N110100%active
SunitinibWINHZLLDWRZWRT-ATVHPVEESA-N21150%exclude
QQWUGDVOUVUTOY-UHFFFAOYSA-N110100%active
UJIAQDJKSXQLIT-UHFFFAOYSA-N110100%active
JOOXLOJCABQBSG-UHFFFAOYSA-N110100%active
VandetanibUHTHHESEBZOYNR-UHFFFAOYSA-N202100%inactive
GCIKSSRWRFVXBI-UHFFFAOYSA-N21150%exclude
VEPKQEUBKLEPRA-UHFFFAOYSA-N101100%inactive
XRKYMMUGXMWDAO-UHFFFAOYSA-N202100%inactive
HLCDNLNLQNYZTK-NRFANRHFSA-N101100%inactive
ABBADGFSRBWENF-UHFFFAOYSA-N202100%inactive
ZGDACLBJJXLKJY-UHFFFAOYSA-N202100%inactive
NAYRELMNTQSBIN-UHFFFAOYSA-M202100%inactive
HOGVTUZUJGHKPL-WRNXMPKJSA-N101100%inactive
-BIWGYFZAEWGBAL-UHFFFAOYSA-N202100%inactive
SVKSJUIYYCQZEC-UHFFFAOYSA-N202100%inactive
OLUKILHGKRVDCT-UHFFFAOYSA-N202100%inactive
UBLFSMURWWWWMH-UHFFFAOYSA-N202100%inactive
-AYIIQABSVDIZSY-UHFFFAOYSA-N202100%inactive
WVMANZPBOBRWCB-UHFFFAOYSA-N101100%inactive
RAMROQQYRRQPDL-OAHLLOKOSA-N101100%inactive
XHBVYDAKJHETMP-UHFFFAOYSA-N101100%inactive
RDTDWGQDFJPTPD-UHFFFAOYSA-N202100%inactive
RWSVQCBZVPWNFM-UHFFFAOYSA-N220100%active
DOEWDSDBFRHVAP-UHFFFAOYSA-N101100%inactive
WEVYNIUIFUYDGI-UHFFFAOYSA-N202100%inactive
QMGUOJYZJKLOLH-UHFFFAOYSA-N202100%inactive
DQYBRTASHMYDJG-UHFFFAOYSA-N202100%inactive
OPQGFIAVPSXOBO-UHFFFAOYSA-N202100%inactive
YAMAGACQNDAKFB-UHFFFAOYSA-N202100%inactive
QJKBRWSJWQVKLY-UHFFFAOYSA-N101100%inactive
UTBSBSOBZHXMHI-GJZGRUSLSA-N101100%inactive
ARIOBGGRZJITQX-UHFFFAOYSA-N110100%active
DWHVZCLBMTZRQM-UHFFFAOYSA-N101100%inactive
DPDZHVCKYBCJHW-UHFFFAOYSA-N101100%inactive
SVJQCVOKYJWUBC-UHFFFAOYSA-N101100%inactive
NMFKDDRQSNVETB-UHFFFAOYSA-N202100%inactive
KFAKESMKRPNZTM-UHFFFAOYSA-N202100%inactive
HFPLHASLIOXVGS-UHFFFAOYSA-N202100%inactive
BGVLELSCIHASRV-UHFFFAOYSA-N101100%inactive
-VQNCIRRXQQTXEL-UHFFFAOYSA-N101100%inactive
WEEFNMFMNMASJY-UHFFFAOYSA-M202100%inactive
UXGJAOIJSROTTN-UHFFFAOYSA-N202100%inactive
XZEFMZCNXDQXOZ-UHFFFAOYSA-N202100%inactive
YXOXHAUUTIOBDA-UHFFFAOYSA-N202100%inactive
NQVIIUBWMBHLOZ-UHFFFAOYSA-N101100%inactive
XHEQSRJCJTWWAH-UHFFFAOYSA-N101100%inactive
KKTZALUTXUZPSN-UHFFFAOYSA-N202100%inactive
YHKSBKQXCWHTQL-UHFFFAOYSA-N202100%inactive
FALILNHGILFDLC-UHFFFAOYSA-N202100%inactive
ZCNBZFRECRPCKU-UHFFFAOYSA-N202100%inactive
UAKWLVYMKBWHMX-UHFFFAOYSA-N101100%inactive
DNOKYISWMVFYFA-UHFFFAOYSA-N202100%inactive
YOHYSYJDKVYCJI-UHFFFAOYSA-N202100%inactive
DLPSDPPZXRJQOY-UHFFFAOYSA-N202100%inactive
XVECMUKVOMUNLE-UHFFFAOYSA-N202100%inactive
RODAAYVFYDKHGT-AUWJEWJLSA-N101100%inactive
PWUOOJVYZQILBG-UHFFFAOYSA-N202100%inactive
FSPQCTGGIANIJZ-UHFFFAOYSA-N202100%inactive
NIMIWWQLOGNYHD-UHFFFAOYSA-N202100%inactive
FNZTULJDGIXMJJ-UHFFFAOYSA-N202100%inactive
JDSJDASOXWCHPN-UHFFFAOYSA-N202100%inactive
ZRHRPGSSSVYBRG-UHFFFAOYSA-N202100%inactive
YAEMHJKFIIIULI-UHFFFAOYSA-N101100%inactive
-WNWSUJQVZJJGLF-UHFFFAOYSA-N101100%inactive
-MENDIXKFTXYTHJ-DMDINBDXSA-N101100%inactive
ZDEJZKULWCZIHL-UHFFFAOYSA-N101100%inactive
VPVLEBIVXZSOMQ-UHFFFAOYSA-N101100%inactive
JYCUVOXSZBECAY-UHFFFAOYSA-N202100%inactive
LLJJDLHGZUOMQP-UHFFFAOYSA-N202100%inactive
DZQLVVLATXPWBK-UHFFFAOYSA-N202100%inactive
-WXUJAQBSBZLVEV-UHFFFAOYSA-N202100%inactive
GELOGQJVGPIKAM-UHFFFAOYSA-N101100%inactive
NOXXIYDYFSNHDF-UHFFFAOYSA-N202100%inactive
-MCAHMSDENAOJFZ-SCUXEZOQSA-N101100%inactive
JBJYTZXCZDNOJW-UHFFFAOYSA-N202100%inactive
SAYGKHKXGCPTLX-UHFFFAOYSA-N202100%inactive
-RKUMZEVCWKZXFV-YOCZKUTFSA-N101100%inactive
-LDEWQRSYYHTQRA-UHFFFAOYSA-N101100%inactive
YBLWOZUPHDKFOT-UHFFFAOYSA-N202100%inactive
QTCFYQHZJIIHBS-UHFFFAOYSA-N202100%inactive
VNDWQCSOSCCWIP-UHFFFAOYSA-N202100%inactive
CBIAKDAYHRWZCU-UHFFFAOYSA-N202100%inactive
ACPOUJIDANTYHO-UHFFFAOYSA-N101100%inactive
NJTUORMLOPXPBY-UHFFFAOYSA-N202100%inactive
ODZGYELAMAOARP-UHFFFAOYSA-N101100%inactive
ZUDPNBZMAJGYTE-UHFFFAOYSA-N110100%active
AVLYNJZZQYEFEA-UHFFFAOYSA-N101100%inactive
KQMPRSZTUSSXND-UHFFFAOYSA-N202100%inactive
ZXVUBPLDUMSDOE-UHFFFAOYSA-N101100%inactive
KOZFSFOOLUUIGY-IYYJOCMQSA-N220100%active
QQUXFYAWXPMDOE-UHFFFAOYSA-N202100%inactive
-BLLBARDQJSOSJD-PGUFJCEWSA-N101100%inactive
LLLQTDSSHZREGW-UHFFFAOYSA-N101100%inactive
FMETVQKSDIOGPX-UHFFFAOYSA-N202100%inactive
CZQHHVNHHHRRDU-UHFFFAOYSA-N202100%inactive
NGAGMBNBKCDCDJ-UHFFFAOYSA-N202100%inactive
-NHBMKTBZZSJUGA-HKRCYGBASA-N101100%inactive
GYQSWJNGTWVFOL-UHFFFAOYSA-N101100%inactive
JLOXTZFYJNCPIS-UHFFFAOYSA-N101100%inactive
FPYJSJDOHRDAMT-UHFFFAOYSA-N101100%inactive
UQPMANVRZYYQMD-UHFFFAOYSA-N101100%inactive
ODYAQBDIXCVKAE-UHFFFAOYSA-N202100%inactive
IBAKVEUZKHOWNG-UHFFFAOYSA-N101100%inactive
VXPWQNBKEIVYIS-OAHLLOKOSA-N101100%inactive
DZFBYHUKZSRPHU-UHFFFAOYSA-N202100%inactive
QFWCYNPOPKQOKV-UHFFFAOYSA-N202100%inactive
BGIYKDUASORTBB-UHFFFAOYSA-N202100%inactive
KFHMLBXBRCITHF-UHFFFAOYSA-N202100%inactive
WUPUZEMRHDROEO-UHFFFAOYSA-N202100%inactive
CZDUJGOCEPWCNA-UHFFFAOYSA-N202100%inactive
INTPTKHSGKBHHW-UHFFFAOYSA-N202100%inactive
ZDNURMVOKAERHZ-UHFFFAOYSA-N202100%inactive
PEPCXHNLEXQQSE-UHFFFAOYSA-N202100%inactive
-DGCXNBUJPWPMJJ-UHFFFAOYSA-N101100%inactive
VFBGXTUGODTSPK-UHFFFAOYSA-N110100%active
ZJFMARHFPUZEKI-UHFFFAOYSA-N101100%inactive
SQWZFLMPDUSYGV-UHFFFAOYSA-N101100%inactive
SRLVNYDXMUGOFI-UHFFFAOYSA-N101100%inactive
KKDPIZPUTYIBFX-UHFFFAOYSA-N202100%inactive
GDQXJQSQYMMKRA-UHFFFAOYSA-N202100%inactive
RONQPWQYDRPRGG-UHFFFAOYSA-N202100%inactive
KIWODJBCHRADND-UHFFFAOYSA-N202100%inactive
PMXCMJLOPOFPBT-OAHLLOKOSA-N101100%inactive
-QFJCIRLUMZQUOT-JRLVRMFHSA-N101100%inactive
LLJRXVHJOJRCSM-UHFFFAOYSA-N202100%inactive
CMKMGFAUKPAOMG-AWEZNQCLSA-N101100%inactive
FXGHOAZJQNLNFD-KRWDZBQOSA-N101100%inactive
-XFXDYDZBKXMGBX-HOTGVXAUSA-N101100%inactive
-NJNKPVPFGLGHPA-UHFFFAOYSA-N101100%inactive
CDMGBJANTYXAIV-MHZLTWQESA-N101100%inactive
VSPFURGQAYMVAN-UHFFFAOYSA-N202100%inactive
OTPNDVKVEAIXTI-IYBDPMFKSA-N110100%active
BHWCZLOXTLWZAQ-UHFFFAOYSA-N202100%inactive
YOELZIQOLWZLQC-UHFFFAOYSA-N202100%inactive
ZFGXZJKLOFCECI-UHFFFAOYSA-N101100%inactive
DMWVGXGXHPOEPT-UHFFFAOYSA-N202100%inactive
HKSZLNNOFSGOKW-HMWZOHBLSA-N220100%active
WNRSTFUVBWNELX-UHFFFAOYSA-N101100%inactive
LOGJQOUIVKBFGH-UHFFFAOYSA-N101100%inactive
QNUKRWAIZMBVCU-UHFFFAOYSA-N110100%active
XPLJEFSRINKZLC-UHFFFAOYSA-N110100%active
MLKHXLFEYOOYEY-UHFFFAOYSA-N101100%inactive
LCACSMNPIITJGG-UHFFFAOYSA-N202100%inactive
KFLWBZPSJQPRDD-UHFFFAOYSA-N101100%inactive
NMEUKWOOQOHUNA-UHFFFAOYSA-N101100%inactive
IBCXZJCWDGCXQT-UHFFFAOYSA-N202100%inactive
BTUOOXPZOVNPMF-UHFFFAOYSA-N202100%inactive
UOHFCPXBKJPCAD-UHFFFAOYSA-N202100%inactive
TUCIOBMMDDOEMM-UHFFFAOYSA-N101100%inactive
DXVJRTIPBNBLLB-UHFFFAOYSA-N101100%inactive
FQNCLVJEQCJWSU-UHFFFAOYSA-N202100%inactive
QNOXYUNHIGOWNY-UHFFFAOYSA-N202100%inactive
GFNNBHLJANVSQV-UHFFFAOYSA-N202100%inactive
PMUJUSJUVIXDQC-UHFFFAOYSA-N101100%inactive
GGPZCOONYBPZEW-UHFFFAOYSA-N202100%inactive
-YUWFTONEHHSMEI-CZUORRHYSA-N101100%inactive
RFHPWPWVGFSLOP-UHFFFAOYSA-N101100%inactive
WUWDLXZGHZSWQZ-UHFFFAOYSA-N101100%inactive
HBWLNACPIFKNIP-UHFFFAOYSA-N202100%inactive
-QDLHCMPXEPAAMD-BLNDMVMCSA-N101100%inactive
-BLQHLDXMMWHXIT-YSZXOBSOSA-N101100%inactive
-AXPBLFXFGVEGKU-UHFFFAOYSA-N101100%inactive
PIQCTGMSNWUMAF-UHFFFAOYSA-N101100%inactive
ZTFBIUXIQYRUNT-MDWZMJQESA-N101100%inactive
BTIHMVBBUGXLCJ-OAHLLOKOSA-N101100%inactive
UJLAWZDWDVHWOW-AAEUAGOBSA-N101100%inactive
FYSRKRZDBHOFAY-UHFFFAOYSA-N101100%inactive
MLKHXLFEYOOYEY-NVNXTCNLSA-N101100%inactive
PMUJUSJUVIXDQC-LCYFTJDESA-N101100%inactive
KFLWBZPSJQPRDD-ONEGZZNKSA-N101100%inactive
HOGVTUZUJGHKPL-UHFFFAOYSA-N101100%inactive
QFJCIRLUMZQUOT-MTKXUJSSSA-N101100%inactive
RFHPWPWVGFSLOP-ZROIWOOFSA-N101100%inactive
VWVYILCFSYNJHF-UHFFFAOYSA-N110100%active
ZUDPNBZMAJGYTE-HYMQDMCPSA-N110100%active
WUWDLXZGHZSWQZ-WQLSENKSSA-N101100%inactive
DPANHMGWPXVBQI-UHFFFAOYSA-N101100%inactive
VFBGXTUGODTSPK-BAQGIRSFSA-N110100%active
NFDQHCCABRRTFB-XJCLVHIMSA-N101100%inactive
TUCIOBMMDDOEMM-RIYZIHGNSA-N101100%inactive
IMYVCWQAHSYYOO-UHFFFAOYSA-N101100%inactive
ZJFMARHFPUZEKI-KMKOMSMNSA-N101100%inactive
BMGQWWVMWDBQGC-UHFFFAOYSA-N110100%active
DXVJRTIPBNBLLB-BJMVGYQFSA-N101100%inactive
UAKWLVYMKBWHMX-RVDMUPIBSA-N101100%inactive
MCAHMSDENAOJFZ-NDSMKMDISA-N101100%inactive
SQWZFLMPDUSYGV-POHAHGRESA-N101100%inactive
FPYJSJDOHRDAMT-KQWNVCNZSA-N110100%active
SRLVNYDXMUGOFI-YWEYNIOJSA-N101100%inactive
XPLJEFSRINKZLC-ATVHPVEESA-N101100%inactive
BLLBARDQJSOSJD-UHFFFAOYSA-N101100%inactive
BLQHLDXMMWHXIT-UYRCGDKNSA-N101100%inactive
LOGJQOUIVKBFGH-YBEGLDIGSA-N101100%inactive
VXPWQNBKEIVYIS-UHFFFAOYSA-N101100%inactive
CDMGBJANTYXAIV-UHFFFAOYSA-N101100%inactive
-HBDSHCUSXQATPO-BGBJRWHRSA-N101100%inactive
HLCDNLNLQNYZTK-UHFFFAOYSA-N101100%inactive
DOEWDSDBFRHVAP-KRXBUXKQSA-N101100%inactive
QMBDONCHHMIWFJ-UHFFFAOYSA-N101100%inactive
OTPNDVKVEAIXTI-UHFFFAOYSA-N101100%inactive
BGVLELSCIHASRV-QPEQYQDCSA-N101100%inactive
QJKBRWSJWQVKLY-UKTHLTGXSA-N101100%inactive
LLLQTDSSHZREGW-AATRIKPKSA-N101100%inactive
UTBSBSOBZHXMHI-LSDHHAIUSA-N101100%inactive
NHBMKTBZZSJUGA-HEHNFIMWSA-N101100%inactive
PMXCMJLOPOFPBT-UHFFFAOYSA-N101100%inactive
ZDRVLAOYDGQLFI-UHFFFAOYSA-N101100%inactive