Q13164 Erk5


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Group: CMGC
Family: MAPK
PDB Structure Num: 7
FDA approved drugs from DrugBank: Fostamatinib






structure FDA kinase druginchikeydata countactive numinactive numsame percentagevote label
BPNUQXPIQBZCMR-LJQANCHMSA-N101100%inactive
WJEOLQLKVOPQFV-UHFFFAOYSA-N101100%inactive
MPVGZUGXCQEXTM-UHFFFAOYSA-N101100%inactive
CVWXJKQAOSCOAB-UHFFFAOYSA-N101100%inactive
RITAVMQDGBJQJZ-UHFFFAOYSA-N101100%inactive
RAHBGWKEPAQNFF-UHFFFAOYSA-N101100%inactive
ODPGGGTTYSGTGO-UHFFFAOYSA-N101100%inactive
OVPNQJVDAFNBDN-UHFFFAOYSA-N110100%active
QYZOGCMHVIGURT-UHFFFAOYSA-N101100%inactive
XXJWYDDUDKYVKI-UHFFFAOYSA-N101100%inactive
CYOHGALHFOKKQC-UHFFFAOYSA-N101100%inactive
XQVVPGYIWAGRNI-QFIPXVFZSA-N101100%inactive
-FCLPVPNWFDOVKL-DQSJHHFOSA-N110100%active
ULXXDDBFHOBEHA-INIZCTEOSA-N101100%inactive
MVCOAUNKQVWQHZ-UHFFFAOYSA-N101100%inactive
PSPFQEBFYXJZEV-UHFFFAOYSA-N110100%active
OUSFTKFNBAZUKL-UHFFFAOYSA-N110100%active
WCWUXEGQKLTGDX-NSHDSACASA-N101100%inactive
UIARLYUEJFELEN-FMLDBKJISA-N110100%active
-KCOYQXZDFIIGCY-CZIZESTLSA-N101100%inactive
YABJJWZLRMPFSI-UHFFFAOYSA-N101100%inactive
OMZCMEYTWSXEPZ-UHFFFAOYSA-N101100%inactive
GFMMXOIFOQCCGU-UHFFFAOYSA-N101100%inactive
UJLAWZDWDVHWOW-DGCLKSJQSA-N101100%inactive
CrizotinibKTEIFNKAUNYNJU-GFCCVEGCSA-N110100%active
DasatinibZBNZXTGUTAYRHI-UHFFFAOYSA-N101100%inactive
ErlotinibAAKJLRGGTJKAMG-UHFFFAOYSA-N101100%inactive
CXQHYVUVSFXTMY-UHFFFAOYSA-N101100%inactive
BIIVYFLTOXDAOV-YVEFUNNKSA-N110100%active
DEZZLWQELQORIU-UHFFFAOYSA-N101100%inactive
LHNIIDJUOCFXAP-UHFFFAOYSA-N101100%inactive
GefitinibXGALLCVXEZPNRQ-UHFFFAOYSA-N101100%inactive
-XWFUWIOJOVXAMS-FXIRQEPWSA-N101100%inactive
ZHJGWYRLJUCMRT-QGZVFWFLSA-N101100%inactive
KGPGFQWBCSZGEL-ZDUSSCGKSA-N101100%inactive
MYQAUKPBNJWPIE-UHFFFAOYSA-N101100%inactive
JWNPDZNEKVCWMY-UHFFFAOYSA-N101100%inactive
ImatinibKTUFNOKKBVMGRW-UHFFFAOYSA-N101100%inactive
RuxolitinibHFNKQEVNSGCOJV-OAHLLOKOSA-N101100%inactive
-OLESUNNHPSUJLS-UHFFFAOYSA-N101100%inactive
SHPFDGWALWEPGS-UHFFFAOYSA-N101100%inactive
YYLKKYCXAOBSRM-UHFFFAOYSA-N110100%active
LapatinibBCFGMOOMADDAQU-UHFFFAOYSA-N101100%inactive
UUADYKVKJIMIPA-UHFFFAOYSA-N101100%inactive
ZCBUQCWBWNUWSU-SFHVURJKSA-N101100%inactive
ZNOLRTPMNMPLHY-UHFFFAOYSA-N101100%inactive
UXXQOJXBIDBUAC-UHFFFAOYSA-N101100%inactive
HHFBDROWDBDFBR-UHFFFAOYSA-N101100%inactive
NilotinibHHZIURLSWUIHRB-UHFFFAOYSA-N101100%inactive
PazopanibCUIHSIWYWATEQL-UHFFFAOYSA-N101100%inactive
VAARYSWULJUGST-UHFFFAOYSA-N101100%inactive
OYONTEXKYJZFHA-OAQYLSRUSA-N110100%active
TUVCWJQQGGETHL-UHFFFAOYSA-N101100%inactive
BMGQWWVMWDBQGC-PZFYLCKJSA-N101100%inactive
YZDJQTHVDDOVHR-UHFFFAOYSA-N101100%inactive
-MTICIDWIKCANDD-UHFFFAOYSA-N101100%inactive
YCOYDOIWSSHVCK-UHFFFAOYSA-N101100%inactive
TamatinibNHHQJBCNYHBUSI-UHFFFAOYSA-N101100%inactive
JRNJNYBQQYBCLE-UHFFFAOYSA-N110100%active
CDMGBJANTYXAIV-HHHXNRCGSA-N101100%inactive
BCZUAADEACICHN-UHFFFAOYSA-N101100%inactive
BosutinibUBPYILGKFZZVDX-UHFFFAOYSA-N110100%active
SorafenibMLDQJTXFUGDVEO-UHFFFAOYSA-N101100%inactive
HKSZLNNOFSGOKW-FYTWVXJKSA-N110100%active
CTNPALGJUAXMMC-PMFHANACSA-N101100%inactive
SunitinibWINHZLLDWRZWRT-ATVHPVEESA-N101100%inactive
QQWUGDVOUVUTOY-UHFFFAOYSA-N110100%active
UJIAQDJKSXQLIT-UHFFFAOYSA-N101100%inactive
JOOXLOJCABQBSG-UHFFFAOYSA-N110100%active
VandetanibUHTHHESEBZOYNR-UHFFFAOYSA-N101100%inactive
GCIKSSRWRFVXBI-UHFFFAOYSA-N101100%inactive
VEPKQEUBKLEPRA-UHFFFAOYSA-N101100%inactive