P42345 FRAP


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Group: Atypical
Family: PIKK
PDB Structure Num: 0
FDA approved drugs from DrugBank: Everolimus Fostamatinib Sirolimus Temsirolimus






structure FDA kinase druginchikeydata countactive numinactive numsame percentagevote label
BPNUQXPIQBZCMR-LJQANCHMSA-N101100%inactive
WJEOLQLKVOPQFV-UHFFFAOYSA-N101100%inactive
MPVGZUGXCQEXTM-UHFFFAOYSA-N101100%inactive
CVWXJKQAOSCOAB-UHFFFAOYSA-N101100%inactive
RITAVMQDGBJQJZ-UHFFFAOYSA-N101100%inactive
RAHBGWKEPAQNFF-UHFFFAOYSA-N101100%inactive
ODPGGGTTYSGTGO-UHFFFAOYSA-N101100%inactive
OVPNQJVDAFNBDN-UHFFFAOYSA-N101100%inactive
QYZOGCMHVIGURT-UHFFFAOYSA-N101100%inactive
XXJWYDDUDKYVKI-UHFFFAOYSA-N101100%inactive
CYOHGALHFOKKQC-UHFFFAOYSA-N101100%inactive
XQVVPGYIWAGRNI-QFIPXVFZSA-N101100%inactive
-FCLPVPNWFDOVKL-DQSJHHFOSA-N101100%inactive
ULXXDDBFHOBEHA-INIZCTEOSA-N101100%inactive
MVCOAUNKQVWQHZ-UHFFFAOYSA-N101100%inactive
PSPFQEBFYXJZEV-UHFFFAOYSA-N101100%inactive
OUSFTKFNBAZUKL-UHFFFAOYSA-N101100%inactive
WCWUXEGQKLTGDX-NSHDSACASA-N101100%inactive
UIARLYUEJFELEN-FMLDBKJISA-N101100%inactive
-KCOYQXZDFIIGCY-CZIZESTLSA-N101100%inactive
YABJJWZLRMPFSI-UHFFFAOYSA-N101100%inactive
OMZCMEYTWSXEPZ-UHFFFAOYSA-N101100%inactive
GFMMXOIFOQCCGU-UHFFFAOYSA-N101100%inactive
UJLAWZDWDVHWOW-DGCLKSJQSA-N101100%inactive
CrizotinibKTEIFNKAUNYNJU-GFCCVEGCSA-N101100%inactive
DasatinibZBNZXTGUTAYRHI-UHFFFAOYSA-N101100%inactive
ErlotinibAAKJLRGGTJKAMG-UHFFFAOYSA-N101100%inactive
CXQHYVUVSFXTMY-UHFFFAOYSA-N101100%inactive
BIIVYFLTOXDAOV-YVEFUNNKSA-N101100%inactive
DEZZLWQELQORIU-UHFFFAOYSA-N101100%inactive
LHNIIDJUOCFXAP-UHFFFAOYSA-N110100%active
GefitinibXGALLCVXEZPNRQ-UHFFFAOYSA-N101100%inactive
-XWFUWIOJOVXAMS-FXIRQEPWSA-N101100%inactive
ZHJGWYRLJUCMRT-QGZVFWFLSA-N101100%inactive
KGPGFQWBCSZGEL-ZDUSSCGKSA-N101100%inactive
MYQAUKPBNJWPIE-UHFFFAOYSA-N202100%inactive
JWNPDZNEKVCWMY-UHFFFAOYSA-N101100%inactive
ImatinibKTUFNOKKBVMGRW-UHFFFAOYSA-N101100%inactive
RuxolitinibHFNKQEVNSGCOJV-OAHLLOKOSA-N101100%inactive
-OLESUNNHPSUJLS-UHFFFAOYSA-N101100%inactive
SHPFDGWALWEPGS-UHFFFAOYSA-N101100%inactive
YYLKKYCXAOBSRM-UHFFFAOYSA-N101100%inactive
LapatinibBCFGMOOMADDAQU-UHFFFAOYSA-N101100%inactive
UUADYKVKJIMIPA-UHFFFAOYSA-N101100%inactive
ZCBUQCWBWNUWSU-SFHVURJKSA-N101100%inactive
ZNOLRTPMNMPLHY-UHFFFAOYSA-N101100%inactive
UXXQOJXBIDBUAC-UHFFFAOYSA-N101100%inactive
HHFBDROWDBDFBR-UHFFFAOYSA-N101100%inactive
NilotinibHHZIURLSWUIHRB-UHFFFAOYSA-N101100%inactive
PazopanibCUIHSIWYWATEQL-UHFFFAOYSA-N101100%inactive
VAARYSWULJUGST-UHFFFAOYSA-N101100%inactive
OYONTEXKYJZFHA-OAQYLSRUSA-N101100%inactive
TUVCWJQQGGETHL-UHFFFAOYSA-N220100%active
BMGQWWVMWDBQGC-PZFYLCKJSA-N101100%inactive
YZDJQTHVDDOVHR-UHFFFAOYSA-N101100%inactive
-MTICIDWIKCANDD-UHFFFAOYSA-N110100%active
YCOYDOIWSSHVCK-UHFFFAOYSA-N101100%inactive
TamatinibNHHQJBCNYHBUSI-UHFFFAOYSA-N101100%inactive
JRNJNYBQQYBCLE-UHFFFAOYSA-N101100%inactive
CDMGBJANTYXAIV-HHHXNRCGSA-N101100%inactive
BCZUAADEACICHN-UHFFFAOYSA-N101100%inactive
BosutinibUBPYILGKFZZVDX-UHFFFAOYSA-N101100%inactive
SorafenibMLDQJTXFUGDVEO-UHFFFAOYSA-N101100%inactive
HKSZLNNOFSGOKW-FYTWVXJKSA-N101100%inactive
CTNPALGJUAXMMC-PMFHANACSA-N101100%inactive
SunitinibWINHZLLDWRZWRT-ATVHPVEESA-N101100%inactive
QQWUGDVOUVUTOY-UHFFFAOYSA-N101100%inactive
UJIAQDJKSXQLIT-UHFFFAOYSA-N110100%active
JOOXLOJCABQBSG-UHFFFAOYSA-N101100%inactive
VandetanibUHTHHESEBZOYNR-UHFFFAOYSA-N101100%inactive
GCIKSSRWRFVXBI-UHFFFAOYSA-N101100%inactive
VEPKQEUBKLEPRA-UHFFFAOYSA-N101100%inactive
ABBADGFSRBWENF-UHFFFAOYSA-N101100%inactive
DQYBRTASHMYDJG-UHFFFAOYSA-N101100%inactive
YOHYSYJDKVYCJI-UHFFFAOYSA-N101100%inactive
YBLWOZUPHDKFOT-UHFFFAOYSA-N101100%inactive
KFHMLBXBRCITHF-UHFFFAOYSA-N101100%inactive
KKDPIZPUTYIBFX-UHFFFAOYSA-N101100%inactive
MLKHXLFEYOOYEY-NVNXTCNLSA-N101100%inactive
GFNNBHLJANVSQV-UHFFFAOYSA-N101100%inactive
ZGDACLBJJXLKJY-UHFFFAOYSA-N101100%inactive
YAMAGACQNDAKFB-UHFFFAOYSA-N101100%inactive
DLPSDPPZXRJQOY-UHFFFAOYSA-N101100%inactive
QTCFYQHZJIIHBS-UHFFFAOYSA-N101100%inactive
WUPUZEMRHDROEO-UHFFFAOYSA-N101100%inactive
GDQXJQSQYMMKRA-UHFFFAOYSA-N101100%inactive
LCACSMNPIITJGG-UHFFFAOYSA-N101100%inactive
PMUJUSJUVIXDQC-LCYFTJDESA-N101100%inactive
NAYRELMNTQSBIN-UHFFFAOYSA-M101100%inactive
WEEFNMFMNMASJY-UHFFFAOYSA-M101100%inactive
FSPQCTGGIANIJZ-UHFFFAOYSA-N101100%inactive
VNDWQCSOSCCWIP-UHFFFAOYSA-N101100%inactive
CZDUJGOCEPWCNA-UHFFFAOYSA-N101100%inactive
RONQPWQYDRPRGG-UHFFFAOYSA-N101100%inactive
KFLWBZPSJQPRDD-ONEGZZNKSA-N101100%inactive
GGPZCOONYBPZEW-UHFFFAOYSA-N101100%inactive
HOGVTUZUJGHKPL-UHFFFAOYSA-N101100%inactive
YXOXHAUUTIOBDA-UHFFFAOYSA-N101100%inactive
NIMIWWQLOGNYHD-UHFFFAOYSA-N101100%inactive
CBIAKDAYHRWZCU-UHFFFAOYSA-N101100%inactive
INTPTKHSGKBHHW-UHFFFAOYSA-N101100%inactive
KIWODJBCHRADND-UHFFFAOYSA-N101100%inactive
IBCXZJCWDGCXQT-UHFFFAOYSA-N101100%inactive
-BIWGYFZAEWGBAL-UHFFFAOYSA-N101100%inactive
KKTZALUTXUZPSN-UHFFFAOYSA-N101100%inactive
NJTUORMLOPXPBY-UHFFFAOYSA-N101100%inactive
ZDNURMVOKAERHZ-UHFFFAOYSA-N101100%inactive
QFJCIRLUMZQUOT-MTKXUJSSSA-N101100%inactive
BTUOOXPZOVNPMF-UHFFFAOYSA-N101100%inactive
RFHPWPWVGFSLOP-ZROIWOOFSA-N101100%inactive
SVKSJUIYYCQZEC-UHFFFAOYSA-N101100%inactive
YHKSBKQXCWHTQL-UHFFFAOYSA-N101100%inactive
VWVYILCFSYNJHF-UHFFFAOYSA-N101100%inactive
ZUDPNBZMAJGYTE-HYMQDMCPSA-N101100%inactive
PEPCXHNLEXQQSE-UHFFFAOYSA-N101100%inactive
LLJRXVHJOJRCSM-UHFFFAOYSA-N101100%inactive
UOHFCPXBKJPCAD-UHFFFAOYSA-N101100%inactive
WUWDLXZGHZSWQZ-WQLSENKSSA-N101100%inactive
DPANHMGWPXVBQI-UHFFFAOYSA-N101100%inactive
LLJJDLHGZUOMQP-UHFFFAOYSA-N101100%inactive
FMETVQKSDIOGPX-UHFFFAOYSA-N101100%inactive
VFBGXTUGODTSPK-BAQGIRSFSA-N101100%inactive
NFDQHCCABRRTFB-XJCLVHIMSA-N101100%inactive
TUCIOBMMDDOEMM-RIYZIHGNSA-N101100%inactive
HBWLNACPIFKNIP-UHFFFAOYSA-N101100%inactive
IMYVCWQAHSYYOO-UHFFFAOYSA-N101100%inactive
ZCNBZFRECRPCKU-UHFFFAOYSA-N101100%inactive
DZQLVVLATXPWBK-UHFFFAOYSA-N101100%inactive
CZQHHVNHHHRRDU-UHFFFAOYSA-N110100%active
ZJFMARHFPUZEKI-KMKOMSMNSA-N101100%inactive
BMGQWWVMWDBQGC-UHFFFAOYSA-N101100%inactive
DXVJRTIPBNBLLB-BJMVGYQFSA-N101100%inactive
FALILNHGILFDLC-UHFFFAOYSA-N101100%inactive
WEVYNIUIFUYDGI-UHFFFAOYSA-N101100%inactive
UAKWLVYMKBWHMX-RVDMUPIBSA-N101100%inactive
MCAHMSDENAOJFZ-NDSMKMDISA-N101100%inactive
NGAGMBNBKCDCDJ-UHFFFAOYSA-N101100%inactive
SQWZFLMPDUSYGV-POHAHGRESA-N110100%active
DMWVGXGXHPOEPT-UHFFFAOYSA-N101100%inactive
FQNCLVJEQCJWSU-UHFFFAOYSA-N101100%inactive
RDTDWGQDFJPTPD-UHFFFAOYSA-N101100%inactive
QMGUOJYZJKLOLH-UHFFFAOYSA-N101100%inactive
DNOKYISWMVFYFA-UHFFFAOYSA-N101100%inactive
FNZTULJDGIXMJJ-UHFFFAOYSA-N101100%inactive
FPYJSJDOHRDAMT-KQWNVCNZSA-N101100%inactive
SRLVNYDXMUGOFI-YWEYNIOJSA-N101100%inactive
XPLJEFSRINKZLC-ATVHPVEESA-N101100%inactive
QNOXYUNHIGOWNY-UHFFFAOYSA-N101100%inactive
HKSZLNNOFSGOKW-HMWZOHBLSA-N101100%inactive
BLLBARDQJSOSJD-UHFFFAOYSA-N101100%inactive
RWSVQCBZVPWNFM-UHFFFAOYSA-N101100%inactive
NMFKDDRQSNVETB-UHFFFAOYSA-N101100%inactive
BLQHLDXMMWHXIT-UYRCGDKNSA-N101100%inactive
LOGJQOUIVKBFGH-YBEGLDIGSA-N101100%inactive
ODYAQBDIXCVKAE-UHFFFAOYSA-N101100%inactive
VXPWQNBKEIVYIS-UHFFFAOYSA-N101100%inactive
CDMGBJANTYXAIV-UHFFFAOYSA-N101100%inactive
XRKYMMUGXMWDAO-UHFFFAOYSA-N101100%inactive
-HBDSHCUSXQATPO-BGBJRWHRSA-N101100%inactive
KFAKESMKRPNZTM-UHFFFAOYSA-N101100%inactive
XVECMUKVOMUNLE-UHFFFAOYSA-N101100%inactive
JYCUVOXSZBECAY-UHFFFAOYSA-N101100%inactive
KQMPRSZTUSSXND-UHFFFAOYSA-N101100%inactive
DZFBYHUKZSRPHU-UHFFFAOYSA-N101100%inactive
NOXXIYDYFSNHDF-UHFFFAOYSA-N101100%inactive
HLCDNLNLQNYZTK-UHFFFAOYSA-N101100%inactive
DOEWDSDBFRHVAP-KRXBUXKQSA-N101100%inactive
HFPLHASLIOXVGS-UHFFFAOYSA-N101100%inactive
QMBDONCHHMIWFJ-UHFFFAOYSA-N101100%inactive
-WXUJAQBSBZLVEV-UHFFFAOYSA-N101100%inactive
KOZFSFOOLUUIGY-IYYJOCMQSA-N101100%inactive
QFWCYNPOPKQOKV-UHFFFAOYSA-N101100%inactive
OTPNDVKVEAIXTI-UHFFFAOYSA-N101100%inactive
OLUKILHGKRVDCT-UHFFFAOYSA-N101100%inactive
OPQGFIAVPSXOBO-UHFFFAOYSA-N101100%inactive
BGVLELSCIHASRV-QPEQYQDCSA-N101100%inactive
PWUOOJVYZQILBG-UHFFFAOYSA-N101100%inactive
JBJYTZXCZDNOJW-UHFFFAOYSA-N101100%inactive
QQUXFYAWXPMDOE-UHFFFAOYSA-N101100%inactive
BGIYKDUASORTBB-UHFFFAOYSA-N101100%inactive
BHWCZLOXTLWZAQ-UHFFFAOYSA-N101100%inactive
UBLFSMURWWWWMH-UHFFFAOYSA-N101100%inactive
QJKBRWSJWQVKLY-UKTHLTGXSA-N101100%inactive
UXGJAOIJSROTTN-UHFFFAOYSA-N101100%inactive
JDSJDASOXWCHPN-UHFFFAOYSA-N101100%inactive
SAYGKHKXGCPTLX-UHFFFAOYSA-N101100%inactive
LLLQTDSSHZREGW-AATRIKPKSA-N101100%inactive
VSPFURGQAYMVAN-UHFFFAOYSA-N101100%inactive
YOELZIQOLWZLQC-UHFFFAOYSA-N101100%inactive
-AYIIQABSVDIZSY-UHFFFAOYSA-N101100%inactive
UTBSBSOBZHXMHI-LSDHHAIUSA-N101100%inactive
XZEFMZCNXDQXOZ-UHFFFAOYSA-N101100%inactive
ZRHRPGSSSVYBRG-UHFFFAOYSA-N101100%inactive
NHBMKTBZZSJUGA-HEHNFIMWSA-N101100%inactive
PMXCMJLOPOFPBT-UHFFFAOYSA-N101100%inactive
ZDRVLAOYDGQLFI-UHFFFAOYSA-N101100%inactive